DANIELA SECCI

Professore ordinario


email: daniela.secci@uniroma1.it
telefono: 0649913763
edificio: CU019
stanza: 103

Direttore Dipartimento di Chimica e Tecnologie del Farmaco
Professore ordinario di Chimica Farmaceutica e Tossicologica (Analisi III) e Biotecnologie Farmaceutiche presso la Facoltà di Farmacia e Medicina della Sapienza Università di Roma.
È membro dall'A.A. 2014-2015 del Collegio dei Docenti del Dottorato di Ricerca in Scienze Farmaceutiche.
È referente per la Facoltà di Farmacia e Medicina - Sezione Chimica Farmaceutica delle attività di tirocinio pre e post laurea.
E' responsabile del Laboratorio Chimico per la Sicurezza Sapienza Università di Roma

È coautrice di oltre 145 pubblicazioni e 3 brevetti.

L'attività scientifica riguarda principalmente:
- Separazione mediante stereo HPLC selettiva di molecole chirali biologicamente attive
- Progettazione, sintesi e valutazione biologica di nuovi composti attivi su Helicobacter pylori, su ceppi di Candida e su altri agenti antimicrobici
- Progettazione, sintesi e valutazione biologica di nuovi inibitori selettivi delle monoamino ossidasi, MAO-A e MAO-B
- Progettazione, sintesi e valutazione biologica di nuovi modulatori epigenetici con particolari inibitori dell'acetiltransferasi (HATs) con attività apoptotica e citodifferenziante
- Progettazione, sintesi e valutazione biologica di nuovi inibitori selettivi delle isoforme IX e XII dell'anidrasi carbonica. XII isoforme dell'anidrasi carbonica per il trattamento di patologie tumorali

Responsabile e coordinatore di un Progetto sullo sviluppo e la caratterizzazione di anticorpi monoclonali per uso terapeutico isolati da piante transgeniche attualmente in corso nell'ambito di un progetto di ricerca POR FESR LAZIO.
Responsabile e coordinatore del Progetto Life 2020 NUCFARNA "Nuove classi di farmaci neurologici e antidepressivi, in forma solida orale, orientate sia alla produzione per conto terzi che a nuove AIC, nuove metodologie di processo, supervisione e controllo, e rapida riparametrizzazione su scala pilota - industriale".


Produzione scientifica

11573/1705144 - 2023 - A Multitarget Approach against Neuroinflammation: Alkyl Substituted Coumarins as Inhibitors of Enzymes Involved in Neurodegeneration
Berrino, E.; Carradori, S.; Carta, F.; Melfi, F.; Gallorini, M.; Poli, G.; Tuccinardi, T.; Fernandez-Bolanos, J. G.; Lopez, O.; Petzer, J. P.; Petzer, A.; Guglielmi, P.; Secci, D.; Supuran, C. T. - 01a Articolo in rivista
rivista: ANTIOXIDANTS (Basel: MDPI) pp. 1-25 - issn: 2076-3921 - wos: WOS:001137805100001 (1) - scopus: 2-s2.0-85180511315 (1)

11573/1666710 - 2023 - Novel Insights on CAI–CORM Hybrids: Evaluation of the CO Releasing Properties and Pain-Relieving Activity of Differently Substituted Coumarins for the Treatment of Rheumatoid Arthritis
Berrino, Emanuela; Micheli, Laura; Carradori, Simone; Di Cesare Mannelli, Lorenzo; Guglielmi, Paolo; De Luca, Alessandro; Carta, Fabrizio; Ghelardini, Carla; Secci, Daniela; Supuran, Claudiu T. - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. - - issn: 0022-2623 - wos: WOS:000925733600001 (3) - scopus: 2-s2.0-85147172354 (3)

11573/1691425 - 2023 - Indoleamine 2,3-dioxygenase
Coluccia, Michele; Secci, Daniela; Guglielmi, Paolo - 02a Capitolo o Articolo
libro: Metalloenzymes: from bench to bedside - (9780128239742)

11573/1693714 - 2023 - Kinetic Study on the Base-Catalyzed Imine-Enamine Tautomerism of a Chiral Biologically Active Isoxazoline Derivative by HPLC on Amylose Tris(3,5-dimethylphenylcarbamate) Chiral Stationary Phase
Sadutto, Daniele; Guglielmi, Paolo; Carradori, Simone; Secci, Daniela; Cirilli, Roberto - 01a Articolo in rivista
rivista: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. - - issn: 1420-3049 - wos: WOS:001077830800001 (0) - scopus: 2-s2.0-85172792347 (1)

11573/1659798 - 2022 - Metal-organic frameworks (MOFs) as biomolecules drug delivery systems for anticancer purposes
Coluccia, Michele; Parisse, Valeria; Guglielmi, Paolo; Giannini, Giuseppe; Secci, Daniela - 01g Articolo di rassegna (Review)
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 114801- - issn: 0223-5234 - wos: WOS:000869750800002 (28) - scopus: 2-s2.0-85139304657 (33)

11573/1659799 - 2022 - Treatment of Toxoplasmosis: An Insight on Epigenetic Drugs
Guglielmi, P.; Secci, D. - 02a Capitolo o Articolo
libro: Topics in Medicinal Chemistry - (978-3-031-06849-2; 978-3-031-06850-8)

11573/1654157 - 2022 - Novel Insights on Human Carbonic Anhydrase Inhibitors Based on Coumalic Acid: Design, Synthesis, Molecular Modeling Investigation, and Biological Studies
Pontecorvi, Virginia; Mori, Mattia; Picarazzi, Francesca; Zara, Susi; Carradori, Simone; Cataldi, Amelia; Angeli, Andrea; Berrino, Emanuela; Chimenti, Paola; Ciogli, Alessia; Secci, Daniela; Guglielmi, Paolo; Supuran, Claudiu T. - 01a Articolo in rivista
rivista: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (Basel: MDPI Center) pp. 7950- - issn: 1422-0067 - wos: WOS:000833202300001 (10) - scopus: 2-s2.0-85135137430 (9)

11573/1638205 - 2022 - A comparative study on the suppression capacity and the environmental impact of different extinguishing agents of lithium-ion battery fires
Ubaldi, Sofia; Di Bari, Cinzia; De Rosa, Armando; Quinterno, Mario; Mazzaro, Michele; Ferrigno, Gianluca; Arrighi, Francesca; Secci, Daniela; Russo, Paola - 04b Atto di convegno in volume
congresso: 10th International Seminar on Fire and Explosion Hazards (Oslo, Norway)
libro: Proceedings of the Tenth International Seminar on Fire and Explosion Hazards, 22-27 May 2022, Oslo, Norway - (978-82-7206-721-1)

11573/1649551 - 2021 - An innovative spectroscopic approach for qualitative and quantitative evaluation of Mb-CO from myoglobin carbonylation reaction through chemometrics methods
Mansoldo, F. R. P.; Berrino, E.; Guglielmi, P.; Carradori, S.; Carta, F.; Secci, D.; Supuran, C. T.; Vermelho, A. B. - 01a Articolo in rivista
rivista: SPECTROCHIMICA ACTA. PART A, MOLECULAR AND BIOMOLECULAR SPECTROSCOPY (Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. 0-0 - issn: 1386-1425 - wos: WOS:000786604400018 (2) - scopus: 2-s2.0-85119982751 (3)

11573/1541961 - 2021 - Synthesis and evaluation of thymol-based synthetic derivatives as dual-action inhibitors against different strains of h. pylori and AGS cell line
Sisto, F.; Carradori, S.; Guglielmi, P.; Spano, M.; Secci, D.; Granese, A.; Sobolev, A. P.; Grande, R.; Campestre, C.; Di Marcantonio, M. C.; Mincione, G. - 01a Articolo in rivista
rivista: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. - - issn: 1420-3049 - wos: WOS:000638744400001 (11) - scopus: 2-s2.0-85103863303 (10)

11573/1325133 - 2020 - High-performance liquid chromatography enantioseparation of chiral 2-(benzylsulfinyl)benzamide derivatives on cellulose tris(3,5-dichlorophenylcarbamate) chiral stationary phase
Carradori, S.; Secci, D.; Guglielmi, P.; Pierini, M.; Cirilli, R. - 01a Articolo in rivista
rivista: JOURNAL OF CHROMATOGRAPHY A ([S.l.] : Elsevier Science) pp. - - issn: 1873-3778 - wos: WOS:000509816200026 (6) - scopus: 2-s2.0-85073049872 (6)

11573/1381665 - 2020 - 1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors
D'ascenzio, M.; Secci, D.; Carradori, S.; Zara, S.; Guglielmi, P.; Cirilli, R.; Pierini, M.; Poli, G.; Tuccinardi, T.; Angeli, A.; Supuran, C. T. - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington DC : ACS Publications) pp. 2470-2488 - issn: 1520-4804 - wos: WOS:000526403900042 (34) - scopus: 2-s2.0-85081944311 (41)

11573/1419599 - 2020 - Inhibition of lysine acetyltransferases impairs tumor angiogenesis acting on both endothelial and tumor cells
Di Martile, Marta; Gabellini, Chiara; Desiderio, Marianna; Matraxia, Marta; Farini, Valentina; Valentini, Elisabetta; Carradori, Simone; Ercolani, Cristiana; Buglioni, Simonetta; Secci, Daniela; Andreazzoli, Massimiliano; Del Bufalo And Daniela Trisciuoglio, Donatella - 01a Articolo in rivista
rivista: JOURNAL OF EXPERIMENTAL & CLINICAL CANCER RESEARCH (London : BioMed Central) pp. - - issn: 1756-9966 - wos: WOS:000540407600001 (2) - scopus: 2-s2.0-85086008098 (4)

11573/1449256 - 2020 - Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation
Guglielmi, P.; Rotondi, G.; Secci, D.; Angeli, A.; Chimenti, P.; Nocentini, A.; Bonardi, A.; Gratteri, P.; Carradori, S.; Supuran, C. T. - 01a Articolo in rivista
rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1891-1905 - issn: 1475-6366 - wos: WOS:000574181700001 (11) - scopus: 2-s2.0-85091861178 (13)

11573/1439431 - 2020 - Chalcones: Unearthing their therapeutic possibility as monoamine oxidase B inhibitors
Guglielmi, Paolo; Mathew, Bijo; Secci, Daniela; Carradori, Simone - 01g Articolo di rassegna (Review)
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. - - issn: 0223-5234 - wos: WOS:000578986400016 (56) - scopus: 2-s2.0-85090769924 (63)

