11573/1716808 - 2024 -
Transmission-Blocking Strategies for Malaria Eradication: Recent Advances in Small-Molecule Drug Development Appetecchia, Federico; Fabbrizi, Emanuele; Fiorentino, Francesco; Consalvi, Sara; Biava, Mariangela; Poce, Giovanna; Rotili, Dante - 01g Articolo di rassegna (Review)
rivista: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. - - issn: 1424-8247 - wos: (0) - scopus: (0)
11573/1711757 - 2024 -
Amino Acid Biosynthesis Inhibitors in Tuberculosis Drug Discovery Guida, Michela; Tammaro, Chiara; Quaranta, Miriana; Salvucci, Benedetta; Biava, Mariangela; Poce, Giovanna; Consalvi, Sara - 01g Articolo di rassegna (Review)
rivista: PHARMACEUTICS (Basel: MDPI, 2009-) pp. 1-36 - issn: 1999-4923 - wos: WOS:001257061500001 (0) - scopus: 2-s2.0-85197351471 (0)
11573/1720626 - 2024 -
SAR Analysis of Novel Coxsackie virus A9 Capsid Binders Tammaro, Chiara; Plavec, Zlatka; Myllymäki, Laura; Mitchell, Cristopher; Consalvi, Sara; Biava, Mariangela; Ciogli, Alessia; Domanska, Aušra; Leppilampi, Valtteri; Buckner, Cienna; Manetto, Simone; Sciò, Pietro; Coluccia, Antonio; Laajala, Mira; Dondio, Giulio M; Bigogno, Chiara; Marjomäki, Varpu; Butcher, Sarah J; Poce, Giovanna - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. - - issn: 0022-2623 - wos: WOS:001315707100001 (0) - scopus: (0)
11573/1668341 - 2023 -
Tannin microcapsules for synergy-enhanced sunscreen formulations Alfonsi, E.; Lange, H.; Zongo, L.; Poce, G.; Sgarzi, M.; Crestini, C. - 01a Articolo in rivista
rivista: INDUSTRIAL CROPS AND PRODUCTS (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598) pp. 116105- - issn: 0926-6690 - wos: WOS:001029319300001 (1) - scopus: 2-s2.0-85143868314 (1)
11573/1675540 - 2023 -
Antiviral Mechanisms of N-Phenyl Benzamides on Coxsackie Virus A9 Laajala, Mira; Kalander, Kerttu; Consalvi, Sara; Sheik Amamuddy, Olivier; Tastan Bishop, Özlem; Biava, Mariangela; Poce, Giovanna; Marjomäki, Varpu - 01a Articolo in rivista
rivista: PHARMACEUTICS (Basel: MDPI, 2009-) pp. - - issn: 1999-4923 - wos: WOS:000957987000001 (2) - scopus: 2-s2.0-85151320878 (1)
11573/1668339 - 2023 -
Direct-Acting Antivirals and Host-Targeting Approaches against Enterovirus B Infections: Recent Advances Tammaro, Chiara; Guida, Michela; Appetecchia, Federico; Biava, Mariangela; Consalvi, Sara; Poce, Giovanna - 01a Articolo in rivista
rivista: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. 203- - issn: 1424-8247 - wos: WOS:000940922000001 (7) - scopus: 2-s2.0-85148952319 (6)
11573/1620087 - 2022 -
Malaria transmission blocking compounds: a patent review Consalvi, Sara; Tammaro, Chiara; Appetecchia, Federico; Biava, Mariangela; Poce, Giovanna - 01a Articolo in rivista
rivista: EXPERT OPINION ON THERAPEUTIC PATENTS (--London United Kingdom:Informa Healthcare
-London, United Kingdom: Ashley Publications Limited) pp. 1-18 - issn: 1354-3776 - wos: WOS:000767678000001 (7) - scopus: 2-s2.0-85126475360 (7)
11573/1655508 - 2022 -
Nano-based drug delivery systems of potent MmpL3 inhibitors for tuberculosis treatment Hanieh, P. N.; Consalvi, S.; Forte, J.; Cabiddu, G.; De Logu, A.; Poce, G.; Rinaldi, F.; Biava, M.; Carafa, M.; Marianecci, C. - 01a Articolo in rivista
rivista: PHARMACEUTICS (Basel: MDPI, 2009-) pp. 1-13 - issn: 1999-4923 - wos: WOS:000774333800001 (6) - scopus: 2-s2.0-85126452255 (6)
11573/1335786 - 2021 -
Dietary flavonoids: Nano delivery and nanoparticles for cancer therapy Aiello, Paola; Consalvi, Sara; Poce, Giovanna; Raguzzini, Anna; Toti, Elisabetta; Palmery, Maura; Biava, Mariangela; Bernardi, Marco; Kamale, Mohammad A.; Perry, George; Peluso, Ilaria - 01g Articolo di rassegna (Review)
rivista: SEMINARS IN CANCER BIOLOGY (Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. 150-165 - issn: 1044-579X - wos: WOS:000631703400011 (71) - scopus: 2-s2.0-85071626772 (79)
11573/1614886 - 2021 -
A novel class of dual-acting DCH-CORMs counteracts oxidative stress-induced inflammation in human primary tenocytes Appetecchia, F.; Consalvi, S.; Berrino, E.; Gallorini, M.; Granese, A.; Campestre, C.; Carradori, S.; Biava, M.; Poce, G. - 01a Articolo in rivista
rivista: ANTIOXIDANTS (Basel: MDPI) pp. - - issn: 2076-3921 - wos: WOS:000728018500001 (5) - scopus: 2-s2.0-85119177792 (6)
11573/1487147 - 2021 -
Therapeutic potential for coxibs-nitric oxide releasing hybrids in cystic fibrosis Consalvi, S.; Poce, G.; Ghelardini, C.; Di Cesare Mannelli, L.; Patrignani, P.; Bruno, A.; Anzini, M.; Calderone, V.; Martelli, A.; Testai, L.; Giordani, A.; Biava, M. - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 112983- - issn: 0223-5234 - wos: WOS:000604903800029 (4) - scopus: 2-s2.0-85096376603 (5)
11573/1614881 - 2021 -
6-Fluorophenylbenzohydrazides inhibit Mycobacterium tuberculosis growth through alteration of tryptophan biosynthesis Consalvi, S.; Venditti, G.; Zhu, J.; Boshoff, H. I.; Arora, K.; De Logu, A.; Ioerger, T. R.; Rubin, E. J.; Biava, M.; Poce, G. - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. - - issn: 0223-5234 - wos: WOS:000703119000027 (2) - scopus: 2-s2.0-85114741985 (2)
11573/1462744 - 2020 -
Sar analysis of small molecules interfering with energy-metabolism in mycobacterium tuberculosis Appetecchia, F.; Consalvi, S.; Scarpecci, C.; Biava, M.; Poce, G. - 01a Articolo in rivista
rivista: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. 1-33 - issn: 1424-8247 - wos: WOS:000580832600001 (10) - scopus: 2-s2.0-85092679912 (12)
