11573/1725663 - 2024 -
Targeting protein disulfide isomerase A with newly designed and synthesized aryl derivatives Albano, A.; Madia, V. N.; Ruggieri, G.; Ialongo, D.; Patacchini, E.; Arpacioglu, M.; Messore, A.; Scipione, L.; Altieri, F.; Paglia, G.; Meschiari, G.; Di Santo, R.; Costi, R. - 04f Poster
conference: EFMC-YMCS 2024 11th EFMC Young Medicinal Chemists' Symposium (Rome)
book: EFMC-YMCS 2024 11th EFMC Young Medicinal Chemists' Symposium - ()
11573/1725672 - 2024 -
Design and synthesis of new aryl derivatives as inhibitors of protein disulfide isomerase Albano, A.; Madia, V. N.; Ruggieri, G.; Ialongo, D.; Patacchini, E.; Arpacioglu, M.; Messore, A.; Scipione, L.; Altieri, F.; Paglia, G.; Meschiari, G.; Di Santo, R.; Costi, R. - 04f Poster
conference: EFMC-ISMC 2024 XXVIII EFMC International Symposium on Medicinal Chemistry (Rome)
book: EFMC-ISMC 2024 XXVIII EFMC International Symposium on Medicinal Chemistry - ()
11573/1725678 - 2024 -
New nitrogen based derivatives as SARS-CoV-2 nsp13 inhibitors Albano, A.; Madia, V. N.; Ruggieri, G.; Ialongo, D.; Patacchini, E.; Arpacioglu, M.; Messore, A.; Scipione, L.; Corona, A.; Esposito, F.; Amatore, D.; Faggioni, G.; De Santis, R.; Lista, F.; Tramontano, E.; Di Santo, R.; Costi, R. - 04f Poster
conference: SCI 2024 Chemistry ELEMENTS OF FUTURE - XXVIII Congresso Nazionale della Società Chimica Italiana (Milan)
book: SCI 2024 Chemistry ELEMENTS OF FUTURE - XXVIII Congresso Nazionale della Società Chimica Italiana - ()
11573/1725682 - 2024 -
New quinolinonyl derivatives as SARS-CoV-2 nsp13 inhibitors Albano, A.; Madia, V. N.; Ruggieri, G.; Ialongo, D.; Patacchini, E.; Arpacioglu, M.; Messore, A.; Scipione, L.; Corona, A.; Esposito, F.; Amatore, D.; Faggioni, G.; De Santis, R.; Lista, F.; Tramontano, E.; Di Santo, R.; Costi, R. - 04f Poster
conference: EFMC-ACSMEDI Medicinal Chemistry Frontiers (Utrecht; Netherlands)
book: EFMC-ACSMEDI Medicinal Chemistry Frontiers - ()
11573/1725811 - 2024 -
DEVELOPING NOVEL COMPOUNDS TARGETING AURKA AND HDAC ENZYMES SIMULTANEOUSLY Arpacioglu, M.; Madia, V. N.; Patacchini, E.; Ialongo, D.; Albano, A.; Messore, A.; Ruggieri, G.; De Leo, A.; Scipione, L.; Rotili, D.; Fiorentino, F.; Paiardini, A.; Di Santo, R.; Costi, R. - 04f Poster
conference: The European Federation for Medicinal Chemistry Young Medicinal Chemists' Symposium (Roma, Italia)
book: The European Federation for Medicinal Chemistry Young Medicinal Chemists' Symposium - ()
11573/1725713 - 2024 -
NEW THIAZOLIDINE-4-ONE DERIVATIVES CAPABLE OF INHIBITING SARS-CoV-2 MPRO Arpacioglu, M.; Patacchini, E.; Messore, A.; Madia, V. N.; Ialongo, D.; Albano, A.; Ruggieri, G.; Esposito, F.; Tramontano, E.; Malune, P.; Sankaranarayanan, M.; Costi, R.; Di Santo, R. - 04f Poster
conference: XXVIII Congresso Nazionale della Società Chimica Italiana (Milano, Italia)
book: XXVIII Congresso Nazionale della Società Chimica Italiana - ()
11573/1725680 - 2024 -
Inhibitors of protein-protein interaction between the human receptor ACE2 and the viral protein spike: a new frontier in the fight against SARS-CoV-2. Ialongo, D.; Madia, V. N.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Albano, A.; Ruggieri, G.; Michelini, Z.; Cara, A.; Scipione, L.; Di Santo, R.; Costi, R. - 04f Poster
conference: EFMC-YMCS 2024 11th EFMC Young Medicinal Chemists' Symposium (Rome, Italy)
book: EFMC-YMCS 2024 11th EFMC Young Medicinal Chemists' Symposium - ()
11573/1725677 - 2024 -
Identification of new heterocyclic compounds as protein disulfide isomerase A inhibitors. Ialongo, D.; Messore, A.; Madia, V. N.; Patacchini, E.; Ruggieri, G.; Albano, A.; Arpacioglu, M.; Scipione, L.; Altieri, F.; Paglia, G.; Meschiari, G.; Di Santo, R.; Costi, R. - 04f Poster
conference: SCI 2024 Chemistry ELEMENTS OF FUTURE - XXVIII Congresso Nazionale della Società Chimica Italiana (Milan, Italy)
book: SCI 2024 Chemistry ELEMENTS OF FUTURE - XXVIII Congresso Nazionale della Società Chimica Italiana - ()
11573/1725690 - 2024 -
Indolyl derivatives as SARS-CoV-2 nsp13 inhibitors active against viral replication Madia, V. N.; Albano, A.; Ruggieri, G.; Ialongo, D.; Patacchini, E.; Arpacioglu, M.; Messore, A.; Saccoliti, F.; Scipione, L.; Corona, A.; Emmolo, R.; Amatore, D.; Faggioni, G.; De Santis, R.; Lista, F.; Tramontano, E.; Di Santo, R.; Costi, R. - 04f Poster
conference: 1NF-ACT Meeting 2024 (Pavia)
book: 1NF-ACT Meeting 2024 - ()
11573/1725695 - 2024 -
Discovery of small molecule derivatives as SARS-CoV-2 nsp13 inhibitors: a new strategy to develop broad-spectrum antiviral agents Madia, V. N.; Albano, A.; Ruggieri, G.; Ialongo, D.; Patacchini, E.; Arpacioglu, M.; Messore, A.; Scipione, L.; Corona, A.; Esposito, F.; Amatore, D.; Faggioni, G.; De Santis, R.; Lista, F.; Tramontano, E.; Di Santo, R.; Costi, R. - 04f Poster
conference: EFMC-YMCS 2024 11th EFMC Young Medicinal Chemists' Symposium (Rome; Italy)
book: EFMC-YMCS 2024 11th EFMC Young Medicinal Chemists' Symposium - ()