11573/1439479 - 2020 - Antimalarial agents from medicinal plant and fungal sources
Luisi, Grazia; Carradori, Simone; Grande, Rossella; Secci, Daniela; Guglielmi, Paolo - 02a Capitolo o Articolo
libro: Plant-derived bioactives. Production, properties and therapeutic applications - (978-981-15-1760-0; 978-981-15-1761-7)

11573/1416201 - 2020 - Metabolic profiling of different wild and cultivated Allium species based on high-resolution mass spectrometry, high-performance liquid chromatography-photodiode array detector, and color analysis
Maccelli, A.; Cesa, S.; Cairone, F.; Secci, D.; Menghini, L.; Chiavarino, B.; Fornarini, S.; Crestoni, M. E.; Locatelli, M. - 01a Articolo in rivista
rivista: JOURNAL OF MASS SPECTROMETRY (John Wiley & Sons Limited:1 Oldlands Way, Bognor Regis, P022 9SA United Kingdom:011 44 1243 779777, EMAIL: cs-journals@wiley.co.uk, INTERNET: http://www.wiley.co.uk, Fax: 011 44 1243 843232) pp. - - issn: 1076-5174 - wos: WOS:000530128000001 (10) - scopus: 2-s2.0-85085141425 (12)

11573/1661131 - 2020 - Innovative pH-interfering agents in association with anticancer agents
Secci, D.; Guglielmi, P. - 02a Capitolo o Articolo
libro: pH-Interfering Agents as Chemosensitizers in Cancer Therapy - (9780128207017)

11573/1575689 - 2020 - Synthesis and biological evaluation of carvacrol-based derivatives as dual inhibitors of H. Pylori strains and ags cell proliferation
Sisto, F.; Carradori, S.; Guglielmi, P.; Traversi, C. B.; Spano, M.; Sobolev, A. P.; Secci, D.; Di Marcantonio, M. C.; Haloci, E.; Grande, R.; Mincione, G. - 01a Articolo in rivista
rivista: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. 1-21 - issn: 1424-8247 - wos: WOS:000594358000001 (19) - scopus: 2-s2.0-85096612970 (20)

11573/1439461 - 2020 - Synthesis and evaluation of a large library of nitroxoline derivatives as pancreatic cancer antiproliferative agents
Veschi, Serena; Carradori, Simone; De Lellis, Laura; Florio, Rosalba; Brocco, Davide; Secci, Daniela; Guglielmi, Paolo; Spano, Mattia; Sobolev, Anatoly P.; Cama, Alessandro - 01a Articolo in rivista
rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1331-1344 - issn: 1475-6366 - wos: WOS:000545146800001 (7) - scopus: 2-s2.0-85087139219 (7)

11573/1349544 - 2019 - Novel approaches to the discovery of selective human monoamine oxidase-B inhibitors: is there room for improvement?
Guglielmi, P.; Carradori, S.; Ammazzalorso, A.; Secci, D. - 01g Articolo di rassegna (Review)
rivista: EXPERT OPINION ON DRUG DISCOVERY (--London United Kingdom:Informa Healthcare -London : Informa Healthcare, 2006-.) pp. 995-1035 - issn: 1746-0441 - wos: WOS:000475153500001 (43) - scopus: 2-s2.0-85070940142 (43)

11573/1237661 - 2019 - Design, synthesis, docking studies and monoamine oxidase inhibition of a small library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1h)-pyrazoles
Guglielmi, Paolo; Carradori, Simone; Poli, Giulio; Secci, Daniela; Cirilli, Roberto; Rotondi, Giulia; Chimenti, Paola; Petzer, Anél; Petzer, Jacobus P. - 01a Articolo in rivista
rivista: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. 1-21 - issn: 1420-3049 - wos: WOS:000458934000108 (20) - scopus: 2-s2.0-85060732811 (24)

11573/1307503 - 2019 - Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity
Guglielmi, Paolo; Secci, Daniela; Petzer, Anél; Bagetta, Donatella; Chimenti, Paola; Rotondi, Giulia; Ferrante, Claudio; Recinella, Lucia; Leone, Sheila; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P; Ortuso, Francesco; Carradori, Simone - 01a Articolo in rivista
rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1511-1525 - issn: 1475-6366 - wos: WOS:000481738100001 (16) - scopus: 2-s2.0-85071029361 (17)

11573/1307498 - 2019 - Design, synthesis and biological activity of selective hCAs inhibitors based on 2-(benzylsulfinyl)benzoic acid scaffold
Rotondi, G.; Guglielmi, P.; Carradori, S.; Secci, D.; De Monte, C.; De Filippis, B.; Maccallini, C.; Amoroso, R.; Cirilli, R.; Akdemir, A.; Angeli, A.; Supuran, C. T. - 01a Articolo in rivista
rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1400-1413 - issn: 1475-6366 - wos: WOS:000480545500001 (20) - scopus: 2-s2.0-85070919829 (22)

11573/1237670 - 2019 - 4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis
Secci, Daniela; Carradori, Simone; Petzer, Anél; Guglielmi, Paolo; D’Ascenzio, Melissa; Chimenti, Paola; Bagetta, Donatella; Alcaro, Stefano; Zengin, Gokhan; Petzer, Jacobus P.; Ortuso, Francesco - 01a Articolo in rivista
rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 597-612 - issn: 1475-6366 - wos: WOS:000457961800001 (33) - scopus: 2-s2.0-85061130350 (36)

11573/1351315 - 2019 - Investigation on the stability of new biologically active thiosemicarbazone-derived compounds by a validated HPLC-PDA method
Secci, Daniela; Locatelli, Marcello; Kabir, Abuzar; Salvatorelli, Erika; Macedonio, Giorgia; Mollica And Simone Carradori, Adriano - 01a Articolo in rivista
rivista: CURRENT ANALYTICAL CHEMISTRY (Netherlands Hilversum : Bentham Science Publishers) pp. 313-320 - issn: 1573-4110 - wos: WOS:000467020900011 (2) - scopus: 2-s2.0-85065572006 (2)

11573/1121984 - 2018 - Magnetic metal−organic framework composite by fast and facile mechanochemical process
Bellusci, M.; Guglielmi, P.; Masi, Andrea; Padella, F.; Singh, G.; Yaacoub, N.; Peddis, D.; Secci, D. - 01a Articolo in rivista
rivista: INORGANIC CHEMISTRY (Washington, D.C. : American Chemical Society, c1962-) pp. 1806-1814 - issn: 1520-510X - wos: WOS:000426014800016 (52) - scopus: 2-s2.0-85042209909 (55)

11573/1212530 - 2018 - Atriplex mollis desf. Aerial parts: extraction procedures, secondary metabolites and color analysis
Boutaoui, Nassima; Zaiter, Lahcene; Benayache, Fadila; Benayache, Samir; Cacciagrano, Francesco; Cesa, Stefania; Secci, Daniela; Carradori, Simone; Giusti, Anna Maria; Campestre, Cristina; Menghini, Luigi; Locatelli, Marcello - 01a Articolo in rivista
rivista: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. 1-12 - issn: 1420-3049 - wos: WOS:000445295500127 (12) - scopus: 2-s2.0-85052379374 (14)

11573/1068937 - 2018 - Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents
Carradori, Simone; Ottuso, Francesco; Petzer, Anèl; Bagetta, Donatella; De Monte, Celeste; Secci, Daniela; De Vita, Daniela; Guglielmi, Paolo; Zengin, Gokhan; Aktumsek, Abdurrahman; Alcaro, Stefano; Petzer, Jacobus P. - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY ([Paris] : Elsevier, [198?]-) pp. 1543-1552 - issn: 1768-3254 - wos: WOS:000423641400032 (38) - scopus: 2-s2.0-85034651451 (40)

11573/1020963 - 2018 - A chromatographic study on the exceptional chiral recognition of 2-(benzylsulfinyl)benzamide by animmobilized-type chiral stationary phase based on cellulose tris(3,5-dichlorophenylcarbamate)
Carradori, Simone; Secci, Daniela; Faggi, Cristina; Cirilli, Roberto - 01a Articolo in rivista
rivista: JOURNAL OF CHROMATOGRAPHY A (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598) pp. 151-156 - issn: 0021-9673 - wos: WOS:000423651300016 (16) - scopus: 2-s2.0-85035053170 (17)

11573/1068947 - 2018 - MAO inhibitors and their wider applications: a patent review
Carradori, Simone; Secci, Daniela; Petzer, Jacques P. - 01g Articolo di rassegna (Review)
rivista: EXPERT OPINION ON THERAPEUTIC PATENTS (--London United Kingdom:Informa Healthcare -London, United Kingdom: Ashley Publications Limited) pp. 211-226 - issn: 1354-3776 - wos: WOS:000424996100005 (84) - scopus: 2-s2.0-85041925798 (85)

11573/1017594 - 2018 - Bioactive isoflavones from Pueraria lobata root and starch: Different extraction techniques and carbonic anhydrase inhibition
Mocan, Andrei; Carradori, Simone; Locatelli, Marcello; Secci, Daniela; Cesa, Stefania; Mollica, Adriano; Riga, Simona; Angeli, Andrea; Supuran, Claudiu T.; Celia, Christian; Di Marzio, Luisa - 01a Articolo in rivista
rivista: FOOD AND CHEMICAL TOXICOLOGY (Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. 441-447 - issn: 0278-6915 - wos: WOS:000425568900050 (39) - scopus: 2-s2.0-85027395216 (41)

11573/1007387 - 2017 - Synthesis, biological evaluation and quantitative structure-active relationships of 1,3-thiazolidin-4-one derivatives. A promising chemical scaffold endowed with high antifungal potency and low cytotoxicity
Carradori, Simone; Bizzarri, Bruna; D'ascenzio, Melissa; De Monte, Celeste; Grande, Rossella; Rivanera, Daniela; Zicari, Alessanda; Mari, Emanuela; Sabatino, Manuela; Patsilinakos, Alexandros; Ragno, Rino; Secci, Daniela - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 274-292 - issn: 0223-5234 - wos: WOS:000414620000022 (19) - scopus: 2-s2.0-85030121237 (19)

11573/974029 - 2017 - Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives
Carradori, Simone; Secci, Daniela; Bizzarri, Bruna; Chimenti, Paola; De Monte, Celeste; Guglielmi, Paolo; Campestre, Cristina; Rivanera, Daniela; Bordón, Claudia; Jones Brando, Lorraine - 01a Articolo in rivista
rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 746-758 - issn: 1475-6366 - wos: WOS:000404271200001 (22) - scopus: 2-s2.0-85019985742 (22)

