DANIELA DE VITA

Researcher


email: daniela.devita@uniroma1.it
phone: 0649912788
building: CU022
room: 319

Part I – General Information
Date of Birth 1st Sept 1977
Place of Birth Tropea (VV)
Citizenship Italian
Permanent Address P.le Aldo Moro, 5 00185 Rome (Italy)
E-mail daniela.devita@uniroma1.it
Spoken Languages Italian, English (Good), Brazilian Portuguese (Basic)

Part II – Education
2004: MSc. in Pharmaceutical Chemistry and Technologies (Sapienza University of Rome, Faculty of Pharmacy); Level in National Classification: 110/110 cum laude with the thesis “D-cycloserine derivatives as potential nootropic agents”
2008: PhD in Pharmaceutical Sciences, Sapienza University of Rome, Faculty of Pharmacy, with the thesis “4-Aminopyridine derivatives as ChE inhibitors”
2005: Qualification for practise pharmacist’s profession, Sapienza University of Rome, Faculty of Pharmacy


Part III – Academic Appointments
15/07/2019 present Dept. Environmental Biology, Sapienza University of Rome Researcher
01/03/2016 30/04/2018 IQSC-USP Sao Carlos (SP, Brazil) Post-doc fellow
01/06/2014 31/05/2015 Dept. Chemistry and Technology of Drug Sapienza University of Rome Research fellow, group of Prof. Di Santo
02/05/2013 01/05/2014 Dept. Chemistry and Technology of Drug, Sapienza University of Rome Research fellow, group of Prof. Silvestri
01/10/2012 31/10/2012 Dept. Chemistry and Technology of Drug Sapienza, University of Rome Reserch fellow, group of Prof.Costi
01/11/2011 30/11/2011 Dept. Chemistry and Technology of Drug Sapienza, University of Rome Research fellow, group of Dr. Di Rienzo
01/03/2011 31/08/2011 Dept. Chemistry and Technology of Drug Sapienza, University of Rome Research fellow, group of Prof. Fornarini
01/09/2010 28/02/2011 Dept. Chemistry and Technology of Drug Sapienza, University of Rome Research fellow, group of Prof. Biava
02/04/2008 02/04/2009 Dept. Chemistry and Technology of Drug Sapienza, University of Rome Research fellow, group of Prof. Biava


Part IV – Teaching experience
AY 2020-2021 Dept. Chemistry and Technology of Drug, Sapienza University of Rome Teaching of Pharmaceutical Botany (SFA and Pharmacy)
AY 2019-2020 Dept. Chemistry and Technology of Drug, Sapienza University of Rome Teaching of Pharmaceutical Botany (SFA)
AY 2012-2013 Dept. “Scienze Ecologiche e Biologiche DEB”, Tuscia University, Viterbo (Italy) Teaching of General and Inorganic Chemistry
AY 2009-2010 Dept.”SBAI-Scienze di Base e Applicate per l'Ingegneria”, Sapienza University of Rome Tutor of General and Inorganic Chemistry


Part V - Society memberberships
2021-present Member of the Italian Botanical Society (SBI)
2014-2015/2019-present Member of the Italian Chemical Society (SCI)

Part VI - Funding Information
2020 Principal investigator in the Program "Development of natural compounds as inhibitors of Mpro, the main protease of SARS-Cov-2" Sapienza Università di Roma- Progetti di Ateneo Medi- (grant Value: 10000 Euro)
2015 Investigator in the Program "Targeting Trypanosomatids sterol biosynthesis and thiol redox metabolism enzymes for lead drug discovery" Sapienza Università di Roma- Grandi progetti di Ateneo- Grant number C26H15WYPW (grant Value: 20000 Euro)

Part VII – Summary of Scientific Achievements
63 papers, Scopus Database, period 2006-present
H index = 16


ADDITIONAL INFORMATION
ORAL COMMUNICATIONS

Nanoinnovation2020, Rome 15-18, September 2020: Bioactive Molecules from Plants: Extraction, Nanoencapsulation and Application

114th Congress of the Italian Botanical Society (VI International Plant Science Conference) Padova (Italy), September, 4-7 2019: Antifungal activity of amaranth seed extract in combination with known antifungal drug

NPCF8 New Prospective in Pharmaceutical Chemistry, Parma (Italy) June 9-11 2014
Imidazole derivatives with in vitro antichagas activity.

XXII NMMC. Rome, September 10-13 2013 (session infectious diseases and drug resistance)
Imidazole derivatives with in vitro antichagas activity: synthesis, biological evaluation and docking studies.

Drug’s day “Antitumoral drugs, orphan drugs and rare diseases”. Salerno (Italy) April 12 2013
New imidazole derivatives in vitro highly active vs T.cruzi.

POSTERS

4th EFMS-YMCS. Vienna (Austria) - August 31-September 1, 2017
DG Silva, JFR Ribeiro, D. De Vita, L. Cianni, JR Rocha, ACB Burtoloso, PW Kenny, CA Montanari. Synthesis of cruzain inhibitors for dipeptidyl nitriles warhead exchange.

IUPAC 2017 - 46th World Chemistry Congress
L. Cianni, G. Sartori, D. De Vita, F. Rosini, CA Montanari, A. Leitão. On the study of halogen bond interaction to increase cruzain affinity of covalently bound reversible inhibitors.

XXIII NMMC. Salerno (Italy) September 6-9 2015
L. Scipione, R. Di Santo, R. Costi, S. Tortorella, G. Simonetti, F. D. D’Auria, F. Pandolfi, and D. De Vita. Cinnamic and caffeic acid derivatives against Candida albicans biofilm.
F. Pandolfi, D. De Vita, R. Di Santo, R. Costi, S. Tortorella, M. Bartolini, V. Andrisano, and L. Scipione. New dual binding site acetylcholinesterase inhibitors.

XXII NMMC. Rome (Italy) September 10-13 2013
D. De Vita, S. Panella, G. Simonetti, F. D. D’Auria, L. Scipione, R. Di Santo, L. Friggeri, S. Tortorella. Synthesis and antifungal activity of a new series of 2-(1H-imidazol-1-yl)-1-phenylethanol derivatives.
L. Friggeri, D. De Vita, F. Pandolfi, S. Tortorella, R. Costi, R. Di Santo, L. Scipione. Synthesis and evaluation of 3,4-dihydroxybenzoic acid derivatives as antioxidants, bio-metal chelating agents and acetylcholinesterase inhibitors.

Drug’s day “Antitumoral drugs, orphan drugs and rare diseases”. Salerno (Italy) April 12 2013
D. De Vita, L. Friggeri, L. Scipione, R. Di Santo, R. Costi, F. Moraca, B. Botta, R. Brun, M. Kaiser, S. Tortorella. New imidazole derivatives in vitro highly active vs T.cruzi.

Cost-CM801 WG1/WG3 Meeting: "New Drugs for Neglected Disease", Siena (Italy) May 31-June 1 2012
D. De Vita, L. Friggeri, P. Mellini, S. Tortorella, L. Scipione, M. Kaiser, R. Brun, R. Di Santo. New 4-aminopyridine and imidazole compounds highly active against T. Cruzi.

XXIV National Congress of the Italian Chemical Society, Lecce (Italy) September 11-16 2011
P. Mellini, D. De Vita, V. Carafa, L. Scipione, B. Di Rienzo and L. Altucci. New carbazole scaffolds as SIRT inhibitors.

