11573/1663401 - 2023 -
Inhibition of Leishmania infantum Trypanothione Reductase by New Aminopropanone Derivatives Interacting with the NADPH Binding Site Madia, Valentina Noemi; Ialongo, Davide; Patacchini, Elisa; Antonelli, Lorenzo; Colotti, Gianni; Messore, Antonella; Tudino, Valeria; Saccoliti, Francesco; Scipione, Luigi; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: MOLECULES (Basel: MDPI
Berlin: Springer, 1996-) pp. 338- - issn: 1420-3049 - wos: WOS:000909976300001 (0) - scopus: 2-s2.0-85145692255 (0)
11573/1668131 - 2023 -
Pyrrolyl and indolyl α-γ-diketo acid derivatives acting as selective inhibitors of human carbonic anhydrases IX and XII Ialongo, Davide; Messore, Antonella; Madia, Valentina Noemi; Tudino, Valeria; Supuran, Claudiu Trandafir; Nicolai, Alice; Scarpa, Susanna; Taurone, Samanta; Camarda, Michele; Artico, Marco; Saccoliti, Francesco; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. - - issn: 1424-8247 - wos: (0) - scopus: (0)
11573/1623281 - 2022 -
Oxidative stress and visual system a review Taurone, Samanta; Ralli, Massimo; Artico, Marco; Madia, Valentina Noemi; Scarpa, Susanna; Nottola, Stefania Annarita; Familiari, Pietro; Nebbioso, Marcella; Costi, Roberta - 01g Articolo di rassegna (Review)
paper: EXCLI JOURNAL (Mainz: EXCLI Journal Business Office c/o 2nd Medical Department, University of Mainz.) pp. 544-553 - issn: 1611-2156 - wos: WOS:000766811300001 (5) - scopus: 2-s2.0-85125850235 (5)
11573/1623472 - 2022 -
The kinesin Eg5 inhibitor K858 exerts antiproliferative and proapoptotic effects and attenuates the invasive potential of head and neck squamous carcinoma cells Nicolai, Alice; Taurone, Samanta; Artico, Marco; Greco, Antonio; Costi, Roberta; Scarpa, Susanna - 01a Articolo in rivista
paper: INVESTIGATIONAL NEW DRUGS (attuale:
-SPRINGER, VAN GODEWIJCKSTRAAT 30, DORDRECHT, NETHERLANDS, 3311 GZ
-Kluwer Academic Publishers / Massachusetts:PO Box 358, Accord Station:Hingham, MA 02018:(617)871-6600) pp. - - issn: 0167-6997 - wos: WOS:000771319900002 (2) - scopus: 2-s2.0-85126822611 (2)
11573/1638210 - 2022 -
Synthesis and evaluation of the antifungal and toxicological activity of Nitrofuran derivatives Pandolfi, Fabiana; De Vita, Daniela; Bortolami, Martina; Tudino, Valeria; Costi, Roberta; Scipione, Luigi - 01a Articolo in rivista
paper: PHARMACEUTICS (Basel: MDPI, 2009-) pp. 1-19 - issn: 1999-4923 - wos: WOS:000774275300001 (1) - scopus: 2-s2.0-85126453264 (1)
11573/1638214 - 2022 -
Evaluation of the Anti-Histoplasma capsulatum activity of Indole and Nitrofuran derivatives and their pharmacological safety in three-dimensional cell cultures Pandolfi, Fabiana; De Vita, Daniela; Bortolami, Martina; Tudino, Valeria; Costi, Roberta; Di Santo, Roberto; Scipione, Luigi - 01a Articolo in rivista
paper: PHARMACEUTICS (Basel: MDPI, 2009-) pp. 1-23 - issn: 1999-4923 - wos: WOS:000803586100001 (0) - scopus: 2-s2.0-85130346777 (0)
11573/1638218 - 2022 -
Design, synthesis, and In vitro, in silico and in cellulo evaluation of new Pyrimidine and Pyridine amide and Carbamate derivatives as multi-functional Cholinesterase Inhibitors Bortolami, Martina; Pandolfi, Fabiana; Tudino, Valeria; Messore, Antonella; Madia, Valentina Noemi; De Vita, Daniela; Di Santo, Roberto; Costi, Roberta; Romeo, Isabella; Scipione, Luigi - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. 1-31 - issn: 1424-8247 - wos: WOS:000818156100001 (1) - scopus: 2-s2.0-85134396743 (1)
11573/1648549 - 2022 -
Ultrastructural damages to H1N1 influenza virus caused by vapor essential oils Madia, Valentina Noemi; Toscanelli, Walter; De Vita, Daniela; De Angelis, Marta; Messore, Antonella; Ialongo, Davide; Scipione, Luigi; Tudino, Valeria; D'auria, Felicia Diodata; Di Santo, Roberto; Garzoli, Stefania; Nencioni, Lucia; Costi, Roberta - 01a Articolo in rivista
paper: MOLECULES (Basel: MDPI
Berlin: Springer, 1996-) pp. 1-14 - issn: 1420-3049 - wos: WOS:000816243700001 (2) - scopus: 2-s2.0-85131746075 (2)
11573/1654141 - 2022 -
New Inhibitors of the human p300/CBP acetyltransferase are selectively active against the Arabidopsis HAC proteins Longo, Chiara; Lepri, Andrea; Messore, Antonella; De Vita, Daniela; Bonaccorsi Di Patti, Maria Carmela; Amadei, Matteo; Madia, Valentina Noemi; Ialongo, Davide; Di Santo, Roberto; Costi, Roberta; Vittorioso, Paola - 01a Articolo in rivista
paper: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (Basel: MDPI Center) pp. 1-18 - issn: 1422-0067 - wos: WOS:000859422800001 (0) - scopus: 2-s2.0-85138734584 (0)
11573/1662952 - 2022 -
Exosomal Functional Cargoes from Liquid Biopsy of Gastric Cancer: A Systematic Review of Studies With Potential Clinical Relevance Virgilio, Edoardo; Giarnieri, Enrico; Montagnini, Monica; Proietti, Antonella; D'urso, Rosaria; Costi, Roberta - 01a Articolo in rivista
paper: ANTICANCER RESEARCH (Kapandriti: International Institute of Anticancer Research, 1995
Earliest publisher: Καπανδρίτι: Ιωάννης Γ. Δεληνάσιος, 1981-1995
Kapandriti: Iōannīs G. Delīnasios, 1981-1995) pp. 2249-2259 - issn: 0250-7005 - wos: WOS:000795123200003 (2) - scopus: 2-s2.0-85129187422 (2)
11573/1404920 - 2021 -
Towards a new application of amaranth seed oil as an agent against Candida albicans De Vita, Daniela; Messore, Antonella; Toniolo, Chiara; Frezza, Claudio; Scipione, Luigi; Madia, Valentina Noemi; Pindinello, Ivano; Simonetti, Giovanna; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: NATURAL PRODUCT RESEARCH (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 4621-4626 - issn: 1478-6419 - wos: WOS:000500457200001 (13) - scopus: 2-s2.0-85075913942 (5)
11573/1490818 - 2021 -
Acetylcholinesterase inhibitors for the treatment of Alzheimer’s disease–a patent review (2016–present) Bortolami, Martina; Rocco, Daniele; Messore, Antonella; Di Santo, Roberto; Costi, Roberta; Madia, Valentina Noemi; Scipione, Luigi; Pandolfi, Fabiana - 01a Articolo in rivista
paper: EXPERT OPINION ON THERAPEUTIC PATENTS (--London United Kingdom:Informa Healthcare
-London, United Kingdom: Ashley Publications Limited) pp. 1-22 - issn: 1354-3776 - wos: WOS:000607685400001 (21) - scopus: 2-s2.0-85099470810 (23)
11573/1493998 - 2021 -
Design, synthesis and biological evaluation of new pyrimidine derivatives as anticancer agents Madia, Valentina Noemi; Nicolai, Alice; Messore, Antonella; De Leo, Alessandro; Ialongo, Davide; Tudino, Valeria; Saccoliti, Francesco; De Vita, Daniela; Scipione, Luigi; Artico, Marco; Taurone, Samanta; Taglieri, Ludovica; Di Santo, Roberto; Scarpa, Susanna; Costi, Roberta - 01a Articolo in rivista
paper: MOLECULES (Basel: MDPI
Berlin: Springer, 1996-) pp. - - issn: 1420-3049 - wos: WOS:000615455300001 (8) - scopus: 2-s2.0-85101195321 (9)
11573/1540215 - 2021 -
Investigation of Commiphora myrrha (Nees) Engl. oil and its main components for antiviral activity Madia, Valentina Noemi; De Angelis, Marta; De Vita, Daniela; Messore, Antonella; De Leo, Alessandro; Ialongo, Davide; Tudino, Valeria; Garzoli, Stefania; Scipione, Luigi; Palamara, Anna Teresa; Di Santo, Roberto; Nencioni, Lucia; Costi, Roberta - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. - - issn: 1424-8247 - wos: WOS:000634055800001 (10) - scopus: 2-s2.0-85102987115 (11)
11573/1540619 - 2021 -
Analytical characterization of an inulin-type fructooligosaccharide from root-tubers of Asphodelus ramosus L Madia, Valentina Noemi; De Vita, Daniela; Messore, Antonella; Toniolo, Chiara; Tudino, Valeria; De Leo, Alessandro; Pindinello, Ivano; Ialongo, Davide; Saccoliti, Francesco; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. - - issn: 1424-8247 - wos: WOS:000634075100001 (2) - scopus: 2-s2.0-85103099178 (2)
11573/1546419 - 2021 -
Design, synthesis and biological evaluation of a series of iron and copper chelating deferiprone derivatives as new agents active against Candida albicans Bortolami, Martina; Pandolfi, Fabiana; Messore, Antonella; Rocco, Daniele; Feroci, Marta; Di Santo, Roberto; De Vita, Daniela; Costi, Roberta; Simonetti, Giovanna; Scipione, Luigi - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. 1-7 - issn: 0960-894X - wos: WOS:000655255700006 (3) - scopus: 2-s2.0-85105482975 (3)
11573/1553152 - 2021 -
Anti-tumoral effects of a (1H-pyrrol-1-yl)methyl-1H-benzoimidazole carbamate ester derivative on head and neck squamous carcinoma cell lines Nicolai, Alice; Madia, Valentina Noemi; Messore, Antonella; De Vita, Daniela; De Leo, Alessandro; Ialongo, Davide; Tudino, Valeria; Tortorella, Elisabetta; Scipione, Luigi; Taurone, Samanta; Artico, Marco; Di Santo, Roberto; Costi, Roberta; Scarpa, Susanna - 01a Articolo in rivista
paper: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. - - issn: 1424-8247 - wos: WOS:000666329400001 (3) - scopus: 2-s2.0-85110773299 (3)
11573/1555182 - 2021 -
Effect of Heparanase inhibitor on Tissue Factor overexpression in platelets and endothelial cells induced by anti-β2-GPI antibodies Capozzi, Antonella; Riitano, Gloria; Recalchi, Serena; Manganelli, Valeria; Costi, Roberta; Saccoliti, Francesco; Pulcinelli, Fabio Maria; Garofalo, Tina; Misasi, Roberta; Longo, Agostina; Di Santo, Roberto; Sorice, Maurizio - 01a Articolo in rivista
paper: JOURNAL OF THROMBOSIS AND HAEMOSTASIS (International Society on Thrombosis and Haemostasis ISTH) pp. 1-12 - issn: 1538-7933 - wos: WOS:000669313100001 (6) - scopus: 2-s2.0-85109019340 (6)
11573/1556284 - 2021 -