11573/1017595 - 2017 - Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms
D'ascenzio, M.; Guglielmi, P.; Carradori, S.; Secci, D.; Florio, R.; Mollica, A.; Ceruso, M.; Akdemir, A.; Sobolev, A. P.; Supuran, C. T. - 01a Articolo in rivista
rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 51-59 - issn: 1475-6366 - wos: WOS:000392591100044 (43) - scopus: 2-s2.0-84992390041 (46)

11573/1017583 - 2017 - Protective effects Induced by microwave-assisted aqueous harpagophytum extract on rat cortex synaptosomes challenged with amyloid β-peptide
Ferrante, Claudio; Recinella, Lucia; Locatelli, Marcello; Guglielmi, Paolo; Secci, Daniela; Leporini, Lidia; Chiavaroli, Annalisa; Leone, Sheila; Martinotti, Sara; Brunetti, Luigi; Vacca, Michele; Meneghini, Luigi; Orlando, Giustino - 01a Articolo in rivista
rivista: PHYTOTHERAPY RESEARCH (New York : J. Wiley) pp. 1257-1264 - issn: 1099-1573 - wos: WOS:000406926800015 (48) - scopus: 2-s2.0-85021271246 (49)

11573/1017599 - 2017 - Optimization of aqueous extraction and biological activity of harpagophytum procumbens root on ex vivo rat Colon inflammatory model
Locatelli, Marcello; Ferrante, Claudio; Carradori, Simone; Secci, Daniela; Leporini, Lidia; Chiavaroli, Annalisa; Leone, Sheila; Recinella, Lucia; Orlando, Giustino; Martinotti, Sara; Brunetti, Luigi; Vacca And Luigi Menghini, Michele - 01a Articolo in rivista
rivista: PHYTOTHERAPY RESEARCH (John Wiley & Sons Limited:1 Oldlands Way, Bognor Regis, P022 9SA United Kingdom:011 44 1243 779777, EMAIL: cs-journals@wiley.co.uk, INTERNET: http://www.wiley.co.uk, Fax: 011 44 1243 843232) pp. 937-944 - issn: 0951-418X - wos: WOS:000402958900013 (54) - scopus: 2-s2.0-85018244260 (55)

11573/925013 - 2017 - Geographical characterization by MAE-HPLC and NIR methodologies and carbonic anhydrase inhibition of Saffron components
Nescatelli, Riccardo; Carradori, Simone; Marini, Federico; Caponigro, Vicky; Bucci, Remo; De Monte, Celeste; Mollica, Adriano; Mannina, Luisa; Ceruso, Mariangela; Supuran, Claudiu Trandafir; Secci, Daniela - 01a Articolo in rivista
rivista: FOOD CHEMISTRY (Elsevier Applied Science:An Imprint of Elsevier Science Ltd, The Boulevard, Langford Lane, Kidlington Oxford OX5 1GB United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: nlinfo-f@elsevier.nl OR usinfo-f@elsevier.com OR forinfo-kyf04035@niftyserve.or.jp, INTERNET: http://www.elsevier.nl/, Fax: 011 44 1865 843010) pp. 855-863 - issn: 0308-8146 - wos: WOS:000389909100109 (41) - scopus: 2-s2.0-85006804608 (51)

11573/955974 - 2017 - 3-(Phenyl-4-oxy)-5-phenyl-4,5-dihydro-(1H)-pyrazole: a fascinating molecular framework to study the enantioseparation ability of the amylose (3,5-dimethylphenylcarbamate) chiral stationary phase. Part II. Solvophobic effects in enantiorecognition process
Pierini, Marco; Carradori, Simone; Menta, Sergio; Secci, Daniela; Cirilli, Roberto - 01a Articolo in rivista
rivista: JOURNAL OF CHROMATOGRAPHY A ([S.l.] : Elsevier Science) pp. 140-148 - issn: 1873-3778 - wos: WOS:000401394200014 (23) - scopus: 2-s2.0-85017477051 (24)

11573/1017596 - 2017 - Neem oil nanoemulsions: characterisation and antioxidant activity
Rinaldi, Federica; Hanieh, Patrizia Nadia; Longhi, Catia; Carradori, Simone; Secci, Daniela; Zengin, Gokhan; Grazia Ammendolia, Maria; Mattia, Elena; Del Favero, Elena; Marianecci, Carlotta; Carafa, Maria - 01a Articolo in rivista
rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1265-1273 - issn: 1475-6366 - wos: WOS:000413901300001 (44) - scopus: 2-s2.0-85030480751 (50)

11573/894544 - 2016 - 3-(Phenyl-4-oxy)-5-phenyl-4,5-dihydro-(1H)-pyrazole: a fascinating molecular framework to study the enantioseparation ability of the amylose (3,5-dimethylphenylcarbamate) chiral stationary phase. Part I. Structure-enantioselectivity relationships
Carradori, Simone; Pierini, Marco; Menta, Sergio; Secci, Daniela; Fioravanti, Rossella; Cirilli, Roberto - 01a Articolo in rivista
rivista: JOURNAL OF CHROMATOGRAPHY A ([S.l.] : Elsevier Science) pp. 221-227 - issn: 1873-3778 - wos: WOS:000385323800017 (12) - scopus: 2-s2.0-84991112085 (13)

11573/851467 - 2016 - A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms
Carradori, Simone; Secci, Daniela; De Monte, Celeste; Mollica, Adriano; Ceruso, Mariangela; Akdemir, Atilla; Sobolev, Anatoly P; Codispoti, Rossella; De Cosmi, Federica; Guglielmi, Paolo; Supuran, Claudiu T. - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 1095-1105 - issn: 0968-0896 - wos: WOS:000369989500020 (44) - scopus: 2-s2.0-84957841303 (51)

11573/851468 - 2016 - Anti-Candida activity and cytotoxicity of a large library of new N-substituted-1,3-thiazolidin-4-one derivatives
De Monte, Celeste; Carradori, Simone; Bizzarri, Bruna; Bolasco, Adriana; Caprara, Federica; Mollica, Adriano; Rivanera, Daniela; Mari, Emanuela; Zicari, Alessandra; Akdemir, Atilla; Secci, Daniela - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 82-96 - issn: 0223-5234 - wos: WOS:000366780500007 (47) - scopus: 2-s2.0-84946782497 (48)

11573/884170 - 2016 - Histone acetyltransferase inhibitor CPTH6 preferentially targets lung cancer stem-like cells
Di Martile, Marta; Desideri, Marianna; De Luca, Teresa; Gabellini, Chiara; Buglioni, Simonetta; Eramo, Adriana; Sette, Giovanni; Milella, Michele Stanislaw; Rotili, Dante; Mai, Antonello; Carradori, Simone; Secci, Daniela; De Maria, Ruggero; Del Bufalo, Donatella; Trisciuoglio, Daniela - 01a Articolo in rivista
rivista: ONCOTARGET (Albany, N.Y. : Impact Journals) pp. 11332-11348 - issn: 1949-2553 - wos: WOS:000375678300047 (36) - scopus: 2-s2.0-84962019515 (37)

11573/1019004 - 2016 - Identification of new anti-Candida compounds by ligand-based pharmacophore virtual screening
Gidaro, Concetta; Alcaro, Stefano; Secci, Daniela; Rivanera, Daniela; Mollica, Adriano; Agamennone, Mariangela; Giampietro, Letizia; Simone Carradori, And - 01a Articolo in rivista
rivista: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1703-1706 - issn: 1475-6366 - wos: WOS:000385270300112 (15) - scopus: 2-s2.0-84961204488 (20)

11573/894545 - 2016 - Elucidation of the mechanisms governing the thermal diastereomerization of bioactive chiral 1,3,4-thiadiazoline spiro-cyclohexyl derivatives towards their anancomeric stereoisomers
Menta, Sergio; Carradori, S.; Siani, G.; Secci, Daniela; Mannina, Luisa; Sobolev, A. P.; Cirilli, R; Pierini, Marco - 01a Articolo in rivista
rivista: RSC ADVANCES (London: Royal Society of Chemistry) pp. 71262-71272 - issn: 2046-2069 - wos: WOS:000381513100064 (1) - scopus: 2-s2.0-84979955372 (1)

11573/906767 - 2016 - Novel 1,3-thiazolidin-4-one derivatives as promising anti-Candida agents endowed with anti-oxidant and chelating properties
Secci, Daniela; Simone, Carradori; Bizzarri, Bruna; Chimenti, Paola; De Monte, Celeste; Adriano, Mollica; Rivanera, Daniela; Zicari, Alessandra; Emanuela, Mari; Gokhan, Zengin; Abdurrahman, Aktumsek - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 144-156 - issn: 0223-5234 - wos: WOS:000376837800012 (41) - scopus: 2-s2.0-84963811487 (46)

11573/951918 - 2015 - Optimization of the microwave-assisted extraction of Azadirachta indica (Neem) leaves Using NMR-based metabolic fingerprinting
Carradori, Simone; Mannina, Luisa; Cosmi, Federica De; Beccarini, Tamara; Secci, Daniela; Sobolevb, Anatoly P. - 01a Articolo in rivista
rivista: CURRENT BIOACTIVE COMPOUNDS (Netherlands Hilversum : Bentham Science Publishers) pp. 142-145 - issn: 1573-4072 - wos: (0) - scopus: 2-s2.0-84947923031 (5)

11573/684853 - 2015 - Out of the active site binding pocket for carbonic anhydrase inhibitors
D'ambrosio, K.; Carradori, S.; Monti, Sm; Buonanno, M.; Secci, Daniela; Vullo, D.; Supuran, Ct; De Simone, G. - 01a Articolo in rivista
rivista: CHEMICAL COMMUNICATIONS (Royal Society of Chemistry:Thomas Graham House, Science Park, Cambridge CB4 0WF United Kingdom:011 44 1223 432360, EMAIL: sales@rsc.org, INTERNET: http://www.rsc.org, http://www.chensoc.org, Fax: 011 44 1223 423429) pp. 302-305 - issn: 1359-7345 - wos: WOS:000345975000012 (99) - scopus: 2-s2.0-84916227702 (109)

11573/851466 - 2015 - Synthesis and pharmacological screening of a large library of 1,3,4-thiadiazolines as innovative therapeutic tools for the treatment of prostate cancer and melanoma
De Monte, Celeste; Carradori, Simone; Secci, Daniela; D'ascenzio, Melissa; Guglielmi, Paolo; Mollica, Adriano; Morrone, Stefania; Scarpa, Susanna; Agliano', Anna Maria; Giantulli, Sabrina; Silvestri, Ida - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 245-262 - issn: 0223-5234 - wos: WOS:000364891400017 (30) - scopus: 2-s2.0-84944886329 (33)