NPCF5 New Prospective in Pharmaceutical Chemistry, Trieste (Italy) March 28-30 2011
L. Pescatori, D. De Vita, G. Cuzzucoli Crucitti, P. Mellini, B. Saint Joanis, R.Brosh, S. Tortorella, L. Scipione, R. Costi, R. Di Santo. Design, synthesis and biological activities of new active agents against mycobacteriun tuberculosis.
L. Pescatori, D. De Vita, P. Mellini, L. Scipione, S. Tortorella, R. Di Santo, G. Cuzzucoli Crucitti, R. Costi, L. Fattorini, G. Piccaro. Activity of drugs against dormant mycobacterium tuberculosis.

Conference on scientific research, faculty of Pharmacy- Rome (Italy), December 9-10 2004
L.Scipione, S Tortorella, V. Fabbri, E.Fabbrini, D. De Vita. Choline derivatives with potential antialzheimer activity.

Research products

11573/1708294 - 2024 - Phytochemical analysis and biological activities of the aerial parts of Odontites vulgaris Moench
Frezza, Claudio; De Vita, Daniela; Venditti, Alessandro; Baldani, Claudia; Giampaoli, Ottavia; Sciubba, Fabio; Dal Bosco, Chiara; Franceschin, Marco; Beccaccioli, Marzia; Reverberi, Massimo; Percaccio, Ester; Di Sotto, Antonella; Foddai, Sebastiano - 01a Articolo in rivista
paper: FITOTERAPIA (Amsterdam Netherlands:Elsevier BV Milano : Inverni & Della Beffa : Elsevier) pp. 1-9 - issn: 1971-551X - wos: (0) - scopus: 2-s2.0-85189551866 (0)

11573/1708695 - 2024 - Occurrence and biological activities of seco-iridoids from Jasminum L.
Frezza, Claudio; Nicolosi, Roberta Maria; Brasili, Elisa; Mura, Francesco; De Vita, Daniela - 01g Articolo di rassegna (Review)
paper: CHEMISTRY & BIODIVERSITY (Zürich: Helvetica chimica acta 2004-) pp. - - issn: 1612-1880 - wos: WOS:001185593300001 (0) - scopus: 2-s2.0-85187722025 (0)

11573/1703448 - 2024 - Evaluation of the antifungal and antiproliferative properties of the lichen Roccella tinctoria DC. Extracts and main components
Frezza, Claudio; Rosa Fraioli, Dalia; Conti, Francesca; Nicolosi, Roberta Maria; Scipione, Luigi; Serafini, Ilaria; Petrucci, Rita; Di Matteo, Paola; Rocco, Daniele; Di Giacomo, Silvia; Di Sotto, Antonella; Bonincontro, Graziana; Simonetti, Giovanna; Garzoli, Stefania; De Vita, Daniela; Foddai, Sebastiano - 01a Articolo in rivista
paper: PHARMACEUTICS (Basel: MDPI, 2009-) pp. - - issn: 1999-4923 - wos: (0) - scopus: (0)

11573/1686128 - 2023 - Phytochemical analysis and In vitro antileukemic activity of alkaloid-enriched extracts from Vinca sardoa (Stearn) Pignatti
De Vita, Daniela; Frezza, Claudio; Sciubba, Fabio; Toniolo, Chiara; Badiali, Camilla; Petrucci, Rita; Bortolami, Martina; Di Matteo, Paola; Rocco, Daniele; Stringaro, Annarita; Colone, Marisa; Maxia, Andrea; Petrucci, Maria Teresa; Serafini, Mauro; Foddai, Sebastiano - 01a Articolo in rivista
paper: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. 1-10 - issn: 1420-3049 - wos: WOS:001045668500001 (0) - scopus: 2-s2.0-85167762463 (0)

11573/1691408 - 2023 - Cellulose nanomaterials: extraction, synthesis, characterization and applications
Fornari, Anastasia; Rossi, Marco; De Vita, Daniela; Mura, Francesco; Mattiello, Leonardo - 04d Abstract in atti di convegno
conference: 21th International Symposium on Wood, Fiber and Pulping Chemistry (ISWFPC2023) (Venice, Italy)
book: 21th International Symposium on Wood, Fiber and Pulping Chemistry. Vol. II Poster Presentations - ()

11573/1691410 - 2023 - Cellulose nanomaterials: extraction, synthesis, characterization and applications
Fornari, Anastasia; Rossi, Marco; De Vita, Daniela; Mura, Francesco; Mattiello, Leonardo - 04f Poster
conference: 21th International Symposium on Wood, Fiber and Pulping Chemistry (ISWFPC2023) (Venice, Italy)
book: 21th International Symposium on Wood, Fiber and Pulping Chemistry - ()

11573/1691411 - 2023 - Chitosan nanocapsules loaded with Aloe-Emodin for cancer treatment
Fornari, Anastasia; Rossi, Marco; Mattiello, Leonardo; Pandolfi, Fabiana; Purificato, Federico; De Vita, Daniela; Colone, Marisa; Stringaro, Annarita - 04d Abstract in atti di convegno
conference: The 9th International Electronic Conference on Medicinal Chemistry (ECMC2023) (online)
book: The 9th International Electronic Conference on Medicinal Chemistry: Book of Abstract - ()

11573/1692697 - 2023 - Comparison of the metabolic profile of pecan nuts cultivars [Carya illinoinensis (Wangenh.) K. Koch] by NMR spectroscopy
Frezza, Claudio; Sciubba, Fabio; Giampaoli, Ottavia; De Salvador, Flavio Roberto; Lucarini, Massimo; Engel, Petra; Patriarca, Adriano; Spagnoli, Mariangela; Gianferri, Raffaella; Delfini, Maurizio; Di Cocco, Maria Enrica; De Vita, Daniela - 01a Articolo in rivista
paper: NATURAL PRODUCT RESEARCH (Milton Park, UK : Taylor & Francis Health Sciences, c2003-) pp. 1-6 - issn: 1478-6427 - wos: WOS:001096252400001 (0) - scopus: 2-s2.0-85175264515 (0)

11573/1692695 - 2023 - Protective effect of procyanidin-rich grape seed extract against Gram-negative virulence factors
Nicolosi, Roberta Maria; Bonincontro, Graziana; Imperia, Elena; Badiali, Camilla; De Vita, Daniela; Sciubba, Fabio; Dugo, Laura; Pier Luca Guarino, Michele; Altomare, Annamaria; Simonetti, Giovanna; Pasqua, Gabriella - 01a Articolo in rivista
paper: ANTIBIOTICS (Basel : MDPI) pp. 1-20 - issn: 2079-6382 - wos: (0) - scopus: 2-s2.0-85178312530 (0)

11573/1669529 - 2023 - Posidonia oceanica (L.) Delile. A Mediterranean seagrass with potential applications but regularly and erroneously referred to as an algal species
Trache, Djalal; Tarchoun, Ahmed Fouzi; De Vita, Daniela; Kennedy, John F - 01a Articolo in rivista
paper: INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES (-Attuale :ELSEVIER SCIENCE BV, PO BOX 211, AMSTERDAM, NETHERLANDS, 1000 AE -Butterworth Heinemann Publishers:Linacre House Jordan Hill, Oxford OX2 8DP United Kingdom:011 44 1865 314569, EMAIL: bhmarketing@repp.co.uk, INTERNET: http://www.laxtonsprices.co.uk, Fax: 011 44 1865 314569) pp. - - issn: 0141-8130 - wos: WOS:000964146400001 (7) - scopus: 2-s2.0-85146081077 (8)

11573/1638218 - 2022 - Design, synthesis, and In vitro, in silico and in cellulo evaluation of new Pyrimidine and Pyridine amide and Carbamate derivatives as multi-functional Cholinesterase Inhibitors
Bortolami, Martina; Pandolfi, Fabiana; Tudino, Valeria; Messore, Antonella; Madia, Valentina Noemi; De Vita, Daniela; Di Santo, Roberto; Costi, Roberta; Romeo, Isabella; Alcaro, Stefano; Colone, Marisa; Stringaro, Annarita; Espargaró, Alba; Sabatè, Raimon; Scipione, Luigi - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. 1-31 - issn: 1424-8247 - wos: WOS:000818156100001 (3) - scopus: 2-s2.0-85134396743 (2)

