PAOLO GUGLIELMI

Professore associato

email: paolo.guglielmi@uniroma1.it
telefono: 3270054538
edificio: CU019
stanza: 101

Produzione scientifica

11573/1745348 - 2025 - Potential of MAO-B Inhibitors with Multi-Target Inhibition and Antioxidant Properties for the Treatment of Neurodegenerative Disorders

A. Shaldam, Moataz; Carradori, Simone; Melfi, Francesco; Guglielmi, Paolo; Diomede, Francesca; Piattelli, Maurizio; O. Tawfik, Haytham - 01g Articolo di rassegna (Review)

rivista: MINI-REVIEWS IN MEDICINAL CHEMISTRY (Bentham Science Publishers BV:PO Box 7917, Exec Ste Y 26, Saif Zone Sharjah Uae:011 971 6 5571132, EMAIL: benthams@emirates.net.ae, INTERNET: http://www.bentham.org, Fax: 011 971 6 5571134) pp. - - issn: 1389-5575 - wos: WOS:001542776900001 (0) - scopus: 2-s2.0-105012435866 (0)

11573/1745344 - 2025 - In Vitro CO-Releasing and Antioxidant Properties of Sulfonamide-Based CAI-CORMs in a H2O2-Stimulated Human Achilles Tendon-Derived Cell Model

Berrino, Emanuela; Guglielmi, Paolo; Carta, Fabrizio; Carradori, Simone; Campestre, Cristina; Angeli, Andrea; Arrighi, Francesca; Pontecorvi, Virginia; Chimenti, Paola; Secci, Daniela; Supuran, Claudiu T.; Gallorini, Marialucia - 01a Articolo in rivista

rivista: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. - - issn: 1420-3049 - wos: (0) - scopus: (0)

11573/1747259 - 2025 - Copper(I)-Anchoring Covalent Organic Polymer for Heterogeneous CuAAC Reaction without Reducing Agents and Copper Leaching

Guarducci, Maria Aurora; Manetto, Simone; Marrani, Andrea Giacomo; Amato, Francesco; Guglielmi, Paolo; Coluccia, Michele; Fontana, Antonella; Pilato, Serena; Villani, Claudio; Ciogli, Alessia; Mazzoccanti, Giulia - 01a Articolo in rivista

rivista: ACS ORGANIC & INORGANIC AU. (Washington DC: American Chemical Society, 2021-) pp. - - issn: 2694-247X - wos: (0) - scopus: (0)

11573/1745347 - 2025 - Design, synthesis, and biological activity of 2-aroylbenzofuran-3-ols and 2-aroylbenzofuran derivatives: A new route towards hMAO-B inhibition

Guglielmi, Paolo; Coluccia, Michele; Marconi, Guya Diletta; Ortuso, Francesco; Procopio, Francesca; Carradori, Simone; Pizzicannella, Jacopo; Arrighi, Francesca; Troiani, Anna; Salvitti, Chiara; Borges, Fernanda; Chavarria, Daniel; Chimenti, Paola; Secci, Daniela; Diomede, Francesca - 01a Articolo in rivista

rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. - - issn: 0223-5234 - wos: (0) - scopus: (0)

11573/1740080 - 2025 - Design, synthesis, molecular modelling investigation and biological studies of novel human carbonic anhydrase inhibitors based on coumalic acid

Pontecorvi, Virginia; Angeli, Andrea; Cutarella, Luigi; Mori, Mattia; Secci, Daniela; Coluccia, Michele; Carradori, Simone; Troiani, Anna; Pepi, Federico; Salvitti, Chiara; Di Noi, Alessia; Spano, Mattia; Arrighi, Francesca; De Falco, Elena; Bordin, Antonella; Berrino, Emanuela; Granese, Arianna; Chimenti, Paola; Guglielmi, Paolo; Supuran, Claudiu T. - 01a Articolo in rivista

rivista: RSC MEDICINAL CHEMISTRY (Cambridge: Royal Society of Chemistry, 2020-) pp. - - issn: 2632-8682 - wos: WOS:001499069400001 (0) - scopus: (0)

11573/1713144 - 2024 - Chiral hydroxy metabolite of Mebendazole. Analytical and semi-preparative high-performance liquid chromatography resolution and chiroptical properties