11573/759322 - 2015 - Metal-chelating salens and tetrahydrosalens and N- and O-substituted acesulfame and saccharin derivatives as selective inhibitors of the cancer-related carbonic anhydrases IX and XII
De Monte, Celeste; Secci, Daniela; Simone, Carradori; Melissa, D’Ascenzio; Mariana, Farella; Claudiu T., Supuran - 04f Poster

11573/837591 - 2015 - The anancomeric character of the pharmacophore 1,3,4-thiadiazoline framework in chiral spiro-cyclohexyl derivatives: effects on stereochemistry and spiro-junction lability. Thermodynamic aspects
Menta, Sergio; Carradori, Simone; Secci, Daniela; Faggi, Cristina; Mannina, Luisa; Cirilli, Roberto; Pierini, Marco - 01a Articolo in rivista
rivista: JOURNAL OF ORGANIC CHEMISTRY ([Washington, D.C: American Chemical Society) pp. 11932-11940 - issn: 0022-3263 - wos: WOS:000366877900004 (7) - scopus: 2-s2.0-84952705860 (6)

11573/685071 - 2014 - Evaluation of a large library of (thiazol-2-yl)hydrazones and analogues as histone acetyltransferase inhibitors: Enzyme and cellular studies.
Carradori, S; Rotili, Dante; De Monte, Celeste; Lenoci, A; D'ascenzio, M; Rodriguez, V; Filetici, Patrizia; Miceli, M; Nebbioso, A; Altucci, L; Secci, Daniela; Mai, Antonello - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 569-578 - issn: 0223-5234 - wos: WOS:000337985400049 (46) - scopus: 2-s2.0-84900559630 (51)

11573/685054 - 2014 - Microwave and Ultrasound-Assisted Synthesis of Thiosemicarbazones and Their Corresponding (4,5-Substituted-thiazol-2-yl)hydrazines
Carradori, S; Secci, Daniela; D'ascenzio, M; Chimenti, Paola; Bolasco, Adriana - 01a Articolo in rivista
rivista: JOURNAL OF HETEROCYCLIC CHEMISTRY (Hetero Corporation:PO Box 170:Provo, UT 84603:(801)400-7373, EMAIL: jhetchem@yahoo.com, Fax: (801)356-7373) pp. 1856-1861 - issn: 0022-152X - wos: WOS:000345457700043 (13) - scopus: 2-s2.0-84915737550 (15)

11573/543217 - 2014 - Selective MAO-B inhibitors: a lesson from natural products
Carradori, Simone; D'ascenzio, Melissa; Chimenti, Paola; Secci, Daniela; Bolasco, Adriana - 01a Articolo in rivista
rivista: MOLECULAR DIVERSITY (Kluwer Academic Publishers:Journals Department, PO Box 322, 3300 AH Dordrecht Netherlands:011 31 78 6576050, EMAIL: frontoffice@wkap.nl, kluweronline@wkap.nl, INTERNET: http://www.kluwerlaw.com, Fax: 011 31 78 6576254) pp. 219-243 - issn: 1381-1991 - wos: WOS:000330978900018 (109) - scopus: 2-s2.0-84894081989 (122)

11573/685073 - 2014 - Design, synthesis and evaluation of N-substituted saccharin derivatives as selective inhibitors of tumor-associated carbonic anhydrase XII
D'ascenzio, M; Carradori, S; De Monte, Celeste; Secci, Daniela; Ceruso, M; Supuran, Ct - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 1821-1831 - issn: 0968-0896 - wos: WOS:000332409700004 (73) - scopus: 2-s2.0-84896720529 (77)

11573/685072 - 2014 - Identification of the stereochemical requirements in the 4-aryl-2-cycloalkylidenhydrazinylthiazole scaffold for the design of selective human monoamine oxidase B inhibitors
D'ascenzio, M; Carradori, S; Secci, Daniela; Mannina, Luisa; Sobolev, Ap; De Monte, Celeste; Cirilli, R; Yanez, M; Alcaro, S; Ortuso, F. - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 2887-2895 - issn: 0968-0896 - wos: WOS:000334744500006 (23) - scopus: 2-s2.0-84899498676 (24)

11573/685062 - 2014 - Selective inhibition of human carbonic anhydrases by novel amide derivatives of probenecid: Synthesis, biological evaluation and molecular modelling studies
D'ascenzio, M; Carradori, S; Secci, Daniela; Vullo, D; Ceruso, M; Akdemir, A; Supuran, Ct - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 3982-3988 - issn: 0968-0896 - wos: WOS:000339859700021 (36) - scopus: 2-s2.0-84905087830 (39)

11573/685057 - 2014 - Design, synthesis and biological characterization of thiazolidin-4-one derivatives as promising inhibitors of Toxoplasma gondii
D'ascenzio, Melissa; Bizzarri, Bruna; De Monte, Celeste; Carradori, S; Bolasco, Adriana; Secci, Daniela; Rivanera, Daniela; Faulhaber, N; Bordon, C; Jones Brando, L. - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 17-30 - issn: 0223-5234 - wos: WOS:000343781800003 (38) - scopus: 2-s2.0-84906328264 (43)

11573/685066 - 2014 - New insights into the biological properties of Crocus sativus L.: chemical modifications, human monoamine oxidases inhibition and molecular modeling studies
De Monte, Celeste; Carradori, Simone; Chimenti, Paola; Secci, Daniela; Mannina, Luisa; Alcaro, F; Petzer, A; N'da, Ci; Gidaro, Mc; Costa, G; Alcaro, S; Petzer, Jp - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 164-171 - issn: 0223-5234 - wos: WOS:000339039100014 (52) - scopus: 2-s2.0-84902213282 (58)

11573/685059 - 2014 - Cyclic tertiary sulfamates: Selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives
De Monte, Celeste; Carradori, Simone; Secci, Daniela; D'ascenzio, Melissa; Vullo, D; Ceruso, M; Supuran, Ct - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 240-246 - issn: 0223-5234 - wos: WOS:000341464500024 (36) - scopus: 2-s2.0-84904288691 (42)

11573/556417 - 2014 - Quinoline-based p300 histone acetyltransferase inhibitors with pro-apoptotic activity in human leukemia U937 cells.
Lenoci, Alessia; Tomassi, S; Conte, M; Benedetti, R; Rodriguez, V; Carradori, Simone; Secci, Daniela; Castellano, S; Sbardella, G; Filetici, P; Novellino, E; Altucci, L; Rotili, Dante; Mai, Antonello - 01a Articolo in rivista
rivista: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. 542-548 - issn: 1860-7187 - wos: WOS:000331795500010 (26) - scopus: 2-s2.0-84896698147 (27)

11573/543220 - 2014 - Effect of the water content on the retention and enantioselectivity of albendazole and fenbendazole sulfoxides using amylose-based chiral stationary phases in organic-acqueous conditions
Materazzo, S.; Carradori, Simone; Ferretti, R.; Gallinella, B.; Secci, Daniela; Cirilli, R. - 01a Articolo in rivista
rivista: JOURNAL OF CHROMATOGRAPHY A (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598) pp. 73-79 - issn: 0021-9673 - wos: WOS:000330910800009 (35) - scopus: 2-s2.0-84892560781 (35)

11573/543278 - 2014 - Synthesis of a novel series of thiazole-based histone acetyltransferase inhibitors
Secci, Daniela; Carradori, S.; Bizzarri, Bruna; Bolasco, Adriana; Ballario, Paola; Patramani, Z.; Fragapane, P.; Vernarecci, S.; Canzonetta, C.; Filetici, P. - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 1680-1689 - issn: 0968-0896 - wos: WOS:000331729500018 (53) - scopus: 2-s2.0-84896716604 (56)

11573/541247 - 2013 - Salen and tetrahydrosalen derivatives act as effective inhibitors of the tumor-associated carbonic anhydrase XII—A new scaffold for designing isoform-selective inhibitors
Carradori, Simone; De Monte, Celeste; D'ascenzio, Melissa; Secci, Daniela; Gulsah, Celik; Mariangela, Ceruso; Daniela, Vullo; Andrea, Scozzafava; Claudiu T., Supuran - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 6759-6763 - issn: 0960-894X - wos: WOS:000327787700044 (45) - scopus: 2-s2.0-84888883083 (44)

11573/555510 - 2013 - Exploring (4-substituted-thiazol-2-yl)hydrazine derivatives of 2-, 3-, and 4-acetylpyridine as selective and reversible hMAO-B inhibitors.
Chimenti, Paola; Petzer, A.; Carradori, S.; D’Ascenzio, M.; Silvestri, Romano; Alcaro, S.; Ortuso, F.; Petzer, J. J.; Secci, Daniela - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 221-227 - issn: 0223-5234 - wos: WOS:000323628500024 (24) - scopus: 2-s2.0-84879467536 (24)

11573/741401 - 2013 - New thiadiazoline and thiadiazole analogues of K858: antiproliferative activity in a model of prostate carcinoma
De Monte, Celeste; Carradori, S.; D’Ascenzio, M.; Chimenti, Paola; Secci, Daniela; Bolasco, Adriana; Nicolazzo, Chiara; Silvestri, Ida - 04f Poster
congresso: 22nd National Meeting on Medicinal Chemistry (Roma)

11573/510197 - 2013 - The thiazole derivative CPTH6 impairs autophagy
Ragazzoni, Ylenia; M., Desideri; C., Gabellini; T., De Luca; Carradori, Simone; Secci, Daniela; Nescatelli, Riccardo; A., Candiloro; M., Condello; S., Meschini; D., Del Bufalo; D., Trisciuoglio - 01a Articolo in rivista
rivista: CELL DEATH & DISEASE (Nature Group) pp. 1-11 - issn: 2041-4889 - wos: WOS:000316868700003 (23) - scopus: 2-s2.0-84875897854 (29)

11573/541244 - 2013 - Synthesis and Selective Human Monoamine Oxidase B Inhibition of Heterocyclic Hybrids Based on Hydrazine and Thiazole Scaffolds
Simone, Carradori; Melissa, D'ascenzio; De Monte, Celeste; Secci, Daniela; Matilde, Yáñez - 01a Articolo in rivista
rivista: ARCHIV DER PHARMAZIE (Wiley-VCH Verlag GmBH:PO Box 101161, D 69451 Weinheim Germany:011 49 6201 606147, EMAIL: service@wiley-vch.de, INTERNET: http://www.wiley-vch.de, Fax: 011 49 6201 606328) pp. 17-22 - issn: 0365-6233 - wos: WOS:000313692000003 (20) - scopus: 2-s2.0-84872226218 (22)