11573/1651261 - 2022 - There is not only Cupressus sempervirens L. A review on the phytochemistry and bioactivities of the other Cupressus L. species
Frezza, Claudio; De Vita, Daniela; Sciubba, Fabio; Toniolo, Chiara; Tomassini, Lamberto; Nicoletti, Marcello; Franceschin, Marco; Guiso, Marcella; Bianco, Armandodoriano; Serafini, Mauro; Foddai, Sebastiano - 01g Articolo di rassegna (Review)
paper: APPLIED SCIENCES (Basel: MDPI AG, 2011-) pp. 1-55 - issn: 2076-3417 - wos: WOS:000834461400001 (6) - scopus: 2-s2.0-85137375749 (5)

11573/1663035 - 2022 - Leucosceptosides A and B. Two phenyl-ethanoid glycosides with important occurrence and biological activities
Frezza, Claudio; De Vita, Daniela; Toniolo, Chiara; Sciubba, Fabio; Tomassini, Lamberto; Venditti, Alessandro; Bianco, Armandodoriano; Serafini, Mauro; Foddai, Sebastiano - 01g Articolo di rassegna (Review)
paper: BIOMOLECULES (Basel: MDPI) pp. 1-27 - issn: 2218-273X - wos: WOS:000900653800001 (0) - scopus: 2-s2.0-85144524418 (1)

11573/1638288 - 2022 - Non-volatile compounds from Araucaria columnaris (G.Forst.) Hook leaves
Frezza, Claudio; Sciubba, Fabio; De Vita, Daniela; Toniolo, Chiara; Foddai, Sebastiano; Tomassini, Lamberto; Petrucci, Rita; Bianco, Armandodoriano; Serafini, Mauro - 01a Articolo in rivista
paper: BIOCHEMICAL SYSTEMATICS AND ECOLOGY (PERGAMON-ELSEVIER SCIENCE LTD, THE BOULEVARD, LANGFORD LANE, KIDLINGTON, OXFORD, ENGLAND, OX5 1GB) pp. 1-5 - issn: 0305-1978 - wos: WOS:000814694200005 (0) - scopus: 2-s2.0-85130963691 (2)

11573/1654141 - 2022 - New Inhibitors of the human p300/CBP acetyltransferase are selectively active against the Arabidopsis HAC proteins
Longo, Chiara; Lepri, Andrea; Paciolla, Andrea; Messore, Antonella; De Vita, Daniela; Bonaccorsi Di Patti, Maria Carmela; Amadei, Matteo; Madia, Valentina Noemi; Ialongo, Davide; Di Santo, Roberto; Costi, Roberta; Vittorioso, Paola - 01a Articolo in rivista
paper: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (Basel: MDPI Center) pp. 1-18 - issn: 1422-0067 - wos: WOS:000859422800001 (3) - scopus: 2-s2.0-85138734584 (3)

11573/1648549 - 2022 - Ultrastructural damages to H1N1 influenza virus caused by vapor essential oils
Madia, Valentina Noemi; Toscanelli, Walter; De Vita, Daniela; De Angelis, Marta; Messore, Antonella; Ialongo, Davide; Scipione, Luigi; Tudino, Valeria; D'auria, Felicia Diodata; Di Santo, Roberto; Garzoli, Stefania; Stringaro, Annarita; Colone, Marisa; Marchetti, Magda; Superti, Fabiana; Nencioni, Lucia; Costi, Roberta - 01a Articolo in rivista
paper: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. 1-14 - issn: 1420-3049 - wos: WOS:000816243700001 (5) - scopus: 2-s2.0-85131746075 (7)

11573/1638214 - 2022 - Evaluation of the Anti-Histoplasma capsulatum activity of Indole and Nitrofuran derivatives and their pharmacological safety in three-dimensional cell cultures
Vaso, C. O.; Bila, N. M.; Pandolfi, F.; De Vita, D.; Bortolami, M.; Bonatti, J. L. C.; De Moraes Silva, R. A.; Goncalves, L. N. C.; Tudino, V.; Costi, R.; Di Santo, R.; Mendes-Giannini, M. J. S.; Costa-Orlandi, C. B.; Scipione, L.; Fusco-Almeida, A. M. - 01a Articolo in rivista
paper: PHARMACEUTICS (Basel: MDPI, 2009-) pp. 1-23 - issn: 1999-4923 - wos: WOS:000803586100001 (4) - scopus: 2-s2.0-85130346777 (4)

11573/1638210 - 2022 - Synthesis and evaluation of the antifungal and toxicological activity of Nitrofuran derivatives
Vaso, C. O.; Pandolfi, F.; Bila, N. M.; De Vita, D.; Bortolami, M.; Mendes-Giannini, M. J. S.; Tudino, V.; Costi, R.; Costa-Orlandi, C. B.; Fusco-Almeida, A. M.; Scipione, L. - 01a Articolo in rivista
paper: PHARMACEUTICS (Basel: MDPI, 2009-) pp. 1-19 - issn: 1999-4923 - wos: WOS:000774275300001 (3) - scopus: 2-s2.0-85126453264 (3)

11573/1564954 - 2021 - Toxicological aspects of cannabinoid, pesticide and metal levels detected in light Cannabis inflorescences grown in Italy
Amendola, G.; Bocca, B.; Picardo, V.; Pelosi, P.; Battistini, B.; Ruggieri, F.; Attard Barbini, D.; De Vita, D.; Madia, V. N.; Messore, A.; Di Santo, R.; Costi, R. - 01a Articolo in rivista
paper: FOOD AND CHEMICAL TOXICOLOGY (Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. - - issn: 0278-6915 - wos: WOS:000696988600002 (6) - scopus: 2-s2.0-85112006002 (8)

11573/1546419 - 2021 - Design, synthesis and biological evaluation of a series of iron and copper chelating deferiprone derivatives as new agents active against Candida albicans
Bortolami, Martina; Pandolfi, Fabiana; Messore, Antonella; Rocco, Daniele; Feroci, Marta; Di Santo, Roberto; De Vita, Daniela; Costi, Roberta; Cascarino, Paola; Simonetti, Giovanna; Scipione, Luigi - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 1-7 - issn: 0960-894X - wos: WOS:000655255700006 (6) - scopus: 2-s2.0-85105482975 (7)

11573/1584588 - 2021 - New pyrimidine and pyridine derivatives as multitarget cholinesterase inhibitors. Design, synthesis, and in vitro and in cellulo evaluation
Bortolami, Martina; Pandolfi, Fabiana; Tudino, Valeria; Messore, Antonella; Madia, Valentina Noemi; De Vita, Daniela; Di Santo, Roberto; Costi, Roberta; Romeo, Isabella; Alcaro, Stefano; Colone, Marisa; Stringaro, Annarita; Espargaró, Alba; Sabatè, Raimon; Scipione, Luigi - 01a Articolo in rivista
paper: ACS CHEMICAL NEUROSCIENCE (Washington, D.C. : American Chemical Society) pp. 4090-4112 - issn: 1948-7193 - wos: WOS:000715842900011 (12) - scopus: 2-s2.0-85118138783 (12)

