ROBERTA COSTI

Associate professor


email: roberta.costi@uniroma1.it
phone: 0649693247
building: CU019
room: 150

Current Position:
Associate Professor in Medicinal Chemistry, University of Rome “La Sapienza”,CTF
Carreer:
2005 – 2024 Associate Professor in Medicinal Chemistry, University of Rome “La Sapienza”, Department Chemistry and Technology of Drug
2000 – 2005 Researcher, University of Rome “La Sapienza”, Department Chemistry and
1999-2000 Research Fellowship, University of Salerno
1995-1998 Post-doc fellow (Istituto Superiore Sanità), AIDS Programme
1994 Post-doc fellow Pasteur Institute / Fondazione Cenci Bolognetti
Education/Training
1994 PhD, University of Rome “La Sapienza ”in Pharmaceutical Science
1994 University of Rome “La Sapienza”; degree with full honours (110 cum lode) inPharmacy
1991University of Rome “La Sapienza”; degree with full honours (110 cum lode) in CTF

A. Personal Statement
I have expertise in the design and synthesis of compounds active against a number of microbial targets. My main research interests lie in the development of enzyme inhibitors (HIV integrase, HIV ribonuclease H, human histone deacetylases and heparanase) with a strong emphasis on target proteins involved in human pathology. My experience in this field led to the discovery of compounds with potent activity against integrase, in particular on the strand transfer step of integration process. After the discovery of aryl diketo acid (ADK) derivatives as selective ST inhibitors endowed of anti-HIV activity, my research team designed and synthesized new ADK compounds characterized by a pyrrole and or quinoline ring that were very useful tools to understand mechanism of action of HIV IN enzyme. I have expertise also in other fields of the medicinal chemistry: anticancer agents , compounds active against HCV polymerase, anti-TBC. I had a number of collaborations with the Biotech companies, to develop antimalarial agents, ligands of the 5-HT receptors, and compounds active against the aggregation of -amyloid fibrils.
Patent:
1) R. Di Santo, Y. Pommier, C. Marchand, M. Artico, R. Costi.
Preparation of quinolin-4-ones as inhibitors of retroviral integrase for the treatment of HIV, AIDS and aids related complex (ARC).
PCT Int. Appl. (2005), 75 pp. WO 2005087759 A1 20050922 CAN 143:326228 AN 2005:1026945.

2) M. A. Alisi, N. Cazzolla, R. Costi, R. Di Santo, G. Furlotti, A. Guglielmotti, L. Polenzani.
Pyrroloquinolines with serotoninergic activity, process for preparing it and pharmaceutical composition comprising it.
PCT/EP2009/059216, WO 2010012611, CAN 152:238937

3) G. Giannini, G. Battistuzzi, R. Di Santo, R. Costi, A. Messore “Symmetrical 2-aminophenyl-benzazolyl-5-acetate compounds and their use as anti-heparanase” EP17163014.8, 27.03.2017

4) G. Giannini, G. Battistuzzi, R. Di Santo, R. Costi, V. N. Madia 2-(4-(4-(Bromomethoxybenzamido)benzylamino)phenyl)benzazole derivatives and their use as anti-heparanase EP17163015.5, 27.03.2017





Main Funding informations:

1. PNRR PE-13 INF-ACT- Spoke 5 Missione 4 Componente 2
2. 2020 Istitut Pasteur International Network Coronavirus Task Force
3. 2012 V National Program of Research on AIDS- Progetti Innovativi
4. 2010 Europian Commision FP7 Programme FP7-HEALTH-2009

ORGANIZER OF MEETINGS:
1) Member of Organizing Committee of XXII National Meeting on Medicinal Chemistry (NMMC 2013), Roma, 2013.
2) Member of the International Scientific Committee (ISC) (2021) of the XXVII International Symposium on Medicinal Chemistry of the European Federation for Medicinal Chemistry and Chemical Biology (ISMC-EFMC) Nice 2022.





Research products

11573/1697149 - 2023 - New blood-brain-barrier permeable compounds as Naegleria Fowleri CYP51 inhibitors.
Arpacioglu, M.; Madia, V. N.; Ialongo, D.; Patacchini, E.; Messore, A.; Tudino, V.; Sharma, V.; Nguyen, J.; Debnath, A.; Podust, L.; Palenca, I.; Basili Franzin, S.; Seguella, L.; Esposito, G.; Petrucci, R.; Di Matteo, P.; Bortolami, M.; Scipione, L.; Costi, R.; Di Santo, R. - 04f Poster
conference: XXVIII edition of the National Meeting on Medicinal Chemistry (Chieti; Italy)
book: XXVIII edition of the National Meeting on Medicinal Chemistry - ()

11573/1697156 - 2023 - Novel nsp13 inhibitors capable of blocking viral replication of SARS-CoV-2.
Arpacioglu, M.; Madia, V. N.; Messore, A.; Patacchini, E.; Ialongo, D.; Tudino, V.; Scipione, L.; Corona, A.; Esposito, F.; Artico, M.; Amatore, D.; Faggioni, G.; De Santis, R.; Lista, F.; Tramontano, E.; Costi, R.; Di Santo, R. - 04f Poster
conference: ESMEC 2023 - European School of Medicinal Chemistry – 42nd Edition (Urbino; Italy)
book: ESMEC 2023 - European School of Medicinal Chemistry – 42nd Edition - ()

11573/1686714 - 2023 - Diketo acid inhibitors of nsp13 of SARS-CoV-2 block viral replication
Corona, Angela; Madia, Valentina Noemi; De Santis, Riccardo; Manelfi, Candida; Emmolo, Roberta; Ialongo, Davide; Patacchini, Elisa; Messore, Antonella; Amatore, Donatella; Faggioni, Giovanni; Artico, Marco; Iaconis, Daniela; Talarico, Carmine; Di Santo, Roberto; Lista, Florigio; Costi, Roberta; Tramontano, Enzo - 01a Articolo in rivista
paper: ANTIVIRAL RESEARCH (Amsterdam: Elsevier Science) pp. - - issn: 1872-9096 - wos: WOS:001062175600001 (0) - scopus: 2-s2.0-85167598331 (0)

11573/1686713 - 2023 - Effects of modified glucosamine on the chondrogenic potential of circulating stem cells under experimental inflammation
Gasparella, Marco; Cenzi, Carola; Piccione, Monica; Madia, Valentina Noemi; Di Santo, Roberto; Tudino, Valeria; Artico, Marco; Taurone, Samanta; De Ponte, Chiara; Costi, Roberta; Di Liddo, Rosa - 01a Articolo in rivista
paper: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (Basel: MDPI Center) pp. - - issn: 1422-0067 - wos: WOS:001020920600001 (0) - scopus: 2-s2.0-85163945199 (0)

11573/1697165 - 2023 - Aminopyrimidine derivatives as new protein kinase inhibitors endowed with anticancer activity.
Ialongo, D.; Madia, V. N.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Scarpa, S.; Rauh, D; Di Santo, R.; Costi, R. - 04f Poster
conference: 10th EFMC Young Medicinal Chemists' Symposium (Zagreb; Croatia.)
book: 10th EFMC Young Medicinal Chemists' Symposium - ()

11573/1697174 - 2023 - Pyrimidine-based compounds as new promising protein kinase inhibitors for cancer treatment.
Ialongo, D.; Madia, V. N.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Scarpa, S.; Rauh, D; Di Santo, R.; Costi, R. - 04f Poster
conference: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry (Zagreb; Croatia.)
book: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry - ()

11573/1697175 - 2023 - Diketo acid heterocyclic derivatives as new SARS-CoV-2 nsp13 inhibitors blocking viral replication.
Ialongo, D.; Madia, V. N.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Tudino, V.; Scipione, L.; Corona, A.; Esposito, F.; Artico, M.; Amatore, D.; Faggioni, G.; De Santis, R.; Lista, F.; Tramontano, E.; Costi, R.; Di Santo, R. - 04f Poster
conference: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry (Zagreb; Croatia.)
book: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry - ()

11573/1697147 - 2023 - Identification of novel aminopyrimidine derivatives as protein kinase inhibitors blocking cell growth.
Ialongo, Davide; Madia, Valentina Noemi; Messore, Antonella; Patacchini, Elisa; Arpacioglu, Merve; Scipione, Luigi; Scarpa, S.; Rauh, D.; Di Santo, R.; Costi, R. - 04f Poster
conference: XXVIII edition of the National Meeting on Medicinal Chemistry (Chieti; Italy)
book: XXVIII edition of the National Meeting on Medicinal Chemistry - ()

11573/1697162 - 2023 - New diketo acid derivatives as dual SARS-CoV-2 nsp13 inhibitors active against viral replication.
Ialongo, Davide; Madia, Valentina Noemi; Messore, Antonella; Patacchini, Elisa; Arpacioglu, Merve; Tudino, Valeria; Scipione, Luigi; Corona, Angela; Esposito, Francesca; Artico, Marco; Amatore, Donatella; Faggioni, Giovanni; De Santis, Riccardo; Lista, Florigio; Tramontano, Enzo; Costi, Roberta; Di Santo, Roberto - 04f Poster
conference: 10th EFMC Young Medicinal Chemists' Symposium (Zagreb; Croatia.)
book: 10th EFMC Young Medicinal Chemists' Symposium - ()

11573/1668131 - 2023 - Pyrrolyl and indolyl α-γ-diketo acid derivatives acting as selective inhibitors of human carbonic anhydrases IX and XII
Ialongo, Davide; Messore, Antonella; Madia, Valentina Noemi; Tudino, Valeria; Nocentini, Alessio; Gratteri, Paola; Giovannuzzi, Simone; Supuran, Claudiu T.; Nicolai, Alice; Scarpa, Susanna; Taurone, Samanta; Camarda, Michele; Artico, Marco; Papa, Veronica; Saccoliti, Francesco; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. - - issn: 1424-8247 - wos: WOS:000941695000001 (0) - scopus: 2-s2.0-85148943598 (0)

11573/1684012 - 2023 - Synergistic Effects of Caffeine in Combination with Conventional Drugs: Perspectives of a Drug That Never Ages
Ialongo, Davide; Tudino, Valeria; Arpacioglu, Merve; Messore, Antonella; Patacchini, Elisa; Costi, Roberta; Di Santo, Roberto; Madia, Valentina Noemi - 01g Articolo di rassegna (Review)
paper: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. 730- - issn: 1424-8247 - wos: WOS:000997931100001 (2) - scopus: 2-s2.0-85160675541 (2)

11573/1678807 - 2023 - Plants and Small Molecules: An Up-and-Coming Synergy
Lepri, A.; Longo, C.; Messore, A.; Kazmi, H.; Madia, V. N.; Di Santo, R.; Costi, R.; Vittorioso, P. - 01g Articolo di rassegna (Review)
paper: PLANTS (Basel: MDPI) pp. - - issn: 2223-7747 - wos: WOS:000977210900001 (2) - scopus: 2-s2.0-85156214656 (1)

11573/1697142 - 2023 - Discovery of new small molecules as anti-SARS-CoV-2 agents inhibiting ACE2-spike binding.
Madia, V. N.; Ialongo, D.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Di Santo, R.; Costi, R. - 04f Poster
conference: XXVIII edition of the National Meeting on Medicinal Chemistry (Chieti; Italy)
book: XXVIII edition of the National Meeting on Medicinal Chemistry - ()

11573/1697168 - 2023 - Dual HIV-1 integrase catalytic site and integrase-RNA interaction inhibitors.
Madia, V. N.; Ialongo, D.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Kvaratskhelia, M.; Di Santo, R.; Costi, R. - 04f Poster
conference: 10th EFMC Young Medicinal Chemists' Symposium (Zagreb; Croatia.)
book: 10th EFMC Young Medicinal Chemists' Symposium - ()

11573/1697179 - 2023 - Quinolinonyl derivatives as dual inhibitors of the HIV-1 integrase catalytic site and integrase-RNA interactions.
Madia, V. N.; Ialongo, D.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Kvaratskhelia, M.; Di Santo, R.; Costi, R. - 04f Poster
conference: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry (Zagreb; Croatia.)
book: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry - ()

11573/1697181 - 2023 - Design and synthesis of brain permeable anti-Naegleria fowleri agents targeting CYP51 for primary amoebic meningoencephalitis treatment.
Madia, V. N.; Ialongo, D.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Tudino, V.; Sharma, V.; Nguyen, J.; Debnath, A.; Podust, L.; Palenca, I.; Basili Franzin, S.; Seguella, L.; Esposito, G.; Petrucci, R.; Di Matteo, P.; Bortolami, M.; Scipione, L.; Costi, R.; Di Santo, R. - 04f Poster
conference: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry (Zagreb; Croatia.)
book: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry - ()

11573/1697153 - 2023 - Small molecule derivatives as dual inhibitors of SARS-CoV-2 nsp13 blocking viral replication.
Madia, V. N.; Ialongo, D.; Patacchini, E.; Arpacioglu, M.; Messore, A.; Tramontano, E.; De Santis, R.; Lista, F.; Costi, R.; Di Santo, R. - 04f Poster
conference: 3rd Synthesis in Drug Discovery and Development (Virtual meeting)
book: 3rd Synthesis in Drug Discovery and Development - ()

11573/1697146 - 2023 - Discovery of quinolinonyl derivatives as anti-HIV-1 inhibitors endowed with an innovative mechanism of action.
Madia, Valentina Noemi; Ialongo, Davide; Messore, Antonella; Patacchini, Elisa; Arpacioglu, Merve; Scipione, Luigi; Di Santo, Roberto; And Costi, Roberta. - 04f Poster
conference: XXVIII edition of the National Meeting on Medicinal Chemistry (Chieti; Italy)
book: XXVIII edition of the National Meeting on Medicinal Chemistry - ()

11573/1663401 - 2023 - Inhibition of Leishmania infantum Trypanothione Reductase by New Aminopropanone Derivatives Interacting with the NADPH Binding Site
Madia, Valentina Noemi; Ialongo, Davide; Patacchini, Elisa; Exertier, Cécile; Antonelli, Lorenzo; Colotti, Gianni; Messore, Antonella; Tudino, Valeria; Saccoliti, Francesco; Scipione, Luigi; Ilari, Andrea; Costi, Roberta; Di Santo, Roberto Di - 01a Articolo in rivista
paper: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. 338- - issn: 1420-3049 - wos: WOS:000909976300001 (0) - scopus: 2-s2.0-85145692255 (0)

11573/1697172 - 2023 - Miconazole-like compounds as brain permeable anti-Naegleria Fowleri agents targeting CYP51.
Madia, Valentina Noemi; Ialongo, Davide; Patacchini, Elisa; Messore, Antonella; Arpacioglu, Merve; Tudino, V.; Sharma, V.; Nguyen, J.; Debnath, A.; Podust, L.; Palenca, I.; Basili Franzin, S.; Seguella, L.; Esposito, G.; Petrucci, R.; Di Matteo, P.; Bortolami, M.; Scipione, L.; Costi, Roberta; Di Santo, Roberto. - 04f Poster
conference: 10th EFMC Young Medicinal Chemists' Symposium (Zagreb; Croatia.)
book: 10th EFMC Young Medicinal Chemists' Symposium - ()

11573/1687531 - 2023 - Role of a Novel Heparanase Inhibitor on the Balance between Apoptosis and Autophagy in U87 Human Glioblastoma Cells
Manganelli, V.; Misasi, R.; Riitano, G.; Capozzi, A.; Mattei, V.; Caglar, T. R.; Ialongo, D.; Madia, V. N.; Messore, A.; Costi, R.; Di Santo, R.; Sorice, M.; Garofalo, T. - 01a Articolo in rivista
paper: CELLS (Basel: mdpi-Molecular Diversity Preservation International) pp. 1-14 - issn: 2073-4409 - wos: WOS:001038054000001 (0) - scopus: 2-s2.0-85165884087 (0)

11573/1697140 - 2023 - Design and synthesis of tetrahydro-β-carbolines derivatives as PDIA inhibitors.
Messore, A.; Madia, V. N.; Ialongo, D.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Altieri, F.; Paglia, G.; Meschiari, G.; Di Santo, R.; Costi, R. - 04f Poster
conference: XXVIII edition of the National Meeting on Medicinal Chemistry (Chieti; Italy)
book: XXVIII edition of the National Meeting on Medicinal Chemistry - ()

11573/1697150 - 2023 - From Iloperidone to new Sigma1 agonists: a structure-based approach for Huntington's disease treatment.
Patacchini, Elisa; Madia, Valentina Noemi; Ialongo, Davide; Messore, Antonella; Ilari, Andrea; Cosconati, Sandro; Di Santo, Roberto; Costi, Roberta. - 04f Poster
conference: ESMEC 2023 - European School of Medicinal Chemistry – 42nd Edition (Urbino; Italy)
book: ESMEC 2023 - European School of Medicinal Chemistry – 42nd Edition - ()