11573/1725699 - 2024 -
Structure-activity relationships of indolyl derivatives as SARS-CoV-2 nsp13 inhibitors Madia, V. N.; Albano, A.; Ruggieri, G.; Ialongo, D.; Patacchini, E.; Arpacioglu, M.; Messore, A.; Scipione, L.; Corona, A.; Esposito, F.; Amatore, D.; Faggioni, G.; De Santis, R.; Lista, F.; Tramontano, E.; Di Santo, R.; Costi, R. - 04f Poster
conference: EFMC-ISMC 2024 XXVIII EFMC International Symposium on Medicinal Chemistry (Rome; Italy)
book: EFMC-ISMC 2024 XXVIII EFMC International Symposium on Medicinal Chemistry - ()
11573/1725701 - 2024 -
Pyrrole derivatives targeting the Endocannabinoid System (ECS) in Prostate Cancer Cells Messore, A.; Madia, V. N.; Ialongo, D.; Patacchini, E.; Arpacioglu, M.; Ruggieri, G.; Albano, A.; Scarpa, S.; Scipione, L.; Di Santo, R.; Costi, R. - 04f Poster
conference: EFMC-YMCS 2024 11th EFMC Young Medicinal Chemists' Symposium (Rome; Italy)
book: EFMC-YMCS 2024 11th EFMC Young Medicinal Chemists' Symposium - ()
11573/1714867 - 2024 -
New Thiazolidine-4-One Derivatives as SARS-CoV-2 Main Protease Inhibitors Messore, A; Malune, P; Patacchini, E; Madia, Vn; Ialongo, D; Arpacioglu, M; Albano, A; Ruggieri, G; Saccoliti, F; Scipione, L; Tramontano, E; Canton, S; Corona, A; Scognamiglio, S; Paulis, A; Suleiman, M; Al-Maqtari, Hm; Abid, Fma; Kawsar, Sma; Sankaranarayanan, M; Di Santo, R; Esposito, F; Costi, R. - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel: MDPI, Molecular Diversity Preservation International, 2004-) pp. 650-673 - issn: 1424-8247 - wos: WOS:001231217500001 (1) - scopus: 2-s2.0-85194037072 (3)
11573/1725693 - 2024 -
From iloperidone to new sigma-1 receptor agonists using a structure-based approach. Patacchini, E.; Albano, A; Ruggieri, G.; Arpacioglu, M.; Ialongo, D.; Madia, V. N.; Messore, A.; Saccoliti, F.; Ilari, A.; Cosconati, S.; Carli, M.; Ciruela, F.; Di Santo, R.; Costi, R. - 04f Poster
conference: EFMC-YMCS 2024 11th EFMC Young Medicinal Chemists' Symposium (Rome, Italy)
book: EFMC-YMCS 2024 11th EFMC Young Medicinal Chemists' Symposium - ()
11573/1725689 - 2024 -
Structure-based drug design of new sigma-1 receptor agonists. Patacchini, E.; Albano, A; Ruggieri, G.; Arpacioglu, M.; Ialongo, D.; Madia, Vn.; Messore, A.; Saccoliti, F.; Ilari, A.; Cosconati, S.; Carli, M.; Ciruela, F.; Di Santo, R.; Costi, R. - 04f Poster
conference: EFMC-ISMC 2024 XXVIII EFMC International Symposium on Medicinal Chemistry (Rome, Italy)
book: EFMC-ISMC 2024 XXVIII EFMC International Symposium on Medicinal Chemistry - ()
11573/1724718 - 2024 -
Quinolinonyl Derivatives as Dual Inhibitors of the HIV-1 Integrase Catalytic Site and Integrase-RNA interactions Patacchini, E.; Madia, V. N.; Albano, A.; Ruggieri, G.; Messore, A.; Ialongo, D.; Saccoliti, F.; Scipione, L.; Cosconati, S.; Koneru, P. C.; Haney, R.; Kvaratskhelia, M.; Di Santo, R.; Costi, R. - 01a Articolo in rivista
paper: ACS MEDICINAL CHEMISTRY LETTERS (USA: ACS Publications) pp. 1533-1540 - issn: 1948-5875 - wos: WOS:001286243200001 (0) - scopus: 2-s2.0-85200556440 (0)
11573/1725687 - 2024 -
From iloperidone to new sigma-1 receptors agonists: a structure-based approach. Patacchini, E.; Madia, Vn.; Albano, A.; Ruggieri, G.; Arpacioglu, M.; Ialongo, D.; Messore, A.; Genovese, I.; Antonelli, L.; Ilari, A.; Ciruela, F.; Carli, M.; Cosconati, S.; Di Santo, R.; Costi, R. - 04f Poster
conference: SCI 2024 Chemistry ELEMENTS OF FUTURE - XXVIII Congresso Nazionale della Società Chimica Italiana (Milan, Italy)
book: SCI 2024 Chemistry ELEMENTS OF FUTURE - XXVIII Congresso Nazionale della Società Chimica Italiana - ()
11573/1725685 - 2024 -
From Iloperidone to new Sigma1 agonists: a structre-based approach for Huntington’s disease treatment. Patacchini, Elisa; Ialongo, Davide; Madia, Valentina Noemi; Messore, Antonella; Ilari, Andrea; Cosconati, Sandro; Di Santo, Roberto; Costi, Roberta - 04f Poster
conference: XIII Meeting Paul Ehrlich Euro-PhD Network & COST ACTION (Rome, Italy)
book: XIII Meeting Paul Ehrlich Euro-PhD Network & COST ACTION - ()
11573/1725675 - 2024 -
Different approaches to target SARS-CoV-2: discovery of new small molecules as antiviral agents. Ruggieri, G.; Madia, V. N.; Patacchini, E.; Albano, A.; Arpacioglu, M.; Ialongo, D.; Messore, A.; Saccoliti, F.; De Leo, A.; Malune, P.; Esposito, F.; Michelini, Z.; Cara, A.; Scipione, L.; Tramontano, E.; Di Santo, R.; Costi, R. - 04f Poster
conference: 1NF-ACT Meeting 2024 (Pavia, Italy)
book: 1NF-ACT Meeting 2024 - ()
11573/1725671 - 2024 -
Design and synthesis of novel compounds targeting both AURKA and HDAC enzymes. Ruggieri, G.; Madia, V. N.; Patacchini, E.; Ialongo, D.; Albano, A.; Messore, A.; Saccoliti, F; Arpacioglu, M.; De Leo, A.; Scipione, L.; Rotili, D.; Fiorentino, F.; Paiardini, A.; Di Santo, R.; Costi, R. - 04f Poster
conference: EFMC-ISMC 2024 XXVIII EFMC International Symposium on Medicinal Chemistry (Rome, Italy)