11573/1404920 - 2021 - Towards a new application of amaranth seed oil as an agent against Candida albicans
De Vita, Daniela; Messore, Antonella; Toniolo, Chiara; Frezza, Claudio; Scipione, Luigi; Bertea, Cinzia Margherita; Micera, Marco; Di Sarno, Veronica; Madia, Valentina Noemi; Pindinello, Ivano; Roscilli, Patrizia; Botto, Alfonso; Simonetti, Giovanna; Orekhova, Anastasia; Manfredini, Stefano; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: NATURAL PRODUCT RESEARCH (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 4621-4626 - issn: 1478-6419 - wos: WOS:000500457200001 (14) - scopus: 2-s2.0-85075913942 (5)

11573/1525063 - 2021 - Phytochemical analysis and biological activities of the ethanolic extract of Daphne sericea Vahl flowering aerial parts collected in Central Italy
Frezza, Claudio; Venditti, Alessandro; De Vita, Daniela; Sciubba, Fabio; Tomai, Pierpaolo; Franceschin, Marco; Di Cecco, Mirella; Ciaschetti, Giampiero; Di Sotto, Antonella; Stringaro, Annarita; Colone, Marisa; Gentili, Alessandra; Serafini, Mauro; Bianco, Armandodoriano - 01a Articolo in rivista
paper: BIOMOLECULES (Basel: MDPI) pp. 1-17 - issn: 2218-273X - wos: WOS:000633395600001 (4) - scopus: 2-s2.0-85101834453 (5)

11573/1540215 - 2021 - Investigation of Commiphora myrrha (Nees) Engl. oil and its main components for antiviral activity
Madia, Valentina Noemi; De Angelis, Marta; De Vita, Daniela; Messore, Antonella; De Leo, Alessandro; Ialongo, Davide; Tudino, Valeria; Saccoliti, Francesco; De Chiara, Giovanna; Garzoli, Stefania; Scipione, Luigi; Palamara, Anna Teresa; Di Santo, Roberto; Nencioni, Lucia; Costi, Roberta - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. - - issn: 1424-8247 - wos: WOS:000634055800001 (16) - scopus: 2-s2.0-85102987115 (19)

11573/1564144 - 2021 - Recent advances in recovery of lycopene from tomato waste. A potent antioxidant with endless benefits
Madia, Valentina Noemi; De Vita, Daniela; Ialongo, Davide; Tudino, Valeria; De Leo, Alessandro; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta; Messore, Antonella - 01a Articolo in rivista
paper: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. 1-18 - issn: 1420-3049 - wos: WOS:000682223800001 (33) - scopus: 2-s2.0-85111602310 (45)

11573/1540619 - 2021 - Analytical characterization of an inulin-type fructooligosaccharide from root-tubers of Asphodelus ramosus L
Madia, Valentina Noemi; De Vita, Daniela; Messore, Antonella; Toniolo, Chiara; Tudino, Valeria; De Leo, Alessandro; Pindinello, Ivano; Ialongo, Davide; Saccoliti, Francesco; D'ursi, Anna Maria; Grimaldi, Manuela; Ceccobelli, Pietro; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. - - issn: 1424-8247 - wos: WOS:000634075100001 (5) - scopus: 2-s2.0-85103099178 (4)

11573/1565318 - 2021 - Small-molecule inhibitors of HIV-1 reverse transcriptase-associated ribonuclease H function. Challenges and recent developments
Madia, Valentina Noemi; Messore, Antonella; De Leo, Alessandro; Tudino, Valeria; Pindinello, Ivano; Saccoliti, Francesco; De Vita, Daniela; Scipione, Luigi; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: CURRENT MEDICINAL CHEMISTRY (Hilversum: Bentham Science Publishers) pp. 1-33 - issn: 1875-533X - wos: WOS:000696992000004 (3) - scopus: 2-s2.0-85115249511 (4)

11573/1493998 - 2021 - Design, synthesis and biological evaluation of new pyrimidine derivatives as anticancer agents
Madia, Valentina Noemi; Nicolai, Alice; Messore, Antonella; De Leo, Alessandro; Ialongo, Davide; Tudino, Valeria; Saccoliti, Francesco; De Vita, Daniela; Scipione, Luigi; Artico, Marco; Taurone, Samanta; Taglieri, Ludovica; Di Santo, Roberto; Scarpa, Susanna; Costi, Roberta - 01a Articolo in rivista
paper: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. - - issn: 1420-3049 - wos: WOS:000615455300001 (11) - scopus: 2-s2.0-85101195321 (16)

11573/1556284 - 2021 - Quinolinonyl non-diketo acid derivatives as Inhibitors of HIV-1 ribonuclease H and polymerase functions of reverse transcriptase
Messore, Antonella; Corona, Angela; Madia, Valentina Noemi; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Ialongo, Davide; Scipione, Luigi; De Vita, Daniela; Amendola, Giorgio; Novellino, Ettore; Cosconati, Sandro; Métifiot, Mathieu; Andreola, Marie-Line; Esposito, Francesca; Grandi, Nicole; Tramontano, Enzo; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 8579-8598 - issn: 0022-2623 - wos: WOS:000668340800039 (9) - scopus: 2-s2.0-85108607601 (8)

11573/1553152 - 2021 - Anti-tumoral effects of a (1H-pyrrol-1-yl)methyl-1H-benzoimidazole carbamate ester derivative on head and neck squamous carcinoma cell lines
Nicolai, Alice; Madia, Valentina Noemi; Messore, Antonella; De Vita, Daniela; De Leo, Alessandro; Ialongo, Davide; Tudino, Valeria; Tortorella, Elisabetta; Scipione, Luigi; Taurone, Samanta; Pergolizzi, Tiziano; Artico, Marco; Di Santo, Roberto; Costi, Roberta; Scarpa, Susanna - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. - - issn: 1424-8247 - wos: WOS:000666329400001 (6) - scopus: 2-s2.0-85110773299 (6)

11573/1408596 - 2021 - A new diterpene and other compounds from the unripe female cones of Wollemia nobilis
Venditti, Alessandro; Frezza, Claudio; Rossi, Giacomo; Sciubba, Fabio; Ornano, Luigi; De Vita, Daniela; Toniolo, Chiara; Tomassini, Lamberto; Foddai, Sebastiano; Nicoletti, Marcello; Di Cocco, Maria Enrica; Bianco, Armandodoriano; Serafini, Mauro - 01a Articolo in rivista
paper: NATURAL PRODUCT RESEARCH (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 3839-3849 - issn: 1478-6419 - wos: WOS:000523315600001 (5) - scopus: 2-s2.0-85082625999 (4)

11573/1482023 - 2020 - On the intrinsic reactivity of highly potent trypanocidal cruzain inhibitors
Bonatto, V.; Batista, P. H. J.; Cianni, L.; De Vita, D.; Silva, D. G.; Cedron, R.; Tezuka, D. Y.; De Albuquerque, S.; Moraes, C. B.; Franco, C. H.; Lameira, J.; Leitao, A.; Montanari, C. A. - 01a Articolo in rivista
paper: RSC MEDICINAL CHEMISTRY (Cambridge: Royal Society of Chemistry, 2020-) pp. 1275-1284 - issn: 2632-8682 - wos: WOS:000591526600007 (7) - scopus: 2-s2.0-85096602811 (7)

11573/1395352 - 2020 - New deferiprone derivatives as multi-functional cholinesterase inhibitors. Design, synthesis and in vitro evaluation
Bortolami, Martina; Pandolfi, Fabiana; De Vita, Daniela.; Carafa, Camilla; Messore, Antonella; Di Santo, Roberto; Feroci, Marta; Costi, Roberta; Chiarotto, Isabella; Bagetta, Donatella; Alcaro, Stefano; Colone, Marisa; Stringaro, Annarita; Scipione, Luigi - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 1-17 - issn: 0223-5234 - wos: WOS:000539425800007 (29) - scopus: 2-s2.0-85084066662 (33)