11573/1696092 - 2023 - Miconazole-like Scaffold is a Promising Lead for Naegleria fowleri-Specific CYP51 Inhibitors
Sharma, Vandna; Madia, Valentina Noemi; Tudino, Valeria; V Nguyen, Jennifer; Debnath, Anjan; Messore, Antonella; Ialongo, Davide; Patacchini, Elisa; Palenca, Irene; Basili Franzin, Silvia; Seguella, Luisa; Esposito, Giuseppe; Petrucci, Rita; Di Matteo, Paola; Bortolami, Martina; Saccoliti, Francesco; Di Santo, Roberto; Scipione, Luigi; Costi, Roberta; M Podust, Larissa - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 17059-17073 - issn: 0022-2623 - wos: WOS:001134079100001 (0) - scopus: 2-s2.0-85180091142 (0)

11573/1638218 - 2022 - Design, synthesis, and In vitro, in silico and in cellulo evaluation of new Pyrimidine and Pyridine amide and Carbamate derivatives as multi-functional Cholinesterase Inhibitors
Bortolami, Martina; Pandolfi, Fabiana; Tudino, Valeria; Messore, Antonella; Madia, Valentina Noemi; De Vita, Daniela; Di Santo, Roberto; Costi, Roberta; Romeo, Isabella; Alcaro, Stefano; Colone, Marisa; Stringaro, Annarita; Espargaró, Alba; Sabatè, Raimon; Scipione, Luigi - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. 1-31 - issn: 1424-8247 - wos: WOS:000818156100001 (3) - scopus: 2-s2.0-85134396743 (2)

11573/1654141 - 2022 - New Inhibitors of the human p300/CBP acetyltransferase are selectively active against the Arabidopsis HAC proteins
Longo, Chiara; Lepri, Andrea; Paciolla, Andrea; Messore, Antonella; De Vita, Daniela; Bonaccorsi Di Patti, Maria Carmela; Amadei, Matteo; Madia, Valentina Noemi; Ialongo, Davide; Di Santo, Roberto; Costi, Roberta; Vittorioso, Paola - 01a Articolo in rivista
paper: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (Basel: MDPI Center) pp. 1-18 - issn: 1422-0067 - wos: WOS:000859422800001 (3) - scopus: 2-s2.0-85138734584 (3)

11573/1648549 - 2022 - Ultrastructural damages to H1N1 influenza virus caused by vapor essential oils
Madia, Valentina Noemi; Toscanelli, Walter; De Vita, Daniela; De Angelis, Marta; Messore, Antonella; Ialongo, Davide; Scipione, Luigi; Tudino, Valeria; D'auria, Felicia Diodata; Di Santo, Roberto; Garzoli, Stefania; Stringaro, Annarita; Colone, Marisa; Marchetti, Magda; Superti, Fabiana; Nencioni, Lucia; Costi, Roberta - 01a Articolo in rivista
paper: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. 1-14 - issn: 1420-3049 - wos: WOS:000816243700001 (5) - scopus: 2-s2.0-85131746075 (5)

11573/1623472 - 2022 - The kinesin Eg5 inhibitor K858 exerts antiproliferative and proapoptotic effects and attenuates the invasive potential of head and neck squamous carcinoma cells
Nicolai, Alice; Taurone, Samanta; Carradori, Simone; Artico, Marco; Greco, Antonio; Costi, Roberta; Scarpa, Susanna - 01a Articolo in rivista
paper: INVESTIGATIONAL NEW DRUGS (attuale: -SPRINGER, VAN GODEWIJCKSTRAAT 30, DORDRECHT, NETHERLANDS, 3311 GZ -Kluwer Academic Publishers / Massachusetts:PO Box 358, Accord Station:Hingham, MA 02018:(617)871-6600) pp. - - issn: 0167-6997 - wos: WOS:000771319900002 (3) - scopus: 2-s2.0-85126822611 (3)

11573/1623281 - 2022 - Oxidative stress and visual system a review
Taurone, S.; Ralli, M.; Artico, M.; Madia, V. N.; Scarpa, S.; Nottola, S. A.; Maconi, A.; Betti, M.; Familiari, P.; Nebbioso, M.; Costi, R.; Micera, A. - 01g Articolo di rassegna (Review)
paper: EXCLI JOURNAL (Mainz: EXCLI Journal Business Office c/o 2nd Medical Department, University of Mainz.) pp. 544-553 - issn: 1611-2156 - wos: WOS:000766811300001 (8) - scopus: 2-s2.0-85125850235 (10)

11573/1638214 - 2022 - Evaluation of the Anti-Histoplasma capsulatum activity of Indole and Nitrofuran derivatives and their pharmacological safety in three-dimensional cell cultures
Vaso, C. O.; Bila, N. M.; Pandolfi, F.; De Vita, D.; Bortolami, M.; Bonatti, J. L. C.; De Moraes Silva, R. A.; Goncalves, L. N. C.; Tudino, V.; Costi, R.; Di Santo, R.; Mendes-Giannini, M. J. S.; Costa-Orlandi, C. B.; Scipione, L.; Fusco-Almeida, A. M. - 01a Articolo in rivista
paper: PHARMACEUTICS (Basel: MDPI, 2009-) pp. 1-23 - issn: 1999-4923 - wos: WOS:000803586100001 (3) - scopus: 2-s2.0-85130346777 (3)

11573/1638210 - 2022 - Synthesis and evaluation of the antifungal and toxicological activity of Nitrofuran derivatives
Vaso, C. O.; Pandolfi, F.; Bila, N. M.; De Vita, D.; Bortolami, M.; Mendes-Giannini, M. J. S.; Tudino, V.; Costi, R.; Costa-Orlandi, C. B.; Fusco-Almeida, A. M.; Scipione, L. - 01a Articolo in rivista
paper: PHARMACEUTICS (Basel: MDPI, 2009-) pp. 1-19 - issn: 1999-4923 - wos: WOS:000774275300001 (3) - scopus: 2-s2.0-85126453264 (3)

11573/1662952 - 2022 - Exosomal Functional Cargoes from Liquid Biopsy of Gastric Cancer. A Systematic Review of Studies With Potential Clinical Relevance
Virgilio, E.; Montali, F.; Annicchiarico, A.; Salvemini, C.; Baldinu, M.; Giarnieri, E.; Montagnini, M.; Villani, S.; Proietti, A.; D'urso, R.; Costi, R. - 01g Articolo di rassegna (Review)
paper: ANTICANCER RESEARCH (Kapandriti: International Institute of Anticancer Research, 1995 Earliest publisher: Καπανδρίτι: Ιωάννης Γ. Δεληνάσιος, 1981-1995 Kapandriti: Iōannīs G. Delīnasios, 1981-1995) pp. 2249-2259 - issn: 0250-7005 - wos: WOS:000795123200003 (2) - scopus: 2-s2.0-85129187422 (3)

11573/1564954 - 2021 - Toxicological aspects of cannabinoid, pesticide and metal levels detected in light Cannabis inflorescences grown in Italy
Amendola, G.; Bocca, B.; Picardo, V.; Pelosi, P.; Battistini, B.; Ruggieri, F.; Attard Barbini, D.; De Vita, D.; Madia, V. N.; Messore, A.; Di Santo, R.; Costi, R. - 01a Articolo in rivista
paper: FOOD AND CHEMICAL TOXICOLOGY (Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. - - issn: 0278-6915 - wos: WOS:000696988600002 (5) - scopus: 2-s2.0-85112006002 (7)

11573/1615167 - 2021 - Pha-680626 is an effective inhibitor of the interaction between aurora-a and n-myc
Boi, D.; Souvalidou, F.; Capelli, D.; Polverino, F.; Marini, G.; Montanari, R.; Pochetti, G.; Tramonti, A.; Contestabile, R.; Trisciuoglio, D.; Carpinelli, P.; Ascanelli, C.; Lindon, C.; De Leo, A.; Saviano, M.; Di Santo, R.; Costi, R.; Guarguaglini, G.; Paiardini, A. - 01a Articolo in rivista
paper: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (Basel (Matthaeustrasse 11) : Molecular Diversity Preservation International MDPI) pp. 13122- - issn: 1661-6596 - wos: WOS:000735123900001 (9) - scopus: 2-s2.0-85120777012 (10)

11573/1490818 - 2021 - Acetylcholinesterase inhibitors for the treatment of Alzheimer’s disease–a patent review (2016–present)
Bortolami, M.; Rocco, D.; Messore, A.; Di Santo, R.; Costi, R.; Madia, V. N.; Scipione, L.; Pandolfi, F. - 01a Articolo in rivista
paper: EXPERT OPINION ON THERAPEUTIC PATENTS (--London United Kingdom:Informa Healthcare -London, United Kingdom: Ashley Publications Limited) pp. 1-22 - issn: 1354-3776 - wos: WOS:000607685400001 (28) - scopus: 2-s2.0-85099470810 (27)

11573/1546419 - 2021 - Design, synthesis and biological evaluation of a series of iron and copper chelating deferiprone derivatives as new agents active against Candida albicans
Bortolami, Martina; Pandolfi, Fabiana; Messore, Antonella; Rocco, Daniele; Feroci, Marta; Di Santo, Roberto; De Vita, Daniela; Costi, Roberta; Cascarino, Paola; Simonetti, Giovanna; Scipione, Luigi - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 1-7 - issn: 0960-894X - wos: WOS:000655255700006 (5) - scopus: 2-s2.0-85105482975 (5)

11573/1584588 - 2021 - New pyrimidine and pyridine derivatives as multitarget cholinesterase inhibitors. Design, synthesis, and in vitro and in cellulo evaluation
Bortolami, Martina; Pandolfi, Fabiana; Tudino, Valeria; Messore, Antonella; Madia, Valentina Noemi; De Vita, Daniela; Di Santo, Roberto; Costi, Roberta; Romeo, Isabella; Alcaro, Stefano; Colone, Marisa; Stringaro, Annarita; Espargaró, Alba; Sabatè, Raimon; Scipione, Luigi - 01a Articolo in rivista
paper: ACS CHEMICAL NEUROSCIENCE (Washington, D.C. : American Chemical Society) pp. 4090-4112 - issn: 1948-7193 - wos: WOS:000715842900011 (10) - scopus: 2-s2.0-85118138783 (12)

11573/1599717 - 2021 - Changes in surgicaL behaviOrs dUring the CoviD-19 pandemic. The SICE CLOUD19 Study
Bracale, U.; Podda, M.; Castiglioni, S.; Peltrini, R.; Sartori, A.; Arezzo, A.; Corcione, F.; Agresta, F.; Antonucci, A.; Zanframundo, C.; Cavallo, F.; Mazzarolo, G.; Agrusa, A.; Di Buono, G.; Aldrighetti, L.; Fiorentini, G.; Lucianetti, A.; Magnone, S.; Alfieri, S.; Rosa, F.; Altomare, D. F.; Picciariello, A.; Parisi, A.; Di Cintio, A.; Amisano, M. F.; Cravero, F.; Ammendola, M.; Ammerata, G.; Anastasi, A.; Canonico, G.; Gattolin, A.; Travaglio, E.; Sartori, A.; De Palma, M.; Angelini, P.; Galante, F.; Benevento, A.; Rausei, S.; Serao, A.; Abbatini, F.; Annecchiarico, M.; Varricchio, A.; Annessi, V.; Tumiati, D.; Annicchiarico, A.; Mirabella, A.; Marino, M. V.; Spinelli, A.; Braun, A.; Santi, H. T.; Romano, L.; Antoniutti, M.; Armellino, M. F.; Argenio, G.; Verzelli, A.; Budassi, A.; Baiocchi, G.; Alfano, M. S.; Balani, A.; Barone, M.; Baldazzi, G.; Cassini, D.; Canger, R. C. B.; Zabbialini, G.; Belli, A.; Izzo, F.; Bertolino, F.; Brunetti, M.; Bianco, F.; Cappiello, A.; Boccia, L.; Boffi, B.; Perna, F.; Bonilauri, S.; Frazzetta, G.; Bordoni, P.; Fleres, F.; Borghi, F.; Giraudo, G.; Bottino, V.; Canfora, A.; Piccoli, F. B.; Calligaris, L.; Nipote, B.; Nasti, A. G.; Bufalari, A.; Bettarini, F.; Buononato, M.; Greco, M.; Calo, P. G.; Medas, F.; Cardamone, E.; Castaldo, P.; Carlini, M.; Spoletini, D.; De Nisco, C.; Pulighe, F.; Feo, C. V.; Fabbri, N.; Antropoli, C.; Foroni, F.; Carnazza, M.; Ragazzi, S.; Cassinotti, E.; Boni, L.; Catena, F.; Giuffrida, M.; Perrone, G.; Ccotsoglou, C.; Granieri, S.; Ceccarelli, G.; Bugiantella, W.; Cedolini, C.; Seriau, L.; Cesari, M.; Contine, A.; Chiara, O.; Cimbanassi, S.; Cocozza, E.; Berselli, M.; Fantini, C.; Costi, R.; Casali, L.; Morini, A.; Crafa, F.; Vanela, S.; Curro, G.; Orsini, V.; Da Lio, C.; Biral, M.; Danelli, P.; Guerci, C.; Scala, D.; Marino, G.; De Carlis, L.; Lauterio, A.; De Giorgi, D.; Sciannamea, G.; De Manzini, N.; Losurdo, P.; De Palma, M.; Sangiuliano, N.; Degiuli, M.; Caterina, F.; Del Rio, P.; Bonati, E.; Di Lernia, S.; Ardizzone, M. V. R.; Di Saverio, S.; Franchi, C.; Di Venere, B.; Miglio, R.; Cuccurullo, D.; Sagnelli, C.; Docimo, L.; Tolone, S.; Longoni, M.; Faillace, G.; Rondelli, F.; Pennella, F. P.; Colucci, V.; Carfora, T.; Muttillo, I. A.; Picardi, B.; Stefano, R.; Campagnacci, R.; Maurizi, A.; Tricarico, F.; Montagna, M.; Amedeo, E.; Scollica, M. C.; Lauro, E.; Laterza, E.; Molinari, E.; Berta, G.; Bono, D.; Fabozzi, M.; Romano, M.; Facci, E.; Parini, D.; Farfaglia, R.; Arizzi, V.; Farsi, M.; Miranda, E.; Fei, L.; Flavio, G.; Pirozzi, F.; Sciuto, A.; Ferrero, A.; Palisi, M.; Filauro, M.; Barberis, A.; Azzinnaro, A.; Fiscon, V.; Vigna, S.; D'ambra, M.; Pontecorvi, E.; Anania, G.; Bombardini, C.; Galizia, G.; Auricchio, A.; Cardella, F.; Genna, M.; Gentilli, S.; Herald, N.; Castagnoli, G.; Bartoli, A.; Gianotti, L.; Garancini, M.; Bellanova, G.; Palazzo, P.; De Palma, G.; Milone, M.; Ferrari, G.; Magistro, C.; Giuliani, A.; Di Natale, G.; Brisinda, G.; Cavallaro, G.; Sammarco, G.; Gallo, G.; Goletti, O.; Macchini, D.; Greco, V.; Amoroso, V.; Guercioni, G.; Benedetti, M.; Guzzo, G.; Pata, F.; Scandroglio, I.; Roscio, F.; Jovine, E.; Lombardi, R.; La Rocca, F.; Di Capua, F.; Lanci, C.; Leli, R.; Borasi, A.; Lepiane, P.; Balla, A.; Liberatore, E.; Morelli, L.; Di Franco, G.; Lucchi, A.; Vittori, L.; Bonavina, L.; Asti, E.; Maggioni, D.; Martino, G.; Manca, G.; Delvecchio, A.; Tedesco, M.; Gambardella, D.; Marafioti, S.; De Marco, M. L.; Guicciardi, M. A.; Motta, M.; Calgaro, M.; Adamo, V.; Guerrieri, M.; Coletta, P.; Ortenzi, M.; Martines, G.; Lantone, G.; Martinotti, M.; Fassardi, G.; Castriconi, M.; Squillante, S.; De Luca, M.; Pavanello, M.; Di Marco, C.; Ronconi, M.; Casiraghi, S.; Mazzaferro, V.; Battiston, C.; Perrotta, M.; Ripa, C.; Giancarlo, M.; Panizzo, V.; Millo, P.; Contul, R. B.; Ferraro, V.; Molino, C.; Crolla, E.; Moretto, G.; Bacchion, M.; Morino, M.; Allaix, M. E.; Motterlini, E.; Petracca, M.; Muratore, A.; Musella, M.; Vitiello, A.; Nardo, B.; Cr - 01a Articolo in rivista
paper: UPDATES IN SURGERY (Milano : Springer-Verlag Italia) pp. 731-744 - issn: 2038-131X - wos: WOS:000625025100002 (25) - scopus: 2-s2.0-85102173717 (30)

11573/1555182 - 2021 - Effect of Heparanase inhibitor on Tissue Factor overexpression in platelets and endothelial cells induced by anti-β2-GPI antibodies
Capozzi, Antonella; Riitano, Gloria; Recalchi, Serena; Manganelli, Valeria; Costi, Roberta; Saccoliti, Francesco; Pulcinelli, Fabio Maria; Garofalo, Tina; Misasi, Roberta; Longo, Agostina; Di Santo, Roberto; Sorice, Maurizio - 01a Articolo in rivista
paper: JOURNAL OF THROMBOSIS AND HAEMOSTASIS (International Society on Thrombosis and Haemostasis ISTH) pp. 1-12 - issn: 1538-7933 - wos: WOS:000669313100001 (8) - scopus: 2-s2.0-85109019340 (8)