book: EFMC-ISMC 2024 XXVIII EFMC International Symposium on Medicinal Chemistry - ()
11573/1725673 - 2024 -
Nitrogen-based derivatives as RNA-dependent RNA polymerase inhibitors of SARS-CoV-2. Ruggieri, G.; Madia, V. N.; Patacchini, E.; Ialongo, D.; Messore, A.; Albano, A.; Arpacioglu, M.; Malune, ; P., Esposito; Scipione, L.; Tramontano, E.; Di Santo, R.; Costi, R. - 04f Poster
conference: EFMC-YMCS 2024 11th EFMC Young Medicinal Chemists' Symposium (Rome, Italy)
book: EFMC-YMCS 2024 11th EFMC Young Medicinal Chemists' Symposium - ()
11573/1725653 - 2024 -
Identification of novel pyrimidine-based compounds as SARS-CoV-2 RNA-dependent RNA polymerase inhibitors. Ruggieri, G.; Madia, V. N.; Patacchini, E.; Ialongo, D.; Messore, A.; Albano, A.; Arpacioglu, M.; Malune, P.; Esposito, F.; Scipione, L.; Tramontano, E.; Di Santo, R.; Costi, R. - 04f Poster
conference: EFMC-ACSMEDI Medicinal Chemistry Frontiers (Utrecht; Netherlands)
book: EFMC-ACSMEDI Medicinal Chemistry Frontiers - ()
11573/1725664 - 2024 -
Unvealing newly discovered small molecules as ACE2-spike inhibitors against SARS-CoV-2. Ruggieri, G.; Madia, Vn.; Patacchini, E.; Ialongo, D.; Messore, A.; Albano, A.; Arpacioglu, M.; De Leo, A.; Saccoliti, F.; Michelini, Z.; Cara, A.; Scipione, L.; Di Santo, R.; Costi, R. - 04f Poster
conference: SCI 2024 Chemistry ELEMENTS OF FUTURE - XXVIII Congresso Nazionale della Società Chimica Italiana (Milan, Italy)
book: SCI 2024 Chemistry ELEMENTS OF FUTURE - XXVIII Congresso Nazionale della Società Chimica Italiana - ()
11573/1697149 - 2023 -
New blood-brain-barrier permeable compounds as Naegleria Fowleri CYP51 inhibitors. Arpacioglu, M.; Madia, V. N.; Ialongo, D.; Patacchini, E.; Messore, A.; Tudino, V.; Sharma, V.; Nguyen, J.; Debnath, A.; Podust, L.; Palenca, I.; Basili Franzin, S.; Seguella, L.; Esposito, G.; Petrucci, R.; Di Matteo, P.; Bortolami, M.; Scipione, L.; Costi, R.; Di Santo, R. - 04f Poster
conference: XXVIII edition of the National Meeting on Medicinal Chemistry (Chieti; Italy)
book: XXVIII edition of the National Meeting on Medicinal Chemistry - ()
11573/1697156 - 2023 -
Novel nsp13 inhibitors capable of blocking viral replication of SARS-CoV-2. Arpacioglu, M.; Madia, V. N.; Messore, A.; Patacchini, E.; Ialongo, D.; Tudino, V.; Scipione, L.; Corona, A.; Esposito, F.; Artico, M.; Amatore, D.; Faggioni, G.; De Santis, R.; Lista, F.; Tramontano, E.; Costi, R.; Di Santo, R. - 04f Poster
conference: ESMEC 2023 - European School of Medicinal Chemistry – 42nd Edition (Urbino; Italy)
book: ESMEC 2023 - European School of Medicinal Chemistry – 42nd Edition - ()
11573/1686714 - 2023 -
Diketo acid inhibitors of nsp13 of SARS-CoV-2 block viral replication Corona, Angela; Madia, Valentina Noemi; De Santis, Riccardo; Manelfi, Candida; Emmolo, Roberta; Ialongo, Davide; Patacchini, Elisa; Messore, Antonella; Amatore, Donatella; Faggioni, Giovanni; Artico, Marco; Iaconis, Daniela; Talarico, Carmine; Di Santo, Roberto; Lista, Florigio; Costi, Roberta; Tramontano, Enzo - 01a Articolo in rivista
paper: ANTIVIRAL RESEARCH (Amsterdam: Elsevier Science) pp. - - issn: 1872-9096 - wos: WOS:001062175600001 (6) - scopus: 2-s2.0-85167598331 (5)
11573/1686713 - 2023 -
Effects of modified glucosamine on the chondrogenic potential of circulating stem cells under experimental inflammation Gasparella, Marco; Cenzi, Carola; Piccione, Monica; Madia, Valentina Noemi; Di Santo, Roberto; Tudino, Valeria; Artico, Marco; Taurone, Samanta; De Ponte, Chiara; Costi, Roberta; Di Liddo, Rosa - 01a Articolo in rivista
paper: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (Basel: MDPI Center) pp. - - issn: 1422-0067 - wos: WOS:001020920600001 (0) - scopus: 2-s2.0-85163945199 (0)
11573/1697165 - 2023 -
Aminopyrimidine derivatives as new protein kinase inhibitors endowed with anticancer activity. Ialongo, D.; Madia, V. N.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Scarpa, S.; Rauh, D; Di Santo, R.; Costi, R. - 04f Poster
conference: 10th EFMC Young Medicinal Chemists' Symposium (Zagreb; Croatia.)
book: 10th EFMC Young Medicinal Chemists' Symposium - ()
11573/1697174 - 2023 -
Pyrimidine-based compounds as new promising protein kinase inhibitors for cancer treatment. Ialongo, D.; Madia, V. N.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Scarpa, S.; Rauh, D; Di Santo, R.; Costi, R. - 04f Poster
conference: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry (Zagreb; Croatia.)
book: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry - ()
11573/1697175 - 2023 -
Diketo acid heterocyclic derivatives as new SARS-CoV-2 nsp13 inhibitors blocking viral replication. Ialongo, D.; Madia, V. N.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Tudino, V.; Scipione, L.; Corona, A.; Esposito, F.; Artico, M.; Amatore, D.; Faggioni, G.; De Santis, R.; Lista, F.; Tramontano, E.; Costi, R.; Di Santo, R. - 04f Poster
conference: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry (Zagreb; Croatia.)