Quinolinonyl non-diketo acid derivatives as Inhibitors of HIV-1 ribonuclease H and polymerase functions of reverse transcriptase Messore, Antonella; Madia, Valentina Noemi; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Ialongo, Davide; Scipione, Luigi; De Vita, Daniela; Esposito, Francesca; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 8579-8598 - issn: 0022-2623 - wos: WOS:000668340800039 (6) - scopus: 2-s2.0-85108607601 (6)
11573/1564144 - 2021 -
Recent advances in recovery of lycopene from tomato waste. A potent antioxidant with endless benefits Madia, Valentina Noemi; De Vita, Daniela; Ialongo, Davide; Tudino, Valeria; De Leo, Alessandro; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta; Messore, Antonella - 01a Articolo in rivista
paper: MOLECULES (Basel: MDPI
Berlin: Springer, 1996-) pp. 1-18 - issn: 1420-3049 - wos: WOS:000682223800001 (20) - scopus: 2-s2.0-85111602310 (20)
11573/1564954 - 2021 -
Toxicological aspects of cannabinoid, pesticide and metal levels detected in light Cannabis inflorescences grown in Italy De Vita, Daniela; Madia, Valentina Noemi; Messore, Antonella; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: FOOD AND CHEMICAL TOXICOLOGY (Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. - - issn: 0278-6915 - wos: WOS:000696988600002 (2) - scopus: 2-s2.0-85112006002 (4)
11573/1565318 - 2021 -
Small-molecule inhibitors of HIV-1 reverse transcriptase-associated ribonuclease H function. Challenges and recent developments Madia, Valentina Noemi; Messore, Antonella; De Leo, Alessandro; Tudino, Valeria; Pindinello, Ivano; De Vita, Daniela; Scipione, Luigi; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: CURRENT MEDICINAL CHEMISTRY (Hilversum: Bentham Science Publishers) pp. 1-33 - issn: 1875-533X - wos: WOS:000696992000004 (1) - scopus: 2-s2.0-85115249511 (1)
11573/1584588 - 2021 -
New pyrimidine and pyridine derivatives as multitarget cholinesterase inhibitors. Design, synthesis, and in vitro and in cellulo evaluation Bortolami, Martina; Pandolfi, Fabiana; Tudino, Valeria; Messore, Antonella; Madia, Valentina Noemi; De Vita, Daniela; Di Santo, Roberto; Costi, Roberta; Scipione, Luigi - 01a Articolo in rivista
paper: ACS CHEMICAL NEUROSCIENCE (Washington, D.C. : American Chemical Society) pp. 4090-4112 - issn: 1948-7193 - wos: WOS:000715842900011 (4) - scopus: 2-s2.0-85118138783 (5)
11573/1594159 - 2021 -
Understanding drivers of ocular fibrosis: current and future therapeutic perspectives Mallone, Fabiana; Costi, Roberta; Marenco, Marco; Plateroti, Rocco; Minni, Antonio; Attanasio, Giuseppe; Artico, Marco; Lambiase, Alessandro - 01g Articolo di rassegna (Review)
paper: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (Basel (Matthaeustrasse 11) : Molecular Diversity Preservation International MDPI) pp. - - issn: 1661-6596 - wos: WOS:000718582700001 (3) - scopus: 2-s2.0-85118118842 (4)
11573/1599717 - 2021 -
Changes in surgicaL behaviOrs dUring the CoviD-19 pandemic. The SICE CLOUD19 Study Abbatini, Francesca; Costi, Roberta; Sciuto, Antonino; Auricchio, Simone Antonio; Gallo, Gaetano; Balla, Andrea; Coletta, Paola; Maida, Paola - 01a Articolo in rivista
paper: UPDATES IN SURGERY (Milano : Springer-Verlag Italia) pp. 731-744 - issn: 2038-131X - wos: WOS:000625025100002 (20) - scopus: 2-s2.0-85102173717 (26)
11573/1615167 - 2021 -
Pha-680626 is an effective inhibitor of the interaction between aurora-a and n-myc Boi, Dalila; Souvalidou, Fani; Polverino, Federica; Montanari, Roberta; Tramonti, Angela; Contestabile, Roberto; Trisciuoglio, Daniela; Saviano, Marialuisa; Costi, Roberta; Guarguaglini, Giulia; Paiardini, Alessandro - 01a Articolo in rivista
paper: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES (Basel (Matthaeustrasse 11) : Molecular Diversity Preservation International MDPI) pp. 13122- - issn: 1661-6596 - wos: WOS:000735123900001 (4) - scopus: 2-s2.0-85120777012 (7)
11573/1274892 - 2020 -
Discovery of a pyrimidine compound endowed with antitumor activity Taglieri, Ludovica; Saccoliti, Francesco; Nicolai, Alice; Peruzzi, Giovanna; Madia, Valentina Noemi; Tudino, Valeria; Messore, Antonella; Di Santo, Roberto; Artico, Marco; Taurone, Samanta; Salvati, Maurizio; Costi, Roberta; Scarpa, Susanna - 01a Articolo in rivista
paper: INVESTIGATIONAL NEW DRUGS (attuale:
-SPRINGER, VAN GODEWIJCKSTRAAT 30, DORDRECHT, NETHERLANDS, 3311 GZ
-Kluwer Academic Publishers / Massachusetts:PO Box 358, Accord Station:Hingham, MA 02018:(617)871-6600) pp. 39-49 - issn: 0167-6997 - wos: WOS:000512107200005 (10) - scopus: 2-s2.0-85063345760 (11)
11573/1389105 - 2020 -
Influence of oral administration mode on the efficacy of commercial bovine Lactoferrin against iron and inflammatory homeostasis disorders Rosa, Luigi; Lepanto, Maria Stefania; Paesano, Rosalba; Costi, Roberta; Valenti, Piera - 01a Articolo in rivista
paper: BIOMETALS (Rapid Science Publishers:2-6 Boundary Row, London SE1 8HN United Kingdom:011 44 207 9407500, EMAIL: rapidcom@vax.oxford.ac.uk, Fax: 011 44 207 8650027) pp. - - issn: 0966-0844 - wos: WOS:000540269500007 (13) - scopus: 2-s2.0-85083453638 (12)
11573/1395352 - 2020 -
New deferiprone derivatives as multi-functional cholinesterase inhibitors. Design, synthesis and in vitro evaluation Bortolami, Martina; Pandolfi, Fabiana; De Vita, Daniela; Messore, Antonella; Di Santo, Roberto; Feroci, Marta; Costi, Roberta; Chiarotto, Isabella; Scipione, Luigi - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 1-17 - issn: 0223-5234 - wos: WOS:000539425800007 (21) - scopus: 2-s2.0-85084066662 (23)
11573/1408850 - 2020 -
Pyrrolyl pyrazoles as non-diketo acid inhibitors of the HIV-1 ribonuclease H function of reverse transcriptase Messore, Antonella; Madia, Valentina Noemi; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Scipione, Luigi; De Vita, Daniela; Valenti, Piera; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: ACS MEDICINAL CHEMISTRY LETTERS (USA: ACS Publications) pp. 798-805 - issn: 1948-5875 - wos: WOS:000535281200029 (19) - scopus: 2-s2.0-85086659986 (21)
11573/1490804 - 2020 -
Recent advancement in the search of innovative antiprotozoal agents targeting trypanothione metabolism Saccoliti, Francesco; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. 2420-2435 - issn: 1860-7179 - wos: WOS:000567909300001 (12) - scopus: 2-s2.0-85091368381 (12)
11573/1205976 - 2019 -
In vitro antiviral activity of new oxazoline derivatives as potent poliovirus inhibitors Madia, Valentina Noemi; Messore, Antonella; Pescatori, Luca; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 798-810 - issn: 0022-2623 - wos: WOS:000457067600026 (6) - scopus: 2-s2.0-85060542889 (8)
11573/1218854 - 2019 -
Searching for new agents active against candida albicans biofilm: a series of indole derivatives, design, synthesis and biological evaluation Pandolfi, Fabiana; D'acierno, Federica; Bortolami, Martina; De Vita, Daniela; Di Santo, Roberto; Costi, Roberta; Simonetti, Giovanna; Scipione, Luigi - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 93-106 - issn: 0223-5234 - wos: WOS:000459358600008 (20) - scopus: 2-s2.0-85060089854 (21)
11573/1222183 - 2019 -
Design, synthesis, and biological evaluation of new 1-(aryl-1H-pyrrolyl)(phenyl)methyl-1H-imidazole derivatives as antiprotozoal agents Saccoliti, Francesco; Madia, Valentina Noemi; Tudino, Valeria; De Leo, Alessandro; Pescatori, Luca; Messore, Antonella; De Vita, Daniela; Scipione, Luigi; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1330-1347 - issn: 0022-2623 - wos: WOS:000459223600016 (20) - scopus: 2-s2.0-85061636363 (22)
11573/1285185 - 2019 -
Comparison of different methods for the extraction of cannabinoids from cannabis De Vita, Daniela; Madia, Valentina Noemi; Tudino, Valeria; Saccoliti, Francesco; De Leo, Alessandro; Messore, Antonella; Pindinello, Ivano; Scipione, Luigi; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: NATURAL PRODUCT RESEARCH (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1-7 - issn: 1478-6419 - wos: WOS:000575920700013 (26) - scopus: 2-s2.0-85065155862 (28)
11573/1321741 - 2019 -
Inhibition of Polycomb Repressive Complex2 activity reduces trimethylation of H3K27 and affects development in Arabidopsis seedlings Ruta, Veronica; Longo, Chiara; Boccaccini, Alessandra; Madia, Valentina Noemi; Saccoliti, Francesco; Tudino, Valeria; Di Santo, Roberto; Lorrai, Riccardo; Dello Ioio, Raffaele; Sabatini, Sabrina; Costi, Roberta; Costantino, Paolo; Vittorioso, Paola - 01a Articolo in rivista
paper: BMC PLANT BIOLOGY (London: BioMed Central.MIDDLESEX HOUSE, 34-42 CLEVELAND ST, LONDON, ENGLAND, W1T 4LB) pp. - - issn: 1471-2229 - wos: WOS:000490716900003 (9) - scopus: 2-s2.0-85073428390 (10)
11573/1336764 - 2019 -
Structure-guided approach to identify a novel class of anti-leishmaniasis diaryl sulfide compounds targeting the trypanothione metabolism Colotti, Gianni; Saccoliti, Francesco; Yadav, Shivangi; Battista, Theo; Mocci, Stefano; Fiorillo, Annarita; Bibi, Aasia; Madia, Valentina Noemi; Messore, Antonella; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: AMINO ACIDS (Wien: Springer Verlag) pp. - - issn: 0939-4451 - wos: WOS:000519385700013 (9) - scopus: 2-s2.0-85065106515 (10)
11573/1405464 - 2019 -
Tegaserod for the treatment of Irritable Bowel syndrome Madia, Valentina Noemi; Messore, Antonella; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; De Vita, Daniela; Bortolami, Martina; Scipione, Luigi; Pindinello, Ivano; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: ANTI-INFLAMMATORY & ANTI-ALLERGY AGENTS IN MEDICINAL CHEMISTRY (Hilversum : Bentham Science Publsihers) pp. 1-28 - issn: 1871-5230 - wos: (0) - scopus: 2-s2.0-85083912835 (0)
11573/1099440 - 2018 -