11573/1404920 - 2021 - Towards a new application of amaranth seed oil as an agent against Candida albicans
De Vita, Daniela; Messore, Antonella; Toniolo, Chiara; Frezza, Claudio; Scipione, Luigi; Bertea, Cinzia Margherita; Micera, Marco; Di Sarno, Veronica; Madia, Valentina Noemi; Pindinello, Ivano; Roscilli, Patrizia; Botto, Alfonso; Simonetti, Giovanna; Orekhova, Anastasia; Manfredini, Stefano; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: NATURAL PRODUCT RESEARCH (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 4621-4626 - issn: 1478-6419 - wos: WOS:000500457200001 (14) - scopus: 2-s2.0-85075913942 (5)

11573/1540215 - 2021 - Investigation of Commiphora myrrha (Nees) Engl. oil and its main components for antiviral activity
Madia, Valentina Noemi; De Angelis, Marta; De Vita, Daniela; Messore, Antonella; De Leo, Alessandro; Ialongo, Davide; Tudino, Valeria; Saccoliti, Francesco; De Chiara, Giovanna; Garzoli, Stefania; Scipione, Luigi; Palamara, Anna Teresa; Di Santo, Roberto; Nencioni, Lucia; Costi, Roberta - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. - - issn: 1424-8247 - wos: WOS:000634055800001 (15) - scopus: 2-s2.0-85102987115 (18)

11573/1564144 - 2021 - Recent advances in recovery of lycopene from tomato waste. A potent antioxidant with endless benefits
Madia, Valentina Noemi; De Vita, Daniela; Ialongo, Davide; Tudino, Valeria; De Leo, Alessandro; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta; Messore, Antonella - 01a Articolo in rivista
paper: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. 1-18 - issn: 1420-3049 - wos: WOS:000682223800001 (33) - scopus: 2-s2.0-85111602310 (40)

11573/1540619 - 2021 - Analytical characterization of an inulin-type fructooligosaccharide from root-tubers of Asphodelus ramosus L
Madia, Valentina Noemi; De Vita, Daniela; Messore, Antonella; Toniolo, Chiara; Tudino, Valeria; De Leo, Alessandro; Pindinello, Ivano; Ialongo, Davide; Saccoliti, Francesco; D'ursi, Anna Maria; Grimaldi, Manuela; Ceccobelli, Pietro; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. - - issn: 1424-8247 - wos: WOS:000634075100001 (4) - scopus: 2-s2.0-85103099178 (3)

11573/1565318 - 2021 - Small-molecule inhibitors of HIV-1 reverse transcriptase-associated ribonuclease H function. Challenges and recent developments
Madia, Valentina Noemi; Messore, Antonella; De Leo, Alessandro; Tudino, Valeria; Pindinello, Ivano; Saccoliti, Francesco; De Vita, Daniela; Scipione, Luigi; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: CURRENT MEDICINAL CHEMISTRY (Hilversum: Bentham Science Publishers) pp. 1-33 - issn: 1875-533X - wos: WOS:000696992000004 (3) - scopus: 2-s2.0-85115249511 (4)

11573/1493998 - 2021 - Design, synthesis and biological evaluation of new pyrimidine derivatives as anticancer agents
Madia, Valentina Noemi; Nicolai, Alice; Messore, Antonella; De Leo, Alessandro; Ialongo, Davide; Tudino, Valeria; Saccoliti, Francesco; De Vita, Daniela; Scipione, Luigi; Artico, Marco; Taurone, Samanta; Taglieri, Ludovica; Di Santo, Roberto; Scarpa, Susanna; Costi, Roberta - 01a Articolo in rivista
paper: MOLECULES (Basel: MDPI Berlin: Springer, 1996-) pp. - - issn: 1420-3049 - wos: WOS:000615455300001 (11) - scopus: 2-s2.0-85101195321 (12)

11573/1594159 - 2021 - Understanding drivers of ocular fibrosis: current and future therapeutic perspectives
Mallone, F.; Costi, R.; Marenco, M.; Plateroti, R.; Minni, A.; Attanasio, G.; Artico, M.; Lambiase, A. - 01g Articolo di rassegna (Review)
paper: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (Basel (Matthaeustrasse 11) : Molecular Diversity Preservation International MDPI) pp. - - issn: 1661-6596 - wos: WOS:000718582700001 (14) - scopus: 2-s2.0-85118118842 (14)

11573/1556284 - 2021 - Quinolinonyl non-diketo acid derivatives as Inhibitors of HIV-1 ribonuclease H and polymerase functions of reverse transcriptase
Messore, Antonella; Corona, Angela; Madia, Valentina Noemi; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Ialongo, Davide; Scipione, Luigi; De Vita, Daniela; Amendola, Giorgio; Novellino, Ettore; Cosconati, Sandro; Métifiot, Mathieu; Andreola, Marie-Line; Esposito, Francesca; Grandi, Nicole; Tramontano, Enzo; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 8579-8598 - issn: 0022-2623 - wos: WOS:000668340800039 (9) - scopus: 2-s2.0-85108607601 (8)

11573/1553152 - 2021 - Anti-tumoral effects of a (1H-pyrrol-1-yl)methyl-1H-benzoimidazole carbamate ester derivative on head and neck squamous carcinoma cell lines
Nicolai, Alice; Madia, Valentina Noemi; Messore, Antonella; De Vita, Daniela; De Leo, Alessandro; Ialongo, Davide; Tudino, Valeria; Tortorella, Elisabetta; Scipione, Luigi; Taurone, Samanta; Pergolizzi, Tiziano; Artico, Marco; Di Santo, Roberto; Costi, Roberta; Scarpa, Susanna - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. - - issn: 1424-8247 - wos: WOS:000666329400001 (6) - scopus: 2-s2.0-85110773299 (6)

11573/1395352 - 2020 - New deferiprone derivatives as multi-functional cholinesterase inhibitors. Design, synthesis and in vitro evaluation
Bortolami, Martina; Pandolfi, Fabiana; De Vita, Daniela.; Carafa, Camilla; Messore, Antonella; Di Santo, Roberto; Feroci, Marta; Costi, Roberta; Chiarotto, Isabella; Bagetta, Donatella; Alcaro, Stefano; Colone, Marisa; Stringaro, Annarita; Scipione, Luigi - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 1-17 - issn: 0223-5234 - wos: WOS:000539425800007 (26) - scopus: 2-s2.0-85084066662 (29)

11573/1408850 - 2020 - Pyrrolyl pyrazoles as non-diketo acid inhibitors of the HIV-1 ribonuclease H function of reverse transcriptase
Messore, Antonella; Corona, Angela; Madia, Valentina Noemi; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Scipione, Luigi; De Vita, Daniela; Amendola, Giorgio; Di Maro, Salvatore; Novellino, Ettore; Cosconati, Sandro; Métifiot, Mathieu; Andreola, Marie-Line; Valenti, Piera; Esposito, Francesca; Grandi, Nicole; Tramontano, Enzo; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: ACS MEDICINAL CHEMISTRY LETTERS (USA: ACS Publications) pp. 798-805 - issn: 1948-5875 - wos: WOS:000535281200029 (22) - scopus: 2-s2.0-85086659986 (23)

11573/1389105 - 2020 - Influence of oral administration mode on the efficacy of commercial bovine Lactoferrin against iron and inflammatory homeostasis disorders
Rosa, L.; Lepanto, M. S.; Cutone, A.; Siciliano, R. A.; Paesano, R.; Costi, R.; Musci, G.; Valenti, P. - 01a Articolo in rivista
paper: BIOMETALS (Rapid Science Publishers:2-6 Boundary Row, London SE1 8HN United Kingdom:011 44 207 9407500, EMAIL: rapidcom@vax.oxford.ac.uk, Fax: 011 44 207 8650027) pp. - - issn: 0966-0844 - wos: WOS:000540269500007 (18) - scopus: 2-s2.0-85083453638 (17)

11573/1490804 - 2020 - Recent advancement in the search of innovative antiprotozoal agents targeting trypanothione metabolism
Saccoliti, F.; Di Santo, R.; Costi, R. - 01a Articolo in rivista
paper: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. 2420-2435 - issn: 1860-7179 - wos: WOS:000567909300001 (13) - scopus: 2-s2.0-85091368381 (13)

11573/1274892 - 2020 - Discovery of a pyrimidine compound endowed with antitumor activity
Taglieri, Ludovica; Saccoliti, Francesco; Nicolai, Alice; Peruzzi, Giovanna; Madia, Valentina Noemi; Tudino, Valeria; Messore, Antonella; Di Santo, Roberto; Artico, Marco; Taurone, Samanta; Salvati, Maurizio; Costi, Roberta; Scarpa, Susanna - 01a Articolo in rivista
paper: INVESTIGATIONAL NEW DRUGS (attuale: -SPRINGER, VAN GODEWIJCKSTRAAT 30, DORDRECHT, NETHERLANDS, 3311 GZ -Kluwer Academic Publishers / Massachusetts:PO Box 358, Accord Station:Hingham, MA 02018:(617)871-6600) pp. 39-49 - issn: 0167-6997 - wos: WOS:000512107200005 (11) - scopus: 2-s2.0-85063345760 (11)

11573/1336764 - 2019 - Structure-guided approach to identify a novel class of anti-leishmaniasis diaryl sulfide compounds targeting the trypanothione metabolism
Colotti, G.; Saccoliti, F.; Gramiccia, M.; Di Muccio, T.; Prakash, J.; Yadav, S.; Dubey, V. K.; Vistoli, G.; Battista, T.; Mocci, S.; Fiorillo, A.; Bibi, Aasia; Madia, V. N.; Messore, A.; Costi, R.; Di Santo, R.; Ilari, A. - 01a Articolo in rivista
paper: AMINO ACIDS (Wien: Springer Verlag) pp. - - issn: 0939-4451 - wos: WOS:000519385700013 (10) - scopus: 2-s2.0-85065106515 (11)

11573/1285185 - 2019 - Comparison of different methods for the extraction of cannabinoids from cannabis
De Vita, D.; Madia, V. N.; Tudino, V.; Saccoliti, F.; De Leo, A.; Messore, A.; Roscilli, P.; Botto, A.; Pindinello, I.; Santilli, G.; Scipione, L.; Costi, R.; Di Santo, R. - 01a Articolo in rivista
paper: NATURAL PRODUCT RESEARCH (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1-7 - issn: 1478-6419 - wos: WOS:000575920700013 (32) - scopus: 2-s2.0-85065155862 (36)

11573/1205976 - 2019 - In vitro antiviral activity of new oxazoline derivatives as potent poliovirus inhibitors
Madia, Valentina Noemi; Messore, Antonella; Pescatori, Luca; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Scipione, Luigi; Fiore, Lucia; Rhoden, Eric; Manetti, Fabrizio; Oberste, M Steven; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 798-810 - issn: 0022-2623 - wos: WOS:000457067600026 (8) - scopus: 2-s2.0-85060542889 (10)

11573/1405464 - 2019 - Tegaserod for the treatment of Irritable Bowel syndrome
Madia, Valentina Noemi; Messore, Antonella; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; De Vita, Daniela; Bortolami, Martina; Scipione, Luigi; Pindinello, Ivano; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: ANTI-INFLAMMATORY & ANTI-ALLERGY AGENTS IN MEDICINAL CHEMISTRY (Hilversum : Bentham Science Publsihers) pp. 1-28 - issn: 1871-5230 - wos: (0) - scopus: 2-s2.0-85083912835 (0)

11573/1218854 - 2019 - Searching for new agents active against candida albicans biofilm: a series of indole derivatives, design, synthesis and biological evaluation
Pandolfi, Fabiana; D'acierno, Federica; Bortolami, Martina; De Vita, Daniela; Gallo, Fabio; De Meo, Alessandra; Di Santo, Roberto; Costi, Roberta; Simonetti, Giovanna; Scipione, Luigi - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 93-106 - issn: 0223-5234 - wos: WOS:000459358600008 (27) - scopus: 2-s2.0-85060089854 (28)

11573/1321741 - 2019 - Inhibition of Polycomb Repressive Complex2 activity reduces trimethylation of H3K27 and affects development in Arabidopsis seedlings
Ruta, Veronica; Longo, Chiara; Boccaccini, Alessandra; Madia, Valentina Noemi; Saccoliti, Francesco; Tudino, Valeria; Di Santo, Roberto; Lorrai, Riccardo; Dello Ioio, Raffaele; Sabatini, Sabrina; Costi, Roberta; Costantino, Paolo; Vittorioso, Paola - 01a Articolo in rivista
paper: BMC PLANT BIOLOGY (London: BioMed Central.MIDDLESEX HOUSE, 34-42 CLEVELAND ST, LONDON, ENGLAND, W1T 4LB) pp. - - issn: 1471-2229 - wos: WOS:000490716900003 (12) - scopus: 2-s2.0-85073428390 (12)

11573/1222183 - 2019 - Design, synthesis, and biological evaluation of new 1-(aryl-1H-pyrrolyl)(phenyl)methyl-1H-imidazole derivatives as antiprotozoal agents
Saccoliti, Francesco; Madia, Valentina Noemi; Tudino, Valeria; De Leo, Alessandro; Pescatori, Luca; Messore, Antonella; De Vita, Daniela; Scipione, Luigi; Brun, Reto; Kaiser, Marcel; Mäser, Pascal; Calvet Alvarez, Claudia Magalhaes; Jennings, Gareth K; Podust, Larissa M; Pepe, Giacomo; Cirilli, Roberto; Faggi, Cristina; Di Marco, Annalise; Battista, Maria Rosaria; Summa, Vincenzo; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1330-1347 - issn: 0022-2623 - wos: WOS:000459223600016 (23) - scopus: 2-s2.0-85061636363 (26)

11573/1176836 - 2018 - Novel benzazole derivatives endowed with potent antiheparanase activity
Madia, Valentina Noemi; Messore, Antonella; Pescatori, Luca; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Bortolami, Martina; Scipione, Luigi; Costi, Roberta; Rivara, Silvia; Scalvini, Laura; Mor, Marco; Fosca Ferrara, Fabiana; Pavoni, Emiliano; Roscilli, Giuseppe; Cassinelli, Giuliana; M Milazzo, Ferdinando; Battistuzzi, Gianfranco; Di Santo, Roberto; Giannin, Giuseppe - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 6918-6936 - issn: 0022-2623 - wos: WOS:000441484300030 (28) - scopus: 2-s2.0-85050088127 (28)

11573/1221546 - 2018 - Novel symmetrical benzazolyl derivatives endowed with potent anti-heparanase activity
Messore, Antonella; Madia, Valentina Noemi; Pescatori, Luca; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Bortolami, Martina; De Vita, Daniela; Scipione, Luigi; Pepi, Federico; Costi, Roberta; Rivara, Silvia; Scalvini, Laura; Mor, Marco; Ferrara, Fabiana Fosca; Pavoni, Emiliano; Roscilli, Giuseppe; Cassinelli, Giuliana; Milazzo, Ferdinando M; Battistuzzi, Gianfranco; Di Santo, Roberto; Giannini, Giuseppe - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 10834-10859 - issn: 0022-2623 - wos: WOS:000453488200031 (17) - scopus: 2-s2.0-85058215116 (16)

11573/1099440 - 2018 - Structure-guided approach identifies a novel class of HIV-1 ribonuclease H inhibitors: binding mode insights through magnesium complexation and site-directed mutagenesis studies
Poongavanam, Vasanthanathan; Corona, Angela; Steinmann, Casper; Scipione, Luigi; Grandi, Nicole; Pandolfi, Fabiana; Di Santo, Roberto; Costi, Roberta; Esposito, Francesca; Tramontano, Enzo; Kongsted, Jacob - 01a Articolo in rivista
paper: MEDCHEMCOMM (Cambridge : Royal Society of Chemistry, 2010-) pp. 562-575 - issn: 2040-2503 - wos: WOS:000428670100016 (17) - scopus: 2-s2.0-85044181388 (17)

11573/1174521 - 2018 - Selective inhibition of the PRC2 methyltransferase activity suppresses trimethylation of H3K27 in Arabidopsis seeds
Ruta, Veronica; Boccaccini, Alessandra; Longo, Chiara; Madia, Valentina Noemi; Tudino, Valeria; Costi, Roberta; Costantino, Paolo; Vittorioso, Paola - 04f Poster
conference: International Plant and Molecular Biology 2018- IPMB2018 (Montpellier)
book: nessuna - ()