book: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry - ()
11573/1697147 - 2023 -
Identification of novel aminopyrimidine derivatives as protein kinase inhibitors blocking cell growth. Ialongo, Davide; Madia, Valentina Noemi; Messore, Antonella; Patacchini, Elisa; Arpacioglu, Merve; Scipione, Luigi; Scarpa, S.; Rauh, D.; Di Santo, R.; Costi, R. - 04f Poster
conference: XXVIII edition of the National Meeting on Medicinal Chemistry (Chieti; Italy)
book: XXVIII edition of the National Meeting on Medicinal Chemistry - ()
11573/1697162 - 2023 -
New diketo acid derivatives as dual SARS-CoV-2 nsp13 inhibitors active against viral replication. Ialongo, Davide; Madia, Valentina Noemi; Messore, Antonella; Patacchini, Elisa; Arpacioglu, Merve; Tudino, Valeria; Scipione, Luigi; Corona, Angela; Esposito, Francesca; Artico, Marco; Amatore, Donatella; Faggioni, Giovanni; De Santis, Riccardo; Lista, Florigio; Tramontano, Enzo; Costi, Roberta; Di Santo, Roberto - 04f Poster
conference: 10th EFMC Young Medicinal Chemists' Symposium (Zagreb; Croatia.)
book: 10th EFMC Young Medicinal Chemists' Symposium - ()
11573/1668131 - 2023 -
Pyrrolyl and indolyl α-γ-diketo acid derivatives acting as selective inhibitors of human carbonic anhydrases IX and XII Ialongo, Davide; Messore, Antonella; Madia, Valentina Noemi; Tudino, Valeria; Nocentini, Alessio; Gratteri, Paola; Giovannuzzi, Simone; Supuran, Claudiu T.; Nicolai, Alice; Scarpa, Susanna; Taurone, Samanta; Camarda, Michele; Artico, Marco; Papa, Veronica; Saccoliti, Francesco; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel: MDPI, Molecular Diversity Preservation International, 2004-) pp. - - issn: 1424-8247 - wos: WOS:000941695000001 (2) - scopus: 2-s2.0-85148943598 (2)
11573/1684012 - 2023 -
Synergistic Effects of Caffeine in Combination with Conventional Drugs: Perspectives of a Drug That Never Ages Ialongo, Davide; Tudino, Valeria; Arpacioglu, Merve; Messore, Antonella; Patacchini, Elisa; Costi, Roberta; Di Santo, Roberto; Madia, Valentina Noemi - 01g Articolo di rassegna (Review)
paper: PHARMACEUTICALS (Basel: MDPI, Molecular Diversity Preservation International, 2004-) pp. 1-23 - issn: 1424-8247 - wos: WOS:000997931100001 (13) - scopus: 2-s2.0-85160675541 (13)
11573/1678807 - 2023 -
Plants and Small Molecules: An Up-and-Coming Synergy Lepri, A.; Longo, C.; Messore, A.; Kazmi, H.; Madia, V. N.; Di Santo, R.; Costi, R.; Vittorioso, P. - 01g Articolo di rassegna (Review)
paper: PLANTS (Basel: MDPI) pp. - - issn: 2223-7747 - wos: WOS:000977210900001 (3) - scopus: 2-s2.0-85156214656 (5)
11573/1697142 - 2023 -
Discovery of new small molecules as anti-SARS-CoV-2 agents inhibiting ACE2-spike binding. Madia, V. N.; Ialongo, D.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Di Santo, R.; Costi, R. - 04f Poster
conference: XXVIII edition of the National Meeting on Medicinal Chemistry (Chieti; Italy)
book: XXVIII edition of the National Meeting on Medicinal Chemistry - ()
11573/1697168 - 2023 -
Dual HIV-1 integrase catalytic site and integrase-RNA interaction inhibitors. Madia, V. N.; Ialongo, D.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Kvaratskhelia, M.; Di Santo, R.; Costi, R. - 04f Poster
conference: 10th EFMC Young Medicinal Chemists' Symposium (Zagreb; Croatia.)
book: 10th EFMC Young Medicinal Chemists' Symposium - ()
11573/1697179 - 2023 -
Quinolinonyl derivatives as dual inhibitors of the HIV-1 integrase catalytic site and integrase-RNA interactions. Madia, V. N.; Ialongo, D.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Kvaratskhelia, M.; Di Santo, R.; Costi, R. - 04f Poster
conference: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry (Zagreb; Croatia.)
book: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry - ()
11573/1697181 - 2023 -
Design and synthesis of brain permeable anti-Naegleria fowleri agents targeting CYP51 for primary amoebic meningoencephalitis treatment. Madia, V. N.; Ialongo, D.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Tudino, V.; Sharma, V.; Nguyen, J.; Debnath, A.; Podust, L.; Palenca, I.; Basili Franzin, S.; Seguella, L.; Esposito, G.; Petrucci, R.; Di Matteo, P.; Bortolami, M.; Scipione, L.; Costi, R.; Di Santo, R. - 04f Poster
conference: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry (Zagreb; Croatia.)
book: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry - ()
11573/1697153 - 2023 -
Small molecule derivatives as dual inhibitors of SARS-CoV-2 nsp13 blocking viral replication. Madia, V. N.; Ialongo, D.; Patacchini, E.; Arpacioglu, M.; Messore, A.; Tramontano, E.; De Santis, R.; Lista, F.; Costi, R.; Di Santo, R. - 04f Poster
conference: 3rd Synthesis in Drug Discovery and Development (Virtual meeting)
book: 3rd Synthesis in Drug Discovery and Development - ()
11573/1697146 - 2023 -
Discovery of quinolinonyl derivatives as anti-HIV-1 inhibitors endowed with an innovative mechanism of action. Madia, Valentina Noemi; Ialongo, Davide; Messore, Antonella; Patacchini, Elisa; Arpacioglu, Merve; Scipione, Luigi; Di Santo, Roberto; And Costi, Roberta. - 04f Poster
conference: XXVIII edition of the National Meeting on Medicinal Chemistry (Chieti; Italy)
book: XXVIII edition of the National Meeting on Medicinal Chemistry - ()
11573/1663401 - 2023 -
Inhibition of Leishmania infantum Trypanothione Reductase by New Aminopropanone Derivatives Interacting with the NADPH Binding Site Madia, Valentina Noemi; Ialongo, Davide; Patacchini, Elisa; Exertier, Cécile; Antonelli, Lorenzo; Colotti, Gianni; Messore, Antonella; Tudino, Valeria; Saccoliti, Francesco; Scipione, Luigi; Ilari, Andrea; Costi, Roberta; Di Santo, Roberto Di - 01a Articolo in rivista
paper: MOLECULES (Basel: MDPI
Berlin: Springer, 1996-) pp. 338- - issn: 1420-3049 - wos: WOS:000909976300001 (1) - scopus: 2-s2.0-85145692255 (3)
11573/1697172 - 2023 -
Miconazole-like compounds as brain permeable anti-Naegleria Fowleri agents targeting CYP51. Madia, Valentina Noemi; Ialongo, Davide; Patacchini, Elisa; Messore, Antonella; Arpacioglu, Merve; Tudino, V.; Sharma, V.; Nguyen, J.; Debnath, A.; Podust, L.; Palenca, I.; Basili Franzin, S.; Seguella, L.; Esposito, G.; Petrucci, R.; Di Matteo, P.; Bortolami, M.; Scipione, L.; Costi, Roberta; Di Santo, Roberto. - 04f Poster
conference: 10th EFMC Young Medicinal Chemists' Symposium (Zagreb; Croatia.)