Guglielmi, Paolo; Pulitelli, Gaia; Arrighi, Francesca; Secci, Daniela; Pierini, Marco; Cirilli, Roberto - 01a Articolo in rivista

rivista: PHARMACEUTICALS (Basel: MDPI, Molecular Diversity Preservation International, 2004-) pp. 1-16 - issn: 1424-8247 - wos: WOS:001256669100001 (0) - scopus: 2-s2.0-85197600100 (0)

11573/1745342 - 2024 - Azo derivatives of monoterpenes as anti-Helicobacter pylori agents: from synthesis to structure-based target investigation

Melfi, Francesco; Fantacuzzi, Marialuigia; Carradori, Simone; D'agostino, Ilaria; Ammazzalorso, Alessandra; Mencarelli, Noemi; Gallorini, Marialucia; Spano, Mattia; Guglielmi, Paolo; Agamennone, Mariangela; Haji Ali, Sazan; Al-Samydai, Ali; Sisto, Francesca - 01a Articolo in rivista

rivista: RSC MEDICINAL CHEMISTRY (Cambridge: Royal Society of Chemistry, 2020-) pp. 346-366 - issn: 2632-8682 - wos: WOS:001345082800001 (2) - scopus: 2-s2.0-85208755250 (2)

11573/1693719 - 2023 - Novel therapeutic opportunities for Toxoplasma gondii, Trichomonas vaginalis, and Giardia intestinalis infections

Arrighi, Francesca; Granese, Arianna; Chimenti, Paola; Guglielmi, Paolo - 01g Articolo di rassegna (Review)

rivista: EXPERT OPINION ON THERAPEUTIC PATENTS (--London United Kingdom:Informa Healthcare -London, United Kingdom: Ashley Publications Limited) pp. 211-245 - issn: 1354-3776 - wos: WOS:000980206000007 (6) - scopus: 2-s2.0-85152473014 (10)

11573/1705144 - 2023 - A multitarget approach against neuroinflammation. Alkyl substituted coumarins as inhibitors of enzymes involved in neurodegeneration

Berrino, E.; Carradori, S.; Carta, F.; Melfi, F.; Gallorini, M.; Poli, G.; Tuccinardi, T.; Fernandez-Bolanos, J. G.; Lopez, O.; Petzer, J. P.; Petzer, A.; Guglielmi, P.; Secci, D.; Supuran, C. T. - 01a Articolo in rivista

rivista: ANTIOXIDANTS (Basel: MDPI) pp. 1-25 - issn: 2076-3921 - wos: WOS:001137805100001 (12) - scopus: 2-s2.0-85180511315 (13)

11573/1666710 - 2023 - Novel Insights on CAI–CORM hybrids. Evaluation of the CO releasing properties and pain-relieving activity of differently substituted coumarins for the treatment of rheumatoid arthritis

Berrino, Emanuela; Micheli, Laura; Carradori, Simone; Di Cesare Mannelli, Lorenzo; Guglielmi, Paolo; De Luca, Alessandro; Carta, Fabrizio; Ghelardini, Carla; Secci, Daniela; Supuran, Claudiu T. - 01a Articolo in rivista

rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1892-1908 - issn: 0022-2623 - wos: WOS:000925733600001 (13) - scopus: 2-s2.0-85147172354 (14)

11573/1691425 - 2023 - Indoleamine 2,3-dioxygenase

Coluccia, Michele; Secci, Daniela; Guglielmi, Paolo - 02a Capitolo o Articolo

libro: Metalloenzymes: from bench to bedside - (9780128239742)

11573/1738930 - 2023 - Drug design and synthesis of new anticancer agents

Mai, A.; Fioravanti, R.; Rotili, D.; Valente, S.; Zwergel, C.; Secci, D.; Chimenti, P.; Granese, A.; Guglielmi, P.; Silvestri, R.; Coluccia, A.; La Regina, G.; Nalli, M. - 04f Poster

congresso: Highlighting the Research Activity of the Sapienza Faculty of Pharmacy and Medicine (Roma, Italy)

libro: Abstract Book - ()

11573/1693714 - 2023 - Kinetic study on the base-catalyzed imine-enamine tautomerism of a chiral biologically active isoxazoline derivative by HPLC on Amylose Tris(3,5-dimethylphenylcarbamate) chiral stationary phase