Structure-guided approach identifies a novel class of HIV-1 ribonuclease H inhibitors: binding mode insights through magnesium complexation and site-directed mutagenesis studies Scipione, Luigi; Pandolfi, Fabiana; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: MEDCHEMCOMM (Cambridge : Royal Society of Chemistry, 2010-) pp. 562-575 - issn: 2040-2503 - wos: WOS:000428670100016 (16) - scopus: 2-s2.0-85044181388 (16)
11573/1174521 - 2018 -
Selective inhibition of the PRC2 methyltransferase activity suppresses trimethylation of H3K27 in Arabidopsis seeds Ruta, Veronica; Boccaccini, Alessandra; Longo, Chiara; Madia, Valentina Noemi; Tudino, Valeria; Costi, Roberta; Costantino, Paolo; Vittorioso, Paola - 04f Poster
conference: International Plant and Molecular Biology 2018- IPMB2018 (Montpellier)
book: nessuna - ()
11573/1176720 - 2018 -
Biological evaluation and structure-activity relationships of imidazole-based compounds as antiprotozoal agents Saccoliti, Francesco; Madia, Valentina Noemi; Tudino, Valeria; De Leo, Alessandro; Pescatori, Luca; Messore, Antonella; De Vita, Daniela; Scipione, Luigi; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 53-60 - issn: 0223-5234 - wos: WOS:000443663200005 (12) - scopus: 2-s2.0-85049312582 (14)
11573/1176836 - 2018 -
Novel benzazole derivatives endowed with potent antiheparanase activity Madia, Valentina Noemi; Messore, Antonella; Pescatori, Luca; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Bortolami, Martina; Scipione, Luigi; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 6918-6936 - issn: 0022-2623 - wos: WOS:000441484300030 (25) - scopus: 2-s2.0-85050088127 (25)
11573/1221546 - 2018 -
Novel symmetrical benzazolyl derivatives endowed with potent anti-heparanase activity Messore, Antonella; Madia, Valentina Noemi; Pescatori, Luca; Saccoliti, Francesco; Tudino, Valeria; De Leo, Alessandro; Bortolami, Martina; De Vita, Daniela; Scipione, Luigi; Pepi, Federico; Costi, Roberta; Mor, Marco; Ferrara, Fabiana Fosca; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 10834-10859 - issn: 0022-2623 - wos: WOS:000453488200031 (14) - scopus: 2-s2.0-85058215116 (13)
11573/1011030 - 2017 -
New pyridine derivatives as inhibitors of acetylcholinesterase and amyloid aggregation Pandolfi, Fabiana; De Vita, Daniela; Bortolami, Martina; Coluccia, Antonio; Di Santo, Roberto; Costi, Roberta; Scipione, Luigi - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 197-210 - issn: 0223-5234 - wos: WOS:000417962900018 (22) - scopus: 2-s2.0-85030860178 (26)
11573/1192249 - 2017 -
Structure-activity relationships on cynnamoyl derivatives as inhibitors of p300 Histone acetyltransferase Madia, Valentina Noemi; Pescatori, Luca; Messore, Antonella; Pupo, Giovanni; Saccoliti, Francesco; Valente, Sergio; Mai, Antonello; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. 1359-1368 - issn: 1860-7187 - wos: WOS:000429592300014 (9) - scopus: 2-s2.0-85017448829 (8)
11573/910059 - 2017 -
Functional roles of Acetylated Histone marks at mouse meiotic recombination hotspots Costi, Roberta - 01a Articolo in rivista
paper: MOLECULAR AND CELLULAR BIOLOGY (American Society for Microbiology / DC:1752 N Street Northwest:Washington, DC 20036:(202)737-3600, EMAIL: jadelman@asmusa.org, INTERNET: http://www.asmusa.org/asm.htm, Fax: (202)942-9342) pp. 1-24 - issn: 0270-7306 - wos: WOS:000392231500009 (15) - scopus: 2-s2.0-85011575217 (14)
11573/929856 - 2017 -
Inhibition of Leishmania infantum trypanothione reductase by diaryl sulfide derivatives Saccoliti, Francesco; Angiulli, Gabriella; Pupo, Giovanni; Pescatori, Luca; Madia, Valentina Noemi; Messore, Antonella; Fiorillo, Annarita; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 304-310 - issn: 1475-6366 - wos: WOS:000392591100025 (38) - scopus: 2-s2.0-85013797723 (42)
11573/972447 - 2017 -
Inhibition of the α-carbonic anhydrase from Vibrio cholerae with amides and sulfonamides incorporating imidazole moieties De Vita, Daniela; Pandolfi, Fabiana; Bortolami, Martina; Costi, Roberta; Di Santo, Roberto; Scipione, Luigi - 01a Articolo in rivista
paper: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 798-804 - issn: 1475-6366 - wos: WOS:000404271200006 (31) - scopus: 2-s2.0-85020209278 (33)
11573/894759 - 2016 -
Diaryl disulfides as novel stabilizers of tumor suppressor Pdcd4 Pescatori, Luca; Scipione, Luigi; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: PLOS ONE (San Francisco, CA : Public Library of Science) pp. 1-14 - issn: 1932-6203 - wos: WOS:000372574900108 (7) - scopus: 2-s2.0-84979088483 (8)
11573/903468 - 2016 -
New N,N-dimethylcarbamate inhibitors of acetylcholinesterase: design synthesis and biological evaluation De Vita, Daniela; Pandolfi, Fabiana; Ornano, Luigi; Feroci, Marta; Chiarotto, Isabella; Pepi, Federico; Costi, Roberta; Di Santo, Roberto; Scipione, Luigi - 01a Articolo in rivista
paper: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1-8 - issn: 1475-6366 - wos: WOS:000391904900013 (11) - scopus: 2-s2.0-84984870776 (11)
11573/910116 - 2016 -
New insights into the interaction between pyrrolyl diketoacids and HIV-1 integrase active site and comparison with RNase H Pescatori, Luca; Madia, Valentina Noemi; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: ANTIVIRAL RESEARCH ([Amsterdam]; [New York]: Elsevier/North-Holland, [c1981]-) pp. 236-243 - issn: 0166-3542 - wos: WOS:000386983800026 (29) - scopus: 2-s2.0-84989205085 (30)
11573/916308 - 2016 -
Exploring the anti-biofilm activity of cinnamic acid derivatives in Candida albicans De Vita, Daniela; Simonetti, Giovanna; Pandolfi, Fabiana; Costi, Roberta; Di Santo, Roberto; D'auria, Felicia Diodata; Scipione, Luigi - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. 5931-5935 - issn: 0960-894X - wos: WOS:000389784500020 (19) - scopus: 2-s2.0-84999015180 (21)
11573/541604 - 2015 -
Design, synthesis and evaluation of 3,4-dihydroxybenzoic acid derivatives as antioxidants, bio-metal chelating agents and acetylcholinesterase inhibitors Friggeri, Laura; De Vita, Daniela; Pandolfi, Fabiana; Tortorella, Silvano; Costi, Roberta; Di Santo, Roberto; Scipione, Luigi - 01a Articolo in rivista
paper: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 166-172 - issn: 1475-6366 - wos: WOS:000347956500024 (7) - scopus: 2-s2.0-84921307137 (7)
11573/783972 - 2015 -
Hypoglycemic activity of curcumin synthetic analogues in alloxan-induced diabetic rats Di Santo, Roberto; Costi, Roberta; Messore, Antonella; Pescatori, Luca; Saso, Luciano - 01a Articolo in rivista
paper: JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY (Taylor & Francis Limited:Rankine Road, Basingstoke RG24 8PR United Kingdom:011 44 1256 813035, EMAIL: madeline.sims@tandf.co.uk, info@tandf.co.uk, INTERNET: http://www.tandf.co.uk, Fax: 011 44 1256 330245) pp. 1-7 - issn: 1475-6366 - wos: WOS:000367555300011 (14) - scopus: 2-s2.0-84953262310 (18)
11573/787196 - 2015 -
N‑substituted quinolinonyl diketo acid derivatives as HIV integrase strand transfer inhibitors and their activity against RNase H function of reverse transcriptase Pescatori, Luca; Messore, Antonella; Pupo, Giovanni; Madia, Valentina Noemi; Saccoliti, Francesco; Scipione, Luigi; Tortorella, Silvano; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 4610-4623 - issn: 0022-2623 - wos: WOS:000356316600015 (36) - scopus: 2-s2.0-84935877076 (42)
11573/852938 - 2015 -
Discovery of N-aryl-naphthylamines as in vitro inhibitors of the interaction between HIV integrase and the cofactor LEDGF/p75 Cuzzucoli Crucitti, Giuliana; Pescatori, Luca; Messore, Antonella; Madia, Valentina Noemi; Pupo, Giovanni; Saccoliti, Francesco; Scipione, Luigi; Tortorella, Silvano; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 288-294 - issn: 0223-5234 - wos: WOS:000360771900026 (12) - scopus: 2-s2.0-84936802596 (12)
11573/895359 - 2015 -
Structure−activity relationship of pyrrolyl diketo acid derivatives as dual Inhibitors of HIV‑1 integrase and reverse transcriptase ribonuclease H domain Pescatori, Luca; Messore, Antonella; Madia, Valentina Noemi; Pupo, Giovanni; Saccoliti, Francesco; Scipione, Luigi; Tortorella, Silvano; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1915-1928 - issn: 0022-2623 - wos: WOS:000351186700021 (68) - scopus: 2-s2.0-84923882396 (73)
11573/541603 - 2014 -
Activity of caffeic acid derivatives against Candida albicans biofilm De Vita, Daniela; Friggeri, Laura; D'auria, Felicia Diodata; Pandolfi, Fabiana; Panella, Simona; Palamara, Anna Teresa; Simonetti, Giovanna; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta; Tortorella, Silvano - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. 1502-1505 - issn: 0960-894X - wos: WOS:000332391900011 (45) - scopus: 2-s2.0-84895795071 (50)
11573/559331 - 2014 -
Basic Quinolinonyl Diketo Acid Derivatives as Inhibitors of HIV
Integrase and their Activity against RNase H Function of Reverse
Transcriptase Costi, Roberta; Cuzzucoli Crucitti, Giuliana; Pescatori, Luca; Messore, Antonella; Madia, Valentina Noemi; Scipione, Luigi; Tortorella, Silvano; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington DC : ACS Publications) pp. 3223-3234 - issn: 1520-4804 - wos: WOS:000335113900005 (48) - scopus: 2-s2.0-84899554749 (52)
11573/579587 - 2014 -
Synthesis, biological evaluation and structure-activity correlation study of a series of imidazol-based compounds as Candida albicans inhibitors De Vita, Daniela; Pandolfi, Fabiana; Di Santo, Roberto; Costi, Roberta; D'auria, Felicia Diodata; Panella, Simona; Palamara, Anna Teresa; Simonetti, Giovanna; Scipione, Luigi - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 665-673 - issn: 0223-5234 - wos: WOS:000340689600059 (20) - scopus: 2-s2.0-84904025140 (20)