book: 10th EFMC Young Medicinal Chemists' Symposium - ()
11573/1687531 - 2023 -
Role of a Novel Heparanase Inhibitor on the Balance between Apoptosis and Autophagy in U87 Human Glioblastoma Cells Manganelli, V.; Misasi, R.; Riitano, G.; Capozzi, A.; Mattei, V.; Caglar, T. R.; Ialongo, D.; Madia, V. N.; Messore, A.; Costi, R.; Di Santo, R.; Sorice, M.; Garofalo, T. - 01a Articolo in rivista
paper: CELLS (Basel: mdpi-Molecular Diversity Preservation International) pp. 1-14 - issn: 2073-4409 - wos: WOS:001038054000001 (4) - scopus: 2-s2.0-85165884087 (4)
11573/1697140 - 2023 -
Design and synthesis of tetrahydro-β-carbolines derivatives as PDIA inhibitors. Messore, A.; Madia, V. N.; Ialongo, D.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Altieri, F.; Paglia, G.; Meschiari, G.; Di Santo, R.; Costi, R. - 04f Poster
conference: XXVIII edition of the National Meeting on Medicinal Chemistry (Chieti; Italy)
book: XXVIII edition of the National Meeting on Medicinal Chemistry - ()
11573/1697150 - 2023 -
From Iloperidone to new Sigma1 agonists: a structure-based approach for Huntington's disease treatment. Patacchini, Elisa; Madia, Valentina Noemi; Ialongo, Davide; Messore, Antonella; Ilari, Andrea; Cosconati, Sandro; Di Santo, Roberto; Costi, Roberta. - 04f Poster
conference: ESMEC 2023 - European School of Medicinal Chemistry – 42nd Edition (Urbino; Italy)
book: ESMEC 2023 - European School of Medicinal Chemistry – 42nd Edition - ()
11573/1696092 - 2023 -
Miconazole-like scaffold is a promising lead for Naegleria fowleri-specific CYP51 inhibitors Sharma, Vandna; Madia, Valentina Noemi; Tudino, Valeria; V Nguyen, Jennifer; Debnath, Anjan; Messore, Antonella; Ialongo, Davide; Patacchini, Elisa; Palenca, Irene; Basili Franzin, Silvia; Seguella, Luisa; Esposito, Giuseppe; Petrucci, Rita; Di Matteo, Paola; Bortolami, Martina; Saccoliti, Francesco; Di Santo, Roberto; Scipione, Luigi; Costi, Roberta; M Podust, Larissa - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 17059-17073 - issn: 0022-2623 - wos: WOS:001134079100001 (5) - scopus: 2-s2.0-85180091142 (4)
11573/1638218 - 2022 -
Design, synthesis, and In vitro, in silico and in cellulo evaluation of new Pyrimidine and Pyridine amide and Carbamate derivatives as multi-functional Cholinesterase Inhibitors Bortolami, Martina; Pandolfi, Fabiana; Tudino, Valeria; Messore, Antonella; Madia, Valentina Noemi; De Vita, Daniela; Di Santo, Roberto; Costi, Roberta; Romeo, Isabella; Alcaro, Stefano; Colone, Marisa; Stringaro, Annarita; Espargaró, Alba; Sabatè, Raimon; Scipione, Luigi - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel: MDPI, Molecular Diversity Preservation International, 2004-) pp. 1-31 - issn: 1424-8247 - wos: WOS:000818156100001 (4) - scopus: 2-s2.0-85134396743 (4)
11573/1654141 - 2022 -
New Inhibitors of the human p300/CBP acetyltransferase are selectively active against the Arabidopsis HAC proteins Longo, Chiara; Lepri, Andrea; Paciolla, Andrea; Messore, Antonella; De Vita, Daniela; Bonaccorsi Di Patti, Maria Carmela; Amadei, Matteo; Madia, Valentina Noemi; Ialongo, Davide; Di Santo, Roberto; Costi, Roberta; Vittorioso, Paola - 01a Articolo in rivista
paper: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (Basel: MDPI Center) pp. 1-18 - issn: 1422-0067 - wos: WOS:000859422800001 (5) - scopus: 2-s2.0-85138734584 (5)
11573/1648549 - 2022 -
Ultrastructural damages to H1N1 influenza virus caused by vapor essential oils Madia, Valentina Noemi; Toscanelli, Walter; De Vita, Daniela; De Angelis, Marta; Messore, Antonella; Ialongo, Davide; Scipione, Luigi; Tudino, Valeria; D'auria, Felicia Diodata; Di Santo, Roberto; Garzoli, Stefania; Stringaro, Annarita; Colone, Marisa; Marchetti, Magda; Superti, Fabiana; Nencioni, Lucia; Costi, Roberta - 01a Articolo in rivista
paper: MOLECULES (Basel: MDPI
Berlin: Springer, 1996-) pp. 1-14 - issn: 1420-3049 - wos: WOS:000816243700001 (11) - scopus: 2-s2.0-85131746075 (12)
11573/1623281 - 2022 -
Oxidative stress and visual system a review Taurone, S.; Ralli, M.; Artico, M.; Madia, V. N.; Scarpa, S.; Nottola, S. A.; Maconi, A.; Betti, M.; Familiari, P.; Nebbioso, M.; Costi, R.; Micera, A. - 01g Articolo di rassegna (Review)
paper: EXCLI JOURNAL (Mainz: EXCLI Journal Business Office c/o 2nd Medical Department, University of Mainz.) pp. 544-553 - issn: 1611-2156 - wos: WOS:000766811300001 (19) - scopus: 2-s2.0-85125850235 (23)
11573/1564954 - 2021 -
Toxicological aspects of cannabinoid, pesticide and metal levels detected in light Cannabis inflorescences grown in Italy Amendola, G.; Bocca, B.; Picardo, V.; Pelosi, P.; Battistini, B.; Ruggieri, F.; Attard Barbini, D.; De Vita, D.; Madia, V. N.; Messore, A.; Di Santo, R.; Costi, R. - 01a Articolo in rivista
paper: FOOD AND CHEMICAL TOXICOLOGY (Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. - - issn: 0278-6915 - wos: WOS:000696988600002 (8) - scopus: 2-s2.0-85112006002 (11)
11573/1490818 - 2021 -
Acetylcholinesterase inhibitors for the treatment of Alzheimer’s disease–a patent review (2016–present) Bortolami, M.; Rocco, D.; Messore, A.; Di Santo, R.; Costi, R.; Madia, V. N.; Scipione, L.; Pandolfi, F. - 01a Articolo in rivista
paper: EXPERT OPINION ON THERAPEUTIC PATENTS (--London United Kingdom:Informa Healthcare
-London, United Kingdom: Ashley Publications Limited) pp. 1-22 - issn: 1354-3776 - wos: WOS:000607685400001 (43) - scopus: 2-s2.0-85099470810 (44)
11573/1584588 - 2021 -
