11573/1714867 - 2024 -
New Thiazolidine-4-One Derivatives as SARS-CoV-2 Main Protease Inhibitors Messore, A; Malune, P; Patacchini, E; Madia, Vn; Ialongo, D; Arpacioglu, M; Albano, A; Ruggieri, G; Saccoliti, F; Scipione, L; Tramontano, E; Canton, S; Corona, A; Scognamiglio, S; Paulis, A; Suleiman, M; Al-Maqtari, Hm; Abid, Fma; Kawsar, Sma; Sankaranarayanan, M; Di Santo, R; Esposito, F; Costi, R. - 01a Articolo in rivista
rivista: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. 650-673 - issn: 1424-8247 - wos: WOS:001231217500001 (1) - scopus: 2-s2.0-85194037072 (0)
11573/1697149 - 2023 -
New blood-brain-barrier permeable compounds as Naegleria Fowleri CYP51 inhibitors. Arpacioglu, M.; Madia, V. N.; Ialongo, D.; Patacchini, E.; Messore, A.; Tudino, V.; Sharma, V.; Nguyen, J.; Debnath, A.; Podust, L.; Palenca, I.; Basili Franzin, S.; Seguella, L.; Esposito, G.; Petrucci, R.; Di Matteo, P.; Bortolami, M.; Scipione, L.; Costi, R.; Di Santo, R. - 04f Poster
congresso: XXVIII edition of the National Meeting on Medicinal Chemistry (Chieti; Italy)
libro: XXVIII edition of the National Meeting on Medicinal Chemistry - ()
11573/1697156 - 2023 -
Novel nsp13 inhibitors capable of blocking viral replication of SARS-CoV-2. Arpacioglu, M.; Madia, V. N.; Messore, A.; Patacchini, E.; Ialongo, D.; Tudino, V.; Scipione, L.; Corona, A.; Esposito, F.; Artico, M.; Amatore, D.; Faggioni, G.; De Santis, R.; Lista, F.; Tramontano, E.; Costi, R.; Di Santo, R. - 04f Poster
congresso: ESMEC 2023 - European School of Medicinal Chemistry – 42nd Edition (Urbino; Italy)
libro: ESMEC 2023 - European School of Medicinal Chemistry – 42nd Edition - ()
11573/1697165 - 2023 -
Aminopyrimidine derivatives as new protein kinase inhibitors endowed with anticancer activity. Ialongo, D.; Madia, V. N.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Scarpa, S.; Rauh, D; Di Santo, R.; Costi, R. - 04f Poster
congresso: 10th EFMC Young Medicinal Chemists' Symposium (Zagreb; Croatia.)
libro: 10th EFMC Young Medicinal Chemists' Symposium - ()
11573/1697174 - 2023 -
Pyrimidine-based compounds as new promising protein kinase inhibitors for cancer treatment. Ialongo, D.; Madia, V. N.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Scarpa, S.; Rauh, D; Di Santo, R.; Costi, R. - 04f Poster
congresso: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry (Zagreb; Croatia.)
libro: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry - ()
11573/1697175 - 2023 -
Diketo acid heterocyclic derivatives as new SARS-CoV-2 nsp13 inhibitors blocking viral replication. Ialongo, D.; Madia, V. N.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Tudino, V.; Scipione, L.; Corona, A.; Esposito, F.; Artico, M.; Amatore, D.; Faggioni, G.; De Santis, R.; Lista, F.; Tramontano, E.; Costi, R.; Di Santo, R. - 04f Poster
congresso: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry (Zagreb; Croatia.)
libro: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry - ()
11573/1697147 - 2023 -
Identification of novel aminopyrimidine derivatives as protein kinase inhibitors blocking cell growth. Ialongo, Davide; Madia, Valentina Noemi; Messore, Antonella; Patacchini, Elisa; Arpacioglu, Merve; Scipione, Luigi; Scarpa, S.; Rauh, D.; Di Santo, R.; Costi, R. - 04f Poster
congresso: XXVIII edition of the National Meeting on Medicinal Chemistry (Chieti; Italy)
libro: XXVIII edition of the National Meeting on Medicinal Chemistry - ()
11573/1697162 - 2023 -
New diketo acid derivatives as dual SARS-CoV-2 nsp13 inhibitors active against viral replication. Ialongo, Davide; Madia, Valentina Noemi; Messore, Antonella; Patacchini, Elisa; Arpacioglu, Merve; Tudino, Valeria; Scipione, Luigi; Corona, Angela; Esposito, Francesca; Artico, Marco; Amatore, Donatella; Faggioni, Giovanni; De Santis, Riccardo; Lista, Florigio; Tramontano, Enzo; Costi, Roberta; Di Santo, Roberto - 04f Poster
congresso: 10th EFMC Young Medicinal Chemists' Symposium (Zagreb; Croatia.)