11573/1477079 - 2020 - Molecular design aided by random forests and synthesis of potent trypanocidal agents as cruzain inhibitors for Chagas disease treatment
De Albuquerque, S.; Cianni, L.; De Vita, D.; Duque, C.; Gomes, A. S. M.; Gomes, P.; Laughton, C.; Leitao, A.; Montanari, C. A.; Montanari, R.; Ribeiro, J. F. R.; Da Silva, J. S.; Teixeira, C. - 01a Articolo in rivista
paper: CHEMICAL BIOLOGY & DRUG DESIGN (Blackwell Munksgaar) pp. 948-960 - issn: 1747-0277 - wos: WOS:000577619900006 (1) - scopus: 2-s2.0-85092586503 (1)

11573/1215347 - 2020 - Secondary metabolites of Tilia tomentosa Moench inflorescences collected in Central Italy: chemotaxonomy relevance and phytochemical rationale of traditional use
Frezza, Claudio; De Vita, Daniela; Spinaci, Giulia; Sarandrea, Marco; Venditti, Alessandro; Bianco, Armandodoriano - 01a Articolo in rivista
paper: NATURAL PRODUCT RESEARCH (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1167-1174 - issn: 1478-6419 - wos: WOS:000526891500018 (9) - scopus: 2-s2.0-85060036247 (12)

11573/1449132 - 2020 - Harpagide.Occurrence in plants and biological activities - A review
Frezza, Claudio; De Vita, Daniela; Toniolo, Chiara; Ventrone, Antonio; Tomassini, Lamberto; Foddai, Sebastiano; Nicoletti, Marcello; Guiso, Marcella; Bianco, Armandodoriano; Serafini, Mauro - 01g Articolo di rassegna (Review)
paper: FITOTERAPIA (Amsterdam Netherlands:Elsevier BV Milano : Inverni & Della Beffa : Elsevier) pp. 1-13 - issn: 1971-551X - wos: WOS:000600721100019 (9) - scopus: 2-s2.0-85094586400 (13)

11573/1431978 - 2020 - Phytochemistry, chemotaxonomy, and biological activities of the Araucariaceae family. A Review
Frezza, Claudio; Venditti, Alessandro; De Vita, Daniela; Toniolo, Chiara; Franceschin, Marco; Ventrone, Antonio; Tomassini, Lamberto; Foddai, Sebastiano; Guiso, Marcella; Nicoletti, Marcello; Bianco, Armandodoriano; Serafini, Mauro - 01g Articolo di rassegna (Review)
paper: PLANTS (Basel: MDPI) pp. 1-73 - issn: 2223-7747 - wos: WOS:000554209800001 (22) - scopus: 2-s2.0-85087986275 (28)

11573/1347864 - 2020 - Nor-lignans. Occurrence in plants and biological activities. A review
Frezza, Claudio; Venditti, Alessandro; Toniolo, Chiara; De Vita, Daniela; Franceschin, Marco; Ventrone, Antonio; Tomassini, Lamberto; Foddai, Sebastiano; Guiso, Marcella; Nicoletti, Marcello; Serafini, Mauro; Bianco, Armandodoriano - 01g Articolo di rassegna (Review)
paper: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. 1-42 - issn: 1420-3049 - wos: WOS:000513770000197 (16) - scopus: 2-s2.0-85077445458 (17)

11573/1477075 - 2020 - N-Sulfonyl dipeptide nitriles as inhibitors of human cathepsin S. In silico design, synthesis and biochemical characterization
Lemke, Carina; Cianni, Lorenzo; Feldmann, Christian; Gilberg, Erik; Yin, Jiafei; Dos Reis Rocho, Fernanda; De Vita, Daniela; Bartz, Ulrike; Bajorath, Jürgen; Montanari, Carlos A.; Gütschow, Michael - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. - - issn: 0960-894X - wos: WOS:000571824300001 (4) - scopus: 2-s2.0-85088941783 (4)

11573/1477077 - 2020 - Synthesis and matched molecular pair analysis of covalent reversible inhibitors of the cysteine protease CPB
Matos, Thiago Kelvin Brito; Batista, Pedro Henrique Jatai; Dos Reis Rocho, Fernanda; De Vita, Daniela; Pearce, Nicholas; Kellam, Barrie; Montanari, Carlos Alberto; Leitão, Andrei - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. - - issn: 0960-894X - wos: WOS:000571829600001 (2) - scopus: 2-s2.0-85089377598 (2)

11573/1408850 - 2020 - Pyrrolyl pyrazoles as non-diketo acid inhibitors of the HIV-1 ribonuclease H function of reverse transcriptase
Messore, Antonella; Corona, Angela; Madia, Valentina Noemi; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Scipione, Luigi; De Vita, Daniela; Amendola, Giorgio; Di Maro, Salvatore; Novellino, Ettore; Cosconati, Sandro; Métifiot, Mathieu; Andreola, Marie-Line; Valenti, Piera; Esposito, Francesca; Grandi, Nicole; Tramontano, Enzo; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: ACS MEDICINAL CHEMISTRY LETTERS (USA: ACS Publications) pp. 798-805 - issn: 1948-5875 - wos: WOS:000535281200029 (22) - scopus: 2-s2.0-85086659986 (24)

11573/1477070 - 2020 - Crystal structure of Leishmania mexicana cysteine protease B in complex with a high-affinity azadipeptide nitrile inhibitor
Ribeiro, Jean F. R.; Cianni, Lorenzo; Li, Chan; Warwick, Thomas G.; De Vita, Daniela; Rosini, Fabiana; Dos Reis Rocho, Fernanda; Martins, Felipe C. P.; Kenny, Peter W.; Lameira, Jeronimo; Leitão, Andrei; Emsley, Jonas; Montanari, Carlos A. - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. - - issn: 0968-0896 - wos: WOS:000596080300010 (5) - scopus: 2-s2.0-85092065887 (6)

11573/1404853 - 2020 - Assessment of the cruzain cysteine protease reversible and Irreversible covalent inhibition mechanism
Silva, José Rogério A; Cianni, Lorenzo; Araujo, Deborah; Batista, Pedro Henrique Jatai; De Vita, Daniela; Rosini, Fabiana; Leitão, Andrei; Lameira, Jerônimo; Montanari, Carlos A - 01a Articolo in rivista
paper: JOURNAL OF CHEMICAL INFORMATION AND MODELING (AMER CHEMICAL SOC, 1155 16TH ST, NW, WASHINGTON, USA, DC, 20036) pp. 1666-1677 - issn: 1549-9596 - wos: WOS:000526390800054 (27) - scopus: 2-s2.0-85082146768 (26)

11573/1404923 - 2019 - Anti-inflammatory and antioxidant properties of dehydrated potato-derived bioactive compounds in intestinal cells
Basilicata, Manuela Giovanna; Pepe, Giacomo; Rapa, Shara Francesca; Merciai, Fabrizio; Ostacolo, Carmine; Manfra, Michele; Di Sarno, Veronica; Autore, Giuseppina; De Vita, Daniela; Marzocco, Stefania; Campiglia, Pietro - 01a Articolo in rivista
paper: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (Basel: MDPI Center) pp. 1-15 - issn: 1422-0067 - wos: WOS:000504428300269 (15) - scopus: 2-s2.0-85076174100 (21)

11573/1285185 - 2019 - Comparison of different methods for the extraction of cannabinoids from cannabis
De Vita, D.; Madia, V. N.; Tudino, V.; Saccoliti, F.; De Leo, A.; Messore, A.; Roscilli, P.; Botto, A.; Pindinello, I.; Santilli, G.; Scipione, L.; Costi, R.; Di Santo, R. - 01a Articolo in rivista
paper: NATURAL PRODUCT RESEARCH (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1-7 - issn: 1478-6419 - wos: WOS:000575920700013 (32) - scopus: 2-s2.0-85065155862 (37)