New pyrimidine and pyridine derivatives as multitarget cholinesterase inhibitors. Design, synthesis, and in vitro and in cellulo evaluation Bortolami, Martina; Pandolfi, Fabiana; Tudino, Valeria; Messore, Antonella; Madia, Valentina Noemi; De Vita, Daniela; Di Santo, Roberto; Costi, Roberta; Romeo, Isabella; Alcaro, Stefano; Colone, Marisa; Stringaro, Annarita; Espargaró, Alba; Sabatè, Raimon; Scipione, Luigi - 01a Articolo in rivista
paper: ACS CHEMICAL NEUROSCIENCE (Washington, D.C. : American Chemical Society) pp. 4090-4112 - issn: 1948-7193 - wos: WOS:000715842900011 (23) - scopus: 2-s2.0-85118138783 (23)
11573/1404920 - 2021 -
Towards a new application of amaranth seed oil as an agent against Candida albicans De Vita, Daniela; Messore, Antonella; Toniolo, Chiara; Frezza, Claudio; Scipione, Luigi; Bertea, Cinzia Margherita; Micera, Marco; Di Sarno, Veronica; Madia, Valentina Noemi; Pindinello, Ivano; Roscilli, Patrizia; Botto, Alfonso; Simonetti, Giovanna; Orekhova, Anastasia; Manfredini, Stefano; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: NATURAL PRODUCT RESEARCH (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 4621-4626 - issn: 1478-6419 - wos: WOS:000500457200001 (17) - scopus: 2-s2.0-85075913942 (10)
11573/1540215 - 2021 -
Investigation of Commiphora myrrha (Nees) Engl. oil and its main components for antiviral activity Madia, Valentina Noemi; De Angelis, Marta; De Vita, Daniela; Messore, Antonella; De Leo, Alessandro; Ialongo, Davide; Tudino, Valeria; Saccoliti, Francesco; De Chiara, Giovanna; Garzoli, Stefania; Scipione, Luigi; Palamara, Anna Teresa; Di Santo, Roberto; Nencioni, Lucia; Costi, Roberta - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel: MDPI, Molecular Diversity Preservation International, 2004-) pp. - - issn: 1424-8247 - wos: WOS:000634055800001 (26) - scopus: 2-s2.0-85102987115 (31)
11573/1564144 - 2021 -
Recent advances in recovery of lycopene from tomato waste. A potent antioxidant with endless benefits Madia, Valentina Noemi; De Vita, Daniela; Ialongo, Davide; Tudino, Valeria; De Leo, Alessandro; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta; Messore, Antonella - 01a Articolo in rivista
paper: MOLECULES (Basel: MDPI
Berlin: Springer, 1996-) pp. 1-18 - issn: 1420-3049 - wos: WOS:000682223800001 (54) - scopus: 2-s2.0-85111602310 (66)
11573/1540619 - 2021 -
Analytical characterization of an inulin-type fructooligosaccharide from root-tubers of Asphodelus ramosus L Madia, Valentina Noemi; De Vita, Daniela; Messore, Antonella; Toniolo, Chiara; Tudino, Valeria; De Leo, Alessandro; Pindinello, Ivano; Ialongo, Davide; Saccoliti, Francesco; D'ursi, Anna Maria; Grimaldi, Manuela; Ceccobelli, Pietro; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel: MDPI, Molecular Diversity Preservation International, 2004-) pp. - - issn: 1424-8247 - wos: WOS:000634075100001 (7) - scopus: 2-s2.0-85103099178 (6)
11573/1565318 - 2021 -
Small-molecule inhibitors of HIV-1 reverse transcriptase-associated ribonuclease H function. Challenges and recent developments Madia, Valentina Noemi; Messore, Antonella; De Leo, Alessandro; Tudino, Valeria; Pindinello, Ivano; Saccoliti, Francesco; De Vita, Daniela; Scipione, Luigi; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: CURRENT MEDICINAL CHEMISTRY (Hilversum: Bentham Science Publishers) pp. 1-33 - issn: 1875-533X - wos: WOS:000696992000004 (5) - scopus: 2-s2.0-85115249511 (6)
11573/1493998 - 2021 -
Design, synthesis and biological evaluation of new pyrimidine derivatives as anticancer agents Madia, Valentina Noemi; Nicolai, Alice; Messore, Antonella; De Leo, Alessandro; Ialongo, Davide; Tudino, Valeria; Saccoliti, Francesco; De Vita, Daniela; Scipione, Luigi; Artico, Marco; Taurone, Samanta; Taglieri, Ludovica; Di Santo, Roberto; Scarpa, Susanna; Costi, Roberta - 01a Articolo in rivista
paper: MOLECULES (Basel: MDPI
Berlin: Springer, 1996-) pp. - - issn: 1420-3049 - wos: WOS:000615455300001 (23) - scopus: 2-s2.0-85101195321 (23)
11573/1556284 - 2021 -
Quinolinonyl non-diketo acid derivatives as Inhibitors of HIV-1 ribonuclease H and polymerase functions of reverse transcriptase Messore, Antonella; Corona, Angela; Madia, Valentina Noemi; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Ialongo, Davide; Scipione, Luigi; De Vita, Daniela; Amendola, Giorgio; Novellino, Ettore; Cosconati, Sandro; Métifiot, Mathieu; Andreola, Marie-Line; Esposito, Francesca; Grandi, Nicole; Tramontano, Enzo; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 8579-8598 - issn: 0022-2623 - wos: WOS:000668340800039 (10) - scopus: 2-s2.0-85108607601 (9)
11573/1553152 - 2021 -
Anti-tumoral effects of a (1H-pyrrol-1-yl)methyl-1H-benzoimidazole carbamate ester derivative on head and neck squamous carcinoma cell lines Nicolai, Alice; Madia, Valentina Noemi; Messore, Antonella; De Vita, Daniela; De Leo, Alessandro; Ialongo, Davide; Tudino, Valeria; Tortorella, Elisabetta; Scipione, Luigi; Taurone, Samanta; Pergolizzi, Tiziano; Artico, Marco; Di Santo, Roberto; Costi, Roberta; Scarpa, Susanna - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel: MDPI, Molecular Diversity Preservation International, 2004-) pp. - - issn: 1424-8247 - wos: WOS:000666329400001 (8) - scopus: 2-s2.0-85110773299 (8)
11573/1408850 - 2020 -