11573/525671 - 2013 - Synthesis and cytotoxicity of novel (thiazol-2-yl)hydrazine derivatives as promising anti-Candida agents
Simone, Carradori; Secci, Daniela; Bolasco, Adriana; Rivanera, Daniela; Mari, Emanuela; Zicari, Alessandra; Lotti, Lavinia Vittoria; Bizzarri, Bruna - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 102-111 - issn: 0223-5234 - wos: WOS:000322850100011 (42) - scopus: 2-s2.0-84878008229 (45)

11573/514588 - 2013 - tert-Butylcarbamate-Containing Histone Deacetylase Inhibitors: Apoptosis Induction, Cytodifferentiation, and Antiproliferative Activities in Cancer Cells.
Valente, Sergio; Trisciuoglio, D; Tardugno, M; Benedetti, R; Labella, Donatella; Secci, Daniela; Mercurio, C; Boggio, R; Tomassi, S; Di Maro, S; Novellino, E; Altucci, L; Del Bufalo, D; Mai, Antonello; Cosconati, S. - 01a Articolo in rivista
rivista: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. - - issn: 1860-7179 - wos: WOS:000318245300013 (15) - scopus: 2-s2.0-84877064105 (17)

11573/495764 - 2012 - MANGANESE IRON OXIDE SUPERPARAMAGNETIC POWDER BY MECHANOCHEMICAL PROCESSING. NANOPARTICLES FUNCTIONALIZATION AND DISPERSION IN A NANOFLUID
Bellusci, Mariangela; Aliotta, C.; Fiorani, D.; La Barbera, A.; Padella, F.; Peddis, D.; Pilloni, M.; Secci, Daniela - 01a Articolo in rivista
rivista: JOURNAL OF NANOPARTICLE RESEARCH (KLUWER ACADEMIC PUBL, VAN GODEWIJCKSTRAAT 30, DORDRECHT, NETHERLANDS, 3311 GZ) pp. 1-11 - issn: 1388-0764 - wos: WOS:000305328900034 (23) - scopus: 2-s2.0-84861742743 (24)

11573/495773 - 2012 - 3-Methylcyclohexanone thiosemicarbazone: Determination of E/Z isomerization barrier by dynamic high-performance liquid chromatography, configuration assignment and theoretical study of the mechanisms involved by the spontaneous, acid and base catalyzed processes
Carradori, Simone; Cirilli, R.; Dei Cicchi, S.; Ferretti, R.; Menta, Sergio; Pierini, Marco; Secci, Daniela - 01a Articolo in rivista
rivista: JOURNAL OF CHROMATOGRAPHY A (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598) pp. 168-177 - issn: 0021-9673 - wos: WOS:000312475300012 (18) - scopus: 2-s2.0-84870314704 (20)

11573/431875 - 2012 - Current and emerging strategies in bladder cancer
Carradori, Simone; Cristini, Cristiano; Secci, Daniela; Caterina, Gulia; Gentile, Vincenzo; Di Pierro, Giovanni Battista - 01a Articolo in rivista
rivista: ANTI-CANCER AGENTS IN MEDICINAL CHEMISTRY (Hilversum : Bentham Science Publishers) pp. 589-603 - issn: 1871-5206 - wos: WOS:000309069000002 (13) - scopus: 2-s2.0-84861678087 (13)

11573/458519 - 2012 - Patent-related survey on new monoamine oxidase inhibitors and their therapeutic potential
Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; D'ascenzio, Melissa - 01a Articolo in rivista
rivista: EXPERT OPINION ON THERAPEUTIC PATENTS (--London United Kingdom:Informa Healthcare -London, United Kingdom: Ashley Publications Limited) pp. 759-801 - issn: 1354-3776 - wos: WOS:000305583200004 (47) - scopus: 2-s2.0-84862867905 (48)

11573/510189 - 2012 - CPTH6, a thiazole derivative, induces histone hypoacetylation and apoptosis in human leukemia cells
D., Trisciuoglio; Ragazzoni, Ylenia; A., Pelosi; M., Desideri; Carradori, Simone; C., Gabellini; G., Maresca; Nescatelli, Riccardo; Secci, Daniela; Bolasco, Adriana; Bizzarri, Bruna; Cavaliere, Chiara; I., D'agnano; Filetici, Patrizia; L., Ricci Vitiani; M. G., Rizzo; D., Del Bufalo - 01a Articolo in rivista
rivista: CLINICAL CANCER RESEARCH (American Association of Cancer Research:150 South Independence Mall West, #826:Philadelphia, PA 19106:(215)440-9300, EMAIL: pubs@aacr.org, INTERNET: http://www.aacr.org, Fax: (215)440-7228) pp. 475-486 - issn: 1078-0432 - wos: WOS:000299320800017 (44) - scopus: 2-s2.0-84856001321 (47)

11573/510205 - 2012 - Modulation of Autophagic Flux by CPTH6, a Gcn5/pCAF Histone Acetyltransferase Inhibitor With Antitumoral Activity
D., Trisciuoglio; Ragazzoni, Ylenia; M., Desideri; C., Gabellini; Nescatelli, Riccardo; Carradori, Simone; Secci, Daniela; D., Del Bufalo - 04d Abstract in atti di convegno
rivista: EUROPEAN JOURNAL OF CANCER (Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. S232-S232 - issn: 0959-8049 - wos: WOS:000313036501427 (0) - scopus: (0)
congresso: 22nd Biennial Congress of the EUROPEAN ASSOCIATION FOR CANCER RESEARCH.From Basic Research to Personalised Cancer Treatment (Barcellona)

11573/455324 - 2012 - Synthesis and biological assessment of novel 2-thiazolylhydrazones and computational analysis of their recognition by monoamine oxidase B
Distinto, S; Yáñez, M; Alcaro, S.; Cardia M., C; Gaspari, M; Sanna M., L; Meleddu, R; Ortuso, F; Kirchmair, J; Markt, P; Bolasco, Adriana; Wolber, G; Secci, Daniela; Maccioni, E. - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 284-295 - issn: 0223-5234 - wos: WOS:000300484900029 (31) - scopus: 2-s2.0-84855994429 (38)

11573/510201 - 2012 - Modulation of autophagic flux by CPTH6, a thiazole derivative with antitumoral activity
Ragazzoni, Ylenia; M., Desideri; C., Gabellini; Carradori, Simone; Nescatelli, Riccardo; Secci, Daniela; A., Candiloro; D., Trisciuoglio; D., Del Bufalo - 04a Atto di comunicazione a congresso
congresso: 25° Convegno Annuale dell’Associazione Italiana di Colture Cellulari (ONLUS-AICC) 3rd International Satellite Symposium AICC–GISM."Controllo dei processi di proliferazione e morte cellulare: nuovi sviluppi della ricerca oncologica preclinica" (Palermo)

11573/733888 - 2012 - Synthesis and selective inhibitory activity against human COX-1 of novel 1-(4-substituted-thiazol-2-yl)-3,5-di(hetero)aryl-pyrazoline derivatives.
S., Carradori; Secci, Daniela; Bolasco, Adriana; De Monte, Celeste; M., Yanez - 01a Articolo in rivista
rivista: ARCHIV DER PHARMAZIE (Weinheim: Wiley-VCH.) pp. 973-979 - issn: 1521-4184 - wos: WOS:000312159900007 (23) - scopus: 2-s2.0-84870558988 (28)

11573/455358 - 2012 - Synthesis, anti-Candida activity, and cytotoxicity of new (4-(4-iodophenyl)thiazol-2-yl)hydrazine derivatives
Secci, Daniela; Bizzarri, Bruna; Bolasco, Adriana; Simone, Carradori; D'ascenzio, Melissa; Rivanera, Daniela; Mari, Emanuela; Polletta, Lucia; Zicari, Alessandra - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 246-253 - issn: 0223-5234 - wos: WOS:000305863100026 (49) - scopus: 2-s2.0-84861626316 (49)

11573/508325 - 2012 - Recent advances in the development of selective human MAO-B inhibitors: (Hetero)arylidene-(4-substituted-thiazol-2- yl)hydrazines
Secci, Daniela; Bolasco, Adriana; Carradori, Simone; D'ascenzio, Melissa; Nescatelli, Riccardo; M., Yáñez - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 405-417 - issn: 0223-5234 - wos: WOS:000312745100043 (39) - scopus: 2-s2.0-84868676600 (44)

11573/438275 - 2012 - Conventional and Microwave-Assisted Synthesis of Benzimidazole Derivatives and their in vitro Inhibition of human Cyclooxygenase.
Secci, Daniela; Bolasco, Adriana; D’Ascenzio, M.; Della Sala, F.; Yáñez, M.; Carradori, Simone - 01a Articolo in rivista
rivista: JOURNAL OF HETEROCYCLIC CHEMISTRY (Hetero Corporation:PO Box 170:Provo, UT 84603:(801)400-7373, EMAIL: jhetchem@yahoo.com, Fax: (801)356-7373) pp. - - issn: 0022-152X - wos: WOS:000310562600032 (36) - scopus: 2-s2.0-84868139326 (44)

11573/525670 - 2012 - Discovery and optimization of pyrazoline derivatives as promising monoamine oxidase inhibitors
Secci, Daniela; Carradori, Simone; Bolasco, Adriana; Bizzarri, Bruna; D'ascenzio, Melissa; E., Maccioni - 01a Articolo in rivista
rivista: CURRENT TOPICS IN MEDICINAL CHEMISTRY (Hilversum : Bentham Science Publishers) pp. 2240-2257 - issn: 1568-0266 - wos: WOS:000314822900009 (44) - scopus: 2-s2.0-84874905503 (48)

11573/458436 - 2011 - EPIGENETIC MODULATION OF PGC-1a ACTIVITY BY GCN5 INHIBITORS: WO2010007085
Carradori, Simone; Secci, Daniela; Mai, Antonello - 01a Articolo in rivista
rivista: EXPERT OPINION ON THERAPEUTIC PATENTS (--London United Kingdom:Informa Healthcare -London, United Kingdom: Ashley Publications Limited) pp. 1651-1656 - issn: 1354-3776 - wos: WOS:000294966800007 (8) - scopus: 2-s2.0-80053007226 (8)

11573/363753 - 2011 - Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents
Franco, Chimenti; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Simone, Carradori; Melissa, D'ascenzio; Lilli, Daniela; Rivanera, Daniela - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 378-382 - issn: 0223-5234 - wos: WOS:000286905400044 (92) - scopus: 2-s2.0-78650509856 (101)