11573/1493983 - 2020 -
Overcoming drug resistance in TB: an update Consalvi, S.; Poce, G.; Scarpecci, C.; Biava, M. - 01m Editorial/Introduzione in rivista
rivista: FUTURE MICROBIOLOGY (London : Future Medicine, 2006-.) pp. 1607-1609 - issn: 1746-0913 - wos: WOS:000591446300001 (1) - scopus: 2-s2.0-85097964343 (1)
11573/1334361 - 2019 -
Mycobacterial tryptophan biosynthesis: a promising target for tuberculosis drug development? Consalvi, Sara; Scarpecci, Cristina; Biava, Mariangela; Poce, Giovanna - 01g Articolo di rassegna (Review)
rivista: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 126731- - issn: 0960-894X - wos: WOS:000495112100015 (11) - scopus: 2-s2.0-85074070157 (11)
11573/1307478 - 2019 -
Novel therapies for glaucoma: a patent review (2013-2019) Guglielmi, Paolo; Carradori, Simone; Campestre, Cristina; Poce, Giovanna - 01g Articolo di rassegna (Review)
rivista: EXPERT OPINION ON THERAPEUTIC PATENTS (--London United Kingdom:Informa Healthcare
-London, United Kingdom: Ashley Publications Limited) pp. 769-780 - issn: 1354-3776 - wos: WOS:000480502600001 (22) - scopus: 2-s2.0-85070821891 (27)
11573/1334375 - 2019 -
Novel pyrazole-containing compounds active against mycobacterium tuberculosis Poce, Giovanna; Consalvi, Sara; Venditti, Giulia; Alfonso, Salvatore; Desideri, Nicoletta; Fernandez-Menendez, Raquel; Bates, Robert H.; Ballell, Lluis; Barros Aguirre, David; Rullas, Joaquin; De Logu, Alessandro; Gardner, Michelle; Ioerger, Thomas R.; Rubin, Eric J.; Biava, Mariangela - 01a Articolo in rivista
rivista: ACS MEDICINAL CHEMISTRY LETTERS (USA: ACS Publications) pp. 1423-1429 - issn: 1948-5875 - wos: WOS:000490355900009 (37) - scopus: 2-s2.0-85073024402 (37)
11573/1655529 - 2019 -
Development of MmpL3 inhibitors for tuberculosis treatment Poce, Giovanna; Consalvi, Sara; Venditti, Giulia; Scarpecci, Cristina; Biava, Mariangela - 02a Capitolo o Articolo
libro: Medicinal Chemistry approaches to tuberculosis and trypanosomiasis - (978-0-12-817556-9)
11573/1334385 - 2019 -
Chocolate consumers and lymphocyte-to-monocyte ratio: a working hypothesis from a preliminary report of a pilot study in celiac subjects Raguzzini, A; Poce, G; Consalvi, S; Toti, E; Palmacci, F; Biava, M; Peluso, I - 01a Articolo in rivista
rivista: ANTIOXIDANTS (Basel: MDPI) pp. - - issn: 2076-3921 - wos: WOS:000500759900023 (4) - scopus: 2-s2.0-85073539054 (4)
11573/1191296 - 2018 -
Stimuli-responsive tannin–feIII hybrid microcapsules demonstrated by the active release of an anti-tuberculosis agent Bartzoka, Elisavet D.; Lange, Heiko; Poce, Giovanna; Crestini, Claudia - 01a Articolo in rivista
rivista: CHEMSUSCHEM (WEINHEIM, GERMANY: WILEY-V C H VERLAG GMBH) pp. 3975-3991 - issn: 1864-5631 - wos: WOS:000451061000015 (20) - scopus: 2-s2.0-85055454631 (20)
11573/1071677 - 2018 -
In vivo potent BM635 analogue with improved drug-like properties Poce, Giovanna; Cocozza, Martina; Alfonso, Salvatore; Consalvi, Sara; Venditti, Giulia; Fernandez-Menendez, Raquel; Bates, Robert H.; Barros Aguirre, David; Ballell, Lluis; De Logu, Alessandro; Vistoli, Giulio; Biava, Mariangela - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 539-550 - issn: 0223-5234 - wos: WOS:000425198200041 (21) - scopus: 2-s2.0-85040337865 (23)
11573/957091 - 2017 -
Pharmaceutical salt of BM635 with improved bioavailability Poce, Giovanna; Consalvi, Sara; Cocozza, Martina; Fernandez Menendez, Raquel; Bates, Robert H.; Ortega Muro, Fátima; Barros Aguirre, David; Ballell, Lluis; Biava, Mariangela - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES (Amsterdam Netherlands: Elsevier BV) pp. 17-23 - issn: 0928-0987 - wos: WOS:000394474200003 (10) - scopus: 2-s2.0-85004187448 (10)
11573/957084 - 2017 -
1,5-Diarylpyrroles as potent antitubercular and anti-inflammatory agents Venditti, Giulia; Poce, Giovanna; Consalvi, Sara; Biava, Mariangela - 01a Articolo in rivista
rivista: CHEMISTRY OF HETEROCYCLIC COMPOUNDS (Consultants Bureau:A Division of Plenum Publishing Corporation, 233 Spring Street, Sixth Floor:New York, NY 10013:(800)221-9369, (212)620-8082, Fax: (212)463-0742) pp. 281-291 - issn: 0009-3122 - wos: WOS:000400545300005 (4) - scopus: 2-s2.0-85018288338 (5)
11573/1071674 - 2017 -
MmpL3 is the flippase for mycolic acids in mycobacteria Xu, Zhujun; Meshcheryakov, Vladimir A.; Poce, Giovanna; Chng, Shu-Sin - 01a Articolo in rivista
rivista: PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA (National Academy of Sciences:2101 Constitution Avenue Northwest:Washington, DC 20418:(877)314-2253, (615)377-3322, EMAIL: subspnas@nas.edu, INTERNET: http://www.pnas.org, Fax: (615)377-0525) pp. 7993-7998 - issn: 0027-8424 - wos: WOS:000406189900070 (138) - scopus: 2-s2.0-85025640419 (142)
11573/891076 - 2016 -
A series of COX-2 inhibitors endowed with NO-releasing properties: synthesis, biological evaluation, and docking analysis Consalvi, Sara; Poce, Giovanna; Ragno, Rino; Sabatino, Manuela; Lamotta, Concettina; Sartini, Stefania; Calderone, Vincenzo; Martelli, Alma; Ghelardini, Carla; Dicesaremannelli, Lorenzo; Biava, Mariangela - 01a Articolo in rivista
rivista: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. 1804-1811 - issn: 1860-7179 - wos: WOS:000383579700016 (5) - scopus: 2-s2.0-84983288442 (7)
11573/869500 - 2016 -