11573/1176720 - 2018 - Biological evaluation and structure-activity relationships of imidazole-based compounds as antiprotozoal agents
Saccoliti, Francesco; Madia, Valentina Noemi; Tudino, Valeria; De Leo, Alessandro; Pescatori, Luca; Messore, Antonella; De Vita, Daniela; Scipione, Luigi; Brun, Reto; Kaiser, Marcel; Mäser, Pascal; Magalhaes Calvet, Claudia; K Jennings, Gareth; M Podust, Larissa; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 53-60 - issn: 0223-5234 - wos: WOS:000443663200005 (16) - scopus: 2-s2.0-85049312582 (20)

11573/972447 - 2017 - Inhibition of the α-carbonic anhydrase from Vibrio cholerae with amides and sulfonamides incorporating imidazole moieties
De Vita, Daniela; Angeli, Andrea; Pandolfi, Fabiana; Bortolami, Martina; Costi, Roberta; Di Santo, Roberto; Suffredini, Elisabetta; Ceruso, Mariangela; Del Prete, Sonia; Capasso, Clemente; Scipione, Luigi; Supuran, Claudiu T. - 01a Articolo in rivista
paper: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 798-804 - issn: 1475-6366 - wos: WOS:000404271200006 (36) - scopus: 2-s2.0-85020209278 (37)

11573/910059 - 2017 - Functional roles of Acetylated Histone marks at mouse meiotic recombination hotspots
Getun, Iv; Wu, Z; Fallahi, M; Ouizem, S; Liu, Q; Li, W; Costi, Roberta; Roush, Wr; Cleveland, Jl; Bois, P. R. - 01a Articolo in rivista
paper: MOLECULAR AND CELLULAR BIOLOGY (American Society for Microbiology / DC:1752 N Street Northwest:Washington, DC 20036:(202)737-3600, EMAIL: jadelman@asmusa.org, INTERNET: http://www.asmusa.org/asm.htm, Fax: (202)942-9342) pp. 1-24 - issn: 0270-7306 - wos: WOS:000392231500009 (16) - scopus: 2-s2.0-85011575217 (15)

11573/1192249 - 2017 - Structure-activity relationships on cynnamoyl derivatives as inhibitors of p300 Histone acetyltransferase
Madia, Valentina Noemi; Benedetti, Rosaria; Letizia Barreca, Maria; Ngo, Liza; Pescatori, Luca; Messore, Antonella; Pupo, Giovanni; Saccoliti, Francesco; Valente, Sergio; Mai, Antonello; Scipione, Luigi; George Zheng, Yujun; Tintori, Cristina; Botta, Maurizio; Cecchetti, Violetta; Altucci, Lucia; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. 1359-1368 - issn: 1860-7187 - wos: WOS:000429592300014 (10) - scopus: 2-s2.0-85017448829 (9)

11573/1011030 - 2017 - New pyridine derivatives as inhibitors of acetylcholinesterase and amyloid aggregation
Pandolfi, Fabiana; De Vita, Daniela; Bortolami, Martina; Coluccia, Antonio; Di Santo, Roberto; Costi, Roberta; Andrisano, Vincenza; Alabiso, Francesco; Bergamini, Christian; Fato, Romana; Bartolini, Manuela; Scipione, Luigi - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 197-210 - issn: 0223-5234 - wos: WOS:000417962900018 (25) - scopus: 2-s2.0-85030860178 (29)

11573/929856 - 2017 - Inhibition of Leishmania infantum trypanothione reductase by diaryl sulfide derivatives
Saccoliti, Francesco; Angiulli, Gabriella; Pupo, Giovanni; Pescatori, Luca; Madia, Valentina Noemi; Messore, Antonella; Colotti, Gianni; Fiorillo, Annarita; Scipione, Luigi; Gramiccia, Marina; Di Muccio, Trentina; Di Santo, Roberto; Costi, Roberta; Ilari, Andrea - 01a Articolo in rivista
paper: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 304-310 - issn: 1475-6366 - wos: WOS:000392591100025 (46) - scopus: 2-s2.0-85013797723 (48)

11573/910116 - 2016 - New insights into the interaction between pyrrolyl diketoacids and HIV-1 integrase active site and comparison with RNase H
Corona, A; Di Leva, Fs; Rigogliuso, G; Pescatori, Luca; Madia, Valentina Noemi; Subra, F; Delelis, O; Esposito, F; Cadeddu, M; Costi, Roberta; Cosconati, S; Novellino, E; Di Santo, Roberto; Tramontano, E. - 01a Articolo in rivista
paper: ANTIVIRAL RESEARCH ([Amsterdam]; [New York]: Elsevier/North-Holland, [c1981]-) pp. 236-243 - issn: 0166-3542 - wos: WOS:000386983800026 (35) - scopus: 2-s2.0-84989205085 (34)

11573/903468 - 2016 - New N,N-dimethylcarbamate inhibitors of acetylcholinesterase: design synthesis and biological evaluation
De Vita, Daniela; Pandolfi, Fabiana; Ornano, Luigi; Feroci, Marta; Chiarotto, Isabella; Sileno, Ilaria; Pepi, Federico; Costi, Roberta; Di Santo, Roberto; Scipione, Luigi - 01a Articolo in rivista
paper: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1-8 - issn: 1475-6366 - wos: WOS:000391904900013 (11) - scopus: 2-s2.0-84984870776 (11)

11573/916308 - 2016 - Exploring the anti-biofilm activity of cinnamic acid derivatives in Candida albicans
De Vita, Daniela; Simonetti, Giovanna; Pandolfi, Fabiana; Costi, Roberta; Di Santo, Roberto; D'auria, Felicia Diodata; Scipione, Luigi - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 5931-5935 - issn: 0960-894X - wos: WOS:000389784500020 (19) - scopus: 2-s2.0-84999015180 (23)

11573/894759 - 2016 - Diaryl disulfides as novel stabilizers of tumor suppressor Pdcd4
Schmid, Tobias; Blees, Johanna S.; Bajer, Magdalena M.; Wild, Janine; Pescatori, Luca; Cuzzucoli Crucitti, Giuliana; Scipione, Luigi; Costi, Roberta; Henrich, Curtis J.; Brüne, Bernhard; Colburn, Nancy H.; Di Santo, Roberto - 01a Articolo in rivista
paper: PLOS ONE (San Francisco, CA : Public Library of Science) pp. 1-14 - issn: 1932-6203 - wos: WOS:000372574900108 (9) - scopus: 2-s2.0-84979088483 (10)

11573/852938 - 2015 - Discovery of N-aryl-naphthylamines as in vitro inhibitors of the interaction between HIV integrase and the cofactor LEDGF/p75
Cuzzucoli Crucitti, G.; Pescatori, L.; Messore, A.; Madia, V. N.; Pupo, G.; Saccoliti, F; Scipione, L; Tortorella, S.; Di Leva, F. S; Cosconati, S; Novellino, E; Debyser, Z; Christ, F; Costi, R; Di Santo, R - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 288-294 - issn: 0223-5234 - wos: WOS:000360771900026 (16) - scopus: 2-s2.0-84936802596 (16)

11573/895359 - 2015 - Structure−activity relationship of pyrrolyl diketo acid derivatives as dual Inhibitors of HIV‑1 integrase and reverse transcriptase ribonuclease H domain
Cuzzucoli Crucitti, Giuliana; Métifiot, Mathieu; Pescatori, Luca; Messore, Antonella; Madia, Valentina Noemi; Pupo, Giovanni; Saccoliti, Francesco; Scipione, Luigi; Tortorella, Silvano; Esposito, Francesca; Corona, Angela; Cadeddu, Marta; Marchand, Christophe; Pommier, Yves; Tramontano, Enzo; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1915-1928 - issn: 0022-2623 - wos: WOS:000351186700021 (72) - scopus: 2-s2.0-84923882396 (76)

11573/783972 - 2015 - Hypoglycemic activity of curcumin synthetic analogues in alloxan-induced diabetic rats
Das, Kk; Razzaghi Asl, N; Tikare, Sn; Di Santo, Roberto; Costi, Roberta; Messore, A; Pescatori, Luca; Crucitti, Gc; Jargar, Jg; Dhundasi, Sa; Saso, Luciano - 01a Articolo in rivista
paper: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1-7 - issn: 1475-6366 - wos: WOS:000367555300011 (18) - scopus: 2-s2.0-84953262310 (22)

11573/541604 - 2015 - Design, synthesis and evaluation of 3,4-dihydroxybenzoic acid derivatives as antioxidants, bio-metal chelating agents and acetylcholinesterase inhibitors
Friggeri, Laura; De Vita, Daniela; Pandolfi, Fabiana; Tortorella, Silvano; Costi, Roberta; Di Santo, Roberto; Scipione, Luigi - 01a Articolo in rivista
paper: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 166-172 - issn: 1475-6366 - wos: WOS:000347956500024 (7) - scopus: 2-s2.0-84921307137 (7)

11573/787196 - 2015 - N‑substituted quinolinonyl diketo acid derivatives as HIV integrase strand transfer inhibitors and their activity against RNase H function of reverse transcriptase
Pescatori, Luca; Metifiot, Mathieu; Chung, Suhman; Masoaka, Takashi; Crucitti Cuzzucoli, Giuliana; Messore, Antonella; Pupo, Giovanni; Madia, Valentina Noemi; Saccoliti, Francesco; Scipione, Luigi; Tortorella, Silvano; Di Leva, Francesco Saverio; Cosconati, Sandro; Marinelli, Luciana; Novellino, Ettore; Le Grice, Stuart F. J.; Pommier, Yves; Marchand, Christophe; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 4610-4623 - issn: 0022-2623 - wos: WOS:000356316600015 (40) - scopus: 2-s2.0-84935877076 (44)

11573/621580 - 2014 - identification of highly conserved residues involved in inhibition of HIV-1 RNase H function by Diketo Acid derivatives
Angela, Corona; Francesco Saverio Di, Leva; Sylvain, Thierry; Pescatori, Luca; Giuliana Cuzzuculi, Crucitti; Frederic, Subra; Olivier, Delelis; Francesca, Esposito; Giuseppe, Rigogliuso; Costi, Roberta; Sandro, Cosconati; Ettore, Novellino; Di Santo, Roberto; Enzo, Tramontano - 01a Articolo in rivista
paper: ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (American Society for Microbiology:PO Box 11127:Birmingham, AL 35201:(800)633-4931, (205)995-1567, EMAIL: asm.nonmembers.subs@ebsco.com, INTERNET: http://www.asm.org, Fax: (205)995-1588) pp. 6101-6110 - issn: 0066-4804 - wos: WOS:000344157500054 (61) - scopus: 2-s2.0-84907266363 (66)

11573/619388 - 2014 - Ptaquiloside in Pteridium aquilinum subsp. aquilinum and corresponding soils from South of Italy: influence of physical and chemical features of soils on its occurrence
Claudio, Zaccone; Ivana, Cavoski; Costi, Roberta; Giorgia, Sarais; Pierluigi, Caboni; Andreina, Traversa; Teodoro, M. Miano - 01a Articolo in rivista
paper: SCIENCE OF THE TOTAL ENVIRONMENT (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598 Tokyo ; Oxford ; Lausanne ; New York ; Shannon ; Amsterdam : Elsevier) pp. 365-372 - issn: 0048-9697 - wos: WOS:000342245600042 (8) - scopus: 2-s2.0-84905460086 (9)

11573/559331 - 2014 - Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV Integrase and their Activity against RNase H Function of Reverse Transcriptase
Costi, Roberta; Mathieu, Metifiot; Suhman, Chung; Cuzzucoli Crucitti, Giuliana; Kasthuraiah, Maddali; Pescatori, Luca; Messore, Antonella; Madia, Valentina Noemi; Giovanni, Pupo; Scipione, Luigi; Tortorella, Silvano; Francesco Saverio Di, Leva; Sandro, Cosconati; Luciana, Marinelli; Ettore, Novellino; Stuart F: J., Le Grice; Angela, Corona; Yves, Pommier; Christophe, Marchand; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington DC : ACS Publications) pp. 3223-3234 - issn: 1520-4804 - wos: WOS:000335113900005 (52) - scopus: 2-s2.0-84899554749 (56)

11573/541603 - 2014 - Activity of caffeic acid derivatives against Candida albicans biofilm
De Vita, Daniela; Friggeri, Laura; D'auria, Felicia Diodata; Pandolfi, Fabiana; Francesco, Piccoli; Panella, Simona; Palamara, Anna Teresa; Simonetti, Giovanna; Scipione, Luigi; R., Santo; Di Santo, Roberto; Costi, Roberta; Tortorella, Silvano - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 1502-1505 - issn: 0960-894X - wos: WOS:000332391900011 (50) - scopus: 2-s2.0-84895795071 (55)

11573/579587 - 2014 - Synthesis, biological evaluation and structure-activity correlation study of a series of imidazol-based compounds as Candida albicans inhibitors
Francesca, Moraca; De Vita, Daniela; Pandolfi, Fabiana; Di Santo, Roberto; Costi, Roberta; Roberto, Cirilli; D'auria, Felicia Diodata; Panella, Simona; Palamara, Anna Teresa; Simonetti, Giovanna; Maurizio, Botta; Scipione, Luigi - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 665-673 - issn: 0223-5234 - wos: WOS:000340689600059 (21) - scopus: 2-s2.0-84904025140 (21)

11573/525948 - 2013 - New Nucleotide-Competitive Non-Nucleoside Inhibitors of Terminal 2 Deoxynucleotidyl Transferase: Discovery, Characterization, and 3 Crystal Structure in Complex with the Target
Costi, Roberta; Cuzzucoli Crucitti, Giuliana; Pescatori, Luca; Messore, Antonella; Scipione, Luigi; Tortorella, Silvano; Alessandra, Amoroso; Emmanuele, Crespan; Pietro, Campiglia; Bruno, Maresca; Amalia, Porta; Ilaria, Granata; Ettore, Novellino; Jérôme, Gouge; Marc, Delarue; Giovanni, Maga; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 7431-7441 - issn: 0022-2623 - wos: WOS:000330097700023 (22) - scopus: 2-s2.0-84885013896 (22)

11573/530616 - 2013 - 6-(1-Benzyl-1H-pyrrol-2-yl)-2,4-dioxo-5-hexenoic acids as dual inhibitors of recombinant HIV-1 integrase and ribonuclease H, synthesized by a parallel synthesis approach.
Costi, Roberta; M., Metifiot; F., Esposito; Cuzzucoli Crucitti, Giuliana; Pescatori, Luca; Messore, Antonella; Scipione, Luigi; Tortorella, Silvano; L., Zinzula; C., Marchand; Y., Pommier; E., Tramontano; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington DC : ACS Publications) pp. 8588-8598 - issn: 1520-4804 - wos: WOS:000327111100029 (54) - scopus: 2-s2.0-84887922481 (57)

11573/515673 - 2013 - Pharmacophore assessment through 3-D QSAR: evaluation of the predictive ability on new derivatives by the application on a series of antitubercular agents
Friggeri, Laura; Ballante, Flavio; Ragno, Rino; Musmuca, Ira; De Vita, Daniela; Manetti, F. .; Biava, Mariangela; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta; Feroci, Marta; Tortorella, Silvano - 01a Articolo in rivista
paper: JOURNAL OF CHEMICAL INFORMATION AND MODELING (AMER CHEMICAL SOC, 1155 16TH ST, NW, WASHINGTON, USA, DC, 20036) pp. 1463-1474 - issn: 1549-9596 - wos: WOS:000321074700019 (7) - scopus: 2-s2.0-84879596019 (10)

11573/516522 - 2013 - New promising compounds with in vitro nanomolar activity against Trypanosoma cruzi
Friggeri, Laura; Scipione, Luigi; Costi, Roberta; Marcel, Kaiser; Francesca, Moraca; Claudio, Zamperini; Botta, Bruno; Di Santo, Roberto; De Vita, Daniela; Reto, Brun; Tortorella, Silvano - 01a Articolo in rivista
paper: ACS MEDICINAL CHEMISTRY LETTERS (USA: ACS Publications) pp. 538-541 - issn: 1948-5875 - wos: WOS:000321883900011 (14) - scopus: 2-s2.0-84879097485 (15)

11573/507015 - 2013 - CONVENIENT ROUTE TO 2H-PYRROLO [3,4-b]QUINOLIN-9(4H)-ONE SKELETON VIA TOSMIC REACTION
Rosi, Federica; Cuzzucoli Crucitti, Giuliana; Alberto, Iacovo; Gaetano, Miele; Pescatori, Luca; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: SYNTHETIC COMMUNICATIONS (New York, NY : Marcel Dekker) pp. 1063-1072 - issn: 1532-2432 - wos: WOS:000313418700015 (6) - scopus: 2-s2.0-84872326307 (6)

11573/485737 - 2012 - Design, Synthesis, and Structure−Activity Relationship of N‑Arylnaphthylamine Derivatives as Amyloid Aggregation Inhibitors
Di Santo, Roberto; Costi, Roberta; Cuzzucoli Crucitti, Giuliana; Pescatori, Luca; Rosi, Federica; Scipione, Luigi; Diana, Celona; Mario, Vertechy; Orlando, Ghirardi; Paola, Piovesan; Mauro, Marzi; Silvio, Caccia; Giovanna, Guiso; Fabrizio, Giorgi; Patrizia, Minetti - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 8538-8548 - issn: 0022-2623 - wos: WOS:000309643500030 (23) - scopus: 2-s2.0-84867382314 (26)

