GIULIA STAZI PhD Graduate PhD program:: XXX Thesis title: From Epigenetics to Lipid Metabolism: different approaches to fight cancer Research products 11573/870518 - 2016 - LSD1 inhibitors: a patent review (2010-2015) (01a Articolo in rivista)STAZI, GIULIA; ZWERGEL, CLEMENS; VALENTE, SERGIO; MAI, ANTONELLO11573/856751 - 2016 - Discovery of a novel inhibitor of histone lysine-specific demethylase 1A (KDM1A/LSD1) as orally active antitumor agent (01a Articolo in rivista)MAI, ANTONELLO; MARROCCO, BIAGINA; STAZI, GIULIA; VALENTE, SERGIO11573/955887 - 2017 - Novel coumarin- and quinolinone-based polycycles as cell division cycle 25-A and -C phosphatases inhibitors induce proliferation arrest and apoptosis in cancer cells (01a Articolo in rivista)ZWERGEL, CLEMENS; STAZI, GIULIA; MORI, MATTIA; PATSILINAKOS, ALEXANDROS; MAI, ANTONELLO; BOTTA, BRUNO; RAGNO, RINO; KIRSCH, GILBERT; VALENTE, SERGIO11573/1017602 - 2017 - EZH2 inhibitors: a patent review (2014-2016) (01a Articolo in rivista)STAZI, GIULIA; ZWERGEL, CLEMENS; MAI, ANTONELLO; VALENTE, SERGIO11573/1070791 - 2018 - From epigenetics to lipid metabolism: different approaches to fight cancer (07a Tesi di Dottorato)STAZI, GIULIA11573/1017610 - 2017 - The histone methyltransferase EZH2 as a druggable target in SHH medulloblastoma cancer stem cells (01a Articolo in rivista)MIELE, EVELINA; VALENTE, SERGIO; ALFANO, VINCENZO; SILVANO, MARIANNA; MELLINI, PAOLO; MARROCCO, BIAGINA; PO, AGNESE; BESHARAT, ZEIN MERSINI; CATANZARO, GIUSEPPINA; BATTAGLIA, GIUSEPPE; ABBALLE, LUANA; ZWERGEL, CLEMENS; STAZI, GIULIA; TAFANI, MARCO; MAI, ANTONELLO; FERRETTI, ELISABETTA11573/1147949 - 2018 - A quinoline-based DNA methyltransferase inhibitor as a possible adjuvant in osteosarcoma therapy (01a Articolo in rivista)VALENTE, SERGIO; ZWERGEL, CLEMENS; MAZZONE, ROBERTA; STAZI, GIULIA; MAI, ANTONELLO11573/1147235 - 2018 - Trends of LSD1 inhibitors in viral infections (01a Articolo in rivista)ZWERGEL, CLEMENS; STAZI, GIULIA; MAI, ANTONELLO; VALENTE, SERGIO11573/1147233 - 2018 - Pyrazole-based inhibitors of enhancer of zeste homologue 2 induce apoptosis and autophagy in cancer cells (01a Articolo in rivista)MELLINI, PAOLO; MARROCCO, BIAGINA; POLLETTA, LUCIA; CARNEVALE, ILARIA; SALADINI, SERENA; STAZI, GIULIA; ZWERGEL, CLEMENS; FERRETTI, ELISABETTA; TAFANI, MARCO; VALENTE, SERGIO; MAI, ANTONELLO11573/779609 - 2015 - Pyrrole- and indole-containing tranylcypromine derivatives as novel lysine-specific demethylase 1 inhibitors active on cancer cells. (01a Articolo in rivista)VALENTE, SERGIO; ROTILI, DANTE; STAZI, GIULIA; LUCIDI, ALESSIA; MAI, ANTONELLO11573/1208206 - 2019 - Development of alkyl glycerone