Sadutto, Daniele; Guglielmi, Paolo; Carradori, Simone; Secci, Daniela; Cirilli, Roberto - 01a Articolo in rivista

rivista: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. 1-12 - issn: 1420-3049 - wos: WOS:001077830800001 (2) - scopus: 2-s2.0-85172792347 (3)

11573/1659798 - 2022 - Metal-organic frameworks (MOFs) as biomolecules drug delivery systems for anticancer purposes

Coluccia, Michele; Parisse, Valeria; Guglielmi, Paolo; Giannini, Giuseppe; Secci, Daniela - 01g Articolo di rassegna (Review)

11573/1659799 - 2022 - Treatment of Toxoplasmosis: An Insight on Epigenetic Drugs

Guglielmi, P.; Secci, D. - 02a Capitolo o Articolo

libro: Topics in medicinal chemistry - (978-3-031-06849-2; 978-3-031-06850-8)

11573/1659800 - 2022 - An updated patent review on monoamine oxidase (MAO) inhibitors

Guglielmi, Paolo; Carradori, Simone; D'agostino, Ilaria; Campestre, Cristina; Petzer, Jacobus P - 01g Articolo di rassegna (Review)

rivista: EXPERT OPINION ON THERAPEUTIC PATENTS (--London United Kingdom:Informa Healthcare -London, United Kingdom: Ashley Publications Limited) pp. 849-883 - issn: 1354-3776 - wos: WOS:000808508300001 (27) - scopus: 2-s2.0-85131672486 (28)

11573/1691261 - 2022 - Aurone Scaffold and Structural Analogues for the Development of Monoamine Oxidase (MAO) Inhibitors

Guglielmi, Paolo; Pontecorvi, Virginia; Akdemir, Atilla - 02a Capitolo o Articolo

libro: Flavonoids and Phenolics - (978-981-5079-10-4)

11573/1654157 - 2022 - Novel insights on human carbonic anhydrase inhibitors based on coumalic acid. Design, synthesis, molecular modeling investigation, and biological studies

Pontecorvi, Virginia; Mori, Mattia; Picarazzi, Francesca; Zara, Susi; Carradori, Simone; Cataldi, Amelia; Angeli, Andrea; Berrino, Emanuela; Chimenti, Paola; Ciogli, Alessia; Secci, Daniela; Guglielmi, Paolo; Supuran, Claudiu T. - 01a Articolo in rivista

rivista: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (Basel: MDPI Center) pp. 1-26 - issn: 1422-0067 - wos: WOS:000833202300001 (16) - scopus: 2-s2.0-85135137430 (17)

11573/1555649 - 2021 - Dual carbonic anhydrase ix/xii inhibitors and carbon monoxide releasing molecules modulate LPS-mediated inflammation in mouse macrophages

Berrino, E.; Carradori, S.; Angeli, A.; Carta, F.; Supuran, C. T.; Guglielmi, P.; Coletti, C.; Paciotti, R.; Schweikl, H.; Maestrelli, F.; Cerbai, E.; Gallorini, M. - 01a Articolo in rivista

rivista: ANTIOXIDANTS (Basel: MDPI) pp. 1-24 - issn: 2076-3921 - wos: WOS:000611142000001 (24) - scopus: 2-s2.0-85099415600 (27)

11573/1649551 - 2021 - An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods

Mansoldo, F. R. P.; Berrino, E.; Guglielmi, P.; Carradori, S.; Carta, F.; Secci, D.; Supuran, C. T.; Vermelho, A. B. - 01a Articolo in rivista

rivista: SPECTROCHIMICA ACTA. PART A, MOLECULAR AND BIOMOLECULAR SPECTROSCOPY (Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. 0-0 - issn: 1386-1425 - wos: WOS:000786604400018 (2) - scopus: 2-s2.0-85119982751 (3)

11573/1575683 - 2021 - New aspects of monoamine oxidase b inhibitors. The key role of halogens to open the golden door