11573/458570 - 2011 - CPTH6, A NOVEL Gcn5/pCAF HISTONE ACETYLTRANSFERASE INHIBITOR, INDUCES BOTH APOPTOSIS AND AUTOPHAGY IN HUMAN LEUKEMIA CELLS
Ragazzoni, Y.; Trisciuoglio, D.; Gabellini, C. .; Pelosi, A.; Desideri, M.; Carradori, Simone; Secci, Daniela; Rizzo, M. G.; Del, Bufalo - 04c Atto di convegno in rivista
rivista: CYTOMETRY. PART A (Hoboken, N.J. : Wiley-Liss, c2002-) pp. 1075-1075 - issn: 1552-4922 - wos: (0) - scopus: (0)
congresso: 29th National Conference of the Italian Society of Cytometry (Salerno)

11573/404480 - 2011 - The State of the Art of Pyrazole Derivatives as Monoamine Oxidase Inhibitors and Antidepressant/Anticonvulsant Agents
Secci, Daniela; Bolasco, Adriana; Carradori, Simone; Chimenti, Paola - 01a Articolo in rivista
rivista: CURRENT MEDICINAL CHEMISTRY (Bentham Science Publishers BV:PO Box 7917, Exec Ste Y 26, Saif Zone Sharjah Uae:011 971 6 5571132, EMAIL: benthams@emirates.net.ae, INTERNET: http://www.bentham.org, Fax: 011 971 6 5571134) pp. 5114-5144 - issn: 0929-8673 - wos: WOS:000299031000010 (92) - scopus: 2-s2.0-80054860498 (98)

11573/543282 - 2011 - Synthesis and selective human monoamine oxidase inhibition of 3-carbonyl, 3-acyl, and 3-carboxyhydrazido coumarin derivatives
Secci, Daniela; Carradori, Simone; Bolasco, Adriana; Chimenti, Paola; Yanez, Matilde; Ortuso, Francesco; Alcaro, Stefano - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 4846-4852 - issn: 0223-5234 - wos: WOS:000296041600006 (86) - scopus: 2-s2.0-80053187018 (87)

11573/358902 - 2010 - Synthesis and anti-Helicobacter pylori activity of 4-(coumarin-3-yl)thiazol-2-ylhydrazone derivatives
Chimenti, F; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, A; Carradori, S; D'ascenzio, M; Scaltrito M., M; Sisto, F. - 01a Articolo in rivista
rivista: JOURNAL OF HETEROCYCLIC CHEMISTRY (Hetero Corporation:PO Box 170:Provo, UT 84603:(801)400-7373, EMAIL: jhetchem@yahoo.com, Fax: (801)356-7373) pp. 1269-1274 - issn: 0022-152X - wos: WOS:000284740700002 (26) - scopus: 2-s2.0-78649674111 (29)

11573/225656 - 2010 - Synthesis, selective anti-Helicobacter pylori activity, and cytotoxicity of novel N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides
Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Rivanera, Daniela; Zicari, Alessandra; M., Maddalena Scaltrito; Francesca, Sisto - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 4922-4926 - issn: 0960-894X - wos: WOS:000280348400041 (109) - scopus: 2-s2.0-77955425222 (113)

11573/228282 - 2010 - Synthesis and characterization of new 3-acyl-7-hydroxy-6,8-substituted-coumarin and 3-acyl-7-benzyloxy-6,8-substituted-coumarin derivatives
Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Bizzarri, Bruna; Chimenti, Paola; Granese, A; Carradori, S. - 01a Articolo in rivista
rivista: JOURNAL OF HETEROCYCLIC CHEMISTRY (Hetero Corporation:PO Box 170:Provo, UT 84603:(801)400-7373, EMAIL: jhetchem@yahoo.com, Fax: (801)356-7373) pp. 729-733 - issn: 0022-152X - wos: WOS:000278638500039 (10) - scopus: 2-s2.0-77953002432 (10)

11573/360184 - 2010 - Investigations on the 2-thiazolylhydrazyne scaffold: Synthesis and molecular modeling of selective human monoamine oxidase inhibitors
Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Arianna, Granese; Simone, Carradori; Matilde, Yanez; Francisco, Orallo; Francesco, Ortuso; Stefano, Alcaro - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 5715-5723 - issn: 0968-0896 - wos: WOS:000280116800027 (84) - scopus: 2-s2.0-77955418391 (86)

11573/360219 - 2010 - Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3,5-di(hetero)aryl-4,5-dihydro-(1H)-pyrazole derivatives
Chimenti, Franco; Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Bizzarri, Bruna; Chimenti, Paola; Arianna, Granese; Matilde, Yanez; Francisco, Orallo - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 800-804 - issn: 0223-5234 - wos: WOS:000274773300047 (79) - scopus: 2-s2.0-73549097080 (95)

11573/365473 - 2010 - A new series of flavones, thioflavones, and flavanones as selective monoamine oxidase-B inhibitors
Chimenti, Franco; Fioravanti, Rossella; Bolasco, Adriana; Chimenti, Paola; Secci, Daniela; Rossi, Francesca; Matilde, Yanez; Francisco, Orallo; Francesco, Ortuso; Stefano, Alcaro; Roberto, Cirilli; Rosella, Ferretti; M., Luisa Sanna - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 1273-1279 - issn: 0968-0896 - wos: WOS:000274153600033 (90) - scopus: 2-s2.0-75149195318 (92)

11573/361775 - 2010 - Synthesis, semipreparative HPLC separation, biological evaluation, and 3D-QSAR of hydrazothiazole derivatives as human monoamine oxidase B inhibitors
Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Arianna, Granese; Simone, Carradori; Elias, Maccioni; M., Cristina Cardia; Matilde, Yanez; Francisco, Orallo; Stefano, Alcaro; Francesco, Ortuso; Roberto, Cirilli; Rosella, Ferretti; Simona, Distinto; Johannes, Kirchmair; Thierry, Langer - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 5063-5070 - issn: 0968-0896 - wos: WOS:000279744700024 (44) - scopus: 2-s2.0-77955325332 (45)

11573/360702 - 2010 - SYNTHESIS, STEREOCHEMICAL SEPARATION, AND BIOLOGICAL EVALUATION OF SELECTIVE INHIBITORS OF HUMAN MAO-B: 1-(4-ARYLTHIAZOL-2-YL)-2-(3-METHYLCYCLOHEXYLIDENE)HYDRAZINES
Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, A; Carradori, S; Yanez, M; Orallo, F; Sanna, Ml; Gallinella, B; Cirilli, R. - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 6516-6520 - issn: 0022-2623 - wos: WOS:000281404200024 (37) - scopus: 2-s2.0-77956305471 (38)

11573/358535 - 2010 - Synthesis and selective inhibition of human monoamine oxidases of a large scaffold of (4,5-substituted-thiazol-2-yl)hydrazones
Chimenti, Franco; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Carradori, Simone; D'ascenzio, Melissa; Matilde, Yanez; Francisco, Orallo; Bolasco, Adriana - 01a Articolo in rivista
rivista: MEDCHEMCOMM (Cambridge : Royal Society of Chemistry, 2010-) pp. 61-72 - issn: 2040-2503 - wos: WOS:000284864200012 (34) - scopus: 2-s2.0-77956325073 (36)

11573/1017684 - 2010 - Synthesis of new 3-aryl-4,5-dihydropyrazole-1-carbothioamide derivatives. An investigation on their ability to inhibit monoamine oxidase
Maccioni, E.; Alcaro, S.; Orallo, F.; Cardia, M. C.; Distinto, S.; Costa, G.; Yanez, M.; Sanna, M. L.; Vigo, S.; Meleddu, R.; Secci, D. - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 4490-4498 - issn: 0223-5234 - wos: WOS:000282112700010 (32) - scopus: 2-s2.0-77956184314 (36)

11573/48936 - 2010 - Semipreparative HPLC Enantioseparation, Chiroptical Properties, and Absolute Configuration of Two Novel Cyclooxygenase-2 Inhibitors
Roberto, Cirilli; Stefano, Fiore; Francesco La, Torre; Elias, Maccioni; Secci, Daniela; Maria Luisa, Sanna; Cristina, Faggi - 01a Articolo in rivista
rivista: CHIRALITY (John Wiley & Sons Incorporated:Customer Service, 111 River Street:Hoboken, NJ 07030:(800)225-5945, (201)748-6000, EMAIL: societyinfo@wiley.com, INTERNET: http://www.wiley.com, Fax: (212)748-6551) pp. 56-62 - issn: 0899-0042 - wos: WOS:000273192200009 (4) - scopus: 2-s2.0-75449101399 (4)

11573/365148 - 2009 - Synthesis and Evaluation of 4-Acyl-2- Thiazolylhydrazone Derivatives for anti-Toxoplasma Efficacy in Vitro
Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Carradori, Simone; A., Granese; Rivanera, Daniela; N., Frishberg; C., Bordón; L., Jones Brando - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 4574-4577 - issn: 0022-2623 - wos: WOS:000268661600002 (18) - scopus: 2-s2.0-68549125302 (20)

11573/359686 - 2009 - A Novel Histone Acetyltransferase Inhibitor Modulating Gcn5 Network: Cyclopentylidene-[4-(4′-chlorophenyl)thiazol-2-yl)hydrazone
Chimenti, Franco; Bizzarri, Bruna; Elias, Maccioni; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Fioravanti, Rossella; Granese, Arianna; Carradori, Simone; Federica, Tosi; Ballario, Paola; S., Vernarecci; Patrizia, Filetici - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 530-536 - issn: 0022-2623 - wos: WOS:000262522100032 (99) - scopus: 2-s2.0-60549085424 (102)

11573/364634 - 2009 - Synthesis and Biological Evaluation of Novel Conjugated Coumarin-Thiazole Systems
Chimenti, Franco; Carradori, Simone; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Bizzarri, Bruna - 01a Articolo in rivista
rivista: JOURNAL OF HETEROCYCLIC CHEMISTRY (Hetero Corporation:PO Box 170:Provo, UT 84603:(801)400-7373, EMAIL: jhetchem@yahoo.com, Fax: (801)356-7373) pp. 575-578 - issn: 0022-152X - wos: WOS:000266844800030 (42) - scopus: 2-s2.0-66349115617 (46)

11573/364118 - 2009 - Synthesis, Molecular Modeling, and Selective Inhibitory Activity against Human Monoamine Oxidases of 3-Carboxamido-7-Substituted Coumarins.
Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Bizzarri, Bruna; Granese, Arianna; Carradori, Simone; Yanez, Matilde; Orallo, Francisco; Ortuso, Francesco; Alcaro, Stefano - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1935-1942 - issn: 0022-2623 - wos: WOS:000264835800015 (155) - scopus: 2-s2.0-64549137053 (160)