phosphate synthase inhibitors: Structure-activity relationship and effects on ether lipids and epithelial-mesenchymal transition in cancer cells (01a Articolo in rivista)STAZI, GIULIA; BATTISTELLI, CECILIA; MAZZONE, ROBERTA; MARROCCO, BIAGINA; ZWERGEL, CLEMENS; ANTONINI, LORENZO; PATSILINAKOS, ALEXANDROS; RAGNO, RINO; CIOGLI, ALESSIA; FABRIZI, GIANCARLO; STRIPPOLI, RAFFAELE; MARCHETTI, ALESSANDRA; TRIPODI, MARCO; MATTEVI, ANDREA; MAI, ANTONELLO; VALENTE, SERGIO11573/1275490 - 2019 - Epigenetic Pharmacology in Regenerative Medicine (Epi-Drugs) (02a Capitolo o Articolo)STAZI, GIULIA; ZWERGEL, CLEMENS; VALENTE, SERGIO; MAI, ANTONELLO11573/1265927 - 2019 - Identification of a novel quinoline-based DNA demethylating compound highly potent in cancer cells (01a Articolo in rivista)ZWERGEL, CLEMENS; BATTISTELLI, CECILIA; STAZI, GIULIA; MAZZONE, ROBERTA; FIORAVANTI, ROSSELLA; STRIPPOLI, RAFFAELE; TRIPODI, MARCO; MAI, ANTONELLO; VALENTE, SERGIO11573/1202973 - 2018 - Application of small epigenetic modulators in pediatric medulloblastoma (01a Articolo in rivista)ZWERGEL, CLEMENS; ROMANELLI, ANNALISA; STAZI, GIULIA; BESHARAT, ZEIN MERSINI; CATANZARO, GIUSEPPINA; TAFANI, MARCO; VALENTE, SERGIO; MAI, ANTONELLO11573/1382317 - 2019 - Lysine methyltransferases and their inhibitors (02a Capitolo o Articolo)STAZI, GIULIA; ZWERGEL, CLEMENS; VALENTE, SERGIO11573/1390392 - 2020 - Altered mitochondrial function in cells carrying a premutation or unmethylated full mutation of the FMR1 gene (01a Articolo in rivista)RAGNO, RINO; STAZI, GIULIA; VALENTE, SERGIO; MAI, ANTONELLO11573/1394955 - 2020 - Design of first-in-class dual EZH2/HDAC inhibitor: biochemical activity and biological evaluation in cancer cells (01a Articolo in rivista)ROMANELLI, ANNALISA; STAZI, GIULIA; FIORAVANTI, ROSSELLA; ZWERGEL, CLEMENS; DI BELLO, ELISABETTA; BATTISTELLI, CECILIA; STRIPPOLI, RAFFAELE; TRIPODI, MARCO; MAI, ANTONELLO; VALENTE, SERGIO11573/1339079 - 2019 - Dissecting the role of novel EZH2 inhibitors in primary glioblastoma cell cultures: effects on proliferation, epithelial-mesenchymal transition, migration, and on the pro-inflammatory phenotype (01a Articolo in rivista)STAZI, GIULIA; TAGLIERI, LUDOVICA; NICOLAI, ALICE; ROMANELLI, ANNALISA; FIORAVANTI, ROSSELLA; MORRONE, STEFANIA; SABATINO, MANUELA; RAGNO, RINO; TAURONE, SAMANTA; NEBBIOSO, MARCELLA; CARLETTI, RAFFAELLA; ARTICO, MARCO; VALENTE, SERGIO; SCARPA, SUSANNA; MAI, ANTONELLO11573/1174048 - 2018 - Six years (2012-2018) of researches on catalytic EZH2 inhibitors: the boom of the 2-pyridone compounds (01a Articolo in rivista)FIORAVANTI, ROSSELLA; STAZI, GIULIA; ZWERGEL, CLEMENS; VALENTE, SERGIO; MAI, ANTONELLO