libro: 10th EFMC Young Medicinal Chemists' Symposium - ()
11573/1684012 - 2023 -
Synergistic Effects of Caffeine in Combination with Conventional Drugs: Perspectives of a Drug That Never Ages Ialongo, Davide; Tudino, Valeria; Arpacioglu, Merve; Messore, Antonella; Patacchini, Elisa; Costi, Roberta; Di Santo, Roberto; Madia, Valentina Noemi - 01g Articolo di rassegna (Review)
rivista: PHARMACEUTICALS (Basel : MDPI, Molecular Diversity Preservation International, 2004-) pp. 1-23 - issn: 1424-8247 - wos: WOS:000997931100001 (4) - scopus: 2-s2.0-85160675541 (9)
11573/1697142 - 2023 -
Discovery of new small molecules as anti-SARS-CoV-2 agents inhibiting ACE2-spike binding. Madia, V. N.; Ialongo, D.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Di Santo, R.; Costi, R. - 04f Poster
congresso: XXVIII edition of the National Meeting on Medicinal Chemistry (Chieti; Italy)
libro: XXVIII edition of the National Meeting on Medicinal Chemistry - ()
11573/1697168 - 2023 -
Dual HIV-1 integrase catalytic site and integrase-RNA interaction inhibitors. Madia, V. N.; Ialongo, D.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Kvaratskhelia, M.; Di Santo, R.; Costi, R. - 04f Poster
congresso: 10th EFMC Young Medicinal Chemists' Symposium (Zagreb; Croatia.)
libro: 10th EFMC Young Medicinal Chemists' Symposium - ()
11573/1697179 - 2023 -
Quinolinonyl derivatives as dual inhibitors of the HIV-1 integrase catalytic site and integrase-RNA interactions. Madia, V. N.; Ialongo, D.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Kvaratskhelia, M.; Di Santo, R.; Costi, R. - 04f Poster
congresso: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry (Zagreb; Croatia.)
libro: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry - ()
11573/1697181 - 2023 -
Design and synthesis of brain permeable anti-Naegleria fowleri agents targeting CYP51 for primary amoebic meningoencephalitis treatment. Madia, V. N.; Ialongo, D.; Messore, A.; Patacchini, E.; Arpacioglu, M.; Tudino, V.; Sharma, V.; Nguyen, J.; Debnath, A.; Podust, L.; Palenca, I.; Basili Franzin, S.; Seguella, L.; Esposito, G.; Petrucci, R.; Di Matteo, P.; Bortolami, M.; Scipione, L.; Costi, R.; Di Santo, R. - 04f Poster
congresso: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry (Zagreb; Croatia.)
libro: IX EFMC International Symposium on Advances in Synthetic and Medicinal Chemistry - ()
11573/1697153 - 2023 -
Small molecule derivatives as dual inhibitors of SARS-CoV-2 nsp13 blocking viral replication. Madia, V. N.; Ialongo, D.; Patacchini, E.; Arpacioglu, M.; Messore, A.; Tramontano, E.; De Santis, R.; Lista, F.; Costi, R.; Di Santo, R. - 04f Poster
congresso: 3rd Synthesis in Drug Discovery and Development (Virtual meeting)
libro: 3rd Synthesis in Drug Discovery and Development - ()
11573/1697146 - 2023 -
Discovery of quinolinonyl derivatives as anti-HIV-1 inhibitors endowed with an innovative mechanism of action. Madia, Valentina Noemi; Ialongo, Davide; Messore, Antonella; Patacchini, Elisa; Arpacioglu, Merve; Scipione, Luigi; Di Santo, Roberto; And Costi, Roberta. - 04f Poster
congresso: XXVIII edition of the National Meeting on Medicinal Chemistry (Chieti; Italy)
libro: XXVIII edition of the National Meeting on Medicinal Chemistry - ()
11573/1697172 - 2023 -
Miconazole-like compounds as brain permeable anti-Naegleria Fowleri agents targeting CYP51. Madia, Valentina Noemi; Ialongo, Davide; Patacchini, Elisa; Messore, Antonella; Arpacioglu, Merve; Tudino, V.; Sharma, V.; Nguyen, J.; Debnath, A.; Podust, L.; Palenca, I.; Basili Franzin, S.; Seguella, L.; Esposito, G.; Petrucci, R.; Di Matteo, P.; Bortolami, M.; Scipione, L.; Costi, Roberta; Di Santo, Roberto. - 04f Poster
congresso: 10th EFMC Young Medicinal Chemists' Symposium (Zagreb; Croatia.)
libro: 10th EFMC Young Medicinal Chemists' Symposium - ()
11573/1697140 - 2023 -
Design and synthesis of tetrahydro-β-carbolines derivatives as PDIA inhibitors. Messore, A.; Madia, V. N.; Ialongo, D.; Patacchini, E.; Arpacioglu, M.; Scipione, L.; Altieri, F.; Paglia, G.; Meschiari, G.; Di Santo, R.; Costi, R. - 04f Poster
congresso: XXVIII edition of the National Meeting on Medicinal Chemistry (Chieti; Italy)
libro: XXVIII edition of the National Meeting on Medicinal Chemistry - ()