11573/457568 - 2012 - Effects of polyphenol compounds on influenza A virus replication and definition of their mechanism of action
Fioravanti, Rossella; Celestino, Ignacio; Costi, Roberta; Cuzzucoli Crucitti, Giuliana; Pescatori, Luca; Mattiello, Leonardo; Ettore, Novellino; Paola, Checconi; Palamara, Anna Teresa; Nencioni, Lucia; Di Santo, Roberto - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 5046-5052 - issn: 0968-0896 - wos: WOS:000307244300020 (38) - scopus: 2-s2.0-84864471453 (42)

11573/482226 - 2012 - Polyphenols as anti-influenza A agents.
Fioravanti, Rossella; Celestino, Ignacio; Costi, Roberta; Cuzzucoli G., Crucitti; Pescatori, Luca; Checconi, Paola; Palamara, Anna Teresa; Nencioni, Lucia; Di Santo, Roberto - 04a Atto di comunicazione a congresso
conference: 21st National Meeting on Medicinal Chemistry. (Palermo, Italy)
book: 21st National Meeting on Medicinal Chemistry. - ()

11573/488191 - 2012 - Discovery and Pharmacological Profile of New 1H‑Indazole-3- carboxamide and 2H‑Pyrrolo[3,4‑c]quinoline Derivatives as SelectiveSerotonin 4 Receptor Ligands
Guido, Furlotti; Maria Alessandra, Alisi; Claudia, Apicella; Alessandra Capezzone De, Joannon; Nicola, Cazzolla; Costi, Roberta; Cuzzucoli Crucitti, Giuliana; Beatrice, Garrone; Alberto, Iacovo; Gabriele, Magaro ; Giorgina, Mangano; Gaetano, Miele; Rosella, Ombrato; Pescatori, Luca; Lorenzo, Polenzani; Federica, Rosi; Marco, Vitiello; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 9446-9466 - issn: 0022-2623 - wos: WOS:000311461500006 (31) - scopus: 2-s2.0-84870052595 (31)

11573/455694 - 2012 - Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells
Valente, Sergio; Ilaria, Lepore; Carmela, Dell'aversa; Maria, Tardugno; Sabrina, Castellano; Gianluca, Sbardella; Stefano, Tomassi; Salvatore Di, Maro; Ettore, Novellino; Di Santo, Roberto; Costi, Roberta; Lucia, Altucci; Mai, Antonello - 01a Articolo in rivista
paper: BIOCHIMIE (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 2308-2313 - issn: 0300-9084 - wos: WOS:000310929200011 (22) - scopus: 2-s2.0-84867395419 (26)

11573/414595 - 2011 - Novel 3,5-bis(bromohydroxybenzylidene)piperidin-4-ones as coactivator-associated arginine methyltransferase 1 inhibitors: Enzyme selectivity and cellular activity
Donghang, Cheng; Valente, Sergio; Sabrina, Castellano; Gianluca, Sbardella; Di Santo, Roberto; Costi, Roberta; Mark T., Bedford; Mai, Antonello - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 4928-4932 - issn: 0022-2623 - wos: WOS:000292479600049 (64) - scopus: 2-s2.0-79960191524 (69)

11573/123490 - 2010 - Evaluation of HIV-1 integrase inhibitors on human primary macrophages using a luciferase-based single-cycle phenotypicassay
Zuleikamichelini, Clementinamariagalluzzo; Negri, D. O. N. A. T. E. L. L. A. R. M.; Pasqualinaleone, Robertaamici; Robertabona, Vincenzosumma; Di Santo, Roberto; Costi, Roberta; Yvespommier, Christophemarchand; Luciapalmisano, Stefanovella; Andreacara, - 01a Articolo in rivista
paper: JOURNAL OF VIROLOGICAL METHODS (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598) pp. 272-276 - issn: 0166-0934 - wos: WOS:000280869400047 (15) - scopus: 2-s2.0-77955092239 (16)

11573/368166 - 2009 - Studio dell’attività antivirale di analoghi del resveratrolo in un modello sperimentale in vitro di infezione da virus influenzale A.
Celestino, Ignacio; Nencioni, Lucia; Di Santo, Roberto; Costi, Roberta; Garaci, E; Palamara, Anna Teresa - 04a Atto di comunicazione a congresso
book: 37° Congresso della Società Italiana di Microbiologia SIM, 11-14 ottobre 2009 pg. 70 - ()

11573/229129 - 2009 - A rational approach to predict and modulate stereolability of chiral alpha-substituted ketones.
Cirilli, R.; Costi, Roberta; Di Santo, Roberto; Gasparrini, Francesco; La Torre, F.; Pierini, Marco; Siani, G. - 01a Articolo in rivista
paper: CHIRALITY (John Wiley & Sons Incorporated:Customer Service, 111 River Street:Hoboken, NJ 07030:(800)225-5945, (201)748-6000, EMAIL: societyinfo@wiley.com, INTERNET: http://www.wiley.com, Fax: (212)748-6551) pp. 24-34 - issn: 0899-0042 - wos: WOS:000261782900006 (15) - scopus: 2-s2.0-59849121710 (15)

11573/227936 - 2009 - Perturbing Effects of Chiral Stationary Phase on Enantiomerization Second-Order Rate Constants Determined by Enantioselective Dynamic High-Performance Liquid Chromatography: A Practical Tool to Quantify the Accessible Acid and Basic Catalytic Sites Bonded on Chromatographic Supports
Roberto, Cirilli; Costi, Roberta; Di Santo, Roberto; Francesco La, Torre; Pierini, Marco; Gabriella, Siani - 01a Articolo in rivista
paper: ANALYTICAL CHEMISTRY (Washington: American Chemical Society, ©1948-) pp. 3560-3570 - issn: 0003-2700 - wos: WOS:000265632400049 (37) - scopus: 2-s2.0-66149097413 (38)

11573/359251 - 2008 - Novel quinolinonyl diketo acid derivatives as HIV-1 integrase inhibitors: Design, synthesis, and biological activities
Di Santo, Roberto; Costi, Roberta; Alessandra, Roux; Gaetano, Miele; Giuliana Cuzzucoli, Crucitti; Alberto, Iacovo; Federica, Rosi; Antonio, Lavecchia; Luciana, Marinelli; Carmen Di, Giovanni; Ettore, Novellino; Lucia, Palmisano; M., Andreaotti; Roberta, Amici; Clementina Maria, Galluzzo; Nencioni, Lucia; Palamara, Anna Teresa; Yves, Pommier; Christophe, Marchand - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 4744-4750 - issn: 0022-2623 - wos: WOS:000258289800043 (49) - scopus: 2-s2.0-49449093292 (53)

11573/122770 - 2008 - Simple synthesis of deuterated pterosines
Gaetano, Miele; Costi, Roberta; Bonadies, Francesco; Rosario, Nicoletti - 01a Articolo in rivista
paper: SYNTHETIC COMMUNICATIONS (New York, NY : Taylor & Francis New York, NY: Marcel Dekker Incorporated) pp. 1553-1559 - issn: 0039-7911 - wos: WOS:000256530800007 (3) - scopus: 2-s2.0-42549109034 (3)

11573/230766 - 2008 - Synthesis and cerebral uptake of 1-(1-[11C]methyl-1H-pyrrol-2-yl)-2-phenyl-2-(1-pyrrolidinyl)ethanone a novel tracer for positron emission tomography studies of monoamine oxidase type A
S. B., Jensen; Di Santo, Roberto; A. K., Olsen; K., Pedersen; Costi, Roberta; R., Cirilli; P., Cumming - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1617-1622 - issn: 0022-2623 - wos: WOS:000254209800011 (12) - scopus: 2-s2.0-41249095463 (10)

11573/228663 - 2008 - HIV-1 Integration: A Potential Target for Microbicides to Prevent Cell-free or Cell-associated Human Immunodeficiency Virus type-1 Infection
Terrazas Aranda, K; Van Herrewege, Y; Hazuda, D; Lewi, P; Costi, Roberta; Di Santo, Roberto; Cara, A; Vanham, G. - 01a Articolo in rivista
paper: ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (American Society for Microbiology:PO Box 11127:Birmingham, AL 35201:(800)633-4931, (205)995-1567, EMAIL: asm.nonmembers.subs@ebsco.com, INTERNET: http://www.asm.org, Fax: (205)995-1588) pp. 2544-2554 - issn: 0066-4804 - wos: WOS:000257183400036 (21) - scopus: 2-s2.0-46249087616 (21)

11573/241523 - 2007 - Probing HIV-1 integrase inhibitor binding sites with position-specific integrase-DNA cross-linking assays
Allison A., Johnson; Christophe, Marchand; Sachindra S., Patil; Costi, Roberta; Di Santo, Roberto; Terrence R., Burke; Yves, Pommier - 01a Articolo in rivista
paper: MOLECULAR PHARMACOLOGY (American Society for Pharmacology and Experimental Therapeutics:9650 Rockville Pike:Bethesda, MD 20814:(301)530-7024, EMAIL: pstoute@aspet.org, INTERNET: http://www.aspet.org, Fax: (301)634-7099) pp. 893-901 - issn: 0026-895X - wos: WOS:000244290400029 (29) - scopus: 2-s2.0-33847098825 (34)

11573/241076 - 2007 - Cynnamoyl compounds as simple molecules that inhibit p300 histone acetyltransferase
Costi, Roberta; Di Santo, Roberto; Artico, Marino; G., Miele; P., Valentini; E., Novellino; A., Cereseto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1973-1977 - issn: 0022-2623 - wos: WOS:000245634500025 (63) - scopus: 2-s2.0-34247281570 (65)

11573/240552 - 2007 - HIV-1 integrase inhibitors are substrates for the multidrug transporter MDR1-P-glycoprotein
M., Cianfriglia; M. L., Dupuis; A., Molinari; A., Verdoliva; Costi, Roberta; C. M., Galluzzo; M., Andreotti; A., Cara; Di Santo, Roberto; L., Palmisano - 01a Articolo in rivista
paper: RETROVIROLOGY (London : BioMed Central) pp. 17-27 - issn: 1742-4690 - wos: WOS:000245096500002 (24) - scopus: 2-s2.0-42049093456 (23)

11573/236938 - 2006 - Arylthiopyrrole (AThP) Derivatives as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors. Synthesis, Structure-Activity Relationships and Docking Studies. Part 1.
Di Santo, Roberto; Costi, Roberta; Artico, Marino; Miele, Gaetano; A., Lavecchia; E., Novellino; A., Bergamini; R., Cancio; G., Maga - 01a Articolo in rivista
paper: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. 1367-1378 - issn: 1860-7179 - wos: WOS:000202946500008 (32) - scopus: 2-s2.0-33846262498 (35)

11573/46567 - 2006 - Arylthiopyrrole (ATP) Derivatives as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors
Di Santo, Roberto; Costi, Roberta; Artico, Marino; Miele, Gaetano; A., Lavecchia; E., Novellino; A., Bergamini; R., Cancio; G., Maga - 01a Articolo in rivista
paper: DRUGS OF THE FUTURE (Prous Science Publishers:Provenza 388, 08025 Barcelona Spain:011 34 3 4592220, EMAIL: service@prous.com, INTERNET: http://www.prous.com, Fax: 011 34 3 4581535) pp. 77-77 - issn: 0377-8282 - wos: (0) - scopus: (0)

11573/237779 - 2006 - Design, Synthesis, Biological Evaluation, and Molecular Modeling Studies on TIBO-Like Cyclic Sulfones as Novel Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors
Di Santo, Roberto; Costi, Roberta; Artico, Marino; Ragno, Rino; Lavecchia, A.; Novellino, E.; Gavuzzo, E.; La Torre, F.; Cirilli, R.; Cancio, R.; Maga, G. - 01a Articolo in rivista
paper: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. 82-95 - issn: 1860-7179 - wos: WOS:000202945500013 (19) - scopus: 2-s2.0-33746322348 (22)

11573/46568 - 2006 - Diketo hexenoic acid (DKHA) derivatives: the first class of selective non-nucleoside inhibitors of mammalian terminal deoxynucleotidyl transferases endowed with cytotoxic effect against leukemic cells
Di Santo, Roberto; Costi, Roberta; G., Miele; G., Maga; U., Hbscher - 01a Articolo in rivista
paper: DRUGS OF THE FUTURE (Prous Science Publishers:Provenza 388, 08025 Barcelona Spain:011 34 3 4592220, EMAIL: service@prous.com, INTERNET: http://www.prous.com, Fax: 011 34 3 4581535) pp. 84-84 - issn: 0377-8282 - wos: (0) - scopus: (0)

11573/46569 - 2006 - Novel Curcumin Derivatives as p300 Histone Acetyltransferases inhibitors
Di Santo, Roberto; Costi, Roberta; Miele, Gaetano; P., Valentini; A., Cereseto - 01a Articolo in rivista
paper: DRUGS OF THE FUTURE (Prous Science Publishers:Provenza 388, 08025 Barcelona Spain:011 34 3 4592220, EMAIL: service@prous.com, INTERNET: http://www.prous.com, Fax: 011 34 3 4581535) pp. 130-130 - issn: 0377-8282 - wos: (0) - scopus: (0)

11573/233551 - 2006 - Novel bifunctional quinolonyl diketo acid derivatives as HIV-1 integrase inhibitors: Design, synthesis, biological activities, and mechanism of action
Di Santo, Roberto; Costi, Roberta; Roux, A; Artico, M; Lavecchia, A; Marinelli, L; Novellino, E; Palmisano, L; Andreotti, M; Amici, R; Galluzzo C., M; Nencioni, Lucia; Palamara, Anna Teresa; Pommier, Y; Marchand, C. - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1939-1945 - issn: 0022-2623 - wos: WOS:000236400100013 (74) - scopus: 2-s2.0-33645405333 (92)

11573/210965 - 2006 - HIV-1 Integrase Inhibitors are potent substrates for the MDR1 multidrug transporter.
M. L., Dupuis; M., Cianfriglia; Costi, Roberta; C., Galluzzo; M., Andreotti; A., Roux; Di Santo, Roberto; L., Palmisano - 04a Atto di comunicazione a congresso
book: 13th Conferente on Retroviruses and Opportunistic Infection (CROI) - ()

11573/236444 - 2006 - Development of a human immunodeficiency virus vector-based, single-cycle assay for evaluation of anti-integrase compounds
R., Bona; M., Andreotti; V., Buffa; P., Leone; C. M., Galluzzo; R., Amici; L., Palmisano; M. G., Mancini; Z., Michelini; Di Santo, Roberto; Costi, Roberta; A., Roux; Y., Pommier; C., Marchand; S., Vella; A., Cara - 01a Articolo in rivista
paper: ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (American Society for Microbiology:PO Box 11127:Birmingham, AL 35201:(800)633-4931, (205)995-1567, EMAIL: asm.nonmembers.subs@ebsco.com, INTERNET: http://www.asm.org, Fax: (205)995-1588) pp. 3407-3417 - issn: 0066-4804 - wos: WOS:000241021700026 (18) - scopus: 2-s2.0-33749515634 (19)

11573/364346 - 2005 - Antifungal agents. 11. N-substituted derivatives of 1-[(aryl)(4-aryl-1H-pyrrol-3-yl)methyl]-1H-imidazole: Synthesis, anti-Candida activity, and QSAR studies
Di Santo, Roberto; A., Tafi; Costi, Roberta; M., Botta; M., Artico; F., Corelli; M., Forte; F., Caporuscio; Angiolella, Letizia; Palamara, Anna Teresa - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 5140-5153 - issn: 0022-2623 - wos: WOS:000231055300011 (115) - scopus: 2-s2.0-23444446586 (130)

11573/46290 - 2005 - 2H-Pyrrolo[3,4-b][1,5] benzothiazepine derivatives as potential inhibitors of HIV-1 reverse transcriptase
Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: IL FARMACO (Attuale:ELSEVIER SCIENCE SA, PO BOX 564, LAUSANNE, SWITZERLAND, 1001 Societa Chimica Italiana:Viale Liegi 48, 00198 Rome Italy:011 39 06 8549691, EMAIL: soc.chim.it@agora.stm.it, Fax: 011 39 06 8548734) pp. 385-392 - issn: 0014-827X - wos: (0) - scopus: 2-s2.0-19444387692 (46)

11573/210963 - 2005 - Quinolinyl-2,4-dioxobutanoic Acids as HIV-1 Integrase Inhibitors: SAR Studies and Binding Mode.
Di Santo, Roberto; Costi, Roberta; A., Roux; M., Artico; A., Lavecchia; E., Novellino; L., Palmisano; C., Galluzzo; M., Andreotti; S., Vella; Nencioni, Lucia; A., Palamara; C., Marchand; Y., Pommier - 04a Atto di comunicazione a congresso
book: Second Joint Italian-Swiss Meeting on Medicinal Chemistry - ()