Synthesis and biological evaluation of fluorinated 1,5-diarylpyrrole-3-alkoxyethyl ether derivatives as selective COX-2 inhibitors endowed with anti-inflammatory activity Di Capua, Angela; Sticozzi, Claudia; Brogi, Simone; Brindisi, Margherita; Cappelli, Andrea; Sautebin, Lidia; Rossi, Antonietta; Pace, Simona; Ghelardini, Carla; Di Cesare Mannelli, Lorenzo; Valacchi, Giuseppe; Giorgi, Gianluca; Giordani, Antonio; Poce, Giovanna; Biava, Mariangela; Anzini, Maurizio - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 99-106 - issn: 0223-5234 - wos: WOS:000375634400009 (27) - scopus: 2-s2.0-84953931791 (30)
11573/1191315 - 2016 -
MmpL3 inhibitors: diverse chemical scaffolds inhibit the same target Poce, Giovanna; Consalvi, Sara; Biava, Mariangela - 01a Articolo in rivista
rivista: MINI-REVIEWS IN MEDICINAL CHEMISTRY (Bentham Science Publishers BV:PO Box 7917, Exec Ste Y 26, Saif Zone Sharjah Uae:011 971 6 5571132, EMAIL: benthams@emirates.net.ae, INTERNET: http://www.bentham.org, Fax: 011 971 6 5571134) pp. 1274-1283 - issn: 1389-5575 - wos: WOS:000385572900002 (24) - scopus: 2-s2.0-84991396425 (28)
11573/870679 - 2016 -
Novel inhibitors of Mycobacterium tuberculosis tryptophan biosynthetic pathway to treat tuberculosis Venditti, Giulia; Consalvi, Sara; Helena, Boshoff; Biava, Mariangela; Poce, Giovanna - 04f Poster
congresso: VI EWDSy (European Workshop in Drug Synthesis) (Siena, Italia)
11573/1668504 - 2015 -
Synthesis, biological evaluation and docking analysis of a new series of methylsulfonyl and sulfamoyl acetamides and ethyl acetates as potent COX-2 inhibitors Consalvi, Sara; Alfonso, Salvatore; Di Capua, Angela; Poce, Giovanna; Pirolli, Adele; Sabatino, Manuela; Ragno, Rino; Anzini, Maurizio; Sartini, Stefania; La Motta, Concettina; Di Cesare Mannelli, Lorenzo; Ghelardini, Carla; Biava, Mariangela - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY ([Oxford]: Elsevier.) pp. 810-820 - issn: 1464-3391 - wos: WOS:000349083100018 (22) - scopus: 2-s2.0-84922322412 (22)
11573/869416 - 2015 -
COX inhibitors: a patent review (2011 - 2014) Consalvi, Sara; Biava, Mariangela; Poce, Giovanna - 01a Articolo in rivista
rivista: EXPERT OPINION ON THERAPEUTIC PATENTS (--London United Kingdom:Informa Healthcare
-London, United Kingdom: Ashley Publications Limited) pp. 1357-1371 - issn: 1354-3776 - wos: WOS:000366526700001 (33) - scopus: 2-s2.0-84949780684 (33)
11573/781378 - 2015 -
A novel antimycobacterial compound acts as an intracellular iron chelator Dragset Marte, S; Poce, Giovanna; Alfonso, Salvatore; Padilla Benavides, T; Ioerger, T. R.; Kaneko, T; Sacchettini, Jc; Biava, Mariangela; Parish, T; Argüello, Jm; Steigedal, M; Rubin, Ej - 01a Articolo in rivista
rivista: ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (American Society for Microbiology:PO Box 11127:Birmingham, AL 35201:(800)633-4931, (205)995-1567, EMAIL: asm.nonmembers.subs@ebsco.com, INTERNET: http://www.asm.org, Fax: (205)995-1588) pp. 2256-2264 - issn: 0066-4804 - wos: WOS:000354993700051 (35) - scopus: 2-s2.0-84928905358 (34)
11573/781382 - 2015 -
Activity of lipophilic and hydrophilic drugs against dormant and replicating mycobacterium tuberculosis Piccaro, G; Poce, Giovanna; Biava, Mariangela; Giannoni, F; Fattorini, L. - 01a Articolo in rivista
rivista: JOURNAL OF ANTIBIOTICS (Japan Antibiotics Research Association:2-20-8 Kamiosaki Shinagawa-ku, Tokyo 141-0021 Japan:011 81 3 34910181, EMAIL: gakkyo@antibotics.or.jp, INTERNET: http://www.anibotics.or.jp, Fax: 011 81 34910179) pp. 711-714 - issn: 0021-8820 - wos: WOS:000365832300010 (52) - scopus: 2-s2.0-84948651608 (57)
11573/869374 - 2015 -
Overcoming drug resistance for tuberculosis Poce, Giovanna; Biava, Mariangela - 01a Articolo in rivista
rivista: FUTURE MICROBIOLOGY (London : Future Medicine, 2006-.) pp. 1735-1741 - issn: 1746-0913 - wos: WOS:000365746000005 (8) - scopus: 2-s2.0-84948137710 (9)
11573/540514 - 2014 -
Enhancing the pharmacodynamic profile of a class of selective COX-2 inhibiting nitric oxide donors Biava, Mariangela; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Consalvi, Sara; Angela Di, Capua; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Lidia, Sautebin; Antonietta, Rossi; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Antonio, Giordani; Stefano, Persiani; Milena, Colovic; Melania, Dovizio; Paola, Patrignani; Maurizio, Anzini - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 772-786 - issn: 0968-0896 - wos: WOS:000329576400011 (25) - scopus: 2-s2.0-84892370910 (26)
11573/639185 - 2014 -
SAR analysis of new anti-TB drugs currently in pre-clinical and clinical development Poce, Giovanna; Cocozza, Martina; Consalvi, Sara; Biava, Mariangela - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 335-351 - issn: 0223-5234 - wos: WOS:000343781800031 (45) - scopus: 2-s2.0-84906997561 (49)
11573/515578 - 2013 -
Novel Analgesic/Anti-inflammatory Agents: 1,5-Diarylpyrrole Nitro-oxyalkyl Ethers and Related Compounds as Cyclooxygenase-2 Inhibiting Nitric Oxide Donors Anzini, M.; Di Capua, A.; Valenti, S.; Brogi, S.; Rovin, M.; Giuliani, G.; Cappelli, A.; Vomero, S.; Chiasserini, L.; Saga, A.; Poce, Giovanna; Giorgi, G.; Calderone, V.; Martelli, A.; Testai, L.; Sautebin, L.; Rossi, A.; Papa, G.; Ghelardini, C.; Di Cesare Mannelli, L.; Benetti, V.; Giordani, A.; Anzellotti, P.; Dovizio, M.; Patrignani, P.; Biava, Mariangela - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 3191-3206 - issn: 0022-2623 - wos: WOS:000318211100005 (45) - scopus: 2-s2.0-84876827778 (47)
11573/523394 - 2013 -