11573/1307384 - 2019 - Pedicularis L. Genus. Systematics, botany, phytochemistry, chemotaxonomy, ethnopharmacology, and other
Frezza, Claudio; Venditti, Alessandro; Toniolo, Chiara; De Vita, Daniela; Serafini, Ilaria; Ciccòla, Alessandro; Franceschin, Marco; Ventrone, Antonio; Tomassini, Lamberto; Foddai, Sebastiano; Guiso, Marcella; Nicoletti, Marcello; Bianco, Armandodoriano; Serafini, Mauro - 01g Articolo di rassegna (Review)
paper: PLANTS (Basel: MDPI) pp. 1-53 - issn: 2223-7747 - wos: WOS:000487958100013 (14) - scopus: 2-s2.0-85073392513 (18)

11573/1404902 - 2019 - Synthesis and structure-activity relationship of nitrile-based cruzain inhibitors incorporating a trifluoroethylamine-based P2 amide replacement
Gomes, Juliana C; Cianni, Lorenzo; Ribeiro, Jean; Dos Reis Rocho, Fernanda; Da Costa Martins Silva, Samelyn; Batista, Pedro Henrique Jatai; Moraes, Carolina Borsoi; Franco, Caio Haddad; Freitas-Junior, Lucio H G; Kenny, Peter W; Leitão, Andrei; Burtoloso, Antonio C B; De Vita, Daniela; Montanari, Carlos A - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 1-14 - issn: 0968-0896 - wos: WOS:000491130200001 (17) - scopus: 2-s2.0-85072563778 (19)

11573/1405464 - 2019 - Tegaserod for the treatment of Irritable Bowel syndrome
Madia, Valentina Noemi; Messore, Antonella; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; De Vita, Daniela; Bortolami, Martina; Scipione, Luigi; Pindinello, Ivano; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: ANTI-INFLAMMATORY & ANTI-ALLERGY AGENTS IN MEDICINAL CHEMISTRY (Hilversum : Bentham Science Publsihers) pp. 1-28 - issn: 1871-5230 - wos: (0) - scopus: 2-s2.0-85083912835 (0)

11573/1218854 - 2019 - Searching for new agents active against candida albicans biofilm: a series of indole derivatives, design, synthesis and biological evaluation
Pandolfi, Fabiana; D'acierno, Federica; Bortolami, Martina; De Vita, Daniela; Gallo, Fabio; De Meo, Alessandra; Di Santo, Roberto; Costi, Roberta; Simonetti, Giovanna; Scipione, Luigi - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 93-106 - issn: 0223-5234 - wos: WOS:000459358600008 (27) - scopus: 2-s2.0-85060089854 (29)

11573/1222183 - 2019 - Design, synthesis, and biological evaluation of new 1-(aryl-1H-pyrrolyl)(phenyl)methyl-1H-imidazole derivatives as antiprotozoal agents
Saccoliti, Francesco; Madia, Valentina Noemi; Tudino, Valeria; De Leo, Alessandro; Pescatori, Luca; Messore, Antonella; De Vita, Daniela; Scipione, Luigi; Brun, Reto; Kaiser, Marcel; Mäser, Pascal; Calvet Alvarez, Claudia Magalhaes; Jennings, Gareth K; Podust, Larissa M; Pepe, Giacomo; Cirilli, Roberto; Faggi, Cristina; Di Marco, Annalise; Battista, Maria Rosaria; Summa, Vincenzo; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1330-1347 - issn: 0022-2623 - wos: WOS:000459223600016 (24) - scopus: 2-s2.0-85061636363 (29)

11573/1068937 - 2018 - Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents
Carradori, Simone; Ottuso, Francesco; Petzer, Anèl; Bagetta, Donatella; De Monte, Celeste; Secci, Daniela; De Vita, Daniela; Guglielmi, Paolo; Zengin, Gokhan; Aktumsek, Abdurrahman; Alcaro, Stefano; Petzer, Jacobus P. - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY ([Paris] : Elsevier, [198?]-) pp. 1543-1552 - issn: 1768-3254 - wos: WOS:000423641400032 (38) - scopus: 2-s2.0-85034651451 (40)

11573/1404906 - 2018 - Leveraging the cruzain S3 subsite to increase affinity for reversible covalent inhibitors
Cianni, Lorenzo; Sartori, Geraldo; Rosini, Fabiana; De Vita, Daniela; Pires, Gabriel; Lopes, Bianca Rebelo; Leitão, Andrei; Burtoloso, Antonio C B; Montanari, Carlos A - 01a Articolo in rivista
paper: BIOORGANIC CHEMISTRY (Academic Press Incorporated:6277 Sea Harbor Drive:Orlando, FL 32887:(800)543-9534, (407)345-4100, EMAIL: ap@acad.com, INTERNET: http://www.idealibrary.com, Fax: (407)352-3445) pp. 285-292 - issn: 0045-2068 - wos: WOS:000436773100031 (18) - scopus: 2-s2.0-85047055263 (19)

11573/1404892 - 2018 - Experimental study and computational modelling of cruzain cysteine protease inhibition by dipeptidyl nitriles
Dos Santos, Alberto Monteiro; Cianni, Lorenzo; De Vita, Daniela; Rosini, Fabiana; Leitão, Andrei; Laughton, Charles A; Lameira, Jerônimo; Montanari, Carlos A - 01a Articolo in rivista
paper: PHYSICAL CHEMISTRY CHEMICAL PHYSICS (Thomas Graham House, Science Park, Cambridge: Royal Society of Chemistry) pp. 24317-24328 - issn: 1463-9076 - wos: WOS:000446766300046 (30) - scopus: 2-s2.0-85054100853 (27)

11573/1221546 - 2018 - Novel symmetrical benzazolyl derivatives endowed with potent anti-heparanase activity
Messore, Antonella; Madia, Valentina Noemi; Pescatori, Luca; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Bortolami, Martina; De Vita, Daniela; Scipione, Luigi; Pepi, Federico; Costi, Roberta; Rivara, Silvia; Scalvini, Laura; Mor, Marco; Ferrara, Fabiana Fosca; Pavoni, Emiliano; Roscilli, Giuseppe; Cassinelli, Giuliana; Milazzo, Ferdinando M; Battistuzzi, Gianfranco; Di Santo, Roberto; Giannini, Giuseppe - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 10834-10859 - issn: 0022-2623 - wos: WOS:000453488200031 (17) - scopus: 2-s2.0-85058215116 (16)

11573/1176720 - 2018 - Biological evaluation and structure-activity relationships of imidazole-based compounds as antiprotozoal agents
Saccoliti, Francesco; Madia, Valentina Noemi; Tudino, Valeria; De Leo, Alessandro; Pescatori, Luca; Messore, Antonella; De Vita, Daniela; Scipione, Luigi; Brun, Reto; Kaiser, Marcel; Mäser, Pascal; Magalhaes Calvet, Claudia; K Jennings, Gareth; M Podust, Larissa; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 53-60 - issn: 0223-5234 - wos: WOS:000443663200005 (16) - scopus: 2-s2.0-85049312582 (21)