Mathew, B.; Carradori, S.; Guglielmi, P.; Uddin, Md. S.; Kim, H. - 01g Articolo di rassegna (Review)

rivista: CURRENT MEDICINAL CHEMISTRY (Bentham Science Publishers BV:PO Box 7917, Exec Ste Y 26, Saif Zone Sharjah Uae:011 971 6 5571132, EMAIL: benthams@emirates.net.ae, INTERNET: http://www.bentham.org, Fax: 011 971 6 5571134) pp. 266-283 - issn: 0929-8673 - wos: WOS:000614610600005 (34) - scopus: 2-s2.0-85099155432 (34)

11573/1541961 - 2021 - Synthesis and evaluation of thymol-based synthetic derivatives as dual-action inhibitors against different strains of h. pylori and AGS cell line

Sisto, F.; Carradori, S.; Guglielmi, P.; Spano, M.; Secci, D.; Granese, A.; Sobolev, A. P.; Grande, R.; Campestre, C.; Di Marcantonio, M. C.; Mincione, G. - 01a Articolo in rivista

rivista: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. - - issn: 1420-3049 - wos: WOS:000638744400001 (16) - scopus: 2-s2.0-85103863303 (16)

11573/1325133 - 2020 - High-performance liquid chromatography enantioseparation of chiral 2-(benzylsulfinyl)benzamide derivatives on cellulose tris(3,5-dichlorophenylcarbamate) chiral stationary phase

Carradori, S.; Secci, D.; Guglielmi, P.; Pierini, M.; Cirilli, R. - 01a Articolo in rivista

rivista: JOURNAL OF CHROMATOGRAPHY A ([S.l.] : Elsevier Science) pp. - - issn: 1873-3778 - wos: WOS:000509816200026 (7) - scopus: 2-s2.0-85073049872 (6)

11573/1381665 - 2020 - 1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors

D'ascenzio, M.; Secci, D.; Carradori, S.; Zara, S.; Guglielmi, P.; Cirilli, R.; Pierini, M.; Poli, G.; Tuccinardi, T.; Angeli, A.; Supuran, C. T. - 01a Articolo in rivista

rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington DC : ACS Publications) pp. 2470-2488 - issn: 1520-4804 - wos: WOS:000526403900042 (37) - scopus: 2-s2.0-85081944311 (44)

11573/1541963 - 2020 - Natural compounds and extracts as novel antimicrobial agents

Guglielmi, P.; Pontecorvi, V.; Rotondi, G. - 01g Articolo di rassegna (Review)

rivista: EXPERT OPINION ON THERAPEUTIC PATENTS (--London United Kingdom:Informa Healthcare -London, United Kingdom: Ashley Publications Limited) pp. 949-962 - issn: 1354-3776 - wos: WOS:000598248100007 (51) - scopus: 2-s2.0-85097552965 (57)

11573/1449256 - 2020 - Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation

Guglielmi, P.; Rotondi, G.; Secci, D.; Angeli, A.; Chimenti, P.; Nocentini, A.; Bonardi, A.; Gratteri, P.; Carradori, S.; Supuran, C. T. - 01a Articolo in rivista

rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1891-1905 - issn: 1475-6366 - wos: WOS:000574181700001 (18) - scopus: 2-s2.0-85091861178 (20)

11573/1439431 - 2020 - Chalcones: Unearthing their therapeutic possibility as monoamine oxidase B inhibitors

Guglielmi, Paolo; Mathew, Bijo; Secci, Daniela; Carradori, Simone - 01g Articolo di rassegna (Review)

11573/1439479 - 2020 - Antimalarial agents from medicinal plant and fungal sources

Luisi, Grazia; Carradori, Simone; Grande, Rossella; Secci, Daniela; Guglielmi, Paolo - 02a Capitolo o Articolo

libro: Plant-derived bioactives. Production, properties and therapeutic applications - (978-981-15-1760-0; 978-981-15-1761-7)

11573/1661131 - 2020 - Innovative pH-interfering agents in association with anticancer agents

Secci, D.; Guglielmi, P. - 02a Capitolo o Articolo

libro: pH-Interfering Agents as Chemosensitizers in Cancer Therapy - (9780128207017)

11573/1575689 - 2020 - Synthesis and biological evaluation of carvacrol-based derivatives as dual inhibitors of H. Pylori strains and ags cell proliferation