11573/210964 - 2005 - Diketo Hexenoic Acid (DKHA) Derivatives as Non-Nucleoside Inhibitors of Mammalian Terminal Deoxynucleotidyl Transferases.
Di Santo, Roberto; Costi, Roberta; A., Roux; M., Artico; E., Crespan; G. A., Locatelli; U., Hbscher; K., Ramadan; I., Shevelev; S., Spadari; G., Maga - 04a Atto di comunicazione a congresso
book: Second Joint Italian-Swiss Meeting on Medicinal Chemistry - ()

11573/210949 - 2005 - Docking Studies on Bifunctional Quinolinyl Diketo Acids as HIV-1 Integrase Ihnhibitors.
Di Santo, Roberto; Costi, Roberta; A., Roux; M., Forte; M., Artico; A., Lavecchia; E., Novellino; L., Palmisano; C., Galluzzo; M., Andreotti; S., Vella; Nencioni, Lucia; A., Palamara; C., Marchand; Y., Pommier - 01a Articolo in rivista
paper: SCIENTIA PHARMACEUTICA (Oesterr Apotheker Verlags GES:Spitalgasse 31, A-1094 Vienna Austria:011 43 1 4023588) pp. 115-115 - issn: 0036-8709 - wos: (0) - scopus: (0)

11573/210960 - 2005 - SAR Studies on Quinolinyl-2,4-Dioxobutanoic Acids, HIV-1 Integrase Inhibitors that Block HIV-1 Replication in Infected Cells.
Di Santo, Roberto; Costi, Roberta; A., Roux; M., Forte; M., Artico; A., Lavecchia; E., Novellino; L., Palmisano; C., Galluzzo; M., Andreotti; S., Vella; Nencioni, Lucia; A., Palamara; C., Marchand; Y., Pommier - 04a Atto di comunicazione a congresso
book: Joint Meeting on Medicinal Chemistry - ()

11573/210962 - 2005 - 2,4-Dioxo-5-hexenoic Acid Derivatives Are Novel Selective Non-Nucleoside Inhibitors of Mammalian Terminal Deoxynucleotidyl Transferases, with Potent Cytotoxic Effect Against Leukemic Cells.
Di Santo, Roberto; Costi, Roberta; A., Roux; M., Forte; M., Artico; E., Crespan; G. A., Locatelli; U., Hbscher; K., Ramadan; I., Shevelev; S., Spadari; G., Maga - 04a Atto di comunicazione a congresso
book: Joint Meeting on Medicinal Chemistry - ()

11573/506757 - 2005 - Design, synthesis, and biological activities of pyrrolylethanoneamine derivatives, a novel class of monoamine oxidases inhibitors
Di Santo, Roberto; Costi, Roberta; Alessandra, Roux; Artico, Marino; Olivia, Befani; Tiziana, Meninno; Agostinelli, Enzo; Paola, Palmegiani; Paola, Turini; Roberto, Cirilli; Rosella, Ferretti; Bruno, Gallinella; Francesco La, Torre - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 4220-4223 - issn: 0022-2623 - wos: WOS:000230121800007 (26) - scopus: 2-s2.0-21244505103 (35)

11573/46061 - 2005 - Regioselectivity of the methyl-TosMIC reaction with substituted ethyl cinnamates
Di Santo, Roberto; Costi, Roberta; Galeffi, C; Forte, M. - 01a Articolo in rivista
paper: ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL (Organic Preparations and Procedures Incorporated:PO Box 610009:Newton Highlands, MA 02161:(617)287-6130, EMAIL: jp.anselme@umb.edu, Fax: (617)287-6030) pp. 110-115 - issn: 0030-4948 - wos: WOS:000228891700003 (2) - scopus: 2-s2.0-19344371166 (2)

11573/210959 - 2005 - Sintesi, saggi enzimatici e attività antivirale di nuovi inibitori dell’integrasi di HIV.
Di Santo, Roberto; Costi, Roberta; M., Artico; A., Roux; M., Forte; G., Miele; A., Palamara; Y., Pommier; C., Marchand; L., Palmisano; M., Andreotti; M. C., Galluzzo; Nencioni, Lucia; E., Novellino - 04a Atto di comunicazione a congresso
book: Fifth National Research Program on AIDS Progress Report,. - ()

11573/239790 - 2005 - Design, synthesis and biological evaluation of heteroaryl diketohexenoic and diketobutanoic acids as HIV-1 integrase inhibitors endowed with antiretroviral activity
Di Santo, Roberto; Costi, Roberta; M., Artico; Ragno, Rino; R., Greco; G., Novellino; E., Marchand; C., Pommier - 01a Articolo in rivista
paper: IL FARMACO (Attuale:ELSEVIER SCIENCE SA, PO BOX 564, LAUSANNE, SWITZERLAND, 1001 Societa Chimica Italiana:Viale Liegi 48, 00198 Rome Italy:011 39 06 8549691, EMAIL: soc.chim.it@agora.stm.it, Fax: 011 39 06 8548734) pp. 409-417 - issn: 0014-827X - wos: (0) - scopus: 2-s2.0-19544380093 (36)

11573/210961 - 2005 - Discovery of Novel Anti-Malarial Agents: 1-[(Aryl)(4-aryl-1H-pyrrol-3-yl)methyl]-1H-imidazoles Targeted to Farnesyl Transferase.
Di Santo, Roberto; Costi, Roberta; M., Forte; C., Galeffi; M., Artico; C., Peters; H., Waldmann; R., Brun - 04a Atto di comunicazione a congresso
book: Joint Meeting on Medicinal Chemistry - ()

11573/210947 - 2005 - Synthesis and Biological Evaluation of Curcumine Analogues as Apoptosis-Inducing Agents.
Di Santo, Roberto; Costi, Roberta; Miele, Gaetano; Artico, Marino; S., Grimaudo; A., Di Cristina; M., Tolomeo - 04a Atto di comunicazione a congresso
book: Joint Meeting on Medicinal Chemistry - ()

11573/210948 - 2005 - Design, Synthesis and Biological Activities of Pyrrolylethanoneamine Derivatives, a Novel Class of MAO Inhibitors.
Di Santo, Roberto; Costi, Roberta; Roux, A.; Artico, M.; Befani, O.; Agostinelli, E.; Turini, P.; Palmegiani, P.; Meninno, T.; La Torre, F.; Cirilli, R.; Ferretti, R.; Gallinella, B. - 04a Atto di comunicazione a congresso
book: Joint Meeting on Medicinal Chemistry - ()

11573/211198 - 2005 - Diaryl Imidazolyl Methanes and Ethanes as Monoamine Oxidase Inhibitors.
Di Santo, Roberto; Costi, Roberta; Roux, A.; Artico, M.; Befani, O.; Agostinelli, E.; Turini, P.; Palmegiani, P.; Meninno, T.; La Torre, F.; Cirilli, R.; Ferretti, R.; Gallinella, B. - 04a Atto di comunicazione a congresso
book: Second Joint Italian-Swiss Meeting on Medicinal Chemistry - ()

11573/238404 - 2005 - Simple but highly effective three-dimensional chemical-feature-based pharmacophore model for diketo acid derivatives as hepatitis C virus RNA-dependent RNA polymerase inhibitors
Di Santo, Roberto; Maurizio, Fermeglia; Marco, Ferrone; Maria Silvia, Paneni; Costi, Roberta; Artico, Marino; Alessandra, Roux; Mirko, Gabriele; Keith D., Tardif; Aleem, Siddiqui; Sabrina, Pricl - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 6304-6314 - issn: 0022-2623 - wos: WOS:000232406600015 (41) - scopus: 2-s2.0-26444491094 (42)

11573/237889 - 2005 - 6-(1-(4-fluorophenyl)methyl-1H-pyrrol-2-yl))-2,4-dioxo-5-hexenoic acid ethyl ester a novel diketo acid derivative which selectively inhibits the HIV-1 viral replication in cell culture and the ribonuclease H activity in vitro
E., Tramontano; F., Esposito; R., Badas; Di Santo, Roberto; Costi, Roberta; P., La Colla - 01a Articolo in rivista
paper: ANTIVIRAL RESEARCH ([Amsterdam]; [New York]: Elsevier/North-Holland, [c1981]-) pp. 117-124 - issn: 0166-3542 - wos: WOS:000227261900007 (118) - scopus: 2-s2.0-13544276913 (127)

11573/234366 - 2005 - Diketo hexenoic acid derivatives are novel selective non-nucleoside inhibitors of mammalian terminal deoxynucleotidyl transferases, with potent cytotoxic effect against leukemic cells
G. A., Locatelli; Di Santo, Roberto; E., Crespan; Costi, Roberta; A., Roux; U., Hbscher; I., Shevelev; G., Blanca; G., Villani; S., Spadai; G., Maga - 01a Articolo in rivista
paper: MOLECULAR PHARMACOLOGY (American Society for Pharmacology and Experimental Therapeutics:9650 Rockville Pike:Bethesda, MD 20814:(301)530-7024, EMAIL: pstoute@aspet.org, INTERNET: http://www.aspet.org, Fax: (301)634-7099) pp. 538-550 - issn: 0026-895X - wos: WOS:000230549900031 (13) - scopus: 2-s2.0-23044491841 (14)

11573/189716 - 2004 - Studio di una nuova classe di derivati pirrol-imidazolici: attività antimicotica e modulazione delle proteine di parete di Candida Albicans.
Angiolella, Letizia; Ciocci, A.; Bonito, M.; Di Santo, Roberto; Costi, Roberta; Forte, Michela; Artico, Marino; Palamara, Anna Teresa - 04a Atto di comunicazione a congresso
book: 1° Congresso Nazionale Società Italiana di Microbiologia Farmaceutica - ()

11573/231135 - 2004 - 6-Aryl-2,4-dioxo-5-hexenoic Acids, Novel Integrase Inhibitors Active Against HIV-1 Multiplication in Cell-Based Assays.
Costi, Roberta; Di Santo, Roberto; Artico, Marino; A., Roux; Ragno, Rino; S., Massa; E., Tramontano; M., La Colla; R., Loddo; M. E., Marongiu; A., Pani; P., La Colla - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 1745-1749 - issn: 0960-894X - wos: WOS:000220411200029 (40) - scopus: 2-s2.0-12144288755 (44)

11573/365225 - 2004 - 2,6-Bis(3,4,5-trihydroxybenzylydene) derivatives of cyclohexanone: novel potent HIV-1 integrase inhibitors that prevent HIV-1 multiplication in cell-based assays
Costi, Roberta; Di Santo, Roberto; Artico, Marino; S., Massa; Ragno, Rino; R., Loddo; M., La Colla; E., Tramomtano; P., La Colla; A., Pani - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 199-215 - issn: 0968-0896 - wos: WOS:000188113400021 (81) - scopus: 2-s2.0-0347301799 (84)

11573/210721 - 2004 - Acidi 6-aril-2,4-dioxo-5-esenoici come inibitori della NS5B polimerasi dell'HCV.
Di Santo, Roberto; Costi, Roberta; A., Roux; Artico, Marino; G., Maga; K., Tardif; A., Siddiqui - 04a Atto di comunicazione a congresso
book: XVII Convegno Nazionale della Divisione di Chimica Farmaceutica della SCI. - ()

11573/210944 - 2004 - Acidi chinolinil-2,4-dioxobutanoici come analoghi conformazionalmente ristretti dei derivati arildichetoesenoici, dotati di potente attività anti-integrasi del virus HIV-1.
Di Santo, Roberto; Costi, Roberta; A., Roux; M., Artico; Ragno, Rino; G., Greco; E., Novellino; C., Marchand; Y., Pommier - 04a Atto di comunicazione a congresso
book: XVII Convegno Nazionale della Divisione di Chimica Farmaceutica della SCI. - ()

11573/210945 - 2004 - 6-Aryl-2,4-dioxo-5-hexenoic acids, Novel HCV NS5b Polymerase Inhibitors.
Di Santo, Roberto; Costi, Roberta; M., Artico; A., Roux; G., Maga; K., Tardif; A., Siddiqui - 04a Atto di comunicazione a congresso
book: COST D28 MC Action, Natural Products as a Source for Discovery, Synthesis, and Application of New Ph - ()

11573/210958 - 2004 - 1[(Aryl)(4-aryl-1H-pyrrol-3-yl)methyl]-1H-imidazoles: a Class of Potent Antifungal Agents. SAR Studies of N-1 Substituted Derivatives.
Di Santo, Roberto; Costi, Roberta; M., Forte; Artico, Marino; Angiolella, Letizia; Palamara, Anna Teresa - 04a Atto di comunicazione a congresso
book: COST D28 MC Action, Natural Products as a Source for Discovery, Synthesis, and Application of New Ph - ()

11573/236844 - 2004 - A General, Versatile Synthesis of 2H-Pyrrolo[3,4-c]quinolines via Tosylmethylisocyanide Reaction
Di Santo, Roberto; Costi, Roberta; M., Forte; C., Galeffi - 01a Articolo in rivista
paper: ARKIVOC (ARKAT USA INC, C/O ALAN R KATRITZKY, UNIV FLORIDA, DEPT CHEMISTRY, PO BOX 117200, GAINESVILLE, USA, FL, 32611) pp. 181-195 - issn: 1551-7004 - wos: (0) - scopus: 2-s2.0-2942694389 (12)

11573/210942 - 2004 - Derivati 1-[(aril)(1(5)-aril-1H-pirrol-2(3)-il)metil]-1H-imidazolici ad attività antifungina.
Di Santo, Roberto; Costi, Roberta; M., Forte; M., Artico; Angiolella, Letizia; A. T., Palamara - 04a Atto di comunicazione a congresso
book: XVII Convegno Nazionale della Divisione di Chimica Farmaceutica della SCI. - ()

11573/210943 - 2004 - 1-((Aril)(4-aril-1H-pirrol-3-il)metil)-1H-imidazoli: studio della relazioni struttura-attività di derivati sostituiti in posizione 1 dell'anello pirrolico.
Di Santo, Roberto; Costi, Roberta; M., Forte; M., Artico; Angiolella, Letizia; Palamara, Anna Teresa - 04a Atto di comunicazione a congresso
book: XVII Convegno Nazionale della Divisione di Chimica Farmaceutica della SCI. - ()

11573/210946 - 2004 - Quinolinyl 2,4-dioxobutanoic Acids, Conformationally Restrained Analogues of Aryldioxohexenoic Acids as HIV-1 Integrase Inhibitors.
Di Santo, Roberto; Costi, Roberta; Roux, Alessandra; Artico, Marino; Ragno, Rino; G., Greco; E., Novellino; C., Marchand; Y., Pommier - 04a Atto di comunicazione a congresso
book: COST D28 MC Action, Natural Products as a Source for Discovery, Synthesis, and Application of New Ph - ()

11573/46059 - 2004 - Enantiomers of new synthetic pyrrolylethanoneamine mono-amino oxidase inhibitor compounds: analytical and semipreparative HPLC separations, and chiroptical characteristics
La Torre, F.; Cirilli, R.; Costi, Roberta; Di Santo, Roberto; Ferretti, R.; Gallinella, B.; Salerno, A.; Zanitti, L. - 01a Articolo in rivista
paper: CHROMATOGRAPHIA (Heidelberg ; Berlin : Springer) pp. 171-178 - issn: 0009-5893 - wos: (0) - scopus: (0)

11573/210706 - 2003 - Derivati Fenilpirroliletanonamminici analoghi del Kathinone dotati di potente e selettiva attività anti-MAO-A.
Agostinelli, Enzo; Turini, P.; Befani, O.; Martone, A.; Di Santo, Roberto; Costi, Roberta; Artico, Marino; Roux, A.; La Torre, F.; Ferretti, R.; Gallinella, B.; Cirilli, R. - 04a Atto di comunicazione a congresso
book: XXI Congresso Nazionale della Società Chimica Italiana - ()

11573/253348 - 2003 - Phenylpyrrolylethanoneamines related to kathinone, endowed with potent and highly selective anti-MAO-A activity.
Agostinelli, Enzo; Turini, P.; Befani, O.; Martone, A.; Di Santo, Roberto; Costi, Roberta; Artico, Marino; Roux, Alessandra; La Torre, F.; Ferretti, R.; Gallinella, B.; Cirilli, R. - 04a Atto di comunicazione a congresso
book: 8th International Congress on Amino Acids and Proteins - ()

11573/253007 - 2003 - Caratterizzazione dell’attività antimicotica di una nuova classe di derivati pirrol-imidazolici
Angiolella, Letizia; A., Ciocci; M. V., Pasceri; Di Santo, Roberto; Costi, Roberta; M., Forte; M., Artico; Palamara, Anna Teresa - 04a Atto di comunicazione a congresso
book: 31° Congresso Nazionale Società Italiana di Microbiologia, - ()

11573/210926 - 2003 - Studies of enantiomerization barrier of 2-[2-(1-methyl-1H-pyrrol-2-yl)-2-oxo-1-phenylethyl]-isoindole-1,3-dione by enantioselective stopped-flow HPLC.
Cirilli, R.; Costi, Roberta; Di Santo, Roberto; Ferretti, R.; La Torre, F.; Gallinella, B.; Salerno, A. - 04a Atto di comunicazione a congresso
book: XXI Congresso Nazionale della Società Chimica Italiana - ()