11573/972447 - 2017 - Inhibition of the α-carbonic anhydrase from Vibrio cholerae with amides and sulfonamides incorporating imidazole moieties
De Vita, Daniela; Angeli, Andrea; Pandolfi, Fabiana; Bortolami, Martina; Costi, Roberta; Di Santo, Roberto; Suffredini, Elisabetta; Ceruso, Mariangela; Del Prete, Sonia; Capasso, Clemente; Scipione, Luigi; Supuran, Claudiu T. - 01a Articolo in rivista
paper: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 798-804 - issn: 1475-6366 - wos: WOS:000404271200006 (36) - scopus: 2-s2.0-85020209278 (38)

11573/1011030 - 2017 - New pyridine derivatives as inhibitors of acetylcholinesterase and amyloid aggregation
Pandolfi, Fabiana; De Vita, Daniela; Bortolami, Martina; Coluccia, Antonio; Di Santo, Roberto; Costi, Roberta; Andrisano, Vincenza; Alabiso, Francesco; Bergamini, Christian; Fato, Romana; Bartolini, Manuela; Scipione, Luigi - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 197-210 - issn: 0223-5234 - wos: WOS:000417962900018 (26) - scopus: 2-s2.0-85030860178 (30)

11573/1404930 - 2017 - A comparative study of warheads for design of cysteine protease inhibitors
Silva, Daniel G; Ribeiro, Jean F R; De Vita, Daniela; Cianni, Lorenzo; Franco, Caio Haddad; Freitas-Junior, Lucio H; Moraes, Carolina Borsoi; Rocha, Josmar R; Burtoloso, Antonio C B; Kenny, Peter W; Leitão, Andrei; Montanari, Carlos A - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 5031-5035 - issn: 0960-894X - wos: WOS:000414000000019 (27) - scopus: 2-s2.0-85031677600 (29)

11573/866932 - 2016 - In vitro screening of 2-(1H-imidazol-1-yl)-1-phenylethanol derivatives as antiprotozoal agents and docking studies on Trypanosoma cruzi CYP51
De Vita, Daniela; Moraca, Francesca; Zamperini, Claudio; Pandolfi, Fabiana; Di Santo, Roberto; Matheeussen, An; Maes, Louis; Tortorella, Silvano; Scipione, Luigi - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 28-33 - issn: 0223-5234 - wos: WOS:000374609000003 (18) - scopus: 2-s2.0-84959016857 (19)

11573/874787 - 2016 - Discovery of in vitro antitubercular agents through in silico ligand-based approaches
De Vita, Daniela; Pandolfi, Fabiana; Cirilli, Roberto; Scipione, Luigi; Di Santo, Roberto; Friggeri, Laura; Mori, Mattia; Fiorucci, Diego; Maccari, Giorgio; Arul Christopher, Robert Selwyne; Zamperini, Claudio; Pau, Valentina; De Logu, Alessandro; Tortorella, Silvano; Botta, Maurizio - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 169-180 - issn: 0223-5234 - wos: WOS:000382269700015 (20) - scopus: 2-s2.0-84971233923 (20)

11573/903468 - 2016 - New N,N-dimethylcarbamate inhibitors of acetylcholinesterase: design synthesis and biological evaluation
De Vita, Daniela; Pandolfi, Fabiana; Ornano, Luigi; Feroci, Marta; Chiarotto, Isabella; Sileno, Ilaria; Pepi, Federico; Costi, Roberta; Di Santo, Roberto; Scipione, Luigi - 01a Articolo in rivista
paper: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1-8 - issn: 1475-6366 - wos: WOS:000391904900013 (11) - scopus: 2-s2.0-84984870776 (11)

11573/916308 - 2016 - Exploring the anti-biofilm activity of cinnamic acid derivatives in Candida albicans
De Vita, Daniela; Simonetti, Giovanna; Pandolfi, Fabiana; Costi, Roberta; Di Santo, Roberto; D'auria, Felicia Diodata; Scipione, Luigi - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 5931-5935 - issn: 0960-894X - wos: WOS:000389784500020 (19) - scopus: 2-s2.0-84999015180 (24)

11573/741200 - 2015 - (Thiazol-2-yl)hydrazone derivatives from acetylpyridines as dual inhibitors of MAO and AChE: synthesis, biological evaluation and molecular modeling studies
D’Ascenzio, M; Chimenti, Paola; Gidaro, Mc; De Monte, Celeste; De Vita, Daniela; Granese, Arianna; Scipione, Luigi; Di Santo, Roberto; Costa, G; Alcaro, S; Yáñez, M; Carradori, S. - 01a Articolo in rivista
paper: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 908-919 - issn: 1475-6366 - wos: WOS:000369915500007 (30) - scopus: 2-s2.0-84945957051 (30)

11573/541604 - 2015 - Design, synthesis and evaluation of 3,4-dihydroxybenzoic acid derivatives as antioxidants, bio-metal chelating agents and acetylcholinesterase inhibitors
Friggeri, Laura; De Vita, Daniela; Pandolfi, Fabiana; Tortorella, Silvano; Costi, Roberta; Di Santo, Roberto; Scipione, Luigi - 01a Articolo in rivista
paper: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 166-172 - issn: 1475-6366 - wos: WOS:000347956500024 (7) - scopus: 2-s2.0-84921307137 (7)

11573/516524 - 2015 - Efficient synthesis of 3,5-dicarbamoyl-1,4-dihydropyridines from pyridinium salts. Key molecules in understanding NAD(P)+/NAD(P)H pathways
Mellini, Paolo; De Vita, Daniela; Di Rienzo, Barbara; La Rosa, Salvatore; Padova, Alessandro; Scipione, Luigi; Tortorella, Silvano; Friggeri, Laura - 01a Articolo in rivista
paper: JOURNAL OF HETEROCYCLIC CHEMISTRY (Hetero Corporation:PO Box 170:Provo, UT 84603:(801)400-7373, EMAIL: jhetchem@yahoo.com, Fax: (801)356-7373) pp. 221-226 - issn: 0022-152X - wos: WOS:000348574100033 (3) - scopus: 2-s2.0-85027932819 (3)

11573/541603 - 2014 - Activity of caffeic acid derivatives against Candida albicans biofilm
De Vita, Daniela; Friggeri, Laura; D'auria, Felicia Diodata; Pandolfi, Fabiana; Francesco, Piccoli; Panella, Simona; Palamara, Anna Teresa; Simonetti, Giovanna; Scipione, Luigi; R., Santo; Di Santo, Roberto; Costi, Roberta; Tortorella, Silvano - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 1502-1505 - issn: 0960-894X - wos: WOS:000332391900011 (50) - scopus: 2-s2.0-84895795071 (57)

11573/541606 - 2014 - Efficient electrochemical N-alkylation of N-boc-protected 4-aminopyridines: towards new biologically active compounds.
Feroci, Marta; Chiarotto, Isabella; Forte, Gianpiero; Simonetti, Giovanna; D'auria, Felicia Diodata; Diodata, ; Maes, Louis; Scipione, Luigi; Friggeri, Laura; Di Santo, Roberto; De Vita, Daniela; Tortorella, Silvano - 01a Articolo in rivista
paper: ISRN ORGANIC CHEMISTRY (Cairo: Hindawi Publishing Corporation) pp. 1-10 - issn: 2090-5149 - wos: (0) - scopus: (0)

11573/579587 - 2014 - Synthesis, biological evaluation and structure-activity correlation study of a series of imidazol-based compounds as Candida albicans inhibitors
Francesca, Moraca; De Vita, Daniela; Pandolfi, Fabiana; Di Santo, Roberto; Costi, Roberta; Roberto, Cirilli; D'auria, Felicia Diodata; Panella, Simona; Palamara, Anna Teresa; Simonetti, Giovanna; Maurizio, Botta; Scipione, Luigi - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 665-673 - issn: 0223-5234 - wos: WOS:000340689600059 (21) - scopus: 2-s2.0-84904025140 (21)