11573/47973 - 2009 - Unusually high enantioselectivity in high-performance liquid chromatography using cellulose tris(4-methylbenzoate) as a chiral phase
Cirilli, R; Alcaro, S; Fioravanti, Rossella; Secci, Daniela; Fiore, S; La Torre, F; Ortuso, F. - 01a Articolo in rivista
rivista: JOURNAL OF CHROMATOGRAPHY A (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598) pp. 4673-4678 - issn: 0021-9673 - wos: WOS:000266307900007 (25) - scopus: 2-s2.0-65449169552 (26)

11573/225849 - 2009 - Chalcones: A Valid Scaffold for Monoamine Oxidases Inhibitors
Franco, Chimenti; Fioravanti, Rossella; Rossella, ; Bolasco, Adriana; Adriana, ; Chimenti, Paola; Paola, ; Secci, Daniela; Daniela, ; Rossi, Francesca - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 2818-2824 - issn: 0022-2623 - wos: WOS:000265911800020 (154) - scopus: 2-s2.0-65649087484 (173)

11573/360667 - 2008 - Synthesis, Stereochemical Identification, and Selective Inhibitory Activity against Human Monoamine Oxidase-B of 2-Methylcyclohexylidene-(4-arylthiazol-2-yl)hydrazones
Chimenti, F.; Maccioni, E.; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Alcaro, S.; Ortuso, F.; Yanez, M.; Orallo, F.; Cirilli, R.; Ferretti, R.; La Torre, F. - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 4874-4880 - issn: 0022-2623 - wos: WOS:000258637400006 (86) - scopus: 2-s2.0-50249143998 (89)

11573/365405 - 2008 - Synthesis, molecular modeling studies and selective inhibitory activity against MAO of N1-propanoyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives
Chimenti, Franco; Fioravanti, Rossella; Bolasco, Adriana; Manna, Fedele; Chimenti, Paola; Secci, Daniela; Rossi, Francesca; Turini, Paola; Francesco, Ortuso; Stefano, Alcaro; Maria Cristina, Cardia - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 2262-2267 - issn: 0223-5234 - wos: WOS:000260898800025 (45) - scopus: 2-s2.0-53149111946 (57)

11573/363673 - 2007 - A novel class of selective anti-Helicobacter pylori agents 2-Oxo-2H-chromene-3-carboxamide derivatives.
Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Carradori, Simone; Granese, Arianna; Rivanera, Daniela; Lilli, Daniela; Zicari, Alessandra; Scaltrito M., M; Sisto, F. - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 3065-3071 - issn: 0960-894X - wos: WOS:000247052900022 (43) - scopus: 2-s2.0-34247869800 (50)

11573/359993 - 2007 - Synthesis and in vitro activity of 2-thiazolylhydrazone derivatives compared with the activity of clotrimazole against clinical isolates of Candida spp.
Chimenti, Franco; Bizzarri, Bruna; Elias, Maccioni; Secci, Daniela; Bolasco, Adriana; Fioravanti, Rossella; Chimenti, Paola; Granese, Arianna; Carradori, Simone; Rivanera, Daniela; Lilli, Daniela; Zicari, Alessandra; Simona, Distinto - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 4635-4640 - issn: 0960-894X - wos: WOS:000248877800043 (77) - scopus: 2-s2.0-34447334808 (78)

11573/231039 - 2007 - Selective inhibitory activity against MAO and molecular modeling studies of 2-thiazolylhydrazone derivatives
Chimenti, Franco; Elias, Maccioni; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Olivia, Befani; Turini, Paola; Stefano, Alcaro; Francesco, Ortuso; Maria C., Cardia; Simona, Distinto - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 707-712 - issn: 0022-2623 - wos: WOS:000244224900013 (79) - scopus: 2-s2.0-33847420851 (83)

11573/233577 - 2007 - Monoamine oxidase isoform-dependent tautomeric influence in the recognition of 3,5-diaryl pyrazole inhibitors.
Chimenti, Franco; Fioravanti, Rossella; Bolasco, Adriana; Manna, Fedele; Chimenti, Paola; Secci, Daniela; Befani, O; Turini, Paola; Ortuso, F; Alcaro, S. - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 425-428 - issn: 0022-2623 - wos: WOS:000243889100002 (65) - scopus: 2-s2.0-33846930800 (70)

11573/360713 - 2007 - High-performance liquid chromatographic separation of enantiomers and diastereomers of 2-methylcyclohexanone thiosemicarbazone, and determination of absolute configuration and configurational stability
Cirilli, R.; Ferretti, R.; Torre, F. La; Secci, Daniela; Bolasco, Adriana; Carradori, Simone; Pierini, Marco - 01a Articolo in rivista
rivista: JOURNAL OF CHROMATOGRAPHY A (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598) pp. 160-169 - issn: 0021-9673 - wos: WOS:000251335300008 (46) - scopus: 2-s2.0-35648952796 (46)

11573/1017717 - 2006 - Synthesis and in vitro selective anti-Helicobacter pylori activity of N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides
Chimenti, Franco; Bizzarri, Bruna; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Carradori, Simone; Granese, Arianna; Rivanera, Daniela; Lilli, Daniela; Maddalena Scaltrito, M.; Immacolata Brenciaglia, M. - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 208-212 - issn: 0223-5234 - wos: WOS:000236643200006 (51) - scopus: 2-s2.0-33644958572 (56)

11573/233573 - 2006 - Synthesis and molecular modelling of novel substituted-4,5-dihydro-(1H)-pyrazole derivatives as potent and highly selective monoamine oxidase-A inhibitors.
Chimenti, Franco; Bolasco, Adriana; Manna, Fedele; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Befani, O; Turini, Paola; Alcaro, S; Ortuso, F. - 01a Articolo in rivista
rivista: CHEMICAL BIOLOGY & DRUG DESIGN (Blackwell Munksgaar) pp. 206-214 - issn: 1747-0277 - wos: WOS:000236241200004 (30) - scopus: 2-s2.0-33645314648 (34)

11573/366526 - 2006 - Synthesis, molecular modeling studies, and selective inhibitory activity against monoamine oxidase of N,N'-bis[2-oxo-2H-benzopyran]-3-carboxamides
Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Carradori, Simone; O., Befani; Turini, Paola; S., Alcaro; F., Ortuso - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 4135-4140 - issn: 0960-894X - wos: WOS:000239291900054 (30) - scopus: 2-s2.0-33745126693 (35)

11573/193860 - 2006 - 2-Methylcyclohexanone thiosemicarbazone: enantio- and diastereoseparation, and isomerization study by dynamic HPLC
Cirilli, R.; Ferretti, R.; La Torre, F.; Bolasco, Adriana; Secci, Daniela; Pierini, Marco - 04a Atto di comunicazione a congresso
libro: XXII Congresso Nazionale della Società Chimica Italiana - ()

11573/232197 - 2006 - Analytical and semipreparative high performance liquid chromatography enantioseparation of new substituted 1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazoles on polysaccharide-based chiral stationary phases in normal-phase, polar organic and reversed-phase conditions.
Cirilli, R; Simonelli, A; Ferretti, R; Bolasco, Adriana; Chimenti, Paola; Secci, Daniela; Maccioni, E; La Torre, F. - 01a Articolo in rivista
rivista: JOURNAL OF CHROMATOGRAPHY A (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598) pp. 198-203 - issn: 0021-9673 - wos: WOS:000234639600021 (55) - scopus: 2-s2.0-28944433830 (57)

11573/233568 - 2006 - Quercetin as the active principle of Hypericum hircinum exerts a selective inhibitory activity against MAO-A: Extraction, biological analysis, and computational study
F., Chimenti; F., Cottiglia; L., Bonsignore; L., Casu; M., Casu; C., Floris; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; O., Befani; Turini, Paola; S., Alcaro; F., Ortuso; G., Trombetta; A., Loizzo; I., Guarino - 01a Articolo in rivista
rivista: JOURNAL OF NATURAL PRODUCTS ([Washington, DC,: American Chemical Society and American Society of Pharmacognosy) pp. 945-949 - issn: 0163-3864 - wos: WOS:000238478800015 (103) - scopus: 2-s2.0-33746514329 (129)

11573/233587 - 2006 - Synthesis, biological evaluation and 3D-QSAR of 1,3,5-trisubstituted-4,5-dihydro-(1H)-pyrazole derivatives as potent and highly selective monoamine oxidase-A inhibitors.
Manna, Fedele; Chimenti, Paola; Granese, Arianna; Befani, O; Turini, Paola; Cirilli, R; La Torre, F; Alcaro, S; Ortuso, F; Langer, T.; Chimenti, Franco; Bolasco, Adriana; Secci, Daniela - 01a Articolo in rivista
rivista: CURRENT MEDICINAL CHEMISTRY (Bentham Science Publishers BV:PO Box 7917, Exec Ste Y 26, Saif Zone Sharjah Uae:011 971 6 5571132, EMAIL: benthams@emirates.net.ae, INTERNET: http://www.bentham.org, Fax: 011 971 6 5571134) pp. 1411-1428 - issn: 0929-8673 - wos: WOS:000237432900005 (60) - scopus: 2-s2.0-33646507688 (64)

11573/233575 - 2005 - Synthesis and In Vitro Selective anti-Helicobacter pylori Activity of Pyrazoline Derivatives
Chimenti, Franco; Bizzarri, Bruna; Manna, Fedele; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna; Rivanera, Daniela; Lilli, Daniela; M. M., Scaltrito; M. I., Brenciaglia - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 603-607 - issn: 0960-894X - wos: WOS:000226935700022 (60) - scopus: 2-s2.0-19944431182 (60)

11573/230760 - 2005 - Synthesis, molecular modeling studies and selective inhibitory activity against MAO of 1-thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1H)-pyrazole derivatives.
Chimenti, Franco; Maccioni, E; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; Befani, Olivia; Turini, Paola; Alcaro, S; Ortuso, F; Cirilli, R; La Torre, F; Cardia, Mc; Distinto, S. - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 7113-7122 - issn: 0022-2623 - wos: WOS:000233399500006 (110) - scopus: 2-s2.0-28544443174 (121)

11573/233604 - 2005 - Cyclization of N ,N’-bis(salicylidene)diamines with Carbon Suboxide.
Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna - 01a Articolo in rivista
rivista: SYNTHETIC COMMUNICATIONS (New York, NY : Taylor & Francis New York, NY: Marcel Dekker Incorporated) pp. 769-773 - issn: 0039-7911 - wos: WOS:000228067400002 (2) - scopus: 2-s2.0-15944413844 (3)