11573/46054 - 2003 - Enantioselective liquid Chromatography of C3-chiral 2,3-dihydro-1,2,5-benzothiadiazepin-4(5H)-one and thione 1,1-dioxides on polyacrylamide- and polysaccaride-based chiral stationary phases
Cirilli, R; Costi, Roberta; Di Santo, Roberto; Artico, Marino; Roux, A; Gallinella, B; Zanitti, L; La Torre, F. - 01a Articolo in rivista
paper: JOURNAL OF CHROMATOGRAPHY A (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598) pp. 17-28 - issn: 0021-9673 - wos: WOS:000182174600002 (29) - scopus: 2-s2.0-0037453478 (33)

11573/46053 - 2003 - HIV-1 Integrase Inhibitors that Block HIV-1 Replication in Infected Cells. Planning Synthetic Derivatives from Natural Products
Di Santo, Roberto; Costi, Roberta; Artico, Marino; Tramontano, E; La Colla, P; Pani, A. - 01a Articolo in rivista
paper: PURE AND APPLIED CHEMISTRY (Editore attuale:INT UNION PURE APPLIED CHEMISTRY, 104 TW ALEXANDER DR, PO BOX 13757, RES TRIANGLE PK, USA, NC, 27709-3757 Blackwell Science Limited:PO Box 88, Oxford OX2 0NE United Kingdom:011 44 1865 776868, 011 44 1865 206038, EMAIL: journals.cs@blacksci.co.uk, INTERNET: http://www.blackwell-science.com, Fax: 011 44 1865 721205) pp. 195-206 - issn: 0033-4545 - wos: WOS:000182416500007 (16) - scopus: 2-s2.0-0037317788 (23)

11573/210707 - 2003 - Acidi 6-Aril-2,4-dioxo-5-esenoici, Nuovi Inibitori dell’Integrasi. Blocco la Replicazione dell’HIV-1 in Cellule Infettate.
Di Santo, Roberto; Costi, Roberta; M., Artico; A., Roux; Ragno, Rino; F., Esposito; L., Onidi; M., Marongiu; M., Atzori; P., La Colla - 04a Atto di comunicazione a congresso
book: XXI Congresso Nazionale della Società Chimica Italiana - ()

11573/210950 - 2003 - 1-[(Aril)(4-aril-1H-pirrol-3-il)metil]-1H-imidazoli: Effetti della Sostituzione all'Azoto Pirrolico sull'Attività anti-Candida.
Di Santo, Roberto; Costi, Roberta; M., Forte; Artico, Marino; Angiolella, Letizia; G., Gigante; M. V., Pasceri; Palamara, Anna Teresa - 04a Atto di comunicazione a congresso
book: XXI Congresso Nazionale della Società Chimica Italiana - ()

11573/210956 - 2003 - Studi SAR su Derivati 2H-Pirrolo[3,4-c]chinolinici quali Potenti e Selettivi Ligandi per i Recettori 5-HT4.
Di Santo, Roberto; Costi, Roberta; M., Forte; M., Artico; C., Saturnino; G., De Martino; F., Dauphin; J. C., Lancelot; S., Rault - 04a Atto di comunicazione a congresso
book: XXI Congresso Nazionale della Società Chimica Italiana - ()

11573/255461 - 2003 - Conversion of a Racemic Mixture of 8-Chloro-2-(2,6-difluorophenylmethyl)-2,3-dihydro-3-methyl-1,2,5-benzothiadiazepin-4(5H)-one 1,1-Dioxide into a Single Enantioemer Via a Chromatographic Resolution/Racemization Method
La Torre, F.; Cirilli, R.; Ferretti, R.; Gallinella, B.; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: CHIRALITY (John Wiley & Sons Incorporated:Customer Service, 111 River Street:Hoboken, NJ 07030:(800)225-5945, (201)748-6000, EMAIL: societyinfo@wiley.com, INTERNET: http://www.wiley.com, Fax: (212)748-6551) pp. 429-432 - issn: 0899-0042 - wos: WOS:000182518000007 (5) - scopus: 2-s2.0-0037277248 (6)

11573/255869 - 2002 - Antifungal Agents. 10. New Derivatives of 1-[(Aryl)[4-aryl-1H-pyrrol-3-yl]methyl]-1H-imidazole, Synthesis, Anti-Candida Activity, and Quantitative Structure-Activity Relationship Studies
A., Tafi; Costi, Roberta; M., Botta; Di Santo, Roberto; F., Corelli; S., Massa; A., Ciacci; F., Manetti; M., Artico - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 2720-2732 - issn: 0022-2623 - wos: WOS:000176204300005 (88) - scopus: 2-s2.0-0037142376 (96)

11573/47152 - 2002 - Derivatives of 2,3-dihydroimidazo[1,5,4-ef][1,2,5]benzothiadiazepin-6(4H,7H)-thione 1,1-dioxide, a new heterocyclic system related to TIBO
Costi, Roberta; Di Santo, Roberto; M., Artico; S., Massa - 01a Articolo in rivista
paper: JOURNAL OF HETEROCYCLIC CHEMISTRY (Hetero Corporation:PO Box 170:Provo, UT 84603:(801)400-7373, EMAIL: jhetchem@yahoo.com, Fax: (801)356-7373) pp. 81-90 - issn: 0022-152X - wos: WOS:000174926800011 (9) - scopus: 2-s2.0-0036185075 (12)

11573/194615 - 2002 - Probing the activity of diketoacids as HCV NS5B polymerase inhibitors via detailed molecular modeling
Di Santo, Roberto; Costi, Roberta; Artico, M; Fermeglia, M; Ferrone, M; Lodi, A; Manfredini, S; Pricl, S. - 04a Atto di comunicazione a congresso
book: 23rd IUPAC - 2002 International Symposium on the Chemistry of Natural Products - ()

11573/194623 - 2002 - Progettazione, Sintesi ed Attività Biologica di 2H-Pirrolo[3,4-c]chinoline, una Nuova Classe di Ligandi Selettivi per i Recettori 5-HT4
Di Santo, Roberto; Costi, Roberta; Artico, M; Forte, M; Satunino, C; De Martino, G; Dauphin, F; Lancelot J., C; Rault, S. - 04a Atto di comunicazione a congresso
book: XVI Convegno Nazionale di Chimica Farmaceutica - ()

11573/194613 - 2002 - Design, Synthesis And Biological Evaluation of 2H-Pyrrolo[3,4-c]quinolines, a New Class of Potent 5-HT4 Ligands.
Di Santo, Roberto; Costi, Roberta; Artico, M; Forte, M; Saturnino, C; De Martino, G; Dauphin, F; Lancelot, J. C.; Rault, S. - 04a Atto di comunicazione a congresso
book: 2ème Congès Combiné de Pharmacochimie - ()

11573/194611 - 2002 - Nuove Classi di Inibitori dell’Integrasi dell’HIV-1 che Bloccano la Replicazione Virale in Cellule Infettate
Di Santo, Roberto; Costi, Roberta; Artico, M; Tramontano, E; La Colla, P; Pani, A. - 04a Atto di comunicazione a congresso
book: XVI Convegno Nazionale di Chimica Farmaceutica - ()

11573/194832 - 2002 - 1-[Aril-(1-aril-1H-pirrol-3-il)metil]-1H-imidazoli, una Nuova Classe di Potenti Inibitori della Farnesiltrasferasi
Di Santo, Roberto; Costi, Roberta; Artico, Marino; Roux, A; Sattler, I. - 04a Atto di comunicazione a congresso
book: XVI Convegno Nazionale di Chimica Farmaceutica - ()

11573/194610 - 2002 - HIV-1 Integrase Inhibitors That Block HIV-1 Replication in Infected Cells: Planning Synthetic Derivatives from Natural Products.
Di Santo, Roberto; Costi, Roberta; Artico, Marino; Tramontano, E; La Colla, P; Pani, A. - 04a Atto di comunicazione a congresso
book: 23rd IUPAC - 2002 International Symposium on the Chemistry of Natural Products - ()

11573/189704 - 2002 - 1-Alchil-3-aril-4[_-(1H-imidazol-1-il)arilmetil]pirroli: una Nuova Classe di Potenti Agenti Anti-Candida
Di Santo, Roberto; Costi, Roberta; Forte, Michela; Artico, Marino; Angiolella, Letizia; Gigante, G.; Pasceri, M. V.; Palamara, Anna Teresa - 04a Atto di comunicazione a congresso
book: 30° Congresso Nazionale Società Italiana di Microbiologia - ()

11573/46051 - 2002 - Design, synthesis and QSAR studies on N-aryl heteroarylisopropanolamines, a new class of non-peptidic HIV-1 protease inhibitors
Di Santo, Roberto; Costi, Roberta; Marino, Artico; Silvio, Massa; Ragno, Rino; G. R., Marshall; P., La Colla - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 2511-2526 - issn: 0968-0896 - wos: WOS:000176294500009 (32) - scopus: 2-s2.0-0036286615 (42)

11573/252637 - 2002 - ARYLTHIOPYRIDYLMETHYLISOPROPYLPYRROLE CARBINOLS, NOVEL NNRTIs ENDOWED WITH POTENT ANTI-HIV-1 ACTIVITY
Di Santo, Roberto; Costi, Roberta; Marino, Artico; Silvio, Massa; Ragno, Rino; Massimiliano La, Colla; Roberta, Loddo; Paolo La, Colla; Alessandra, Pani - 01a Articolo in rivista
paper: MEDICINAL CHEMISTRY RESEARCH (Birkhauser Boston Incorporated:c/o Springer Verlag, PO Box 2485:Secaucus, NJ 07096:(800)777-4643, (973)348-4033, Fax: (973)348-4505) pp. 153-167 - issn: 1054-2523 - wos: WOS:000176370900002 (7) - scopus: 2-s2.0-0036056712 (7)

11573/194609 - 2001 - 3,4,5-Trihydroxycynnamoyl moiety: a Potent Pharmacophore for Anti-Integrase Agents Active Either in Enzymatic or in Cell-Based Assays.
Artico, M; Di Santo, Roberto; Costi, Roberta; Massa, S; Murgioni, C; Setzu, M. G.; Loddo, R; Serra, I. - 04a Atto di comunicazione a congresso
book: Third National Research Program on AIDS Progress Report - ()

11573/254828 - 2001 - 1-[4-(4-Chlorophenyl)-1H-pyrrol-3-yl](2,4-dichlorophenyl)methyl-1H-imidazole (RDS 416)
Camalli, M.; Pifferi, A.; Costi, Roberta; Di Santo, Roberto; Massa, S.; Artico, Marino - 01a Articolo in rivista
paper: ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE (Pubblicata da BLACKWELL MUNKSGAARD, 35 NORRE SOGADE, PO BOX 2148, COPENHAGEN, DENMARK, DK-1016) pp. 096-098 - issn: 1600-5368 - wos: (0) - scopus: (0)

11573/125012 - 2001 - Analytical and semipreparative enantiomeric separation of azole antifungal agents by high-performance liquid chromatography on polysaccharide-based chiral stationary phases Application to in vitro biological studies
Cirilli, R.; Costi, R.; Di Santo, R.; Ferretti, R.; La Torre, F.; Angiolella, L.; Micocci, M. - 01a Articolo in rivista
paper: JOURNAL OF CHROMATOGRAPHY A (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598) pp. 107-114 - issn: 0021-9673 - wos: WOS:000173120900010 (18) - scopus: 2-s2.0-0037016285 (19)

11573/194612 - 2001 - Arylthiopyrroles (ATPs) A New Class of Potent NNRTIs Active either Against HIV-1 WT or Resistant Strains.
Costi, Roberta; Artico, M; Di Santo, Roberto; Massa, S; Piacciau, A; Serra, I; La Colla, P; Loddo, R. - 04a Atto di comunicazione a congresso
book: Hungarian-German-Italian-Polish Joint Meeting on Medicinal Chemistry - ()

11573/254827 - 2000 - Structure-activity relationship studies on potential non-nucleoside DABO-like inhibitors of HIV-1 reverse transcriptase.
Costi, Roberta; Di Santo, Roberto; Artico, Marino; Massa, S.; La Vecchia, A.; Marceddu, T.; Sanna, L.; La Colla, P.; Marongiu, M. E. - 01a Articolo in rivista
paper: ANTIVIRAL CHEMISTRY & CHEMOTHERAPY (International Medical Press:2-4 Idol Lane, London EC3R 5DD United Kingdom:011 44 207 3980700, EMAIL: imp@intmedpress.com, INTERNET: http://www.intmedpress.com, Fax: 011 44 207 3980701) pp. 117-133 - issn: 0956-3202 - wos: WOS:000086782000004 (14) - scopus: 2-s2.0-0034017027 (13)

11573/194608 - 2000 - Derivati del 2H-pirrolo[3,4-c]chinolin-4(5H)-one: Nuovi Potenziali Agonisti dei Recettori 5-HT3
Costi, Roberta; Di Santo, Roberto; Artico, Marino; Massa, Silvio; De Martino, G.; Saturnino, C. - 04a Atto di comunicazione a congresso
book: XX Congresso Nazionale della Società Chimica Italiana (SCI 2000) - ()

11573/249530 - 2000 - Antimycobacterial Pyrroles: Synthesis, Anti-Mycobacterium tuberculosis Activity and QSAR Studies.
Ragno, Rino; Marshall, G. R.; Di Santo, Roberto; Costi, Roberta; Massa, S.; Pompei, R.; Artico, Marino - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 1423-1432 - issn: 0968-0896 - wos: WOS:000087742300019 (138) - scopus: 2-s2.0-0034131292 (145)

11573/244906 - 1999 - Pyridinylpyrrolyl Analogs of Isoniazid: Synthesis and Antimycobacterial Activities.
Costi, Roberta; Artico, Marino; Di Santo, Roberto; De Martino, G.; Massa, S.; Deidda, D.; Lampis, G.; Pompei, R. - 01a Articolo in rivista
paper: MEDICINAL CHEMISTRY RESEARCH (Birkhauser Boston Incorporated:c/o Springer Verlag, PO Box 2485:Secaucus, NJ 07096:(800)777-4643, (973)348-4033, Fax: (973)348-4505) pp. 408-423 - issn: 1054-2523 - wos: WOS:000084511600004 (3) - scopus: 2-s2.0-0033399508 (2)

11573/194595 - 1999 - 3,4,5-Trioxycinnamoyl Moiety: a Potent Pharmacophore for anti-HIV-1 Integrase Activity either in Enzyme or in Cell-Based Assays.
Di Santo, Roberto; Costi, Roberta; Artico, M.; Massa, S.; Novellino, E.; Greco, G.; Tramontano, E.; Marceddu, T.; Serra, I.; La Colla, P. - 04a Atto di comunicazione a congresso
book: Italian-Hungarian-Polish Joint Meeting on Medicinal Chemistry - ()

11573/244226 - 1999 - Structure Based Design of N-aryl-heteroarylpropanolamines, a new class of simple HIV-1 Protease Inhibitors
Di Santo, Roberto; Costi, Roberta; Artico, M.; Massa, S.; Ragno, Rino; Vargiu, L.; Demontis, F.; Sanna, L.; Lostia, S.; La Colla, P. - 04a Atto di comunicazione a congresso
book: Italian – hungarian – Polish Joint Meeting on Medicinal Chemistry - ()

11573/194597 - 1999 - Trihydroxy-cinnamoyl derivatives targeted at the integrase inhibit the HIV-1 multiplication in cell-based assays
Marceddu, T.; Di Santo, Roberto; Costi, Roberta; Artico, M.; La Colla, P. - 04a Atto di comunicazione a congresso
book: Second National program on AIDS Progress Repor - ()

11573/194594 - 1999 - Different kinetics of inhibition of the HIV-1 integrase activities by different classes of derivatives.
Tramontano, E.; Marceddu, T.; Di Santo, Roberto; Costi, Roberta; Artico, M.; La Colla, P. - 04a Atto di comunicazione a congresso
book: Italian-Hungarian-Polish Joint Meeting on Medicinal Chemistry - ()

11573/194601 - 1998 - 3D QSAR and Molecular Modeling on a Set of New Anti Mycobacterial Compounds.
Artico, M.; Di Santo, Roberto; Costi, Roberta; Massa, S.; Marshall, G. R.; Ragno, Rino - 04a Atto di comunicazione a congresso
book: Second research project on Tuberculosis (1998) Progress report - ()

11573/247184 - 1998 - Geometrically and Conformationally Restrained Cinnamoyl-Compounds as Inhibitors of HIV-1 Integrase: Synthesis, Biological Evaluation and Molecular Modeling
Artico, Marino; Di Santo, Roberto; Costi, Roberta; Novellino, E.; Greco, G.; Massa, S.; Tramontano, E.; Marongiu, M. E.; De Montis, A.; La Colla, P: - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 3948-3960 - issn: 0022-2623 - wos: WOS:000076374300005 (170) - scopus: 2-s2.0-15144355755 (169)

