11573/1744255 - 2025 -
Beyond Antibodies: Reinventing Alzheimer’s Treatment for the Next Decade Garbo, Sabrina; Raucci, Alessia; Zwergel, Clemens; Handzlik, Jadwiga; Battistelli, Cecilia - 01m Editorial/Introduzione in rivista
rivista: DRUG DISCOVERY TODAY (Elsevier Science Limited Trends Journals:PO Box 331, Haywards Heath RH16 3FG United Kingdom:011 44 1444 475651, EMAIL: ct.subs@rbi.co.uk, Fax: 011 44 1444 445423) pp. - - issn: 1359-6446 - wos: (0) - scopus: (0)
11573/1735469 - 2025 -
Procognitive Potential of Neuroprotective Triazine 5-HT6 Receptor Antagonists Tested on Chronic Activity In Vivo in Rats: Computer-Aided Insight into the Role of Chalcogen-Differences on the Pharmacological Profile Jastrzębska-Więsek, Magdalena; Garbo, Sabrina; Cios, Agnieszka; Wilczyńska-Zawal, Natalia; Partyka, Anna; Honkisz-Orzechowska, Ewelina; Żesławska, Ewa; Handzlik, Jarosław; Mordyl, Barbara; Głuch-Lutwin, Monika; Raucci, Alessia; Hittinger, Marius; Starek, Małgorzata; Dąbrowska, Monika; Nitek, Wojciech; Karcz, Tadeusz; Skórkowska, Alicja; Gdula-Argasińska, Joanna; Czarnota-Łydka, Kinga; Pyka, Patryk; Szymańska, Ewa; Kucwaj-Brysz, Katarzyna; Zwergel, Clemens; Wesołowska, Anna; Battistelli, Cecilia; Handzlik, Jadwiga - 01a Articolo in rivista
rivista: ACS CHEMICAL NEUROSCIENCE (Washington, D.C. : American Chemical Society) pp. 1190-1209 - issn: 1948-7193 - wos: WOS:001436003400001 (0) - scopus: 2-s2.0-86000144563 (1)
11573/1746317 - 2025 -
Design of Benzyl-triazolopyrimidine-Based NADPH Oxidase Inhibitors Leads to the Discovery of a Potent Dual Covalent NOX2/MAOB Inhibitor Noce, Beatrice; Marchese, Sara; Massari, Marta; Lambona, Chiara; Reis, Joana; Fiorentino, Francesco; Raucci, Alessia; Fioravanti, Rossella; Castelôa, Mariana; Mormino, Alessandro; Garofalo, Stefano; Limatola, Cristina; Basile, Lorenzo; Gottinger, Andrea; Binda, Claudia; Mattevi, Andrea; Mai, Antonello; Valente, Sergio - 01a Articolo in rivista
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington DC : ACS Publications) pp. 6292-6311 - issn: 1520-4804 - wos: WOS:001437973800001 (1) - scopus: 2-s2.0-86000188474 (1)
11573/1742842 - 2025 -
Advancements in hydrazide-based HDAC inhibitors. A review of recent developments and therapeutic potential Raucci, Alessia; Zwergel, Clemens; Valente, Sergio; Mai, Antonello - 01g Articolo di rassegna (Review)
rivista: JOURNAL OF MEDICINAL CHEMISTRY (Washington, DC: American Chemical Society) pp. 14171-14194 - issn: 0022-2623 - wos: WOS:001525998800001 (3) - scopus: 2-s2.0-105010245358 (3)
11573/1710159 - 2024 -
Uracil- and Pyridine-containing HDAC inhibitors displayed cytotoxicity in colorectal and glioblastoma cancer stem cells Fiorentino, Francesco; Fabbrizi, Emanuele; Raucci, Alessia; Noce, Beatrice; Fioravanti, Rossella; Valente, Sergio; Paolini, Chantal; De Maria, Ruggero; Steinkühler, Christian; Gallinari, Paola; Rotili, Dante; Mai, Antonello - 01a Articolo in rivista
rivista: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. - - issn: 1860-7187 - wos: WOS:001214621100001 (8) - scopus: 2-s2.0-85191719139 (9)
11573/1716603 - 2024 -
Unlocking the potential of higher-molecular-weight 5-HT7R ligands. Synthesis, affinity, and ADMET examination Pyka, Patryk; Garbo, Sabrina; Murzyn, Aleksandra; Satała, Grzegorz; Janusz, Artur; Górka, Michał; Pietruś, Wojciech; Mituła, Filip; Popiel, Delfina; Wieczorek, Maciej; Palmisano, Biagio; Raucci, Alessia; Bojarski, Andrzej J.; Zwergel, Clemens; Szymańska, Ewa; Kucwaj-Brysz, Katarzyna; Battistelli, Cecilia; Handzlik, Jadwiga; Podlewska, Sabina - 01a Articolo in rivista
rivista: BIOORGANIC CHEMISTRY (Academic Press Incorporated:6277 Sea Harbor Drive:Orlando, FL 32887:(800)543-9534, (407)345-4100, EMAIL: ap@acad.com, INTERNET: http://www.idealibrary.com, Fax: (407)352-3445) pp. 1-20 - issn: 0045-2068 - wos: WOS:001284368500001 (2) - scopus: 2-s2.0-85199923673 (2)
11573/1710160 - 2024 -
Heterocycles-containing HDAC inhibitors active in cancer. An overview of the last fifteen years Raucci, Alessia; Castiello, Carola; Mai, Antonello; Zwergel, Clemens; Valente, Sergio - 01g Articolo di rassegna (Review)
rivista: CHEMMEDCHEM (Weinheim : Wiley-VCH-Verl..) pp. 1-53 - issn: 1860-7179 - wos: WOS:001300014900001 (3) - scopus: 2-s2.0-85202594031 (6)