11573/143386 - 2005 - LC Determination of Coumarin-3-acyl Derivatives for Evaluation of the Stability and Monoamine Oxidase Inhibition Mechanism.
Chimenti, Paola; Granese, Arianna; Gagliardi, L; De Orsi, D.; Chimenti, Franco; Secci, Daniela; Bolasco, Adriana - 01a Articolo in rivista
rivista: CHROMATOGRAPHIA (Heidelberg ; Berlin : Springer) pp. 519-522 - issn: 0009-5893 - wos: WOS:000229283800013 (7) - scopus: 2-s2.0-20044366228 (7)

11573/231009 - 2005 - Pyrazole Derivatives as Potential Anticancer agents and their Affinity Binding to P-Glycoprotein
F., Manna; Chimenti, Franco; Fioravanti, Rossella; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; C., Ferlini; G., Scambia - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 4632-4635 - issn: 0960-894X - wos: WOS:000231936700048 (146) - scopus: 2-s2.0-24344507274 (156)

11573/233580 - 2004 - Synthesis and selective inhibitory activity against MAO of 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives.
Chimenti, Franco; Bolasco, Adriana; Manna, Fedele; Secci, Daniela; Chimenti, Paola; Befani, O.; Turini, P.; Giovannini, V.; Mondovi', B.; Cirilli, R.; La Torre, F. - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 2071-2074 - issn: 0022-2623 - wos: WOS:000220642100020 (117) - scopus: 2-s2.0-11144358502 (122)

11573/232010 - 2004 - Synthesis of New Diethynylbenzene Derivatives.
Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Granese, Arianna - 01a Articolo in rivista
rivista: SYNTHETIC COMMUNICATIONS (New York, NY : Taylor & Francis New York, NY: Marcel Dekker Incorporated) pp. 2549-2555 - issn: 0039-7911 - wos: WOS:000223207400006 (7) - scopus: 2-s2.0-3843067540 (9)

11573/233608 - 2004 - Inhibition of Monoamine Oxidases by Coumarin-3-Acyl Derivatives: Biological Activity and Computational Study
Chimenti, Franco; Secci, Daniela; Bolasco, Adriana; Chimenti, Paola; Granese, Arianna; O., Befani; Turini, Paola; S., Alcaro; F., Ortuso - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 3697-3703 - issn: 0960-894X - wos: WOS:000222367300016 (93) - scopus: 2-s2.0-2942527408 (94)

11573/239216 - 2004 - Enantiomers of C5-chiral 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives: analytical and semipreparative HPLC separation, chiroptical properties, absolute configuration and inhibitory activity against monoamino oxidase
Cirilli, R.; Ferretti, R.; Gallinella, B.; Turchetto, L.; Bolasco, Adriana; Secci, Daniela; Chimenti, Paola; Pierini, Marco; Fares, V.; Befani, O.; La Torre, F. - 01a Articolo in rivista
rivista: CHIRALITY (John Wiley & Sons Incorporated:Customer Service, 111 River Street:Hoboken, NJ 07030:(800)225-5945, (201)748-6000, EMAIL: societyinfo@wiley.com, INTERNET: http://www.wiley.com, Fax: (212)748-6551) pp. 625-636 - issn: 0899-0042 - wos: WOS:000224693700008 (33) - scopus: 2-s2.0-7044235090 (35)

11573/253216 - 2002 - Inhibition of amine oxidases activity by 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives.
Manna, Fedele; Chimenti, Franco; Bolasco, Adriana; Secci, Daniela; Bizzarri, Bruna; Befani, Olivia; Turini, Paola; Mondovi', Bruno; Alcaro, Stefano; Tafi, Andrea - 01a Articolo in rivista
rivista: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 3629-3633 - issn: 0960-894X - wos: WOS:000179735200029 (96) - scopus: 2-s2.0-18744407545 (116)

11573/253228 - 2001 - Efficacy of Hypericum and Calendula oils in the epithelial reconstruction of surgical wounds in childbirth with cesarean section.
Lavagna, Silvio Massimo; Secci, Daniela; Chimenti, Paola; Bonsignore, L.; Ottaviani, A.; Bizzarri, Bruna - 01a Articolo in rivista
rivista: IL FARMACO (Attuale:ELSEVIER SCIENCE SA, PO BOX 564, LAUSANNE, SWITZERLAND, 1001 Societa Chimica Italiana:Viale Liegi 48, 00198 Rome Italy:011 39 06 8549691, EMAIL: soc.chim.it@agora.stm.it, Fax: 011 39 06 8548734) pp. 451-453 - issn: 0014-827X - wos: (0) - scopus: 2-s2.0-0035395343 (83)

11573/253214 - 2000 - Synthesis of the 4-hydroxymino-3-carboxamide-2-quinolone with a new heterocyclization mechanism of the reaction between carbon suboxide and 2-aminobenzamidoxime.
Secci, Daniela; Chimenti, Franco; Lavagna, Silvio Massimo; F., Manna; A., Bolasco; S., Alcaro; L., Bonsignore - 01a Articolo in rivista
rivista: HETEROCYCLES (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598) pp. 2789-2793 - issn: 0385-5414 - wos: (0) - scopus: (0)

11573/254362 - 2000 - Synthesis of the 4-hydroxyimino-3-carboxamide-2-quinolone with a new heterocyclization mechanism of the reaction between carbon suboxide and 2-aminobenzamidoxime
Secci, Daniela; Chimenti, Franco; Lavagna, Silvio Massimo; Manna, Fedele; Bolasco, Adriana; Alcaro, S. - 01a Articolo in rivista
rivista: HETEROCYCLES (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598) pp. 2789-2793 - issn: 0385-5414 - wos: WOS:000165941900021 (1) - scopus: 2-s2.0-0034387709 (1)

11573/244922 - 1999 - Synthesis of coumarin-3-O-acylisoureas by different carbodiimides
L., Bonsignore; F., Cottiglia; Lavagna, Silvio Massimo; G., Loy; Secci, Daniela - 01a Articolo in rivista
rivista: HETEROCYCLES (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598) pp. 469-472 - issn: 0385-5414 - wos: (0) - scopus: (0)

11573/157330 - 1999 - Controllo e sicurezza degli impianti medico-ospedalieri finalizzati alla tutela della salute
Secci, Daniela - 03a Saggio, Trattato Scientifico

11573/245383 - 1998 - Synthesis via carbon suboxide and pharmacological activity of coumarin derivatives
L., Bonsignore; F., Cottiglia; Lavagna, Silvio Massimo; G., Loy; Secci, Daniela - 01a Articolo in rivista
rivista: IL FARMACO (Attuale:ELSEVIER SCIENCE SA, PO BOX 564, LAUSANNE, SWITZERLAND, 1001 Societa Chimica Italiana:Viale Liegi 48, 00198 Rome Italy:011 39 06 8549691, EMAIL: soc.chim.it@agora.stm.it, Fax: 011 39 06 8548734) pp. 693-697 - issn: 0014-827X - wos: (0) - scopus: (0)

11573/16250 - 1998 - Synthesis and antimicrobial activity of coumarin 7-substituted cephalosporin and sulfones
Lavagna, Silvio Massimo; Jehl, F.; Monteil, H.; Secci, Daniela; Elkhaili, H. - 01a Articolo in rivista
rivista: IL FARMACO (Attuale:ELSEVIER SCIENCE SA, PO BOX 564, LAUSANNE, SWITZERLAND, 1001 Societa Chimica Italiana:Viale Liegi 48, 00198 Rome Italy:011 39 06 8549691, EMAIL: soc.chim.it@agora.stm.it, Fax: 011 39 06 8548734) pp. 425-430 - issn: 0014-827X - wos: (0) - scopus: (0)

11573/27483 - 1998 - Synthesis and antimicrobial activity of coumarin 7-substituted cephalosporins and sulfones
Leonardo, Bonsignore; Filippo, Cottiglia; Elkhaili, H.; Françoise, Jehl; Lavagna, Silvio Massimo; Giuseppe, Loy; Manna, Fedele; Henry, Monteil; Davide, Pompei; Secci, Daniela - 01a Articolo in rivista
rivista: IL FARMACO (Attuale:ELSEVIER SCIENCE SA, PO BOX 564, LAUSANNE, SWITZERLAND, 1001 Societa Chimica Italiana:Viale Liegi 48, 00198 Rome Italy:011 39 06 8549691, EMAIL: soc.chim.it@agora.stm.it, Fax: 011 39 06 8548734) pp. 425-430 - issn: 0014-827X - wos: WOS:000075823400009 (35) - scopus: 2-s2.0-0032580912 (36)

11573/48434 - 1998 - Nucleophilic aromatic substitutionreactions promoted by aryl and heteroaryl amine nitranions
Secci, Daniela; D., Landini; A., Maia; V. M., Vlasov; I., Os'kina - 01a Articolo in rivista
rivista: NEW JOURNAL OF CHEMISTRY (Royal Society of Chemistry:Thomas Graham House, Science Park, Cambridge CB4 0WF United Kingdom:011 44 1223 432360, EMAIL: sales@rsc.org, INTERNET: http://www.rsc.org, http://www.chensoc.org, Fax: 011 44 1223 423429) pp. 71-74 - issn: 1144-0546 - wos: (0) - scopus: (0)

11573/48432 - 1998 - One-step synthesis of new 3-oxa- or 3-azabicyclo(5.3.0)dec-1-en-3-methyliden-6,8-dione derivatives
Secci, Daniela; L., Bonsignore; F., Cottiglia; G., Loy - 01a Articolo in rivista
rivista: IL FARMACO (Attuale:ELSEVIER SCIENCE SA, PO BOX 564, LAUSANNE, SWITZERLAND, 1001 Societa Chimica Italiana:Viale Liegi 48, 00198 Rome Italy:011 39 06 8549691, EMAIL: soc.chim.it@agora.stm.it, Fax: 011 39 06 8548734) pp. 680-683 - issn: 0014-827X - wos: (0) - scopus: 2-s2.0-0032462093 (2)

11573/151712 - 1995 - Pyrogen and depyrogenation
Secci, Daniela - 02a Capitolo o Articolo
libro: Injectables and water for pharmaceutica use - ()

11573/16693 - 1994 - Synthesis and antimicrobial activity of coumarin and benzodioxazepine, diazepine and benzoxazepine substituted penicillins
Lavagna, Silvio Massimo; Secci, Daniela; Alessandro De, Logu; Leonardo, Bonsignore - 01a Articolo in rivista
rivista: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 479-485 - issn: 0223-5234 - wos: (0) - scopus: (0)

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