Inhibition of Leishmania infantum trypanothione reductase by azole-based compounds: a comparative analysis with its physiological substrate by X-ray crystallography Baiocco, P.; Poce, Giovanna; Alfonso, Salvatore; Cocozza, Martina; Porretta, Giulio Cesare; Colotti, G.; Biava, Mariangela; Moraca, F.; Botta, M.; Yardley, V.; Fiorillo, A.; Lantella, A.; Malatesta, Francesco; Ilari, Andrea - 01a Articolo in rivista
rivista: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. 1175-1183 - issn: 1860-7179 - wos: WOS:000320928400012 (57) - scopus: 2-s2.0-84879786172 (61)
11573/516096 - 2013 -
A class of pyrrole derivatives endowed with analgesic/anti-inflammatory activity Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; Consalvi, Sara; L., Sautebin; S., Pace; A., Rossi; C., Ghelardini; L., Di Cesare Mannelli; S., Schenone; A., Giordani; L., Di Francesco; P., Patrignani; Biava, Mariangela - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY ([Oxford]: Elsevier.) pp. 3695-3701 - issn: 1464-3391 - wos: WOS:000320347100007 (83) - scopus: 2-s2.0-84878612651 (88)
11573/526248 - 2013 -
The novel anti-inflammatory agent VA694, endowed with both
NO-releasing and COX2-selective inhibiting properties, exhibits
NO-mediated positive effects on blood pressure, coronary flow and endothelium in an experimental model of hypertension and
endothelial dysfunction Martelli, A; Testai, L; Anzini, M; Cappelli, A; Di Capua, A; Biava, Mariangela; Poce, Giovanna; Consalvi, Sara; Giordani, A; Caselli, G; Rovati, L; Ghelardini, C; Patrignani, P; Sautebin, L; Breschi, Mc; Calderone, V. - 01a Articolo in rivista
rivista: PHARMACOLOGICAL RESEARCH (Attuale:ACADEMIC PRESS LTD ELSEVIER SCIENCE LTD, 24-28 OVAL RD, LONDON, ENGLAND, NW1 7DX
Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. 1-9 - issn: 1043-6618 - wos: WOS:000328874100001 (22) - scopus: 2-s2.0-84886005479 (25)
11573/515576 - 2013 -
Improved BM212 MmpL3 Inhibitor Analogue Shows Efficacy in Acute Murine Model of Tuberculosis Infection Poce, Giovanna; H. R., Bates; Alfonso, Salvatore; Cocozza, Martina; Porretta, Giulio Cesare; L., Ballel; Joaquin, Rullas; Alessandro De, Logu; Emanuela, Agus; Valentina La, Rosa; Maria Rosalia, Pasca; Edda De, Rossi; Baojie, Wae; S. J., Franzblau; Fabrizio, Manetti; Maurizio, Botta; Biava, Mariangela - 01a Articolo in rivista
rivista: PLOS ONE (San Francisco, CA : Public Library of Science) pp. e56980-e56980 - issn: 1932-6203 - wos: WOS:000315186000063 (91) - scopus: 2-s2.0-84874297088 (97)
11573/492770 - 2012 -
New 1,5 diarylpyrrole derivatives as antimycobacterial agents: Design, synthesis, biological evaluation and study of their mode of action Alfonso, Salvatore; Poce, Giovanna; Porretta, Giulio Cesare; Battilocchio, Claudio; Rubin, E. J.; De Rossi, E.; De Logu, A.; Franzblau, S. C.; Botta, M.; Biava, Mariangela - 04a Atto di comunicazione a congresso
congresso: NPCF6 (Riccione)
11573/490950 - 2012 -
Improving the solubility of a new class of antiinflammatory pharmacodynamic hybrids, that release nitric oxide and inhibit cycloxygenase-2 isoenzyme Biava, Mariangela; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; Consalvi, Sara; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Lidia, Sautebin; Antonietta, Rossi; Antonio, Giordani; Paola, Patrignani; Maurizio, Anzini - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 287-298 - issn: 0223-5234 - wos: WOS:000312745100029 (14) - scopus: 2-s2.0-84868249710 (16)
11573/492768 - 2012 -
New Heterocyclic Compounds Targeting Trypanothyione Metabolism in Leishmania Parasites Biava, Mariangela; Cocozza, Martina; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; Colotti, G.; Malatesta, F.; Baiocco, P.; Ilari, Andrea - 04d Abstract in atti di convegno
congresso: NPCF6 (Riccione)
11573/492764 - 2012 -
New Pyrrole Derivatives as Anti-inflammatory and Analgesic Agents: Design, Synthesis and Biological Evaluation Biava, Mariangela; Consalvi, Sara; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Ghelardini, C.; Sautebin, L. - 04a Atto di comunicazione a congresso
congresso: NPCF6 (Riccione)
11573/492117 - 2012 -
Analogs of BM 212: a new chemical class of antimycobacterial agents acting upon a new target Biava, Mariangela; Poce, Giovanna; Porretta, Giulio Cesare; Alfonso, Salvatore; Cocozza, Martina; De Logu, A; De Rossi, E; Ballel, L; Franzblau, S; Rubin E., J; Botta, M. - 04a Atto di comunicazione a congresso
congresso: 21st National Meeting on Medicinal Chemistry (Palermo)
11573/492120 - 2012 -
Identification of a new chemical class of potent antimycobacterial compounds derived from BM 212: design, synthesis, biological evaluation and study of their mode of action. Biava, Mariangela; Poce, Giovanna; Porretta, Giulio Cesare; Alfonso, Salvatore; De Logu, A; De Rossi, E; Ballel, L; Franzblau, S; Manetti, ; Rubin, Ej; Botta, M. - 04a Atto di comunicazione a congresso
congresso: XXIInd International Symposium on Medicinal Chemistry (EFMC-ISMC) (Berlino, Germania)
11573/509516 - 2012 -
New 1,5-diphenyl pyrrole derivatives as anti-inflammatory COX-2 selective compounds and their use as potential antitumoral agents. Consalvi, Sara; Battilocchio, Claudio; Poce, Giovanna; Alfonso, Salvatore; Porretta, Giulio Cesare; M., Anzini; L., Sautebin; C., Ghelardini; A., Giordani; P., Patrignani; V., Calderone; Biava, Mariangela - 04a Atto di comunicazione a congresso
congresso: IV European Workshop in Drug Synthesis (Siena)