Pyrrolyl pyrazoles as non-diketo acid inhibitors of the HIV-1 ribonuclease H function of reverse transcriptase Messore, Antonella; Corona, Angela; Madia, Valentina Noemi; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Scipione, Luigi; De Vita, Daniela; Amendola, Giorgio; Di Maro, Salvatore; Novellino, Ettore; Cosconati, Sandro; Métifiot, Mathieu; Andreola, Marie-Line; Valenti, Piera; Esposito, Francesca; Grandi, Nicole; Tramontano, Enzo; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: ACS MEDICINAL CHEMISTRY LETTERS (USA: ACS Publications) pp. 798-805 - issn: 1948-5875 - wos: WOS:000535281200029 (28) - scopus: 2-s2.0-85086659986 (28)
11573/1274892 - 2020 -
Discovery of a pyrimidine compound endowed with antitumor activity Taglieri, Ludovica; Saccoliti, Francesco; Nicolai, Alice; Peruzzi, Giovanna; Madia, Valentina Noemi; Tudino, Valeria; Messore, Antonella; Di Santo, Roberto; Artico, Marco; Taurone, Samanta; Salvati, Maurizio; Costi, Roberta; Scarpa, Susanna - 01a Articolo in rivista
paper: INVESTIGATIONAL NEW DRUGS (attuale:
-SPRINGER, VAN GODEWIJCKSTRAAT 30, DORDRECHT, NETHERLANDS, 3311 GZ
-Kluwer Academic Publishers / Massachusetts:PO Box 358, Accord Station:Hingham, MA 02018:(617)871-6600) pp. 39-49 - issn: 0167-6997 - wos: WOS:000512107200005 (16) - scopus: 2-s2.0-85063345760 (17)
11573/1336764 - 2019 -
Structure-guided approach to identify a novel class of anti-leishmaniasis diaryl sulfide compounds targeting the trypanothione metabolism Colotti, G.; Saccoliti, F.; Gramiccia, M.; Di Muccio, T.; Prakash, J.; Yadav, S.; Dubey, V. K.; Vistoli, G.; Battista, T.; Mocci, S.; Fiorillo, A.; Bibi, Aasia; Madia, V. N.; Messore, A.; Costi, R.; Di Santo, R.; Ilari, A. - 01a Articolo in rivista
paper: AMINO ACIDS (Wien: Springer Verlag) pp. - - issn: 0939-4451 - wos: WOS:000519385700013 (16) - scopus: 2-s2.0-85065106515 (17)
11573/1285185 - 2019 -
Comparison of different methods for the extraction of cannabinoids from cannabis De Vita, D.; Madia, V. N.; Tudino, V.; Saccoliti, F.; De Leo, A.; Messore, A.; Roscilli, P.; Botto, A.; Pindinello, I.; Santilli, G.; Scipione, L.; Costi, R.; Di Santo, R. - 01a Articolo in rivista
paper: NATURAL PRODUCT RESEARCH (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1-7 - issn: 1478-6419 - wos: WOS:000575920700013 (36) - scopus: 2-s2.0-85065155862 (39)
11573/1205976 - 2019 -
In vitro antiviral activity of new oxazoline derivatives as potent poliovirus inhibitors Madia, Valentina Noemi; Messore, Antonella; Pescatori, Luca; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Scipione, Luigi; Fiore, Lucia; Rhoden, Eric; Manetti, Fabrizio; Oberste, M Steven; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 798-810 - issn: 0022-2623 - wos: WOS:000457067600026 (11) - scopus: 2-s2.0-85060542889 (13)
11573/1405464 - 2019 -
Tegaserod for the treatment of Irritable Bowel syndrome Madia, Valentina Noemi; Messore, Antonella; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; De Vita, Daniela; Bortolami, Martina; Scipione, Luigi; Pindinello, Ivano; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: ANTI-INFLAMMATORY & ANTI-ALLERGY AGENTS IN MEDICINAL CHEMISTRY (Hilversum : Bentham Science Publsihers) pp. 1-28 - issn: 1871-5230 - wos: (0) - scopus: 2-s2.0-85083912835 (0)
11573/1321741 - 2019 -
Inhibition of Polycomb Repressive Complex2 activity reduces trimethylation of H3K27 and affects development in Arabidopsis seedlings Ruta, Veronica; Longo, Chiara; Boccaccini, Alessandra; Madia, Valentina Noemi; Saccoliti, Francesco; Tudino, Valeria; Di Santo, Roberto; Lorrai, Riccardo; Dello Ioio, Raffaele; Sabatini, Sabrina; Costi, Roberta; Costantino, Paolo; Vittorioso, Paola - 01a Articolo in rivista
paper: BMC PLANT BIOLOGY (London: BioMed Central.MIDDLESEX HOUSE, 34-42 CLEVELAND ST, LONDON, ENGLAND, W1T 4LB) pp. - - issn: 1471-2229 - wos: WOS:000490716900003 (15) - scopus: 2-s2.0-85073428390 (15)
11573/1222183 - 2019 -
Design, synthesis, and biological evaluation of new 1-(aryl-1H-pyrrolyl)(phenyl)methyl-1H-imidazole derivatives as antiprotozoal agents Saccoliti, Francesco; Madia, Valentina Noemi; Tudino, Valeria; De Leo, Alessandro; Pescatori, Luca; Messore, Antonella; De Vita, Daniela; Scipione, Luigi; Brun, Reto; Kaiser, Marcel; Mäser, Pascal; Calvet Alvarez, Claudia Magalhaes; Jennings, Gareth K; Podust, Larissa M; Pepe, Giacomo; Cirilli, Roberto; Faggi, Cristina; Di Marco, Annalise; Battista, Maria Rosaria; Summa, Vincenzo; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1330-1347 - issn: 0022-2623 - wos: WOS:000459223600016 (31) - scopus: 2-s2.0-85061636363 (32)
11573/1176836 - 2018 -
Novel benzazole derivatives endowed with potent antiheparanase activity Madia, Valentina Noemi; Messore, Antonella; Pescatori, Luca; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Bortolami, Martina; Scipione, Luigi; Costi, Roberta; Rivara, Silvia; Scalvini, Laura; Mor, Marco; Fosca Ferrara, Fabiana; Pavoni, Emiliano; Roscilli, Giuseppe; Cassinelli, Giuliana; M Milazzo, Ferdinando; Battistuzzi, Gianfranco; Di Santo, Roberto; Giannin, Giuseppe - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 6918-6936 - issn: 0022-2623 - wos: WOS:000441484300030 (28) - scopus: 2-s2.0-85050088127 (28)
11573/1221546 - 2018 -
Novel symmetrical benzazolyl derivatives endowed with potent anti-heparanase activity Messore, Antonella; Madia, Valentina Noemi; Pescatori, Luca; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Bortolami, Martina; De Vita, Daniela; Scipione, Luigi; Pepi, Federico; Costi, Roberta; Rivara, Silvia; Scalvini, Laura; Mor, Marco; Ferrara, Fabiana Fosca; Pavoni, Emiliano; Roscilli, Giuseppe; Cassinelli, Giuliana; Milazzo, Ferdinando M; Battistuzzi, Gianfranco; Di Santo, Roberto; Giannini, Giuseppe - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 10834-10859 - issn: 0022-2623 - wos: WOS:000453488200031 (18) - scopus: 2-s2.0-85058215116 (17)