11573/619388 - 2014 -
Ptaquiloside in Pteridium aquilinum subsp. aquilinum and corresponding soils from South of
Italy: influence of physical and chemical features of soils on its occurrence Costi, Roberta - 01a Articolo in rivista
paper: SCIENCE OF THE TOTAL ENVIRONMENT (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598
Tokyo ; Oxford ; Lausanne ; New York ; Shannon ; Amsterdam : Elsevier) pp. 365-372 - issn: 0048-9697 - wos: WOS:000342245600042 (7) - scopus: 2-s2.0-84905460086 (7)
11573/621580 - 2014 -
identification of highly conserved residues involved in inhibition of HIV-1 RNase H function by Diketo Acid derivatives Pescatori, Luca; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (American Society for Microbiology:PO Box 11127:Birmingham, AL 35201:(800)633-4931, (205)995-1567, EMAIL: asm.nonmembers.subs@ebsco.com, INTERNET: http://www.asm.org, Fax: (205)995-1588) pp. 6101-6110 - issn: 0066-4804 - wos: WOS:000344157500054 (56) - scopus: 2-s2.0-84907266363 (61)
11573/507015 - 2013 -
CONVENIENT ROUTE TO 2H-PYRROLO
[3,4-b]QUINOLIN-9(4H)-ONE SKELETON
VIA TOSMIC REACTION Rosi, Federica; Cuzzucoli Crucitti, Giuliana; Pescatori, Luca; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: SYNTHETIC COMMUNICATIONS (New York, NY : Marcel Dekker) pp. 1063-1072 - issn: 1532-2432 - wos: WOS:000313418700015 (6) - scopus: 2-s2.0-84872326307 (6)
11573/515673 - 2013 -
Pharmacophore assessment through 3-D QSAR: evaluation of the predictive ability on new
derivatives by the application on a series of antitubercular agents Friggeri, Laura; Ballante, Flavio; Ragno, Rino; Musmuca, Ira; De Vita, Daniela; Biava, Mariangela; Scipione, Luigi; Di Santo, Roberto; Costi, Roberta; Feroci, Marta; Tortorella, Silvano - 01a Articolo in rivista
paper: JOURNAL OF CHEMICAL INFORMATION AND MODELING (AMER CHEMICAL SOC, 1155 16TH ST, NW, WASHINGTON, USA, DC, 20036) pp. 1463-1474 - issn: 1549-9596 - wos: WOS:000321074700019 (5) - scopus: 2-s2.0-84879596019 (10)
11573/516522 - 2013 -
New promising compounds with in vitro
nanomolar activity against Trypanosoma cruzi Friggeri, Laura; Scipione, Luigi; Costi, Roberta; Botta, Bruno; Di Santo, Roberto; De Vita, Daniela; Tortorella, Silvano - 01a Articolo in rivista
paper: ACS MEDICINAL CHEMISTRY LETTERS (USA: ACS Publications) pp. 538-541 - issn: 1948-5875 - wos: WOS:000321883900011 (14) - scopus: 2-s2.0-84879097485 (14)
11573/525948 - 2013 -
New Nucleotide-Competitive Non-Nucleoside Inhibitors of Terminal
2 Deoxynucleotidyl Transferase: Discovery, Characterization, and
3 Crystal Structure in Complex with the Target Costi, Roberta; Cuzzucoli Crucitti, Giuliana; Pescatori, Luca; Messore, Antonella; Scipione, Luigi; Tortorella, Silvano; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 7431-7441 - issn: 0022-2623 - wos: WOS:000330097700023 (16) - scopus: 2-s2.0-84885013896 (15)
11573/530616 - 2013 -
6-(1-Benzyl-1H-pyrrol-2-yl)-2,4-dioxo-5-hexenoic acids as dual inhibitors of recombinant HIV-1 integrase and ribonuclease H, synthesized by a parallel synthesis approach. Costi, Roberta; Cuzzucoli Crucitti, Giuliana; Pescatori, Luca; Messore, Antonella; Scipione, Luigi; Tortorella, Silvano; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington DC : ACS Publications) pp. 8588-8598 - issn: 1520-4804 - wos: WOS:000327111100029 (50) - scopus: 2-s2.0-84887922481 (54)
11573/455694 - 2012 -
Identification of PR-SET7 and EZH2 selective inhibitors inducing cell death in human leukemia U937 cells Valente, Sergio; Di Santo, Roberto; Costi, Roberta; Mai, Antonello - 01a Articolo in rivista
paper: BIOCHIMIE (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 2308-2313 - issn: 0300-9084 - wos: WOS:000310929200011 (22) - scopus: 2-s2.0-84867395419 (26)
11573/457568 - 2012 -
Effects of polyphenol compounds on influenza A virus replication and definition of their mechanism of action Fioravanti, Rossella; Celestino, Ignacio; Costi, Roberta; Cuzzucoli Crucitti, Giuliana; Pescatori, Luca; Mattiello, Leonardo; Palamara, Anna Teresa; Nencioni, Lucia; Di Santo, Roberto - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 5046-5052 - issn: 0968-0896 - wos: WOS:000307244300020 (37) - scopus: 2-s2.0-84864471453 (40)
11573/482226 - 2012 -
Polyphenols as anti-influenza A agents. Fioravanti, Rossella; Celestino, Ignacio; Costi, Roberta; Pescatori, Luca; Checconi, Paola; Palamara, Anna Teresa; Nencioni, Lucia; Di Santo, Roberto - 04a Atto di comunicazione a congresso
conference: 21st National Meeting on Medicinal Chemistry. (Palermo, Italy)
book: 21st National Meeting on Medicinal Chemistry. - ()
11573/485737 - 2012 -
Design, Synthesis, and Structure−Activity Relationship of
N‑Arylnaphthylamine Derivatives as Amyloid Aggregation Inhibitors Di Santo, Roberto; Costi, Roberta; Cuzzucoli Crucitti, Giuliana; Pescatori, Luca; Rosi, Federica; Scipione, Luigi - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 8538-8548 - issn: 0022-2623 - wos: WOS:000309643500030 (21) - scopus: 2-s2.0-84867382314 (25)
11573/488191 - 2012 -
Discovery and Pharmacological Profile of New 1H‑Indazole-3-
carboxamide and 2H‑Pyrrolo[3,4‑c]quinoline Derivatives as SelectiveSerotonin 4 Receptor Ligands Costi, Roberta; Cuzzucoli Crucitti, Giuliana; Pescatori, Luca; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 9446-9466 - issn: 0022-2623 - wos: WOS:000311461500006 (29) - scopus: 2-s2.0-84870052595 (31)
11573/414595 - 2011 -
Novel 3,5-bis(bromohydroxybenzylidene)piperidin-4-ones as coactivator-associated arginine methyltransferase 1 inhibitors: Enzyme selectivity and cellular activity Valente, Sergio; Di Santo, Roberto; Costi, Roberta; Mai, Antonello - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 4928-4932 - issn: 0022-2623 - wos: WOS:000292479600049 (61) - scopus: 2-s2.0-79960191524 (67)
11573/123490 - 2010 -
Evaluation of HIV-1 integrase inhibitors on human primary macrophages using a luciferase-based single-cycle phenotypicassay Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: JOURNAL OF VIROLOGICAL METHODS (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598) pp. 272-276 - issn: 0166-0934 - wos: WOS:000280869400047 (14) - scopus: 2-s2.0-77955092239 (15)
11573/227936 - 2009 -
Perturbing Effects of Chiral Stationary Phase on Enantiomerization Second-Order Rate Constants Determined by Enantioselective Dynamic High-Performance Liquid Chromatography: A Practical Tool to Quantify the Accessible Acid and Basic Catalytic Sites Bonded on Chromatographic Supports Costi, Roberta; Di Santo, Roberto; Pierini, Marco - 01a Articolo in rivista
paper: ANALYTICAL CHEMISTRY (Washington: American Chemical Society, ©1948-) pp. 3560-3570 - issn: 0003-2700 - wos: WOS:000265632400049 (35) - scopus: 2-s2.0-66149097413 (34)
11573/229129 - 2009 -
A rational approach to predict and modulate stereolability of chiral alpha-substituted ketones. Costi, Roberta; Di Santo, Roberto; Gasparrini, Francesco; La Torre, Filippo; Pierini, Marco - 01a Articolo in rivista
paper: CHIRALITY (John Wiley & Sons Incorporated:Customer Service, 111 River Street:Hoboken, NJ 07030:(800)225-5945, (201)748-6000, EMAIL: societyinfo@wiley.com, INTERNET: http://www.wiley.com, Fax: (212)748-6551) pp. 24-34 - issn: 0899-0042 - wos: WOS:000261782900006 (15) - scopus: 2-s2.0-59849121710 (14)
11573/368166 - 2009 -
Studio dell’attività antivirale di analoghi del resveratrolo in un modello sperimentale in vitro di infezione da virus influenzale A. Celestino, Ignacio; Nencioni, Lucia; Di Santo, Roberto; Costi, Roberta; Palamara, Anna Teresa - 04a Atto di comunicazione a congresso
book: 37° Congresso della Società Italiana di Microbiologia SIM, 11-14 ottobre 2009 pg. 70 - ()
11573/122770 - 2008 -
Simple synthesis of deuterated pterosines Costi, Roberta; Bonadies, Francesco - 01a Articolo in rivista
paper: SYNTHETIC COMMUNICATIONS (New York, NY : Taylor & Francis
New York, NY: Marcel Dekker Incorporated) pp. 1553-1559 - issn: 0039-7911 - wos: WOS:000256530800007 (3) - scopus: 2-s2.0-42549109034 (3)
11573/228663 - 2008 -
HIV-1 Integration: A Potential Target for Microbicides to Prevent Cell-free or Cell-associated Human Immunodeficiency Virus type-1 Infection Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (American Society for Microbiology:PO Box 11127:Birmingham, AL 35201:(800)633-4931, (205)995-1567, EMAIL: asm.nonmembers.subs@ebsco.com, INTERNET: http://www.asm.org, Fax: (205)995-1588) pp. 2544-2554 - issn: 0066-4804 - wos: WOS:000257183400036 (21) - scopus: 2-s2.0-46249087616 (21)
11573/230766 - 2008 -
Synthesis and cerebral uptake of 1-(1-[11C]methyl-1H-pyrrol-2-yl)-2-phenyl-2-(1-pyrrolidinyl)ethanone a novel tracer for positron emission tomography studies of monoamine oxidase type A Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1617-1622 - issn: 0022-2623 - wos: WOS:000254209800011 (12) - scopus: 2-s2.0-41249095463 (10)
11573/359251 - 2008 -
Novel quinolinonyl diketo acid derivatives as HIV-1 integrase inhibitors: Design, synthesis, and biological activities Di Santo, Roberto; Costi, Roberta; Nencioni, Lucia; Palamara, Anna Teresa - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 4744-4750 - issn: 0022-2623 - wos: WOS:000258289800043 (46) - scopus: 2-s2.0-49449093292 (51)
11573/240552 - 2007 -
HIV-1 integrase inhibitors are substrates for the multidrug transporter MDR1-P-glycoprotein Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: RETROVIROLOGY (London : BioMed Central) pp. 17-27 - issn: 1742-4690 - wos: WOS:000245096500002 (23) - scopus: 2-s2.0-42049093456 (22)