11573/492772 - 2012 -
1,5-Diphenyl pyrroles as new antimycobacterial agents. Hit-to-lead development and target validation, New drugs for neglected diseases Poce, Giovanna; Porretta, Giulio Cesare; De Logu, A; De Rossi, A; Rubin, Ej; Ballel, L; Botta, M; Biava, Mariangela - 04a Atto di comunicazione a congresso
congresso: , CM0801 – (Siena,)
11573/434001 - 2012 -
MmpL3 Is the Cellular Target of the Antitubercular Pyrrole Derivative BM212 V., La Rosa; Poce, Giovanna; J., Ortiz Canseco; S., Buroni; M. R., Pasca; Biava, Mariangela; R. M., Raju; Porretta, Giulio Cesare; Alfonso, Salvatore; C., Battilocchio; B., Javid; F., Sorrentino; T. R., Ioerger; J. C., Sacchettini; F., Manetti; M., Botta; A., De Logu; E. J., Rubin - 01a Articolo in rivista
rivista: ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (American Society for Microbiology:PO Box 11127:Birmingham, AL 35201:(800)633-4931, (205)995-1567, EMAIL: asm.nonmembers.subs@ebsco.com, INTERNET: http://www.asm.org, Fax: (205)995-1588) pp. 324-331 - issn: 0066-4804 - wos: WOS:000298404900040 (186) - scopus: 2-s2.0-84455173193 (200)
11573/492740 - 2011 -
Pyrrole-based selective COX-2 inhibiting nitric oxide donors: synthesis, in vitro and in vivo evaluation Battilocchio, Claudio; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Calderone, V.; Sautebin, L.; Ghelardini, C.; Giordani, A.; Anzini, M.; Biava, Mariangela - 04a Atto di comunicazione a congresso
congresso: 5° Meeting NPCF (Trieste)
libro: 5° Meeting
NUOVE PROSPETTIVE IN
CHIMICA FARMACEUTICA - ()
11573/492752 - 2011 -
New Pyrrole-based selective COX-2 inhibiting nitric oxide donors: synthesis, in vitro and in vivo evaluation Battilocchio, Claudio; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Giordani, A.; Sautebin, L.; Ghelardini, C.; Calderone, V.; Patrignani, P.; Anzini, M.; Biava, Mariangela - 04a Atto di comunicazione a congresso
congresso: XXIV Congresso Naionale della Società Chimica Italiana (Lecce)
11573/492735 - 2011 -
Synthesis and biological evaluation of new heterocyclic derivatives with potential antimycobacterial activity: systematic approach to lead compound optimization Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A; Manetti, F; Botta, M. - 04a Atto di comunicazione a congresso
congresso: NPCF5 (Trieste)
11573/357725 - 2011 -
Developing Pyrrole-Derived Antimycobacterial Agents: a Rational Lead Optimization Approach Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; A., De Logu; Fabrizio, Manetti; Maurizio, Botta - 01a Articolo in rivista
rivista: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. 593-599 - issn: 1860-7179 - wos: WOS:000288814900004 (43) - scopus: 2-s2.0-79953052237 (43)
11573/427797 - 2011 -
Novel Analgesic/Anti-Inflammatory Agents: Diarylpyrrole Acetic Esters Endowed with Nitric Oxide Releasing Properties Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Michele, Rovini; Salvatore, Valenti; Gianluca, Giorgi; Vincenzo, Calderone; Alma, Martelli; Lara, Testai; Lidia, Sautebin; Antonietta, Rossi; Giuseppina, Papa; Carla, Ghelardini; Lorenzo Di Cesare, Mannelli; Antonio, Giordani; Paola, Anzellotti; Annalisa, Bruno; Paola, Patrignani; Anzini, - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 7759-7771 - issn: 0022-2623 - wos: WOS:000297001600003 (41) - scopus: 2-s2.0-81555218668 (42)
11573/356131 - 2011 -
Enlarging the NSAIDs Family: Ether, Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Novel Anti-Inflammatory and Analgesic Agents Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Botta, M; Manetti, F; Rovini, M; Cappelli, A; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Galeotti, N; Makovec, F; Giordani, A; Anzellotti, P; Tacconelli, S; Patrignani, P; Anzini, M. - 01a Articolo in rivista
rivista: CURRENT MEDICINAL CHEMISTRY (Bentham Science Publishers BV:PO Box 7917, Exec Ste Y 26, Saif Zone Sharjah Uae:011 971 6 5571132, EMAIL: benthams@emirates.net.ae, INTERNET: http://www.bentham.org, Fax: 011 971 6 5571134) pp. 1540-1554 - issn: 0929-8673 - wos: WOS:000289781000012 (13) - scopus: 2-s2.0-79955005080 (14)
11573/492747 - 2011 -
BM212 targets MmpL3, Gordon Research Conference on Tuberculosis Drug Development Poce, Giovanna; Biava, Mariangela; Porretta, Giulio Cesare; Battilocchio, Claudio; Alfonso, Salvatore; Botta, M.; Javid, B.; Sorrentino, F.; Ioerger, T. R.; Sacchettini, J. R.; Rubin, E. - 04a Atto di comunicazione a congresso
congresso: Gordon Research Conference on Tuberculosis Drug Development (Lucca (Barga))
11573/492710 - 2010 -
New pyrrole derivatives of BM 212: a new class of antimycobacterial agents. Design, synthesis, biological evaluation and study of their mode of action Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; De Rossi, E.; Manetti, F; Botta, M. - 04a Atto di comunicazione a congresso
congresso: COST Action Meeting CM0801 (Siena)
libro: CM0801-New Drugs For Neglected Diseases - ()
11573/492446 - 2010 -
BM 579: a novel pyrrole derivative with improved antimycobacterial activity Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A.; Manetti, F; Botta, M. - 04a Atto di comunicazione a congresso
congresso: NPCF4 (Santa Margherita di Pula (Ca))
libro: IV Meeting "Nuove Prospettive in Chimica Farmaceutica" - ()
11573/172075 - 2010 -
1,5-Diaryl-Pyrroles as New Generation of Anti-Inflammatory and Analgesic Agents: Design, Synthesis, in vitro and in vivo Evaluation Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, S; Battilocchio, Claudio; De Logu, A; Manetti, F; Botta, M. - 04a Atto di comunicazione a congresso