Sisto, F.; Carradori, S.; Guglielmi, P.; Traversi, C. B.; Spano, M.; Sobolev, A. P.; Secci, D.; Di Marcantonio, M. C.; Haloci, E.; Grande, R.; Mincione, G. - 01a Articolo in rivista

rivista: PHARMACEUTICALS (Basel: MDPI, Molecular Diversity Preservation International, 2004-) pp. 1-21 - issn: 1424-8247 - wos: WOS:000594358000001 (27) - scopus: 2-s2.0-85096612970 (30)

11573/1439461 - 2020 - Synthesis and evaluation of a large library of nitroxoline derivatives as pancreatic cancer antiproliferative agents

Veschi, Serena; Carradori, Simone; De Lellis, Laura; Florio, Rosalba; Brocco, Davide; Secci, Daniela; Guglielmi, Paolo; Spano, Mattia; Sobolev, Anatoly P.; Cama, Alessandro - 01a Articolo in rivista

rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1331-1344 - issn: 1475-6366 - wos: WOS:000545146800001 (11) - scopus: 2-s2.0-85087139219 (11)

11573/1381672 - 2019 - Mechanisms of action of carbonic anhydrase inhibitors: compounds that bind “out of the binding site” and compounds with an unknown mechanism of action

Carradori, Simone; Guglielmi, Paolo - 02a Capitolo o Articolo

libro: Carbonic anhydrases biochemistry and pharmacology of an evergreen pharmaceutical target - (9780128164761)

11573/1349544 - 2019 - Novel approaches to the discovery of selective human monoamine oxidase-B inhibitors: is there room for improvement?

Guglielmi, P.; Carradori, S.; Ammazzalorso, A.; Secci, D. - 01g Articolo di rassegna (Review)

rivista: EXPERT OPINION ON DRUG DISCOVERY (--London United Kingdom:Informa Healthcare -London : Informa Healthcare, 2006-.) pp. 995-1035 - issn: 1746-0441 - wos: WOS:000475153500001 (49) - scopus: 2-s2.0-85070940142 (50)

11573/1307478 - 2019 - Novel therapies for glaucoma: a patent review (2013-2019)

Guglielmi, Paolo; Carradori, Simone; Campestre, Cristina; Poce, Giovanna - 01g Articolo di rassegna (Review)

rivista: EXPERT OPINION ON THERAPEUTIC PATENTS (--London United Kingdom:Informa Healthcare -London, United Kingdom: Ashley Publications Limited) pp. 769-780 - issn: 1354-3776 - wos: WOS:000480502600001 (24) - scopus: 2-s2.0-85070821891 (30)

11573/1237661 - 2019 - Design, synthesis, docking studies and monoamine oxidase inhibition of a small library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1h)-pyrazoles

Guglielmi, Paolo; Carradori, Simone; Poli, Giulio; Secci, Daniela; Cirilli, Roberto; Rotondi, Giulia; Chimenti, Paola; Petzer, Anél; Petzer, Jacobus P. - 01a Articolo in rivista

rivista: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. 1-21 - issn: 1420-3049 - wos: WOS:000458934000108 (27) - scopus: 2-s2.0-85060732811 (31)

11573/1307503 - 2019 - Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity

Guglielmi, Paolo; Secci, Daniela; Petzer, Anél; Bagetta, Donatella; Chimenti, Paola; Rotondi, Giulia; Ferrante, Claudio; Recinella, Lucia; Leone, Sheila; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P; Ortuso, Francesco; Carradori, Simone - 01a Articolo in rivista

rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1511-1525 - issn: 1475-6366 - wos: WOS:000481738100001 (23) - scopus: 2-s2.0-85071029361 (24)

11573/1349548 - 2019 - Kinesin Eg5 targeting inhibitors as a new strategy for gastric adenocarcinoma treatment

Marconi, G. D.; Carradori, S.; Ricci, A.; Guglielmi, P.; Cataldi, A.; Zara, S. - 01a Articolo in rivista

rivista: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. - - issn: 1420-3049 - wos: WOS:000498055500137 (22) - scopus: 2-s2.0-85074344175 (24)

11573/1307480 - 2019 - The up-regulation of oxidative stress as a potential mechanism of novel MAO-B inhibitors for glioblastoma treatment