11573/241076 - 2007 -
Cynnamoyl compounds as simple molecules that inhibit p300 histone acetyltransferase Costi, Roberta; Di Santo, Roberto; Artico, Marino - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1973-1977 - issn: 0022-2623 - wos: WOS:000245634500025 (61) - scopus: 2-s2.0-34247281570 (64)
11573/241523 - 2007 -
Probing HIV-1 integrase inhibitor binding sites with position-specific integrase-DNA cross-linking assays Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: MOLECULAR PHARMACOLOGY (American Society for Pharmacology and Experimental Therapeutics:9650 Rockville Pike:Bethesda, MD 20814:(301)530-7024, EMAIL: pstoute@aspet.org, INTERNET: http://www.aspet.org, Fax: (301)634-7099) pp. 893-901 - issn: 0026-895X - wos: WOS:000244290400029 (29) - scopus: 2-s2.0-33847098825 (34)
11573/210965 - 2006 -
HIV-1 Integrase Inhibitors are potent substrates for the MDR1 multidrug transporter. Costi, Roberta; Di Santo, Roberto - 04a Atto di comunicazione a congresso
book: 13th Conferente on Retroviruses and Opportunistic Infection (CROI) - ()
11573/233551 - 2006 -
Novel bifunctional quinolonyl diketo acid derivatives as HIV-1 integrase inhibitors: Design, synthesis, biological activities, and mechanism of action Di Santo, Roberto; Costi, Roberta; Nencioni, Lucia; Palamara, Anna Teresa - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1939-1945 - issn: 0022-2623 - wos: WOS:000236400100013 (70) - scopus: 2-s2.0-33645405333 (90)
11573/236444 - 2006 -
Development of a human immunodeficiency virus vector-based, single-cycle assay for evaluation of anti-integrase compounds Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: ANTIMICROBIAL AGENTS AND CHEMOTHERAPY (American Society for Microbiology:PO Box 11127:Birmingham, AL 35201:(800)633-4931, (205)995-1567, EMAIL: asm.nonmembers.subs@ebsco.com, INTERNET: http://www.asm.org, Fax: (205)995-1588) pp. 3407-3417 - issn: 0066-4804 - wos: WOS:000241021700026 (18) - scopus: 2-s2.0-33749515634 (19)
11573/236938 - 2006 -
Arylthiopyrrole (AThP) Derivatives as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors. Synthesis, Structure-Activity Relationships and Docking Studies. Part 1. Di Santo, Roberto; Costi, Roberta; Artico, Marino; Miele, Gaetano - 01a Articolo in rivista
paper: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. 1367-1378 - issn: 1860-7179 - wos: WOS:000202946500008 (31) - scopus: 2-s2.0-33846262498 (34)
11573/237779 - 2006 -
Design, Synthesis, Biological Evaluation, and Molecular Modeling Studies on TIBO-Like Cyclic Sulfones as Novel Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors Di Santo, Roberto; Costi, Roberta; Artico, Marino; Ragno, Rino; La Torre, Filippo - 01a Articolo in rivista
paper: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. 82-95 - issn: 1860-7179 - wos: WOS:000202945500013 (18) - scopus: 2-s2.0-33746322348 (21)
11573/46567 - 2006 -
Arylthiopyrrole (ATP) Derivatives as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors Di Santo, Roberto; Costi, Roberta; Artico, Marino; Miele, Gaetano - 01a Articolo in rivista
paper: DRUGS OF THE FUTURE (Prous Science Publishers:Provenza 388, 08025 Barcelona Spain:011 34 3 4592220, EMAIL: service@prous.com, INTERNET: http://www.prous.com, Fax: 011 34 3 4581535) pp. 77-77 - issn: 0377-8282 - wos: (0) - scopus: (0)
11573/46568 - 2006 -
Diketo hexenoic acid (DKHA) derivatives: the first class of selective non-nucleoside inhibitors of mammalian terminal deoxynucleotidyl transferases endowed with cytotoxic effect against leukemic cells Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: DRUGS OF THE FUTURE (Prous Science Publishers:Provenza 388, 08025 Barcelona Spain:011 34 3 4592220, EMAIL: service@prous.com, INTERNET: http://www.prous.com, Fax: 011 34 3 4581535) pp. 84-84 - issn: 0377-8282 - wos: (0) - scopus: (0)
11573/46569 - 2006 -
Novel Curcumin Derivatives as p300 Histone Acetyltransferases inhibitors Di Santo, Roberto; Costi, Roberta; Miele, Gaetano - 01a Articolo in rivista
paper: DRUGS OF THE FUTURE (Prous Science Publishers:Provenza 388, 08025 Barcelona Spain:011 34 3 4592220, EMAIL: service@prous.com, INTERNET: http://www.prous.com, Fax: 011 34 3 4581535) pp. 130-130 - issn: 0377-8282 - wos: (0) - scopus: (0)
11573/210947 - 2005 -
Synthesis and Biological Evaluation of Curcumine Analogues as Apoptosis-Inducing Agents. Di Santo, Roberto; Costi, Roberta; Miele, Gaetano; Artico, Marino - 04a Atto di comunicazione a congresso
book: Joint Meeting on Medicinal Chemistry - ()
11573/210948 - 2005 -
Design, Synthesis and Biological Activities of Pyrrolylethanoneamine Derivatives, a Novel Class of MAO Inhibitors. Di Santo, Roberto; Costi, Roberta; La Torre, Filippo - 04a Atto di comunicazione a congresso
book: Joint Meeting on Medicinal Chemistry - ()
11573/210949 - 2005 -
Docking Studies on Bifunctional Quinolinyl Diketo Acids as HIV-1 Integrase Ihnhibitors. Di Santo, Roberto; Costi, Roberta; Nencioni, Lucia - 01a Articolo in rivista
paper: SCIENTIA PHARMACEUTICA (Oesterr Apotheker Verlags GES:Spitalgasse 31, A-1094 Vienna Austria:011 43 1 4023588) pp. 115-115 - issn: 0036-8709 - wos: (0) - scopus: (0)
11573/210959 - 2005 -
Sintesi, saggi enzimatici e attività antivirale di nuovi inibitori dell’integrasi di HIV. Di Santo, Roberto; Costi, Roberta; Nencioni, Lucia - 04a Atto di comunicazione a congresso
book: Fifth National Research Program on AIDS Progress Report,. - ()
11573/210960 - 2005 -
SAR Studies on Quinolinyl-2,4-Dioxobutanoic Acids, HIV-1 Integrase Inhibitors that Block HIV-1 Replication in Infected Cells. Di Santo, Roberto; Costi, Roberta; Nencioni, Lucia - 04a Atto di comunicazione a congresso
book: Joint Meeting on Medicinal Chemistry - ()
11573/210961 - 2005 -
Discovery of Novel Anti-Malarial Agents: 1-[(Aryl)(4-aryl-1H-pyrrol-3-yl)methyl]-1H-imidazoles Targeted to Farnesyl Transferase. Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: Joint Meeting on Medicinal Chemistry - ()
11573/210962 - 2005 -
2,4-Dioxo-5-hexenoic Acid Derivatives Are Novel Selective Non-Nucleoside Inhibitors of Mammalian Terminal Deoxynucleotidyl Transferases, with Potent Cytotoxic Effect Against Leukemic Cells. Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: Joint Meeting on Medicinal Chemistry - ()
11573/210963 - 2005 -
Quinolinyl-2,4-dioxobutanoic Acids as HIV-1 Integrase Inhibitors: SAR Studies and Binding Mode. Di Santo, Roberto; Costi, Roberta; Nencioni, Lucia - 04a Atto di comunicazione a congresso
book: Second Joint Italian-Swiss Meeting on Medicinal Chemistry - ()
11573/210964 - 2005 -
Diketo Hexenoic Acid (DKHA) Derivatives as Non-Nucleoside Inhibitors of Mammalian Terminal Deoxynucleotidyl Transferases. Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: Second Joint Italian-Swiss Meeting on Medicinal Chemistry - ()
11573/211198 - 2005 -
Diaryl Imidazolyl Methanes and Ethanes as Monoamine Oxidase Inhibitors. Di Santo, Roberto; Costi, Roberta; La Torre, Filippo - 04a Atto di comunicazione a congresso
book: Second Joint Italian-Swiss Meeting on Medicinal Chemistry - ()
11573/234366 - 2005 -
Diketo hexenoic acid derivatives are novel selective non-nucleoside inhibitors of mammalian terminal deoxynucleotidyl transferases, with potent cytotoxic effect against leukemic cells Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: MOLECULAR PHARMACOLOGY (American Society for Pharmacology and Experimental Therapeutics:9650 Rockville Pike:Bethesda, MD 20814:(301)530-7024, EMAIL: pstoute@aspet.org, INTERNET: http://www.aspet.org, Fax: (301)634-7099) pp. 538-550 - issn: 0026-895X - wos: WOS:000230549900031 (12) - scopus: 2-s2.0-23044491841 (13)
11573/237889 - 2005 -
6-(1-(4-fluorophenyl)methyl-1H-pyrrol-2-yl))-2,4-dioxo-5-hexenoic acid ethyl ester a novel diketo acid derivative which selectively inhibits the HIV-1 viral replication in cell culture and the ribonuclease H activity in vitro Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: ANTIVIRAL RESEARCH ([Amsterdam]; [New York]: Elsevier/North-Holland, [c1981]-) pp. 117-124 - issn: 0166-3542 - wos: WOS:000227261900007 (113) - scopus: 2-s2.0-13544276913 (124)
11573/238404 - 2005 -
Simple but highly effective three-dimensional chemical-feature-based pharmacophore model for diketo acid derivatives as hepatitis C virus RNA-dependent RNA polymerase inhibitors Di Santo, Roberto; Costi, Roberta; Artico, Marino - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 6304-6314 - issn: 0022-2623 - wos: WOS:000232406600015 (41) - scopus: 2-s2.0-26444491094 (42)
11573/239790 - 2005 -
Design, synthesis and biological evaluation of heteroaryl diketohexenoic and diketobutanoic acids as HIV-1 integrase inhibitors endowed with antiretroviral activity Di Santo, Roberto; Costi, Roberta; Ragno, Rino - 01a Articolo in rivista
paper: IL FARMACO (Attuale:ELSEVIER SCIENCE SA, PO BOX 564, LAUSANNE, SWITZERLAND, 1001
Societa Chimica Italiana:Viale Liegi 48, 00198 Rome Italy:011 39 06 8549691, EMAIL: soc.chim.it@agora.stm.it, Fax: 011 39 06 8548734) pp. 409-417 - issn: 0014-827X - wos: (0) - scopus: 2-s2.0-19544380093 (36)
11573/364346 - 2005 -
Antifungal agents. 11. N-substituted derivatives of 1-[(aryl)(4-aryl-1H-pyrrol-3-yl)methyl]-1H-imidazole: Synthesis, anti-Candida activity, and QSAR studies Di Santo, Roberto; Costi, Roberta; Angiolella, Letizia; Palamara, Anna Teresa - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 5140-5153 - issn: 0022-2623 - wos: WOS:000231055300011 (109) - scopus: 2-s2.0-23444446586 (124)
11573/46061 - 2005 -