congresso: NPCF IV (Santa Margherita di Pula)
libro: NPCF IV - ()
11573/492727 - 2010 -
Identification of a new Chemical Class of Potent Antimycobacterial Compounds Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Alfonso, Salvatore; Battilocchio, Claudio; De Logu, A; Manetti, F; Botta, M. - 04a Atto di comunicazione a congresso
congresso: XX Meeting on Medicinal Chemistry (Abano Terme (PD))
11573/364093 - 2010 -
Identification of a novel pyrrole derivative endowed with antimycobacterial activity and protection index comparable to that of the current antitubercular drugs streptomycin and rifampin Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; A., De Logu; Nadia, Serra; Fabrizio, Manetti; Maurizio, Botta - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 8076-8084 - issn: 0968-0896 - wos: WOS:000283649900045 (44) - scopus: 2-s2.0-78449242124 (50)
11573/492716 - 2010 -
Developing New Antiinflammatory and Analgesic Agents: Design, Synthesis, Biological and harmacological Evaluation Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Alfonso, Salvatore; Botta, M.; Manetti, F.; Sautebin, L; Ghelardini, C; Makovec, F; Giordani, A; Patrignani, P; Anzini, M. - 04a Atto di comunicazione a congresso
congresso: III European Workshop in Drug Synthesis (Siena)
11573/362423 - 2010 -
Novel Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Anti-inflammatory and Analgesic Agents. Synthesis, in vitro and in vivo Biological Evaluation Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; Manetti, F; Botta, M; Sautebin, L; Rossi, A; Pergola, C; Ghelardini, C; Norcini, M; Makovec, F; Anzellotti, P; Cirilli, R; Ferretti, R; Patrignani, P; Anzini, M. - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 723-733 - issn: 0022-2623 - wos: WOS:000273672100019 (45) - scopus: 2-s2.0-77249138784 (49)
11573/361148 - 2010 -
New heterocyclic compounds with potential activity against parasitic protozoan: Trypanosoma and Leishmania Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Battilocchio, Claudio; V., Yardley; Alfonso, Salvatore - 04a Atto di comunicazione a congresso
congresso: COST Action Meeting CM0801 (Certosa di Pontignano, Siena, Italia)
libro: CM0801-New Drugs For Neglected Diseases - ()
11573/341214 - 2010 -
One-pot conversions of olefins to cyclic carbonates and secondary allylic and homoallylic amines to cyclic carbamates Stephen G., Davies; Ai M., Fletcher; Wataru, Kurosawa; James A., Lee; Poce, Giovanna; Paul M., Roberts; James E., Thomson; David M., Williamson - 01a Articolo in rivista
rivista: JOURNAL OF ORGANIC CHEMISTRY ([Washington, D.C: American Chemical Society) pp. 7745-7756 - issn: 0022-3263 - wos: WOS:000284080300027 (39) - scopus: 2-s2.0-78449236740 (41)
11573/341213 - 2010 -
Doubly diastereoselective conjugate addition of enantiopure lithium amides to enantiopure N-enoyl oxazolidin-2-ones: a mechanistic probe Stephen G., Davies; M. A., Fletcher; Gesine J., Hermann; Poce, Giovanna; Paul M., Roberts; Andrew D., Smith; Miles J., Sweet; James E., Thomson - 01a Articolo in rivista
rivista: TETRAHEDRON-ASYMMETRY (PERGAMON-ELSEVIER SCIENCE LTD, THE BOULEVARD, LANGFORD LANE, KIDLINGTON, OXFORD, ENGLAND, OX5 1GB) pp. 1635-1648 - issn: 0957-4166 - wos: WOS:000281356000001 (27) - scopus: 2-s2.0-77956264668 (21)
11573/225700 - 2009 -
New pyrrole derivatives of BM 212: a new class of antimycobacterial agents.Design, synthesis, biological evaluation and study of their mode of action. Biava, Mariangela; Porretta, G. C.; Poce, G; De Logu, A; Manetti, F; Botta, M. - 04a Atto di comunicazione a congresso
libro: NUOVE PROSPETTIVE IN CHIMICA FARMACEUTICA - ()
11573/368481 - 2009 -
Pyrrole derivatives of BM212 as novel antimycobacterial agents Design, synthesis, biological evaluation and study of their mode of action Biava, Mariangela; Porretta, Giulio Cesare; Battilocchio, Claudio; Poce, G; Pompei, R; De Logu, A; Manetti, F; Botta, M. - 04a Atto di comunicazione a congresso
libro: XXVIII CONGRESSO NAZIONALE DELLA SOCIETÀ DI MICROBIOLOGIA GENERALE E BIOTECNOLOGIE MICROBICHE - ()
11573/359624 - 2009 -
1,5-Diaryl-2-ethyl pyrrole derivatives as antimycobacterial agents: design, synthesis, and microbiological evaluation Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; De Logu, A; Saddi, M; Meleddu, R; Manetti, F; De Rossi, E; Botta, M. - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 4734-4738 - issn: 0223-5234 - wos: WOS:000271225800057 (72) - scopus: 2-s2.0-70349765643 (77)
11573/224933 - 2009 -
Derivatives of BM 212: synthesis and biological evaluation of new derivatives with improved antimycobacterial activity. Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Pompei, R; De Logu, A; Manetti, F; Botta, M. - 04a Atto di comunicazione a congresso
congresso: 10th Drug Development Seminar in conjunction with the COST Action CM0801 (Rauischholzhausen Castle, Germany)
libro: 10th Drug Development Seminar in conjunction with the COST Action CM0801 - ()
11573/172394 - 2009 -
Potent in vitro and in vivo novel 1,5-Diarylpyrrole-3-acetic Esters COX-2 inhibitors. Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Sautebin, L; Patrignani, P; Ghelardini, C; Giordani, A; Anzini, M. - 04a Atto di comunicazione a congresso
congresso: XXIII CONGRESSO NAZIONALE DELLA SOCIETÀ CHIMICA ITALIANA (Sorrento)