Marconi, G. D.; Gallorini, M.; Carradori, S.; Guglielmi, P.; Cataldi, A.; Zara, S. - 01a Articolo in rivista

rivista: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. - - issn: 1420-3049 - wos: WOS:000470996600163 (30) - scopus: 2-s2.0-85066285276 (31)

11573/1307498 - 2019 - Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold

Rotondi, G.; Guglielmi, P.; Carradori, S.; Secci, D.; De Monte, C.; De Filippis, B.; Maccallini, C.; Amoroso, R.; Cirilli, R.; Akdemir, A.; Angeli, A.; Supuran, C. T. - 01a Articolo in rivista

rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1400-1413 - issn: 1475-6366 - wos: WOS:000480545500001 (23) - scopus: 2-s2.0-85070919829 (24)

11573/1237670 - 2019 - 4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis

Secci, Daniela; Carradori, Simone; Petzer, Anél; Guglielmi, Paolo; D’Ascenzio, Melissa; Chimenti, Paola; Bagetta, Donatella; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P.; Ortuso, Francesco - 01a Articolo in rivista

rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 597-612 - issn: 1475-6366 - wos: WOS:000457961800001 (40) - scopus: 2-s2.0-85061130350 (46)

11573/1121984 - 2018 - Magnetic metal−organic framework composite by fast and facile mechanochemical process

Bellusci, M.; Guglielmi, P.; Masi, Andrea; Padella, F.; Singh, G.; Yaacoub, N.; Peddis, D.; Secci, D. - 01a Articolo in rivista

rivista: INORGANIC CHEMISTRY (Washington, D.C. : American Chemical Society, c1962-) pp. 1806-1814 - issn: 1520-510X - wos: WOS:000426014800016 (66) - scopus: 2-s2.0-85042209909 (72)

11573/1068937 - 2018 - Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents

Carradori, Simone; Ottuso, Francesco; Petzer, Anèl; Bagetta, Donatella; De Monte, Celeste; Secci, Daniela; De Vita, Daniela; Guglielmi, Paolo; Zengin, Gokhan; Aktumsek, Abdurrahman; Alcaro, Stefano; Petzer, Jacobus P. - 01a Articolo in rivista

rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY ([Paris] : Elsevier, [198?]-) pp. 1543-1552 - issn: 1768-3254 - wos: WOS:000423641400032 (46) - scopus: 2-s2.0-85034651451 (52)

11573/1194382 - 2018 - Crystal structure of the Eg5 - K858 complex and implications for structure-based design of thiadiazole-containing inhibitors

Talapatra, Sandeep K.; Tham, Chuin Lean; Guglielmi, Paolo; Cirilli, Roberto; Chandrasekaran, Balakumar; Karpoormath, Rajshekhar; Carradori, Simone; Kozielski, Frank - 01a Articolo in rivista

11573/1194522 - 2017 - Analysis of imidazoles and triazoles in biological samples after MicroExtraction by packed sorbent

Campestre, Cristina; Locatelli, Marcello; Guglielmi, Paolo; De Luca, Elisa; Bellagamba, Giuseppe; Menta, Sergio; Zengin, Gokhan; Celia, Christian; Di Marzio, Luisa; Carradori, Simone - 01a Articolo in rivista

rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1-11 - issn: 1475-6366 - wos: WOS:000416951100001 (41) - scopus: 2-s2.0-85026870702 (46)

11573/974029 - 2017 - Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives

Carradori, Simone; Secci, Daniela; Bizzarri, Bruna; Chimenti, Paola; De Monte, Celeste; Guglielmi, Paolo; Campestre, Cristina; Rivanera, Daniela; Bordón, Claudia; Jones Brando, Lorraine - 01a Articolo in rivista

rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 746-758 - issn: 1475-6366 - wos: WOS:000404271200001 (24) - scopus: 2-s2.0-85019985742 (25)

11573/1194466 - 2017 - The sodium salt of the enantiomers of ricobendazole: preparation, solubility and chiroptical properties

Cirilli, Roberto; Guglielmi, Paolo; Formica, Francesca Romana; Casulli, Adriano; Carradori, Simone - 01a Articolo in rivista

rivista: JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS (Oxford ; New York : Pergamon Press Amsterdam : Elsevier Science) pp. 1-7 - issn: 0731-7085 - wos: WOS:000399865900001 (27) - scopus: 2-s2.0-85014043891 (30)