Regioselectivity of the methyl-TosMIC reaction with substituted ethyl cinnamates Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL (Organic Preparations and Procedures Incorporated:PO Box 610009:Newton Highlands, MA 02161:(617)287-6130, EMAIL: jp.anselme@umb.edu, Fax: (617)287-6030) pp. 110-115 - issn: 0030-4948 - wos: WOS:000228891700003 (2) - scopus: 2-s2.0-19344371166 (2)
11573/46290 - 2005 -
2H-Pyrrolo[3,4-b][1,5] benzothiazepine derivatives as potential inhibitors of HIV-1 reverse transcriptase Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: IL FARMACO (Attuale:ELSEVIER SCIENCE SA, PO BOX 564, LAUSANNE, SWITZERLAND, 1001
Societa Chimica Italiana:Viale Liegi 48, 00198 Rome Italy:011 39 06 8549691, EMAIL: soc.chim.it@agora.stm.it, Fax: 011 39 06 8548734) pp. 385-392 - issn: 0014-827X - wos: (0) - scopus: 2-s2.0-19444387692 (44)
11573/506757 - 2005 -
Design, synthesis, and biological activities of pyrrolylethanoneamine derivatives, a novel class of monoamine oxidases inhibitors Di Santo, Roberto; Costi, Roberta; Agostinelli, Enzo - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 4220-4223 - issn: 0022-2623 - wos: WOS:000230121800007 (26) - scopus: 2-s2.0-21244505103 (34)
11573/189716 - 2004 -
Studio di una nuova classe di derivati pirrol-imidazolici: attività antimicotica e modulazione delle proteine di parete di Candida Albicans. Angiolella, Letizia; Di Santo, Roberto; Costi, Roberta; Forte, Michela; Artico, Marino; Palamara, Anna Teresa - 04a Atto di comunicazione a congresso
book: 1° Congresso Nazionale Società Italiana di Microbiologia Farmaceutica - ()
11573/210721 - 2004 -
Acidi 6-aril-2,4-dioxo-5-esenoici come inibitori della NS5B polimerasi dell'HCV. Di Santo, Roberto; Costi, Roberta; Artico, Marino - 04a Atto di comunicazione a congresso
book: XVII Convegno Nazionale della Divisione di Chimica Farmaceutica della SCI. - ()
11573/210942 - 2004 -
Derivati 1-[(aril)(1(5)-aril-1H-pirrol-2(3)-il)metil]-1H-imidazolici ad attività antifungina. Di Santo, Roberto; Costi, Roberta; Angiolella, Letizia - 04a Atto di comunicazione a congresso
book: XVII Convegno Nazionale della Divisione di Chimica Farmaceutica della SCI. - ()
11573/210943 - 2004 -
1-((Aril)(4-aril-1H-pirrol-3-il)metil)-1H-imidazoli: studio della relazioni struttura-attività di derivati sostituiti in posizione 1 dell'anello pirrolico. Di Santo, Roberto; Costi, Roberta; Angiolella, Letizia; Palamara, Anna Teresa - 04a Atto di comunicazione a congresso
book: XVII Convegno Nazionale della Divisione di Chimica Farmaceutica della SCI. - ()
11573/210944 - 2004 -
Acidi chinolinil-2,4-dioxobutanoici come analoghi conformazionalmente ristretti dei derivati arildichetoesenoici, dotati di potente attività anti-integrasi del virus HIV-1. Di Santo, Roberto; Costi, Roberta; Ragno, Rino - 04a Atto di comunicazione a congresso
book: XVII Convegno Nazionale della Divisione di Chimica Farmaceutica della SCI. - ()
11573/210945 - 2004 -
6-Aryl-2,4-dioxo-5-hexenoic acids, Novel HCV NS5b Polymerase Inhibitors. Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: COST D28 MC Action, Natural Products as a Source for Discovery, Synthesis, and Application of New Ph - ()
11573/210946 - 2004 -
Quinolinyl 2,4-dioxobutanoic Acids, Conformationally Restrained Analogues of Aryldioxohexenoic Acids as HIV-1 Integrase Inhibitors. Di Santo, Roberto; Costi, Roberta; Roux, Alessandra; Artico, Marino; Ragno, Rino - 04a Atto di comunicazione a congresso
book: COST D28 MC Action, Natural Products as a Source for Discovery, Synthesis, and Application of New Ph - ()
11573/210958 - 2004 -
1[(Aryl)(4-aryl-1H-pyrrol-3-yl)methyl]-1H-imidazoles: a Class of Potent Antifungal Agents. SAR Studies of N-1 Substituted Derivatives. Di Santo, Roberto; Costi, Roberta; Artico, Marino; Angiolella, Letizia; Palamara, Anna Teresa - 04a Atto di comunicazione a congresso
book: COST D28 MC Action, Natural Products as a Source for Discovery, Synthesis, and Application of New Ph - ()
11573/231135 - 2004 -
6-Aryl-2,4-dioxo-5-hexenoic Acids, Novel Integrase Inhibitors Active Against HIV-1 Multiplication in Cell-Based Assays. Costi, Roberta; Di Santo, Roberto; Artico, Marino; Ragno, Rino - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. 1745-1749 - issn: 0960-894X - wos: WOS:000220411200029 (39) - scopus: 2-s2.0-12144288755 (44)
11573/236844 - 2004 -
A General, Versatile Synthesis of 2H-Pyrrolo[3,4-c]quinolines via Tosylmethylisocyanide Reaction Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: ARKIVOC (ARKAT USA INC, C/O ALAN R KATRITZKY, UNIV FLORIDA, DEPT CHEMISTRY, PO BOX 117200, GAINESVILLE, USA, FL, 32611) pp. 181-195 - issn: 1551-7004 - wos: (0) - scopus: 2-s2.0-2942694389 (12)
11573/365225 - 2004 -
2,6-Bis(3,4,5-trihydroxybenzylydene) derivatives of cyclohexanone: novel potent HIV-1 integrase inhibitors that prevent HIV-1 multiplication in cell-based assays Costi, Roberta; Di Santo, Roberto; Artico, Marino; Ragno, Rino - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 199-215 - issn: 0968-0896 - wos: WOS:000188113400021 (78) - scopus: 2-s2.0-0347301799 (81)
11573/46059 - 2004 -
Enantiomers of new synthetic pyrrolylethanoneamine mono-amino oxidase inhibitor compounds: analytical and semipreparative HPLC separations, and chiroptical characteristics La Torre, Filippo; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: CHROMATOGRAPHIA (Heidelberg ; Berlin : Springer) pp. 171-178 - issn: 0009-5893 - wos: (0) - scopus: (0)
11573/210706 - 2003 -
Derivati Fenilpirroliletanonamminici analoghi del Kathinone dotati di potente e selettiva attività anti-MAO-A. Agostinelli, Enzo; Di Santo, Roberto; Costi, Roberta; Artico, Marino; La Torre, Filippo - 04a Atto di comunicazione a congresso
book: XXI Congresso Nazionale della Società Chimica Italiana - ()
11573/210707 - 2003 -
Acidi 6-Aril-2,4-dioxo-5-esenoici, Nuovi Inibitori dell’Integrasi. Blocco la Replicazione dell’HIV-1 in Cellule Infettate. Di Santo, Roberto; Costi, Roberta; Ragno, Rino - 04a Atto di comunicazione a congresso
book: XXI Congresso Nazionale della Società Chimica Italiana - ()
11573/210926 - 2003 -
Studies of enantiomerization barrier of 2-[2-(1-methyl-1H-pyrrol-2-yl)-2-oxo-1-phenylethyl]-isoindole-1,3-dione by enantioselective stopped-flow HPLC. Costi, Roberta; Di Santo, Roberto; La Torre, Filippo - 04a Atto di comunicazione a congresso
book: XXI Congresso Nazionale della Società Chimica Italiana - ()
11573/210950 - 2003 -
1-[(Aril)(4-aril-1H-pirrol-3-il)metil]-1H-imidazoli: Effetti della Sostituzione all'Azoto Pirrolico sull'Attività anti-Candida. Di Santo, Roberto; Costi, Roberta; Artico, Marino; Angiolella, Letizia; Palamara, Anna Teresa - 04a Atto di comunicazione a congresso
book: XXI Congresso Nazionale della Società Chimica Italiana - ()
11573/210956 - 2003 -
Studi SAR su Derivati 2H-Pirrolo[3,4-c]chinolinici quali Potenti e Selettivi Ligandi per i Recettori 5-HT4. Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: XXI Congresso Nazionale della Società Chimica Italiana - ()
11573/253007 - 2003 -
Caratterizzazione dell’attività antimicotica di una nuova classe di derivati pirrol-imidazolici Angiolella, Letizia; Di Santo, Roberto; Costi, Roberta; Palamara, Anna Teresa - 04a Atto di comunicazione a congresso
book: 31° Congresso Nazionale Società Italiana di Microbiologia, - ()
11573/253348 - 2003 -
Phenylpyrrolylethanoneamines related to kathinone, endowed with potent and highly selective anti-MAO-A activity. Agostinelli, Enzo; Di Santo, Roberto; Costi, Roberta; Artico, Marino; Roux, Alessandra; La Torre, Filippo - 04a Atto di comunicazione a congresso
book: 8th International Congress on Amino Acids and Proteins - ()
11573/255461 - 2003 -
Conversion of a Racemic Mixture of 8-Chloro-2-(2,6-difluorophenylmethyl)-2,3-dihydro-3-methyl-1,2,5-benzothiadiazepin-4(5H)-one 1,1-Dioxide into a Single Enantioemer Via a Chromatographic Resolution/Racemization Method La Torre, Filippo; Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: CHIRALITY (John Wiley & Sons Incorporated:Customer Service, 111 River Street:Hoboken, NJ 07030:(800)225-5945, (201)748-6000, EMAIL: societyinfo@wiley.com, INTERNET: http://www.wiley.com, Fax: (212)748-6551) pp. 429-432 - issn: 0899-0042 - wos: WOS:000182518000007 (4) - scopus: 2-s2.0-0037277248 (5)
11573/46053 - 2003 -
HIV-1 Integrase Inhibitors that Block HIV-1 Replication in Infected Cells. Planning Synthetic Derivatives from Natural Products Di Santo, Roberto; Costi, Roberta; Artico, Marino - 01a Articolo in rivista
paper: PURE AND APPLIED CHEMISTRY (Editore attuale:INT UNION PURE APPLIED CHEMISTRY, 104 TW ALEXANDER DR, PO BOX 13757, RES TRIANGLE PK, USA, NC, 27709-3757
Blackwell Science Limited:PO Box 88, Oxford OX2 0NE United Kingdom:011 44 1865 776868, 011 44 1865 206038, EMAIL: journals.cs@blacksci.co.uk, INTERNET: http://www.blackwell-science.com, Fax: 011 44 1865 721205) pp. 195-206 - issn: 0033-4545 - wos: WOS:000182416500007 (16) - scopus: 2-s2.0-0037317788 (23)
11573/46054 - 2003 -
Enantioselective liquid Chromatography of C3-chiral 2,3-dihydro-1,2,5-benzothiadiazepin-4(5H)-one and thione 1,1-dioxides on polyacrylamide- and polysaccaride-based chiral stationary phases Costi, Roberta; Di Santo, Roberto; Artico, Marino; La Torre, Filippo - 01a Articolo in rivista
paper: JOURNAL OF CHROMATOGRAPHY A (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598) pp. 17-28 - issn: 0021-9673 - wos: WOS:000182174600002 (28) - scopus: 2-s2.0-0037453478 (32)
11573/189704 - 2002 -