11573/43958 - 1998 - 1,2,5-Benzothiadiazepine and Pyrrolo[2,1-d][1,2,5]Benzothiadiazepine Derivatives with Anti-HIV-1 Activity.
Di Santo, Roberto; Costi, Roberta; Artico, M.; Massa, S.; Marongiu, M. E.; Loi, A. G.; Putzolu, M.; La Colla, P. - 01a Articolo in rivista
paper: ANTIVIRAL CHEMISTRY & CHEMOTHERAPY (International Medical Press:2-4 Idol Lane, London EC3R 5DD United Kingdom:011 44 207 3980700, EMAIL: imp@intmedpress.com, INTERNET: http://www.intmedpress.com, Fax: 011 44 207 3980701) pp. 127-137 - issn: 0956-3202 - wos: WOS:000072685800004 (35) - scopus: 2-s2.0-0031954544 (39)

11573/194599 - 1998 - Synthesis and Antimycobacterial Activities of Pyrrole Derivatives Related to Pyrrolnitrin.
Di Santo, Roberto; Costi, Roberta; Artico, M.; Massa, S.; Maullu, C.; Deidda, D.; Pompei, R. - 04a Atto di comunicazione a congresso
book: XIV CONVEGNO NAZIONALE Divisione di Chimica Farmaceutica SCI - ()

11573/194598 - 1998 - SAR Studies on 1-Alkyl-3-aryl-4-[a-(1H-imidazol-1-yl)arylmethyl]pyrroles a Class of Potent Anti-Candida Agents.
Di Santo, Roberto; Costi, Roberta; Artico, M.; Massa, S.; Vargiu, L.; Congiu, D.; Musiu, C.; La Colla, P. - 04a Atto di comunicazione a congresso
book: XIV CONVEGNO NAZIONALE Divisione di Chimica Farmaceutica SCI - ()

11573/245377 - 1998 - Pyrrolnitrin and Related Pyrroles Endowed with Antibacterial Activities against Mycobacterium Tuberculosis.
Di Santo, Roberto; Costi, Roberta; Artico, Marino; Massa, S.; Lampis, G.; Deidda, D.; Pompei, R. - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 2931-2936 - issn: 0960-894X - wos: (0) - scopus: (0)

11573/243326 - 1998 - ARYLSULFONYL PYRROLES FROM REACTION OF TOSYLMETHYL ISOCIANIDE (TOSMIC) WITH 3-ARYLSULFONYL ACRYLATES AS MICHAEL ACCEPTORS.
Di Santo, Roberto; Costi, Roberta; Massa, S.; Artico, M. - 01a Articolo in rivista
paper: SYNTHETIC COMMUNICATIONS (New York, NY : Taylor & Francis New York, NY: Marcel Dekker Incorporated) pp. 1801-1815 - issn: 0039-7911 - wos: (0) - scopus: 2-s2.0-0031807811 (9)

11573/247003 - 1998 - PYRROLE-ANNULATED HETEROCYCLIC SYSTEMS. SYNTHESIS OF 2H-PYRROLO[3,4-b][1,5]BENZOTHIAZEPINE 4,4-DIOXIDE DERIVATIVES
Di Santo, Roberto; Costi, Roberta; Massa, S.; Artico, M. - 01a Articolo in rivista
paper: SYNTHETIC COMMUNICATIONS (New York, NY : Taylor & Francis New York, NY: Marcel Dekker Incorporated) pp. 2517-2530 - issn: 0039-7911 - wos: (0) - scopus: (0)

11573/245262 - 1997 - 1-Arylsulfonyl-3-(a-hydroxybenzyl)-1H-pyrroles, a novel class of anti-HIV-1 reverse transcriptase inhibitors.
Artico, M.; Di Santo, Roberto; Costi, Roberta; Massa, S.; Scintu, F.; Loi, A. G.; De Montis, A.; La Colla, P. - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Oxford: Pergamon, Amsterdam the Netherlands: Elsevier) pp. 1931-1936 - issn: 0960-894X - wos: WOS:A1997XP63900026 (13) - scopus: 2-s2.0-0030804024 (12)

11573/194604 - 1997 - Synthesis of Curcumin-like Derivatives with Potent Activity Against the HIV-1 Integrase.
Artico, M.; Di Santo, Roberto; Costi, Roberta; Massa, S.; Tramontano, E.; Putzolu, M.; Fadda, D.; La Colla, P. - 04a Atto di comunicazione a congresso
book: First Italian-Swiss meeting on Medicinal Chemistry - ()

11573/244912 - 1997 - N-(1-Naphthylmethyl)-N-(1-alkyl-4-aryl-1H-pyrrol-3-ylmethyl)methylamines Related to Naftifine. Synthesis and Antifungal Activity.
Di Santo, Roberto; Costi, Roberta; Artico, M.; Massa, S.; Musiu, C.; Milia, C.; Putzolu, M.; La Colla, P. - 01a Articolo in rivista
paper: MEDICINAL CHEMISTRY RESEARCH (Birkhauser Boston Incorporated:c/o Springer Verlag, PO Box 2485:Secaucus, NJ 07096:(800)777-4643, (973)348-4033, Fax: (973)348-4505) pp. 98-108 - issn: 1054-2523 - wos: (0) - scopus: 2-s2.0-0003066751 (4)

11573/194606 - 1997 - Pyrrolo[2,1-d][1,2,5]benzothiadiazepine derivatives with anti-HIV-1 activity.
Di Santo, Roberto; Costi, Roberta; Artico, M.; Massa, S.; Puddu, I.; Corrias, S.; Loi, A. G.; La Colla, P. - 04a Atto di comunicazione a congresso
book: Ninth research project on AIDS (1996) Progress report - ()

11573/245525 - 1997 - Antifungal estrogen-like imidazoles. Synthesis and antifungal activities of thienyl and 1H-pyrrolyl derivatives of 1-aryl-2-(1H-imidazol-1-yl)ethane.
Di Santo, Roberto; Costi, Roberta; Artico, Marino; Massa, S.; Musiu, C.; Scintu, F.; Putzolu, M.; La Colla, P. - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 143-149 - issn: 0223-5234 - wos: (0) - scopus: (0)

11573/245204 - 1997 - Heterocycles with a benzothiadiazepine moiety .5. Derivatives of pyrrolo[2,1-d][1,2,5]benzothiadiazepine, a novel tricyclic ring
Di Santo, Roberto; Costi, Roberta; Marino, Artico; Silvio, Massa - 01a Articolo in rivista
paper: IL FARMACO (Attuale:ELSEVIER SCIENCE SA, PO BOX 564, LAUSANNE, SWITZERLAND, 1001 Societa Chimica Italiana:Viale Liegi 48, 00198 Rome Italy:011 39 06 8549691, EMAIL: soc.chim.it@agora.stm.it, Fax: 011 39 06 8548734) pp. 375-378 - issn: 0014-827X - wos: WOS:A1997YD01000006 (9) - scopus: 2-s2.0-0030665610 (13)

11573/122334 - 1996 - Molecular Modeling of Azole Antifungal Agents Active.Againts Candida Albicans.I: a CoMFA Study.
A., Tafi; Y., Anastassopoulou; T., Theophanides; M., Botta; F., Corelli; Artico, Marino; Costi, Roberta; Di Santo, Roberto; S., Massa; Ragno, Rino - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1227-1235 - issn: 0022-2623 - wos: WOS:A1996UA57700006 (60) - scopus: 2-s2.0-13344282738 (66)

11573/194607 - 1996 - Aryl-(1-benzenesulfonyl-1H-pyrrol-3yl)-carbinols: a new class of non-nucleoside inhibitors of HIV-1 RT.
Di Santo, Roberto; Costi, Roberta; Artico, M.; Massa, S.; Putzolu, M.; Puddu, I.; Pinna, N.; La Colla, P. - 04a Atto di comunicazione a congresso
book: XIII Convegno Nazionale Divisione di Chimica Farmaceutica SCI - ()

11573/242453 - 1996 - Novel pyrrole-annulated heterocyclic systems. Synthesis of 10H-pyrrolo[1,2-b][1,2,6]benzothiadiazocin-11(12H)-one 5,5-dioxide.
Di Santo, Roberto; Costi, Roberta; M., Artico; Massa, S. - 01a Articolo in rivista
paper: JOURNAL OF HETEROCYCLIC CHEMISTRY (Hetero Corporation:PO Box 170:Provo, UT 84603:(801)400-7373, EMAIL: jhetchem@yahoo.com, Fax: (801)356-7373) pp. 2019-2023 - issn: 0022-152X - wos: WOS:A1996WE32000073 (5) - scopus: 2-s2.0-2742517067 (9)

11573/246926 - 1996 - Synthesis of Pyrrolo[3,4-c][1]benzazepine-4,10(2H,5H)-dione, a Model System Useful for the Design of 11-Oxosibiromycinone Analogues.
Di Santo, Roberto; Costi, Roberta; Massa, S.; Artico, M. - 01a Articolo in rivista
paper: SYNTHETIC COMMUNICATIONS (New York, NY : Taylor & Francis New York, NY: Marcel Dekker Incorporated) pp. 1839-1847 - issn: 0039-7911 - wos: (0) - scopus: 2-s2.0-0029952695 (13)

11573/244100 - 1995 - Antifungal Agents. 9. 3-Aryl-4-[a-(1H-imidazol-1-yl)arylmethyl]pyrroles: A New Class of Potent Anti-Candida Agents.
Artico, M.; Di Santo, Roberto; Costi, Roberta; Massa, S.; Retico, Augusta; Artico, M.; Apuzzo, G.; Simonetti, Giovanna; Strippoli, V. - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 4223-4233 - issn: 0022-2623 - wos: WOS:A1995TA40700011 (46) - scopus: 2-s2.0-0028791168 (49)

11573/44023 - 1995 - Novel Heterocyclic Systems. Synthesis of 10H-Pyrrolo[1,2-b][1,2,5]benzothiadiazocine 5,5-Dioxide and Related Derivatives.
Di Santo, Roberto; Costi, Roberta; Artico, M.; Massa, S. - 01a Articolo in rivista
paper: JOURNAL OF HETEROCYCLIC CHEMISTRY (Hetero Corporation:PO Box 170:Provo, UT 84603:(801)400-7373, EMAIL: jhetchem@yahoo.com, Fax: (801)356-7373) pp. 1779-1782 - issn: 0022-152X - wos: WOS:A1995TQ34800019 (6) - scopus: 2-s2.0-84993876560 (8)

11573/44025 - 1995 - Simple Synthetic Approach to Arylacetic NSAIAs via TosMIC Procedure.
Di Santo, Roberto; Costi, Roberta; Massa, S.; Artico, M. - 01a Articolo in rivista
paper: SYNTHETIC COMMUNICATIONS (New York, NY : Taylor & Francis New York, NY: Marcel Dekker Incorporated) pp. 787-793 - issn: 0039-7911 - wos: (0) - scopus: 2-s2.0-0028837973 (6)

11573/255643 - 1995 - 4-Substituted 2-phenyl- and 2-phenyl-3-aryl pyrroles by reaction of tosylbenzyl isocyanide (TosBIC) with Michael acceptors.
Di Santo, Roberto; Costi, Roberta; Massa, S.; M., Artico - 01a Articolo in rivista
paper: SYNTHETIC COMMUNICATIONS (New York, NY : Taylor & Francis New York, NY: Marcel Dekker Incorporated) pp. 795-802 - issn: 0039-7911 - wos: (0) - scopus: 2-s2.0-0028799586 (12)

11573/253762 - 1994 - ANTIFUNGAL AGENTS .8. SYNTHESIS AND ANTIFUNGAL ACTIVITIES OF BIPYRRYL ANALOGS OF BIFONAZOLE
Di Santo, Roberto; Silvio, Massa; Costi, Roberta; Simonetti, Giovanna; Retico, Augusta; G., Apuzzo; F., Troccoli - 01a Articolo in rivista
paper: IL FARMACO (Attuale:ELSEVIER SCIENCE SA, PO BOX 564, LAUSANNE, SWITZERLAND, 1001 Societa Chimica Italiana:Viale Liegi 48, 00198 Rome Italy:011 39 06 8549691, EMAIL: soc.chim.it@agora.stm.it, Fax: 011 39 06 8548734) pp. 229-236 - issn: 0014-827X - wos: WOS:A1994NN69600001 (8) - scopus: 2-s2.0-0028361653 (12)

11573/44027 - 1994 - Synthesis of Novel HEPT Analogues with Anti-HIV-1 Activity.
Massa, S.; Di Santo, Roberto; Costi, Roberta; Artico, M.; Loi, A. G.; Doa, M.; Scano, P.; La Colla, P. - 01a Articolo in rivista
paper: MEDICINAL CHEMISTRY RESEARCH (Birkhauser Boston Incorporated:c/o Springer Verlag, PO Box 2485:Secaucus, NJ 07096:(800)777-4643, (973)348-4033, Fax: (973)348-4505) pp. 554-562 - issn: 1054-2523 - wos: (0) - scopus: (0)

11573/44268 - 1993 - Antifungal Agents. 5. Chloro and Amino Derivatives of 1,2-Diaryl-1-(1H-imidazol-1-yl)ethane with Potent Antifungal Activities.
Artico, M.; Massa, S.; Di Santo, Roberto; Costi, Roberta; Retico, Augusta; Apuzzo, G.; Simonetti, N. - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 715-720 - issn: 0223-5234 - wos: WOS:A1993MC71600008 (9) - scopus: 2-s2.0-0027449161 (10)

11573/47093 - 1993 - Research on Nitrogen Containing Heterocyclic Compounds. XX. Synthesis of 8H-Imidazo[5,1-c]pyrrolo[1,2-a][1,4]benzodiazepine and its 6-Derivatives.
Massa, S.; Di Santo, Roberto; Costi, Roberta; Artico, M. - 01a Articolo in rivista
paper: JOURNAL OF HETEROCYCLIC CHEMISTRY (Hetero Corporation:PO Box 170:Provo, UT 84603:(801)400-7373, EMAIL: jhetchem@yahoo.com, Fax: (801)356-7373) pp. 749-753 - issn: 0022-152X - wos: WOS:A1993LL38300025 (8) - scopus: 2-s2.0-0343779409 (9)

11573/247026 - 1993 - Antifungal Agents. 4. Synthesis of neo-Isopyrrolnitrin and other 3-Aryl-4-nitro-1H-pyrroles via TosMIC.
Massa, S; Di Santo, Roberto; Costi, Roberta; Mai, Antonello; Artico, M; Retico, A; Apuzzo, G; Artico, M; Simonetti, Giovanna - 01a Articolo in rivista
paper: MEDICINAL CHEMISTRY RESEARCH (Birkhauser Boston Incorporated:c/o Springer Verlag, PO Box 2485:Secaucus, NJ 07096:(800)777-4643, (973)348-4033, Fax: (973)348-4505) pp. 192-199 - issn: 1054-2523 - wos: (0) - scopus: (0)

11573/470052 - 1993 - Antifungal agents. III. Naphthyl and thienyl derivatives of 1H-imidazol-1-yl-4-phenyl-1H-pyrrol-3-ylmethane.
Massa, S; Di Santo, Roberto; Costi, Roberta; Simonetti, Giovanna; Retico, Augusta; Apuzzo, G; Artico, Marco - 01a Articolo in rivista
paper: IL FARMACO (Attuale:ELSEVIER SCIENCE SA, PO BOX 564, LAUSANNE, SWITZERLAND, 1001 Societa Chimica Italiana:Viale Liegi 48, 00198 Rome Italy:011 39 06 8549691, EMAIL: soc.chim.it@agora.stm.it, Fax: 011 39 06 8548734) pp. 725-736 - issn: 0014-827X - wos: WOS:A1993LQ31800002 (8) - scopus: 2-s2.0-0027170720 (7)

11573/47097 - 1992 - Novel In Vitro Highly Active Antifungal Agents With Pyrrole and Imidazole Moieties.
Massa, S.; Di Santo, Roberto; Artico, Marco; Costi, Roberta; Apuzzo, G.; Simonetti, Giovanna; Artico, M. - 01a Articolo in rivista
paper: MEDICINAL CHEMISTRY RESEARCH (Birkhauser Boston Incorporated:c/o Springer Verlag, PO Box 2485:Secaucus, NJ 07096:(800)777-4643, (973)348-4033, Fax: (973)348-4505) pp. 148-153 - issn: 1054-2523 - wos: (0) - scopus: (0)

11573/47098 - 1992 - Researches on Antibacterial and Antifungal Agents. XV. 3-Aryl-4-[a-(1H-imidazol-1-yl)benzyl]pyrroles with Potent Antifungal Activity.
Massa, S.; Di Santo, Roberto; Retico, Augusta; Costi, Roberta; Di Filippo, C.; Simonetti, Giovanna; Retico, A.; Artico, M. - 01a Articolo in rivista
paper: EUROPEAN BULLETIN OF DRUG RESEARCH (Firenze: Europharma 2000.) pp. 12-17 - issn: 1122-2441 - wos: (0) - scopus: (0)

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