libro: XXIII CONGRESSO NAZIONALE DELLA SOCIETÀ CHIMICA ITALIANA - ()
11573/428134 - 2009 -
C-9 Alkenylidine bridged macrolides: WO2008061189. Poce, Giovanna; Porretta, Giulio Cesare; Biava, Mariangela - 01a Articolo in rivista
rivista: EXPERT OPINION ON THERAPEUTIC PATENTS (--London United Kingdom:Informa Healthcare
-London, United Kingdom: Ashley Publications Limited) pp. 901-906 - issn: 1354-3776 - wos: WOS:000267103900010 (2) - scopus: 2-s2.0-67649383643 (2)
11573/55507 - 2009 -
New pyrrole derivatives of BM 212: lead compound optimization strategy, Tuberculosis drug development. Targets, technologies and trials Poce, Giovanna; Porretta, Giulio Cesare; Borzi, F; De Logu, A; De Rossi, E; Manetti, F; Botta, M; Biava, Mariangela - 04a Atto di comunicazione a congresso
congresso: Gordon Conference (Magdalen College, Oxford)
libro: -- - ()
11573/52493 - 2009 -
BM212 and its derivatives: lead optimization of a new class of antimycobacterial agents. Poce, Giovanna; Porretta, Giulio Cesare; De Logu, A; De Rossi, E; Manetti, F; Botta, M; Biava, Mariangela - 04a Atto di comunicazione a congresso
congresso: 10th Drug Development Seminar in conjunction with the COST Action CM0801 (Rauischholzhausen Castle, Germania)
libro: none - ()
11573/228858 - 2008 -
HPLC Enantioseparation and Absolute Configuration of Novel Antiinflammatory Pyrrole Derivatives Biava, Mariangela; Cirilli, R; Fares, V; Ferretti, R; Gallinella, B; Poce, Giovanna; Porretta, Giulio Cesare; Supino, Sibilla; Villani, Claudio - 01a Articolo in rivista
rivista: CHIRALITY (John Wiley & Sons Incorporated:Customer Service, 111 River Street:Hoboken, NJ 07030:(800)225-5945, (201)748-6000, EMAIL: societyinfo@wiley.com, INTERNET: http://www.wiley.com, Fax: (212)748-6551) pp. 775-780 - issn: 0899-0042 - wos: WOS:000256777400003 (12) - scopus: 2-s2.0-45849083178 (13)
11573/368120 - 2008 -
Design and Synthesis of novel diarylpyrroles as p38 MAP kinase inhibitors Biava, Mariangela; Porretta, G. C.; Poce, Giovanna; Giordani, A; Menziani, C. - 04a Atto di comunicazione a congresso
libro: XIX NATIONAL MEETING ON MEDICINAL CHEMISTRY DIVISION OF ITALIAN CHEMICAL SOCIETY (SCI) - ()
11573/367352 - 2008 -
Design and synthesis of 1,5-diaryl-2-ethyl pyrrole derivatives and their evaluation as antimycobacterial agents Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; De Logu, A; Maleddu, R; De Rossi, E; Manetti, F; Botta, M. - 04a Atto di comunicazione a congresso
libro: XIX NATIONAL MEETING ON MEDICINAL CHEMISTRY DIVISION OF ITALIAN CHEMICAL SOCIETY (SCI) - ()
11573/362033 - 2008 -
1,5-Diphenyl Pyrrole Derivatives as Antimycobacterial Agents. Probing the Influence on Antimycobacterial Activity of Lipophilic Substituents at the Phenyl Rings Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; De Logu, A; Saddi, M; Meleddu, R; Manetti, F; De Rossi, E; Botta, M. - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 3644-3648 - issn: 0022-2623 - wos: WOS:000256922800031 (83) - scopus: 2-s2.0-45749084929 (86)
11573/55497 - 2008 -
New derivatives of BM 212 with improved antimycobacterial activity. Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Pompei, R; De Logu, A; Manetti, F; Botta, M. - 04a Atto di comunicazione a congresso
libro: 2nd World Conference on Magic Bullets - ()
11573/228277 - 2008 -
Synthesis, in vitro, and in vivo biological evaluation and molecular docking simulations of chiral alcohol and ether derivatives of the 1,5-diarylpyrrole scaffold as novel anti-inflammatory and analgesic agents Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Sibilla, Supino; Fabrizio, Manetti; Stefano, Forli; Maurizio, Botta; Lidia, Sautebin; Antonietta, Rossi; Carlo, Pergola; Carla, Ghelardini; Monica, Norcini; Francesco, Makovec; Paola, Anzellotti; Roberto, Cirilli; Rosella, Ferretti; Bruno, Gallinella; F., La Torre; Maurizio, Anzini; Paola, Patrignani - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 8072-8081 - issn: 0968-0896 - wos: WOS:000258827800024 (20) - scopus: 2-s2.0-50349084855 (21)
11573/364227 - 2008 -
New oxazolidinone derivatives as antibacterial agents with improved activity Poce, Giovanna; Giovanni, Zappia; Porretta, Giulio Cesare; Botta, Bruno; Biava, Mariangela - 01a Articolo in rivista
rivista: EXPERT OPINION ON THERAPEUTIC PATENTS (--London United Kingdom:Informa Healthcare
-London, United Kingdom: Ashley Publications Limited) pp. 97-121 - issn: 1354-3776 - wos: WOS:000253670500001 (28) - scopus: 2-s2.0-40749136990 (32)
11573/366568 - 2008 -
BM212 and new derivatives as a new class of antimycobacterial agents. Poce, Giovanna; Porretta, G. C.; Borzi, F; De Logu, A; De Rossi, E; Manetti, F; Botta, M; Biava, M. - 04a Atto di comunicazione a congresso
libro: First IRBM workshop on Medicinal & Organic Chemistry. - ()
11573/368289 - 2007 -
New 1,5-diphenyl Pyrrole Derived from BM 212: a New class of Antimycobacterial Agents. Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; De Logu, A; Manetti, F; Botta, M. - 04a Atto di comunicazione a congresso
congresso: TUBERCULOSIS DRUG DEVELOPMENT. GORDON RESEARCH CONFERENCE (OXFORD)
11573/55496 - 2007 -
New 1,5-diarylpyrrole with improved antimycobacterial activity Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; De Logu, A; Saddi, M; Botta, M. - 04a Atto di comunicazione a congresso
libro: XVIII Convegno Nazionale della Divisione di Chimica Farmaceutica della Società Chimica Italiana - ()
11573/492438 - 2007 -
