11573/1771634 - 2026 -
(S,S)-5-Chloro-3-((3,5-dimethylphenyl)sulfonyl)-N-(1-oxo-1-((1-(pyridin-4-yl)ethyl)amino)propan-2-yl)-1H-indole-2-carboxamide, a New Dishevelled 1 and P-glycoprotein Dual Inhibitor as Anticancer Agent Puxeddu, Michela; Cui, Zeyu; Colla, Claudia; Nalli, Marianna; Manetto, Simone; Ciogli, Alessia; Cuřínová, Petra; Bufano, Marianna; Toto, Angelo; Gianni, Stefano; Pastore, Arianna; Stornaiuolo, Mariano; Baldini, Enke; Ulisse, Salvatore; Kopecka, Joanna; Riganti, Chiara; Bigogno, Chiara; Dondio, Giulio; Liu, Te; Coluccia, Antonio; Regina, Giuseppe La; Silvestri, Romano - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 14667-14690 - issn: 0022-2623 - wos: WOS:001792658700001 (0) - scopus: 2-s2.0-105043709893 (0)
11573/1762833 - 2026 -
4-(5-Chloro-3-(3,4,5-trimethoxybenzoyl)-1h-indol-1-yl) benzenesulfonamide. A novel polypharmacology agent to target carbonic anhydrase IX and XII with Improved selectivity, wnt/β-catenin signaling pathway, and p-glycoprotein Puxeddu, Michela; Bordone, Rosa; Colla, Claudia; Rotili, Gabriele; Coluccia, Antonio; Sciò, Pietro; Cuřínová, Petra; Nocentini, Alessio; Supuran, Claudiu T.; Filiberti, Serena; Turati, Marta; Ronca, Roberto; Kopecka, Joanna; Riganti, Chiara; Jimenez, Lucia; Link, Wolfgang; Bigogno, Chiara; Dondio, Giulio; Barba, Martina; Canettieri, Gianluca; Silvestri, Romano; La Regina, Giuseppe - 01a Articolo in rivista
paper: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. 1-19 - issn: 1860-7179 - wos: WOS:001705396000005 (0) - scopus: 2-s2.0-105031001806 (0)
11573/1748729 - 2025 -
Ferroptosis Induction by a New Pyrrole Derivative in Triple Negative Breast Cancer and Colorectal Cancer Masci, Domiziana; Ling, Lele; Yang, Lian; Puxeddu, Michela; Colla, Claudia; Coluccia, Antonio; Santelli, Martina; Scio', Pietro; Cuřínová, Petra; Ansari, Mohammad Salik Zeya; Naro, Chiara; Sette, Claudio; Jimenez, Lucia; Link, Wolfgang; Bigogno, Chiara; Dondio, Giulio; Hamel, Ernest; Liu, Te; Silvestri, Romano; La Regina, Giuseppe - 01a Articolo in rivista
paper: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 17840-17858 - issn: 0022-2623 - wos: WOS:001547406200001 (4) - scopus: 2-s2.0-105014469330 (3)
11573/1748751 - 2025 -
Microwave-assisted synthesis of tubulin assembly inhibitors as anticancer agents by aryl ring reversal and conjunctive approach Masci, Domiziana; Puxeddu, Michela; Colla, Claudia; Coluccia, Antonio; Santelli, Martina; Scio', Pietro; Mariotto, Elena; Viola, Giampietro; Hamel, Ernest; Lerose, Rosa; Mazzoccoli, Carmela; Silvestri, Romano; La Regina, Giuseppe - 01a Articolo in rivista
paper: RSC MEDICINAL CHEMISTRY (Cambridge: Royal Society of Chemistry, 2020-) pp. - - issn: 2632-8682 - wos: WOS:001538325300001 (2) - scopus: 2-s2.0-105018766780 (2)