11573/684252 - 2014 - Structural basis for rational design of inhibitors targeting Trypanosoma cruzi sterol 14α-demethylase: two regions of the enzyme molecule potentiate its inhibition
Friggeri, L.; Hargrove, T. Y.; Rachakonda, G.; Williams, A. D.; Wawrzak, Z.; Di Santo, Roberto; De Vita, Daniela; Waterman, M. R.; Tortorella, Silvano; Villalta, F.; Lepesheva, G. I. - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 6704-6717 - issn: 0022-2623 - wos: WOS:000340445900033 (36) - scopus: 2-s2.0-84906302973 (41)

11573/515673 - 2013 - Pharmacophore assessment through 3-D QSAR: evaluation of the predictive ability on new derivatives by the application on a series of antitubercular agents
Friggeri, Laura; Ballante, Flavio; Ragno, Rino; Musmuca, Ira; De Vita, Daniela; Manetti, F. .; Biava, Mariangela; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta; Feroci, Marta; Tortorella, Silvano - 01a Articolo in rivista
paper: JOURNAL OF CHEMICAL INFORMATION AND MODELING (AMER CHEMICAL SOC, 1155 16TH ST, NW, WASHINGTON, USA, DC, 20036) pp. 1463-1474 - issn: 1549-9596 - wos: WOS:000321074700019 (7) - scopus: 2-s2.0-84879596019 (10)

11573/516522 - 2013 - New promising compounds with in vitro nanomolar activity against Trypanosoma cruzi
Friggeri, Laura; Scipione, Luigi; Costi, Roberta; Marcel, Kaiser; Francesca, Moraca; Claudio, Zamperini; Botta, Bruno; Di Santo, Roberto; De Vita, Daniela; Reto, Brun; Tortorella, Silvano - 01a Articolo in rivista
paper: ACS MEDICINAL CHEMISTRY LETTERS (USA: ACS Publications) pp. 538-541 - issn: 1948-5875 - wos: WOS:000321883900011 (15) - scopus: 2-s2.0-84879097485 (15)

11573/434328 - 2012 - Synthesis and antifungal activity of a new series of 2-(1H-imidazol-1-yl)-1-phenylethanol derivatives
De Vita, Daniela; Scipione, Luigi; Tortorella, Silvano; Mellini, Paolo; Di Rienzo, Barbara; Simonetti, Giovanna; D'auria, Felicia Diodata; Panella, Simona; Roberto, Cirilli; Di Santo, Roberto; Palamara, Anna Teresa - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 334-342 - issn: 0223-5234 - wos: WOS:000302033300033 (32) - scopus: 2-s2.0-84857239066 (38)

11573/440836 - 2012 - Electrogenerated acetonitrile anion induced selective N-alkylation of bifunctional compounds
Feroci, Marta; De Vita, Daniela; Scipione, Luigi; Sotgiu, Giovanni; Tortorella, Silvano - 01a Articolo in rivista
paper: TETRAHEDRON LETTERS (Oxford; New York; Paris; Frankfurt: Pergamon Press, 1959-) pp. 2564-2567 - issn: 0040-4039 - wos: WOS:000303372200020 (6) - scopus: 2-s2.0-84859779446 (7)

11573/495328 - 2012 - Carprofen Analogues as Sirtuin Inhibitors: Enzyme and Cellular Studies
Paolo, Mellini; Vincenzo, Carafa; Barbara Di, Rienzo; Rotili, Dante; De Vita, Daniela; Roberto, Cirilli; Bruno, Gallinella; Donatella Paola, Provvisiero; Salvatore Di, Maro; Ettore, Novellino; Lucia, Altucci; Mai, Antonello - 01a Articolo in rivista
paper: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. 1905-1908 - issn: 1860-7187 - wos: WOS:000310485200005 (14) - scopus: 2-s2.0-84868149996 (15)

11573/357392 - 2011 - Activity of Drugs Against Dormant Mycobacterium tuberculosis
G., Piccaro; P., Filippini; F., Giannoni; Scipione, Luigi; Tortorella, Silvano; De Vita, Daniela; Mellini, Paolo; L., Fattorini - 01a Articolo in rivista
paper: JOURNAL OF CHEMOTHERAPY (ESIFT Srl:Casella Postale 147, I 50018 Scandicci Fi Italy:011 39 055 4271516, EMAIL: mary@jchemother.it, Fax: 011 39 055 4271280) pp. 28-31 - issn: 1120-009X - wos: WOS:000294584500012 (4) - scopus: 2-s2.0-80052780950 (4)

11573/46397 - 2010 - Facile and Efficient Synthesis of 4-Alkyl Derivatives of 3-Carbamoyl- and 3,5-Dicarbamoylpyridines as Nicotinamide Mimetics
Di Rienzo, Barbara; Mellini, Paolo; Tortorella, Silvano; De Vita, Daniela; Scipione, Luigi - 01a Articolo in rivista
paper: SYNTHESIS (Stuttgart : Thieme Verlag) pp. 3835-3839 - issn: 0039-7881 - wos: WOS:000284533700007 (1) - scopus: 2-s2.0-78149465862 (3)

11573/46403 - 2010 - Simple Choline Esters as Potential Anti-Alzheimer Agents
Stefano, Alcaro; Rosaria, Arcone; Giosue, Costa; De Vita, Daniela; Michelangelo, Iannone; Francesco, Ortuso; Antonio, Procopio; Raffaele, Pasceri; Domenicantonio, Rotiroti; Scipione, Luigi - 01a Articolo in rivista
paper: CURRENT PHARMACEUTICAL DESIGN (Bentham Science Publishers BV:PO Box 7917, Exec Ste Y 26, Saif Zone Sharjah Uae:011 971 6 5571132, EMAIL: benthams@emirates.net.ae, INTERNET: http://www.bentham.org, Fax: 011 971 6 5571134) pp. 692-697 - issn: 1381-6128 - wos: WOS:000274032700013 (9) - scopus: 2-s2.0-77950241009 (13)

11573/358977 - 2008 - Choline pivaloyl ester enhances brain expression of both nerve growth factor and high-affinity receptor TrkA, and reverses memory and cognitive deficits, in rats with excitotoxic lesion of nucleus basalis magnocellularis
Rispoli, V.; Marra, R.; Costa, N.; Rotiroti, D.; Tirassa, P.; Scipione, Luigi; De Vita, Daniela; Liberatore, F.; Carelli, V. - 01a Articolo in rivista
paper: BEHAVIOURAL BRAIN RESEARCH (Amsterdam; London; New York NY; Tokyo: Elsevier) pp. 22-32 - issn: 0166-4328 - wos: WOS:000255766800003 (7) - scopus: 2-s2.0-41949132598 (6)

11573/366237 - 2008 - 4-aminopyridine derivatives with anticholinesterase and antiamnesic activity
Scipione, Luigi; De Vita, Daniela; Alessandra, Musella; Lisa, Flammini; Simona, Bertoni; Elisabetta, Barocelli - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 309-312 - issn: 0960-894X - wos: WOS:000253720300056 (13) - scopus: 2-s2.0-37549036692 (14)

11573/366509 - 2006 - Choline pivaloyl ester strengthened the benefit effects of Tacrine and Galantamine on electroencephalographic and cognitive performances in nucleus basalis magnocellularis-lesioned and aged rats
V., Rispoli; R., Marra; N., Costa; D., Rotiroti; Scipione, Luigi; De Vita, Daniela; Felice, Liberatore; Vincenzo, Carelli - 01a Articolo in rivista
paper: PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR (Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. 453-467 - issn: 0091-3057 - wos: WOS:000240707000009 (9) - scopus: 2-s2.0-33748712915 (11)

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