11573/1017595 - 2017 - Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms

D'ascenzio, M.; Guglielmi, P.; Carradori, S.; Secci, D.; Florio, R.; Mollica, A.; Ceruso, M.; Akdemir, A.; Sobolev, A. P.; Supuran, C. T. - 01a Articolo in rivista

rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 51-59 - issn: 1475-6366 - wos: WOS:000392591100044 (45) - scopus: 2-s2.0-84992390041 (48)

11573/1017583 - 2017 - Protective effects Induced by microwave-assisted aqueous harpagophytum extract on rat cortex synaptosomes challenged with amyloid β-peptide

Ferrante, Claudio; Recinella, Lucia; Locatelli, Marcello; Guglielmi, Paolo; Secci, Daniela; Leporini, Lidia; Chiavaroli, Annalisa; Leone, Sheila; Martinotti, Sara; Brunetti, Luigi; Vacca, Michele; Meneghini, Luigi; Orlando, Giustino - 01a Articolo in rivista

rivista: PHYTOTHERAPY RESEARCH (New York : J. Wiley) pp. 1257-1264 - issn: 1099-1573 - wos: WOS:000406926800015 (53) - scopus: 2-s2.0-85021271246 (57)

11573/956728 - 2017 - Enantiomers of triclabendazole sulfoxide: analytical and semipreparative HPLC separation, absolute configuration assignment, and transformation into sodium salt

Ferretti, Rosella; Carradori, Simone; Guglielmi, Paolo; Pierini, Marco; Casulli, Adriano; Cirilli, Roberto - 01a Articolo in rivista

rivista: JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS (Oxford ; New York : Pergamon Press Amsterdam : Elsevier Science) pp. 38-44 - issn: 0731-7085 - wos: WOS:000402850500005 (20) - scopus: 2-s2.0-85015734029 (22)

11573/1122262 - 2016 - Inhibition of human monoamine oxidase: biological and molecular modeling studies on selected natural flavonoids

Carradori, Simone; Gidaro, Maria Concetta; Petzer, Anél; Costa, Giosuè; Guglielmi, Paolo; Chimenti, Paola; Alcaro, Stefano; Petzer, Jacobus P. - 01a Articolo in rivista

rivista: JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY (American Chemical Society:1155 Sixteenth Street Northwest:Washington, DC 20036:(800)227-5558, EMAIL: service@acs.org, INTERNET: http://www.pubs.acs.org, Fax: (614)447-3671) pp. 9004-9011 - issn: 0021-8561 - wos: WOS:000389161900006 (85) - scopus: 2-s2.0-85002627776 (94)

11573/851467 - 2016 - A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms

Carradori, Simone; Secci, Daniela; De Monte, Celeste; Mollica, Adriano; Ceruso, Mariangela; Akdemir, Atilla; Sobolev, Anatoly P; Codispoti, Rossella; De Cosmi, Federica; Guglielmi, Paolo; Supuran, Claudiu T. - 01a Articolo in rivista

rivista: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 1095-1105 - issn: 0968-0896 - wos: WOS:000369989500020 (48) - scopus: 2-s2.0-84957841303 (54)

11573/851466 - 2015 - Synthesis and pharmacological screening of a large library of 1,3,4-thiadiazolines as innovative therapeutic tools for the treatment of prostate cancer and melanoma

De Monte, Celeste; Carradori, Simone; Secci, Daniela; D'ascenzio, Melissa; Guglielmi, Paolo; Mollica, Adriano; Morrone, Stefania; Scarpa, Susanna; Agliano', Anna Maria; Giantulli, Sabrina; Silvestri, Ida - 01a Articolo in rivista

11573/789264 - 2015 - Opening new scenarios for human MAO inhibitors

De Monte, Celeste; D'ascenzio, Melissa; Guglielmi, Paolo; Mancini, Veronica; Carradori, Simone - 01a Articolo in rivista

rivista: CENTRAL NERVOUS SYSTEM AGENTS IN MEDICINAL CHEMISTRY (Hilversum : Bentham Science Publishers) pp. - - issn: 1875-6166 - wos: (0) - scopus: 2-s2.0-84973659371 (16)