11573/1174521 - 2018 -
Selective inhibition of the PRC2 methyltransferase activity suppresses trimethylation of H3K27 in Arabidopsis seeds Ruta, Veronica; Boccaccini, Alessandra; Longo, Chiara; Madia, Valentina Noemi; Tudino, Valeria; Costi, Roberta; Costantino, Paolo; Vittorioso, Paola - 04f Poster
conference: International Plant and Molecular Biology 2018- IPMB2018 (Montpellier)
book: nessuna - ()
11573/1176720 - 2018 -
Biological evaluation and structure-activity relationships of imidazole-based compounds as antiprotozoal agents Saccoliti, Francesco; Madia, Valentina Noemi; Tudino, Valeria; De Leo, Alessandro; Pescatori, Luca; Messore, Antonella; De Vita, Daniela; Scipione, Luigi; Brun, Reto; Kaiser, Marcel; Mäser, Pascal; Magalhaes Calvet, Claudia; K Jennings, Gareth; M Podust, Larissa; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 53-60 - issn: 0223-5234 - wos: WOS:000443663200005 (21) - scopus: 2-s2.0-85049312582 (23)
11573/1192249 - 2017 -
Structure-activity relationships on cynnamoyl derivatives as inhibitors of p300 Histone acetyltransferase Madia, Valentina Noemi; Benedetti, Rosaria; Letizia Barreca, Maria; Ngo, Liza; Pescatori, Luca; Messore, Antonella; Pupo, Giovanni; Saccoliti, Francesco; Valente, Sergio; Mai, Antonello; Scipione, Luigi; George Zheng, Yujun; Tintori, Cristina; Botta, Maurizio; Cecchetti, Violetta; Altucci, Lucia; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. 1359-1368 - issn: 1860-7187 - wos: WOS:000429592300014 (10) - scopus: 2-s2.0-85017448829 (9)
11573/929856 - 2017 -
Inhibition of Leishmania infantum trypanothione reductase by diaryl sulfide derivatives Saccoliti, Francesco; Angiulli, Gabriella; Pupo, Giovanni; Pescatori, Luca; Madia, Valentina Noemi; Messore, Antonella; Colotti, Gianni; Fiorillo, Annarita; Scipione, Luigi; Gramiccia, Marina; Di Muccio, Trentina; Di Santo, Roberto; Costi, Roberta; Ilari, Andrea - 01a Articolo in rivista
paper: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 304-310 - issn: 1475-6366 - wos: WOS:000392591100025 (50) - scopus: 2-s2.0-85013797723 (57)
11573/910116 - 2016 -
New insights into the interaction between pyrrolyl diketoacids and HIV-1 integrase active site and comparison with RNase H Corona, A; Di Leva, Fs; Rigogliuso, G; Pescatori, Luca; Madia, Valentina Noemi; Subra, F; Delelis, O; Esposito, F; Cadeddu, M; Costi, Roberta; Cosconati, S; Novellino, E; Di Santo, Roberto; Tramontano, E. - 01a Articolo in rivista
paper: ANTIVIRAL RESEARCH ([Amsterdam]; [New York]: Elsevier/North-Holland, [c1981]-) pp. 236-243 - issn: 0166-3542 - wos: WOS:000386983800026 (38) - scopus: 2-s2.0-84989205085 (36)
11573/852938 - 2015 -
Discovery of N-aryl-naphthylamines as in vitro inhibitors of the interaction between HIV integrase and the cofactor LEDGF/p75 Cuzzucoli Crucitti, G.; Pescatori, L.; Messore, A.; Madia, V. N.; Pupo, G.; Saccoliti, F; Scipione, L; Tortorella, S.; Di Leva, F. S; Cosconati, S; Novellino, E; Debyser, Z; Christ, F; Costi, R; Di Santo, R - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 288-294 - issn: 0223-5234 - wos: WOS:000360771900026 (17) - scopus: 2-s2.0-84936802596 (17)
11573/895359 - 2015 -
Structure−activity relationship of pyrrolyl diketo acid derivatives as dual Inhibitors of HIV‑1 integrase and reverse transcriptase ribonuclease H domain Cuzzucoli Crucitti, Giuliana; Métifiot, Mathieu; Pescatori, Luca; Messore, Antonella; Madia, Valentina Noemi; Pupo, Giovanni; Saccoliti, Francesco; Scipione, Luigi; Tortorella, Silvano; Esposito, Francesca; Corona, Angela; Cadeddu, Marta; Marchand, Christophe; Pommier, Yves; Tramontano, Enzo; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1915-1928 - issn: 0022-2623 - wos: WOS:000351186700021 (76) - scopus: 2-s2.0-84923882396 (80)
11573/787196 - 2015 -
N‑substituted quinolinonyl diketo acid derivatives as HIV integrase strand transfer inhibitors and their activity against RNase H function of reverse transcriptase Pescatori, Luca; Metifiot, Mathieu; Chung, Suhman; Masoaka, Takashi; Crucitti Cuzzucoli, Giuliana; Messore, Antonella; Pupo, Giovanni; Madia, Valentina Noemi; Saccoliti, Francesco; Scipione, Luigi; Tortorella, Silvano; Di Leva, Francesco Saverio; Cosconati, Sandro; Marinelli, Luciana; Novellino, Ettore; Le Grice, Stuart F. J.; Pommier, Yves; Marchand, Christophe; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 4610-4623 - issn: 0022-2623 - wos: WOS:000356316600015 (43) - scopus: 2-s2.0-84935877076 (46)
11573/559331 - 2014 -
Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV
Integrase and their Activity against RNase H Function of Reverse
Transcriptase Costi, Roberta; Mathieu, Metifiot; Suhman, Chung; Cuzzucoli Crucitti, Giuliana; Kasthuraiah, Maddali; Pescatori, Luca; Messore, Antonella; Madia, Valentina Noemi; Giovanni, Pupo; Scipione, Luigi; Tortorella, Silvano; Francesco Saverio Di, Leva; Sandro, Cosconati; Luciana, Marinelli; Ettore, Novellino; Stuart F: J., Le Grice; Angela, Corona; Yves, Pommier; Christophe, Marchand; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington DC : ACS Publications) pp. 3223-3234 - issn: 1520-4804 - wos: WOS:000335113900005 (54) - scopus: 2-s2.0-84899554749 (59)