Design, synthesis and screening of new antitubercular agents derived from BM 212 Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Deidda, D.; Pompei, R.; Manetti, F; Botta, M. - 04a Atto di comunicazione a congresso
congresso: VI Laboratorio di Metodologie Sintetiche in Chimica Farmaceutica (Siena)
libro: VI LABORATORIO DI METODOLOGIE SINTETICHE IN CHIMICA FARMACEUTICA - ()
11573/121312 - 2007 -
New pyrroles with potential antimycobacterial, antifungal and COX-2 selective inhibiting activities. Synthetic methodologies Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Supino, S; Sleiter, G. - 01a Articolo in rivista
rivista: CURRENT ORGANIC CHEMISTRY (Bentham Science Publishers BV:PO Box 7917, Exec Ste Y 26, Saif Zone Sharjah Uae:011 971 6 5571132, EMAIL: benthams@emirates.net.ae, INTERNET: http://www.bentham.org, Fax: 011 971 6 5571134) pp. 1092-1112 - issn: 1385-2728 - wos: WOS:000249103400005 (13) - scopus: 2-s2.0-34548247237 (14)
11573/364538 - 2007 -
Cyclooxygenase-2 Inhibitors. 1,5-Diarylpyrrol-3-acetic Esters with Enhanced Inhibitory Activity toward Cyclooxygenase-2 and Improved Cyclooxygenase-2/Cyclooxygenase-1 Selectivity Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Supino, Sibilla; Cappelli, A; Vomero, S; Manetti, F; Botta, M; Sautebin, L; Rossi, A; Ghelardini, C; Vivoli, E; Makovec, F; Anzellotti, P; Patrignani, P; Anzini, M. - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 5403-5411 - issn: 0022-2623 - wos: WOS:000250557100018 (53) - scopus: 2-s2.0-35948946191 (58)
11573/364230 - 2006 -
Antimycobacterial agents. Novel diarylpirrole derivatives of BM212 endowed with high activity toward Mycobacterium tuberculosis and low cytotoxicity Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Supino, S; Deidda, D; Pompei, R; Molicotti, P; Manetti, F; Botta, M. - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 4946-4952 - issn: 0022-2623 - wos: WOS:000239459800018 (116) - scopus: 2-s2.0-33746924405 (126)
11573/52491 - 2006 -
New 1,5-diphenyl pyrrole derived from BM 212: a new class of antimycobacterial Agents Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Supino, S; Pompei, R; Manetti, F; Botta, M. - 04a Atto di comunicazione a congresso
libro: “Tuberculosis 2006" - ()
11573/492426 - 2006 -
Synthesis of new pyrrole derivatives of BM 212, a potent antimycobacterial compound Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Supino, Sibilla; Deidda, D.; Pompei, R.; Manetti, F.; Botta, M. - 04a Atto di comunicazione a congresso
congresso: XXII Convegno Nazionale della Divisione di Chimica Farmaceutica della SCI (Firenze)
libro: Atti del XXII Convegno Nazionale della Divisione di Chimica Farmaceutica della SCI - ()
11573/242012 - 2005 -
ENANTIOMERS OF NOVEL ANTIINFLAMMATORY PYRROLE DERIVATIVES:ANALYTICAL AND SEMIPREPARATIVE HPLC SEPARATION AND CHIROPTICAL PROPERTIES. Biava, Mariangela; Cirilli, R.; Ferretti, R.; Poce, Giovanna; Porretta, Giulio Cesare; Villani, C. . - 04a Atto di comunicazione a congresso
libro: 17th International Symposium on Chiral Discrimination - ()
11573/365959 - 2005 -
Antimycobacterial compounds. Optimization of the BM 212 structure, the lead compound for a new pyrrole derivative class Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Delia, Deidda; Raffaello, Pompei; Andrea, Tafi; Fabrizio, Manetti - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 1221-1230 - issn: 0968-0896 - wos: WOS:000226967900030 (57) - scopus: 2-s2.0-12844266203 (62)
11573/368576 - 2005 -
1,5-DIARYLPYRROLE DERIVATIVESAS NOVEL CLASSES OF ACTIVE AND SELECTIVE COX-2 INHIBITORS. Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Tibuzzi, D; Cappelli, A; Vomero, S; Botta, M; Manetti, F; Sautebin, L; Rossi, A; Makovec, F; Anzini, A. - 04a Atto di comunicazione a congresso
libro: XVIII NATIONAL MEETING OF MEDICINAL CHEMISTRY DIVISION OF ITALIAN CHEMICAL SOCIETY (SCI) - ()
11573/368160 - 2004 -
Nuovi derivati 1,5-difenilpirrolici derivati del BM212 attivi come agenti antitubercolari Biava, M; Porretta, G. C.; Poce, Giovanna; Deidda, D; Pompei, R; Tafi, A; Manetti, F. - 04a Atto di comunicazione a congresso
libro: XVII Convegno Nazionale della Divisione di Chimica Farmaceutica - ()
11573/368453 - 2004 -
1,5-diarylpyrrole-3-acetic acids and esters as novel class of potent and selective COX-2 inhibitors. Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Cappelli, A.; Vomero, S.; Botta, M.; Manetti, F.; Giorni, G.; Sautebin, L.; Rossi, A.; Makovec, F.; Anzini, M. . - 04a Atto di comunicazione a congresso
libro: Twelfth FECHEM Conference on Heterocycles in Bio-organic Chemistry - ()
11573/327339 - 2004 -
1,5-DIARYLPYRROLE-3-ACETIC ACIDS AND ESTERS AS NOVEL CLASSES OF POTENT AND SELECTIVE COX-2 INHIBITORS. Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Cappelli, A; Vomero, S; Botta, M; Manetti, F; Giorni, G; Sautebin, L; Rossi, A; Makovec, F; Anzini, M. - 04a Atto di comunicazione a congresso
libro: CONFERENZA SULLA RICERCA SCIENTIFICA. FACOLTÀ DI FARMACIA . “DALLE MOLECOLE AGLI ORGANISMI” - ()
11573/52488 - 2004 -
Pyrrole Derivatives as New Antimycobacterial Class: Synthesis, S.A.R., Molecular Modelling Considerations and Microbiological Activity Biava, Mariangela; Porretta, Giulio Cesare; Poce, Giovanna; Pompei, R; Deidda, D; Tafi, A.; Manetti, F.; Botta, M. - 04a Atto di comunicazione a congresso
libro: Conferenza sulla Ricerca Scientifica, Facoltà di Farmacia, dalle Molecole agli Organismi - ()