1-Alchil-3-aril-4[_-(1H-imidazol-1-il)arilmetil]pirroli: una Nuova Classe di Potenti Agenti Anti-Candida Di Santo, Roberto; Costi, Roberta; Forte, Michela; Artico, Marino; Angiolella, Letizia; Palamara, Anna Teresa - 04a Atto di comunicazione a congresso
book: 30° Congresso Nazionale Società Italiana di Microbiologia - ()
11573/194610 - 2002 -
HIV-1 Integrase Inhibitors That Block HIV-1 Replication in Infected Cells: Planning Synthetic Derivatives from Natural Products. Di Santo, Roberto; Costi, Roberta; Artico, Marino - 04a Atto di comunicazione a congresso
book: 23rd IUPAC - 2002 International Symposium on the Chemistry of Natural Products - ()
11573/194611 - 2002 -
Nuove Classi di Inibitori dell’Integrasi dell’HIV-1 che Bloccano la Replicazione Virale in Cellule Infettate Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: XVI Convegno Nazionale di Chimica Farmaceutica - ()
11573/194613 - 2002 -
Design, Synthesis And Biological Evaluation of 2H-Pyrrolo[3,4-c]quinolines, a New Class of Potent 5-HT4 Ligands. Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: 2ème Congès Combiné de Pharmacochimie - ()
11573/194615 - 2002 -
Probing the activity of diketoacids as HCV NS5B polymerase inhibitors via detailed molecular modeling Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: 23rd IUPAC - 2002 International Symposium on the Chemistry of Natural Products - ()
11573/194623 - 2002 -
Progettazione, Sintesi ed Attività Biologica di 2H-Pirrolo[3,4-c]chinoline, una Nuova Classe di Ligandi Selettivi per i Recettori 5-HT4 Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: XVI Convegno Nazionale di Chimica Farmaceutica - ()
11573/194832 - 2002 -
1-[Aril-(1-aril-1H-pirrol-3-il)metil]-1H-imidazoli, una Nuova Classe di Potenti Inibitori della Farnesiltrasferasi Di Santo, Roberto; Costi, Roberta; Artico, Marino - 04a Atto di comunicazione a congresso
book: XVI Convegno Nazionale di Chimica Farmaceutica - ()
11573/252637 - 2002 -
ARYLTHIOPYRIDYLMETHYLISOPROPYLPYRROLE CARBINOLS, NOVEL NNRTIs ENDOWED WITH POTENT ANTI-HIV-1 ACTIVITY Di Santo, Roberto; Costi, Roberta; Ragno, Rino - 01a Articolo in rivista
paper: MEDICINAL CHEMISTRY RESEARCH (Birkhauser Boston Incorporated:c/o Springer Verlag, PO Box 2485:Secaucus, NJ 07096:(800)777-4643, (973)348-4033, Fax: (973)348-4505) pp. 153-167 - issn: 1054-2523 - wos: WOS:000176370900002 (7) - scopus: 2-s2.0-0036056712 (7)
11573/255869 - 2002 -
Antifungal Agents. 10. New Derivatives of 1-[(Aryl)[4-aryl-1H-pyrrol-3-yl]methyl]-1H-imidazole, Synthesis, Anti-Candida Activity, and Quantitative Structure-Activity Relationship Studies Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 2720-2732 - issn: 0022-2623 - wos: WOS:000176204300005 (86) - scopus: 2-s2.0-0037142376 (94)
11573/46051 - 2002 -
Design, synthesis and QSAR studies on N-aryl heteroarylisopropanolamines, a new class of non-peptidic HIV-1 protease inhibitors Di Santo, Roberto; Costi, Roberta; Ragno, Rino - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 2511-2526 - issn: 0968-0896 - wos: WOS:000176294500009 (32) - scopus: 2-s2.0-0036286615 (42)
11573/47152 - 2002 -
Derivatives of 2,3-dihydroimidazo[1,5,4-ef][1,2,5]benzothiadiazepin-6(4H,7H)-thione 1,1-dioxide, a new heterocyclic system related to TIBO Costi, Roberta; Di Santo, Roberto - 01a Articolo in rivista
paper: JOURNAL OF HETEROCYCLIC CHEMISTRY (Hetero Corporation:PO Box 170:Provo, UT 84603:(801)400-7373, EMAIL: jhetchem@yahoo.com, Fax: (801)356-7373) pp. 81-90 - issn: 0022-152X - wos: WOS:000174926800011 (9) - scopus: 2-s2.0-0036185075 (12)
11573/125012 - 2001 -
Analytical and semipreparative enantiomeric separation of azole antifungal agents by high-performance liquid chromatography on polysaccharide-based chiral stationary phases Application to in vitro biological studies Costi, Roberta; Di Santo, Roberto; Angiolella, Letizia - 01a Articolo in rivista
paper: JOURNAL OF CHROMATOGRAPHY A (Elsevier BV:PO Box 211, 1000 AE Amsterdam Netherlands:011 31 20 4853757, 011 31 20 4853642, 011 31 20 4853641, EMAIL: nlinfo-f@elsevier.nl, INTERNET: http://www.elsevier.nl, Fax: 011 31 20 4853598) pp. 107-114 - issn: 0021-9673 - wos: WOS:000173120900010 (17) - scopus: 2-s2.0-0037016285 (18)
11573/194609 - 2001 -
3,4,5-Trihydroxycynnamoyl moiety: a Potent Pharmacophore for Anti-Integrase Agents Active Either in Enzymatic or in Cell-Based Assays. Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: Third National Research Program on AIDS Progress Report - ()
11573/194612 - 2001 -
Arylthiopyrroles (ATPs) A New Class of Potent NNRTIs Active either Against HIV-1 WT or Resistant Strains. Costi, Roberta; Di Santo, Roberto - 04a Atto di comunicazione a congresso
book: Hungarian-German-Italian-Polish Joint Meeting on Medicinal Chemistry - ()
11573/254828 - 2001 -
1-[4-(4-Chlorophenyl)-1H-pyrrol-3-yl](2,4-dichlorophenyl)methyl-1H-imidazole (RDS 416) Costi, Roberta; Di Santo, Roberto; Artico, Marino - 01a Articolo in rivista
paper: ACTA CRYSTALLOGRAPHICA SECTION E-STRUCTURE REPORTS ONLINE (Pubblicata da
BLACKWELL MUNKSGAARD, 35 NORRE SOGADE, PO BOX 2148, COPENHAGEN, DENMARK, DK-1016) pp. 096-098 - issn: 1600-5368 - wos: (0) - scopus: (0)
11573/194608 - 2000 -
Derivati del 2H-pirrolo[3,4-c]chinolin-4(5H)-one: Nuovi Potenziali Agonisti dei Recettori 5-HT3 Costi, Roberta; Di Santo, Roberto; Artico, Marino - 04a Atto di comunicazione a congresso
book: XX Congresso Nazionale della Società Chimica Italiana (SCI 2000) - ()
11573/249530 - 2000 -
Antimycobacterial Pyrroles: Synthesis, Anti-Mycobacterium tuberculosis Activity and QSAR Studies. Ragno, Rino; Di Santo, Roberto; Costi, Roberta; Artico, Marino - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY (Oxford: Pergamon, 1993-) pp. 1423-1432 - issn: 0968-0896 - wos: WOS:000087742300019 (132) - scopus: 2-s2.0-0034131292 (137)
11573/254827 - 2000 -
Structure-activity relationship studies on potential non-nucleoside DABO-like inhibitors of HIV-1 reverse transcriptase. Costi, Roberta; Di Santo, Roberto; Artico, Marino - 01a Articolo in rivista
paper: ANTIVIRAL CHEMISTRY & CHEMOTHERAPY (International Medical Press:2-4 Idol Lane, London EC3R 5DD United Kingdom:011 44 207 3980700, EMAIL: imp@intmedpress.com, INTERNET: http://www.intmedpress.com, Fax: 011 44 207 3980701) pp. 117-133 - issn: 0956-3202 - wos: WOS:000086782000004 (14) - scopus: 2-s2.0-0034017027 (13)
11573/194594 - 1999 -
Different kinetics of inhibition of the HIV-1 integrase activities by different classes of derivatives. Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: Italian-Hungarian-Polish Joint Meeting on Medicinal Chemistry - ()
11573/194595 - 1999 -
3,4,5-Trioxycinnamoyl Moiety: a Potent Pharmacophore for anti-HIV-1 Integrase Activity either in Enzyme or in Cell-Based Assays. Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: Italian-Hungarian-Polish Joint Meeting on Medicinal Chemistry - ()
11573/194597 - 1999 -
Trihydroxy-cinnamoyl derivatives targeted at the integrase inhibit the HIV-1 multiplication in cell-based assays Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: Second National program on AIDS Progress Repor - ()
11573/244226 - 1999 -
Structure Based Design of N-aryl-heteroarylpropanolamines, a new class of simple HIV-1 Protease Inhibitors Di Santo, Roberto; Costi, Roberta; Ragno, Rino - 04a Atto di comunicazione a congresso
book: Italian – hungarian – Polish Joint Meeting on Medicinal Chemistry - ()
11573/244906 - 1999 -
Pyridinylpyrrolyl Analogs of Isoniazid: Synthesis and Antimycobacterial Activities. Costi, Roberta; Artico, Marino; Di Santo, Roberto - 01a Articolo in rivista
paper: MEDICINAL CHEMISTRY RESEARCH (Birkhauser Boston Incorporated:c/o Springer Verlag, PO Box 2485:Secaucus, NJ 07096:(800)777-4643, (973)348-4033, Fax: (973)348-4505) pp. 408-423 - issn: 1054-2523 - wos: WOS:000084511600004 (3) - scopus: 2-s2.0-0033399508 (2)
11573/194598 - 1998 -
SAR Studies on 1-Alkyl-3-aryl-4-[a-(1H-imidazol-1-yl)arylmethyl]pyrroles a Class of Potent Anti-Candida Agents. Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: XIV CONVEGNO NAZIONALE Divisione di Chimica Farmaceutica SCI - ()
11573/194599 - 1998 -
Synthesis and Antimycobacterial Activities of Pyrrole Derivatives Related to Pyrrolnitrin. Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: XIV CONVEGNO NAZIONALE Divisione di Chimica Farmaceutica SCI - ()
11573/194601 - 1998 -
3D QSAR and Molecular Modeling on a Set of New Anti Mycobacterial Compounds. Di Santo, Roberto; Costi, Roberta; Ragno, Rino - 04a Atto di comunicazione a congresso
book: Second research project on Tuberculosis (1998) Progress report - ()
11573/243326 - 1998 -
ARYLSULFONYL PYRROLES FROM REACTION OF TOSYLMETHYL ISOCIANIDE (TOSMIC) WITH 3-ARYLSULFONYL ACRYLATES AS MICHAEL ACCEPTORS. Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: SYNTHETIC COMMUNICATIONS (New York, NY : Taylor & Francis
New York, NY: Marcel Dekker Incorporated) pp. 1801-1815 - issn: 0039-7911 - wos: (0) - scopus: 2-s2.0-0031807811 (9)
11573/245377 - 1998 -
Pyrrolnitrin and Related Pyrroles Endowed with Antibacterial Activities against Mycobacterium Tuberculosis. Di Santo, Roberto; Costi, Roberta; Artico, Marino - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. 2931-2936 - issn: 0960-894X - wos: (0) - scopus: (0)
11573/247003 - 1998 -
PYRROLE-ANNULATED HETEROCYCLIC SYSTEMS. SYNTHESIS OF 2H-PYRROLO[3,4-b][1,5]BENZOTHIAZEPINE 4,4-DIOXIDE DERIVATIVES Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: SYNTHETIC COMMUNICATIONS (New York, NY : Taylor & Francis
New York, NY: Marcel Dekker Incorporated) pp. 2517-2530 - issn: 0039-7911 - wos: (0) - scopus: (0)
11573/247184 - 1998 -
Geometrically and Conformationally Restrained Cinnamoyl-Compounds as Inhibitors of HIV-1 Integrase: Synthesis, Biological Evaluation and Molecular Modeling Artico, Marino; Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 3948-3960 - issn: 0022-2623 - wos: WOS:000076374300005 (169) - scopus: 2-s2.0-15144355755 (166)
11573/43958 - 1998 -
1,2,5-Benzothiadiazepine and Pyrrolo[2,1-d][1,2,5]Benzothiadiazepine Derivatives with Anti-HIV-1 Activity. Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: ANTIVIRAL CHEMISTRY & CHEMOTHERAPY (International Medical Press:2-4 Idol Lane, London EC3R 5DD United Kingdom:011 44 207 3980700, EMAIL: imp@intmedpress.com, INTERNET: http://www.intmedpress.com, Fax: 011 44 207 3980701) pp. 127-137 - issn: 0956-3202 - wos: WOS:000072685800004 (35) - scopus: 2-s2.0-0031954544 (39)
11573/194604 - 1997 -
Synthesis of Curcumin-like Derivatives with Potent Activity Against the HIV-1 Integrase. Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: First Italian-Swiss meeting on Medicinal Chemistry - ()
11573/194606 - 1997 -
Pyrrolo[2,1-d][1,2,5]benzothiadiazepine derivatives with anti-HIV-1 activity. Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: Ninth research project on AIDS (1996) Progress report - ()
11573/244912 - 1997 -
N-(1-Naphthylmethyl)-N-(1-alkyl-4-aryl-1H-pyrrol-3-ylmethyl)methylamines Related to Naftifine. Synthesis and Antifungal Activity. Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: MEDICINAL CHEMISTRY RESEARCH (Birkhauser Boston Incorporated:c/o Springer Verlag, PO Box 2485:Secaucus, NJ 07096:(800)777-4643, (973)348-4033, Fax: (973)348-4505) pp. 98-108 - issn: 1054-2523 - wos: (0) - scopus: 2-s2.0-0003066751 (4)
11573/245204 - 1997 -
Heterocycles with a benzothiadiazepine moiety .5. Derivatives of pyrrolo[2,1-d][1,2,5]benzothiadiazepine, a novel tricyclic ring Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: IL FARMACO (Attuale:ELSEVIER SCIENCE SA, PO BOX 564, LAUSANNE, SWITZERLAND, 1001
Societa Chimica Italiana:Viale Liegi 48, 00198 Rome Italy:011 39 06 8549691, EMAIL: soc.chim.it@agora.stm.it, Fax: 011 39 06 8548734) pp. 375-378 - issn: 0014-827X - wos: WOS:A1997YD01000006 (9) - scopus: 2-s2.0-0030665610 (13)
11573/245262 - 1997 -
1-Arylsulfonyl-3-(a-hydroxybenzyl)-1H-pyrroles, a novel class of anti-HIV-1 reverse transcriptase inhibitors. Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS (Elsevier Science Limited:Oxford Fulfillment Center, PO Box 800, Kidlington Oxford OX5 1DX United Kingdom:011 44 1865 843000, 011 44 1865 843699, EMAIL: asianfo@elsevier.com, tcb@elsevier.co.UK, INTERNET: http://www.elsevier.com, http://www.elsevier.com/locate/shpsa/, Fax: 011 44 1865 843010) pp. 1931-1936 - issn: 0960-894X - wos: WOS:A1997XP63900026 (12) - scopus: 2-s2.0-0030804024 (11)
11573/245525 - 1997 -
Antifungal estrogen-like imidazoles. Synthesis and antifungal activities of thienyl and 1H-pyrrolyl derivatives of 1-aryl-2-(1H-imidazol-1-yl)ethane. Di Santo, Roberto; Costi, Roberta; Artico, Marino - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 143-149 - issn: 0223-5234 - wos: (0) - scopus: (0)
11573/122334 - 1996 -
Molecular Modeling of Azole Antifungal Agents Active.Againts Candida Albicans.I: a CoMFA Study. Artico, Marino; Costi, Roberta; Di Santo, Roberto; Ragno, Rino - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 1227-1235 - issn: 0022-2623 - wos: WOS:A1996UA57700006 (59) - scopus: 2-s2.0-13344282738 (66)
11573/194607 - 1996 -
Aryl-(1-benzenesulfonyl-1H-pyrrol-3yl)-carbinols: a new class of non-nucleoside inhibitors of HIV-1 RT. Di Santo, Roberto; Costi, Roberta - 04a Atto di comunicazione a congresso
book: XIII Convegno Nazionale Divisione di Chimica Farmaceutica SCI - ()
11573/242453 - 1996 -
Novel pyrrole-annulated heterocyclic systems. Synthesis of 10H-pyrrolo[1,2-b][1,2,6]benzothiadiazocin-11(12H)-one 5,5-dioxide. Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: JOURNAL OF HETEROCYCLIC CHEMISTRY (Hetero Corporation:PO Box 170:Provo, UT 84603:(801)400-7373, EMAIL: jhetchem@yahoo.com, Fax: (801)356-7373) pp. 2019-2023 - issn: 0022-152X - wos: WOS:A1996WE32000073 (5) - scopus: 2-s2.0-2742517067 (8)
11573/246926 - 1996 -
Synthesis of Pyrrolo[3,4-c][1]benzazepine-4,10(2H,5H)-dione, a Model System Useful for the Design of 11-Oxosibiromycinone Analogues. Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: SYNTHETIC COMMUNICATIONS (New York, NY : Taylor & Francis
New York, NY: Marcel Dekker Incorporated) pp. 1839-1847 - issn: 0039-7911 - wos: (0) - scopus: 2-s2.0-0029952695 (13)
11573/244100 - 1995 -
Antifungal Agents. 9. 3-Aryl-4-[a-(1H-imidazol-1-yl)arylmethyl]pyrroles: A New Class of Potent Anti-Candida Agents. Artico, Marco; Di Santo, Roberto; Costi, Roberta; Simonetti, Giovanna - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 4223-4233 - issn: 0022-2623 - wos: WOS:A1995TA40700011 (45) - scopus: 2-s2.0-0028791168 (48)
11573/255643 - 1995 -
4-Substituted 2-phenyl- and 2-phenyl-3-aryl pyrroles by reaction of tosylbenzyl isocyanide (TosBIC) with Michael acceptors. Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: SYNTHETIC COMMUNICATIONS (New York, NY : Taylor & Francis
New York, NY: Marcel Dekker Incorporated) pp. 795-802 - issn: 0039-7911 - wos: (0) - scopus: 2-s2.0-0028799586 (12)
11573/44023 - 1995 -
Novel Heterocyclic Systems. Synthesis of 10H-Pyrrolo[1,2-b][1,2,5]benzothiadiazocine 5,5-Dioxide and Related Derivatives. Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: JOURNAL OF HETEROCYCLIC CHEMISTRY (Hetero Corporation:PO Box 170:Provo, UT 84603:(801)400-7373, EMAIL: jhetchem@yahoo.com, Fax: (801)356-7373) pp. 1779-1782 - issn: 0022-152X - wos: WOS:A1995TQ34800019 (6) - scopus: 2-s2.0-84993876560 (8)
11573/44025 - 1995 -
Simple Synthetic Approach to Arylacetic NSAIAs via TosMIC Procedure. Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: SYNTHETIC COMMUNICATIONS (New York, NY : Taylor & Francis
New York, NY: Marcel Dekker Incorporated) pp. 787-793 - issn: 0039-7911 - wos: (0) - scopus: 2-s2.0-0028837973 (5)
11573/253762 - 1994 -
ANTIFUNGAL AGENTS .8. SYNTHESIS AND ANTIFUNGAL ACTIVITIES OF BIPYRRYL ANALOGS OF BIFONAZOLE Di Santo, Roberto; Costi, Roberta; Simonetti, Giovanna - 01a Articolo in rivista
paper: IL FARMACO (Attuale:ELSEVIER SCIENCE SA, PO BOX 564, LAUSANNE, SWITZERLAND, 1001
Societa Chimica Italiana:Viale Liegi 48, 00198 Rome Italy:011 39 06 8549691, EMAIL: soc.chim.it@agora.stm.it, Fax: 011 39 06 8548734) pp. 229-236 - issn: 0014-827X - wos: WOS:A1994NN69600001 (8) - scopus: 2-s2.0-0028361653 (12)
11573/44027 - 1994 -
Synthesis of Novel HEPT Analogues with Anti-HIV-1 Activity. Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: MEDICINAL CHEMISTRY RESEARCH (Birkhauser Boston Incorporated:c/o Springer Verlag, PO Box 2485:Secaucus, NJ 07096:(800)777-4643, (973)348-4033, Fax: (973)348-4505) pp. 554-562 - issn: 1054-2523 - wos: (0) - scopus: (0)
11573/247026 - 1993 -
Antifungal Agents. 4. Synthesis of neo-Isopyrrolnitrin and other 3-Aryl-4-nitro-1H-pyrroles via TosMIC. Di Santo, Roberto; Costi, Roberta; Mai, Antonello; Simonetti, Giovanna - 01a Articolo in rivista
paper: MEDICINAL CHEMISTRY RESEARCH (Birkhauser Boston Incorporated:c/o Springer Verlag, PO Box 2485:Secaucus, NJ 07096:(800)777-4643, (973)348-4033, Fax: (973)348-4505) pp. 192-199 - issn: 1054-2523 - wos: (0) - scopus: (0)
11573/44268 - 1993 -
Antifungal Agents. 5. Chloro and Amino Derivatives of 1,2-Diaryl-1-(1H-imidazol-1-yl)ethane with Potent Antifungal Activities. Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY (Editions Scientifique & Medical Elsevier:23 Rue Linois, F 75724 Paris Cedex 15 France:011 33 1 71724646, INTERNET: http://www.elsevier.fr, Fax: 011 33 1 71724664) pp. 715-720 - issn: 0223-5234 - wos: WOS:A1993MC71600008 (9) - scopus: 2-s2.0-0027449161 (9)
11573/470052 - 1993 -
Antifungal agents. III. Naphthyl and thienyl derivatives of 1H-imidazol-1-yl-4-phenyl-1H-pyrrol-3-ylmethane. Di Santo, Roberto; Costi, Roberta; Simonetti, Giovanna; Artico, Marco - 01a Articolo in rivista
paper: IL FARMACO (Attuale:ELSEVIER SCIENCE SA, PO BOX 564, LAUSANNE, SWITZERLAND, 1001
Societa Chimica Italiana:Viale Liegi 48, 00198 Rome Italy:011 39 06 8549691, EMAIL: soc.chim.it@agora.stm.it, Fax: 011 39 06 8548734) pp. 725-736 - issn: 0014-827X - wos: WOS:A1993LQ31800002 (8) - scopus: 2-s2.0-0027170720 (7)
11573/47093 - 1993 -
Research on Nitrogen Containing Heterocyclic Compounds. XX. Synthesis of 8H-Imidazo[5,1-c]pyrrolo[1,2-a][1,4]benzodiazepine and its 6-Derivatives. Di Santo, Roberto; Costi, Roberta - 01a Articolo in rivista
paper: JOURNAL OF HETEROCYCLIC CHEMISTRY (Hetero Corporation:PO Box 170:Provo, UT 84603:(801)400-7373, EMAIL: jhetchem@yahoo.com, Fax: (801)356-7373) pp. 749-753 - issn: 0022-152X - wos: WOS:A1993LL38300025 (8) - scopus: 2-s2.0-0343779409 (9)
11573/47097 - 1992 -
Novel In Vitro Highly Active Antifungal Agents With Pyrrole and Imidazole Moieties. Di Santo, Roberto; Artico, Marco; Costi, Roberta; Simonetti, Giovanna - 01a Articolo in rivista
paper: MEDICINAL CHEMISTRY RESEARCH (Birkhauser Boston Incorporated:c/o Springer Verlag, PO Box 2485:Secaucus, NJ 07096:(800)777-4643, (973)348-4033, Fax: (973)348-4505) pp. 148-153 - issn: 1054-2523 - wos: (0) - scopus: (0)
11573/47098 - 1992 -
Researches on Antibacterial and Antifungal Agents. XV. 3-Aryl-4-[a-(1H-imidazol-1-yl)benzyl]pyrroles with Potent Antifungal Activity. Di Santo, Roberto; Costi, Roberta; Simonetti, Giovanna; Artico, Marco - 01a Articolo in rivista
paper: EUROPEAN BULLETIN OF DRUG RESEARCH (Firenze: Europharma 2000.) pp. 12-17 - issn: 1122-2441 - wos: (0) - scopus: (0)